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buparvaquone and naphthoquinones

buparvaquone has been researched along with naphthoquinones in 100 studies

Research

Studies (100)

TimeframeStudies, this research(%)All Research%
pre-19908 (8.00)18.7374
1990's32 (32.00)18.2507
2000's24 (24.00)29.6817
2010's31 (31.00)24.3611
2020's5 (5.00)2.80

Authors

AuthorsStudies
Ahmed, JS; Dobbelaere, D; Rintelen, M; Schein, E; Williams, RO1
Dolan, TT; Gisemba, F; Injairu, R; Maina, JN; Mbadi, G; Mbwiria, SK; Mulela, GH; Othieno, DA1
Kariuki, DP; Lampard, D; Lesan, AC; Linyonyi, A; Mining, SK; Ndungu, SG; Ngumi, PN; Williamson, SM; Young, AS1
Lane, VM; Zaugg, JL2
McHardy, N1
Coquerelle, TM; Dobbelaere, DA; Eichhorn, M; Kelke, C; Roditi, IJ; Williams, RO1
Kocan, AA; Mitema, ES; Mukolwe, SW; Sangiah, S; Sherban, D1
Kariuki, DP; Morzaria, SP; Mutugi, JJ; Tameno, JM; Young, AS1
Hashemi-Fesharki, R1
Motzel, SL; Wagner, JE1
de Vos, AJ; McHardy, N; Standfast, NF; Stewart, NP1
Ahmed, JS; Rintelen, M; Schein, E1
Mishra, AK; Sharma, NN1
Bhushan, C; Dhar, S; Gautam, OP; Malhotra, DV3
el Refaii, AH; McHardy, N; Michael, SA; Rae, DG1
Bansal, GC; Sharma, NN1
Bogan, JA; Kinabo, LD1
Leitch, BL; Linyonyi, A; Maritim, AC; Mbogo, SK; Mutugi, JJ; Young, AS1
Hudson, AT; McHardy, N; Randall, AW; Wekesa, LS1
Mishra, AK; Sharma, NN; Viswanathan, CB1
Gill, JS; Kwatra, MS; Sharma, KK; Singh, J1
Armson, A; Grubb, WB; Mendis, AH; Reynoldson, JA; Thompson, RC1
Raghav, PR; Singh, DK; Thakur, M; Varshney, BC1
Hagiwara, K; Ishihara, C; Iwai, H; Kurosawa, T; Tajima, M; Takahashi, K; Tsuji, M1
Kariuki, DP; Mbogo, SK; McHardy, N; Ngumi, PN1
Davis, WC; Dobbelaere, DA; Jungi, TW; Sager, H1
Davis, W; Dobbelaere, D; Eichhorn, M; Galley, Y; Glaser, I; Hagens, G1
Ahmed, JS; Shayan, P1
Croft, SL; Furtado Campos, JH; Miles, MA; Vexenat, JA1
Brown, CG; Ilhan, T; Kirvar, E; Shiels, B; Williamson, S1
Bell-Sakyi, LJ; Brown, CG; Kirvar, BE; Sparagano, O; Thomas, M; Wilkie, GM; Williamson, SM1
Bröker, BM; Fich, C; Fleischer, B; Klauenberg, U1
Brown, CG; Kirvar, E; Sparagano, O; Thomas, EM; Wilkie, GM1
Beniwal, RK; Nichani, AK; Sharma, RD1
el-Metenawy, TM1
Naziroğlu, M; Saki, CE; Sevgili, M1
Kiara, HK; McHardy, N; Muraguri, GR1
Lewis, BD; López-Rebollar, LM; Penzhorn, BL; Swan, GE1
Croft, SL; Luque-Ortega, JR; Rivas, L; Rivero-Lezcano, OM1
Jacobs, C; Kayser, O; Müller, RH1
