bw 245c has been researched along with dinoprostone in 17 studies
Studies (bw 245c) | Trials (bw 245c) | Recent Studies (post-2010) (bw 245c) | Studies (dinoprostone) | Trials (dinoprostone) | Recent Studies (post-2010) (dinoprostone) |
---|---|---|---|---|---|
96 | 3 | 10 | 29,105 | 1,346 | 6,357 |
Protein | Taxonomy | bw 245c (IC50) | dinoprostone (IC50) |
---|---|---|---|
Prostaglandin E2 receptor EP1 subtype | Homo sapiens (human) | 0.0155 | |
Prostaglandin E2 receptor EP4 subtype | Homo sapiens (human) | 0.0031 | |
Prostaglandin E2 receptor EP4 subtype | Rattus norvegicus (Norway rat) | 0.0021 | |
Prostaglandin E2 receptor EP3 subtype | Homo sapiens (human) | 0.002 | |
Prostaglandin E2 receptor EP2 subtype | Homo sapiens (human) | 0.0087 | |
Prostacyclin receptor | Homo sapiens (human) | 0.26 | |
Prostaglandin E2 receptor EP2 subtype | Rattus norvegicus (Norway rat) | 0.0052 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (11.76) | 18.7374 |
1990's | 6 (35.29) | 18.2507 |
2000's | 7 (41.18) | 29.6817 |
2010's | 2 (11.76) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Abramovitz, M; Boie, Y; Metters, KM; Sawyer, N; Slipetz, DM | 1 |
Hirata, M; Kiriyama, M; Kobayashi, T; Narumiya, S; Sugimoto, Y; Ushikubi, F | 1 |
Abramovitz, M; Ford-Hutchinson, AW; Metters, KM; Wright, DH | 1 |
Ivanyi, J; Kay, JE; Kingston, AE | 1 |
Andersen, NH; Hanson, SR; Harker, LA; Tynan, SS; Wills, MT | 1 |
Lawrence, RA; Woodward, DF | 1 |
Leff, P; Lydford, SJ; McKechnie, KC | 1 |
Eguchi, N; Hayaishi, O; Ito, S; Kanaoka, Y; Minami, T; Nagata, A; Shirafuji, N; Tanaka, T; Urade, Y; Yoshida, N | 1 |
Hu, DN; McCormick, SA; Woodward, DF | 1 |
Cao, J; Kitazawa, T; Shayibuzhati, M; Tajima, T; Taneike, T | 1 |
Heinemann, A; Holzer, P; Peskar, BA; Shahbazian, A | 1 |
DeMasi, GM; Hardwick, JC; Jelson, GS; Sager, KL | 1 |
Sharif, NA; Xu, SX | 1 |
Jones, RL; Kan, KK; Ngan, MP; Rudd, JA | 1 |
de Brum-Fernandes, AJ; Gallant, MA; Miousse, MC; Parent, JL; Samadfam, R | 1 |
Devillier, P; Grassin-Delyle, S; Mechiche, H; Nazeyrollas, P; Robinet, A | 1 |
Arai, T; Awata, A; Fujino, H; Murayama, T; Okura, I; Oyama, S; Regan, JW; Yamazaki, R | 1 |
17 other study(ies) available for bw 245c and dinoprostone
Article | Year |
---|---|
Molecular cloning and characterization of the human prostanoid DP receptor.
Topics: Amino Acid Sequence; Base Sequence; Blotting, Northern; Calcium; Cells, Cultured; Cloning, Molecular; Cyclic AMP; Humans; Molecular Sequence Data; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin | 1995 |
Ligand binding specificities of the eight types and subtypes of the mouse prostanoid receptors expressed in Chinese hamster ovary cells.
Topics: Animals; CHO Cells; Cricetinae; Ligands; Mice; Prostaglandins; Receptors, Prostaglandin; Transfection | 1997 |
Characterization of the recombinant human prostanoid DP receptor and identification of L-644,698, a novel selective DP agonist.
Topics: Adenine Nucleotides; Benzoates; Binding, Competitive; Cell Line; Cyclic AMP; Dinoprostone; Guanine Nucleotides; Humans; Kinetics; Receptors, Immunologic; Receptors, Prostaglandin; Recombinant Proteins; Thiazoles; Thiazolidines; Tritium | 1998 |
The effects of prostaglandin E and I analogues on lymphocyte stimulation.
Topics: Dinoprostone; Dose-Response Relationship, Drug; Epoprostenol; Humans; Hydantoins; In Vitro Techniques; Leucine; Lymphocyte Activation; Lymphocytes; Phytohemagglutinins; Prostaglandins E; Prostaglandins E, Synthetic; Protein Biosynthesis | 1985 |
On the multiplicity of platelet prostaglandin receptors. II. The use of N-0164 for distinguishing the loci of action for PGI2, PGD2, PGE2 and hydantoin analogs.
Topics: Blood Platelets; Dinoprostone; Epoprostenol; Humans; Hydantoins; Organophosphonates; Organophosphorus Compounds; Platelet Aggregation; Prostaglandin Antagonists; Prostaglandin D2; Prostaglandins; Prostaglandins D; Prostaglandins E; Receptors, Cell Surface; Receptors, Prostaglandin; Structure-Activity Relationship | 1984 |
Identification of a single (FP) receptor associated with prostanoid-induced Ca2+ signals in Swiss 3T3 cells.
Topics: 3T3 Cells; Animals; Binding, Competitive; Calcium; Dinoprostone; Hydantoins; Mice; Prostaglandin D2; Prostaglandins F; Prostaglandins F, Synthetic; Receptors, Prostaglandin; Second Messenger Systems | 1994 |
Interaction of BW A868C, a prostanoid DP-receptor antagonist, with two receptor subtypes in the rabbit isolated saphenous vein.
Topics: Animals; Anti-Arrhythmia Agents; Biphenyl Compounds; Dinoprostone; Dose-Response Relationship, Drug; Hydantoins; Male; Potassium Chloride; Prostaglandin D2; Rabbits; Receptors, Immunologic; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP4 Subtype; Saphenous Vein | 1996 |
Lack of tactile pain (allodynia) in lipocalin-type prostaglandin D synthase-deficient mice.
Topics: Anesthesia; Animals; Bicuculline; Central Nervous System; Dinoprost; Dinoprostone; GABA Antagonists; Gene Targeting; Hydantoins; Hyperalgesia; Immunohistochemistry; Intramolecular Oxidoreductases; Lipocalins; Mice; Mice, Knockout; Molecular Sequence Data; Pain; Prostaglandin D2; Receptors, Prostaglandin | 1999 |
A functional study on prostanoid receptors involved in cultured human iridal melanocyte stimulation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Cell Count; Cells, Cultured; Cyclic AMP; Dinoprostone; Epoprostenol; Fibroblast Growth Factor 2; Humans; Hydantoins; Iris; Melanins; Melanocytes; Prostaglandin Antagonists; Prostanoic Acids; Receptors, Prostaglandin | 2001 |
In vitro pharmacological characterization of the prostanoid receptor population in the non-pregnant porcine myometrium.
Topics: Animals; Cloprostenol; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Epoprostenol; Female; Hydantoins; Iloprost; In Vitro Techniques; Muscle Contraction; Myometrium; Prostaglandin D2; Receptors, Prostaglandin; Swine | 2002 |
Differential peristaltic motor effects of prostanoid (DP, EP, IP, TP) and leukotriene receptor agonists in the guinea-pig isolated small intestine.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Alprostadil; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dinoprostone; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Female; Guinea Pigs; Hydantoins; Hydrazines; Iloprost; In Vitro Techniques; Intestine, Small; Leukotriene Antagonists; Leukotriene D4; Male; Oxazepines; Peristalsis; Prostaglandin D2; Prostaglandins A; Receptors, Leukotriene; Receptors, Prostaglandin; Xanthenes; Xanthones; Yohimbine | 2002 |
Modulation of guinea pig intrinsic cardiac neurons by prostaglandins.
Topics: Animals; Dinoprostone; Female; Ganglia, Parasympathetic; Guinea Pigs; Heart; Hydantoins; Male; Mast Cells; Membrane Potentials; Phospholipases A; Phospholipases A2; Potassium Channel Blockers; Prostaglandin D2; Receptors, Prostaglandin; Xanthenes; Xanthones | 2003 |
Pharmacological characterization and identification of EP3 prostanoid receptor binding sites in hamster uterus homogenates.
Topics: Animals; Binding Sites; Biphenyl Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cloprostenol; Cricetinae; Dinoprost; Dinoprostone; Enprostil; Epoprostenol; Fatty Acids, Unsaturated; Female; Hydantoins; Hydrazines; Iloprost; Latanoprost; Misoprostol; Prostaglandins; Prostaglandins E, Synthetic; Prostaglandins F, Synthetic; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP3 Subtype; Tritium; Uterus | 2004 |
Excitatory action of prostanoids on the ferret isolated vagus nerve preparation.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Biguanides; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Electrophysiology; Epoprostenol; Ferrets; Hydantoins; Iloprost; In Vitro Techniques; Male; Prostaglandins; Prostaglandins F, Synthetic; Serotonin; Vagus Nerve | 2004 |
Implication of prostaglandin receptors in the accumulation of osteoprotegerin in human osteoblast cultures.
Topics: Cell Line, Transformed; Cell Line, Tumor; Dinoprostone; Dose-Response Relationship, Drug; Drug Combinations; Enzyme-Linked Immunosorbent Assay; Gene Expression; Glycoproteins; Humans; Hydantoins; Osteoblasts; Osteoprotegerin; Prostaglandin-Endoperoxide Synthases; Prostaglandins F, Synthetic; Receptors, Cytoplasmic and Nuclear; Receptors, Prostaglandin; Receptors, Tumor Necrosis Factor; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2006 |
Prostanoid receptors involved in regulation of the beating rate of neonatal rat cardiomyocytes.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Animals, Newborn; Blotting, Western; Cells, Cultured; Cloprostenol; Dibenz(b,f)(1,4)oxazepine-10(11H)-carboxylic acid, 8-chloro-, 2-acetylhydrazide; Dinoprostone; Dose-Response Relationship, Drug; Epoprostenol; Hydantoins; Iloprost; Latanoprost; Myocytes, Cardiac; Prostaglandin D2; Prostaglandins F, Synthetic; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Thromboxane | 2012 |
A novel indole compound, AWT-489, inhibits prostaglandin D2-induced CD55 expression by acting on DP prostanoid receptors as an antagonist in LS174T human colon cancer cells.
Topics: Carcinogenesis; CD55 Antigens; Cell Line, Tumor; Colonic Neoplasms; Cyclic AMP; Dinoprostone; Drug Design; Gene Expression Regulation, Neoplastic; Humans; Hydantoins; Indoles; Prostaglandin D2; Receptors, Immunologic; Receptors, Prostaglandin; RNA, Messenger | 2014 |