Jacobs, C; Müller, RH1
Angelisová, P; Baumgartner, M; Horejsí, V; Langsley, G; Mooney, N; Setterblad, N; Werling, D1
Chen, ZJ; Dobbelaere, DA; Fernandez, PC; Heussler, VT; Küenzi, P; McKellar, S; Orth, K; Rottenberg, S; Schwab, R; Shiels, B; Wallach, D1
Anson, CE; Croft, SL; Davies, W; Gokhale, NH; Kendrick, HD; Padhye, SB; Powell, AK1
Dobbelaere, DA; Küenzi, P; Schneider, P1
Dessauge, F; Garcia, A; Guergnon, J; Langsley, G1
Dwivedi, SK; Gupta, AK; Kumar, S; Pal, Y1
Croft, SL; Garnier, T; Järvinen, T; Koskinen, A; Mäntylä, A; Nevalainen, T; Rautio, J; Vepsälainen, J1
Aktas, M; Dabak, DO; Dabak, M1
Croft, SL; Garnier, T; Järvinen, T; Juvonen, R; Kendrick, H; Mäntylä, A; Nevalainen, T; Rautio, J; Vepsälainen, J1
Boniphace, S; Gwamaka, M; Maselle, RM; Matovelo, JA; Mbassa, GK; Mtambo, MM1
Järvinen, T; Keski-Rahkonen, P; Mäntylä, A; Nevalainen, T; Rautio, J; Vepsälainen, J1
Bang, K; Dunne, J; Fox, A; McHardy, N; Muraguri, GR; Ndungu, SG; Ngumi, PN; Wanjohi, JM; Wesonga, D1
Magwisha, HB; Mbwambo, HA; Mfinanga, JM1
Croft, SL; Mansor, SM; Nair, NK; Navaratnam, V; Ramanathan, S; Sattar, MA; Venkatesh, G1
Brown, MB; Croft, SL; Garnier, T; Järvinen, T; Lawrence, MJ; Mäntylä, A1
Al-Gaabary, MH; Osman, SA1
Brown, M; Croft, S; Garnier, T; Järvinen, T; Lawrence, J; Mäntylä, A1
Croft, SL; Majid, MI; Mansor, SM; Nair, NK; Navaratnam, V; Ramanathan, S; Venkatesh, G1
Paşa, S; Saruhan, B1
Glass, EJ; Hulme, MJ; Jensen, K; Kaliszewska, A; Makins, GD; Paxton, E1
Croft, SL; Majid, MI; Mansor, SM; Nair, NK; Navaratnam, V; Venkatesh, G1
BenAbderazzak, S; Boumiza, A; Chaabani, MF; Darghouth, MA; Mhadhbi, M; Naouach, A1
Ahmed, JS; Beyer, D; Gerber, S; Haller, D; Kullmann, B; Mackiewicz, M; Schneider, I; Seitzer, U1
Ding, F; Guo, J; Li, LY; Li, Z; Lian, J; Song, WH; Zhang, JH; Zhang, JY; Zhu, L1
Colombo, FA; Pereira-Chioccola, VL; Reimão, JQ; Tempone, AG1
Namazi, F; Oryan, A; Razavi, M; Shahriari, R; Sharifiyazdi, H1
Aguiar, MG; Carneiro, G; Fernandes, AP; Ferreira, LA1
Greene, MI; Hattori, M; Hayashida, K; Kajino, K; Morrison, I; Sugimoto, C; Wallace, M1
Lawrence, JA; Prozesky, L; Steyl, JC; Stoltsz, WH1
Baird, M; Durrani, Z; Kinnaird, JH; Pillai, SS; Shiels, BR; Weir, W1
Ait-Si-Ali, S; Chluba, J; DeBarry, JD; Fritsch, L; Garrido, C; Lopez, T; Lu, KP; Marsolier, J; Medjkane, S; Mhadhbi, M; Perichon, M; Villoutreix, BO; Weitzman, JB; Zhou, XZ1
Awan, MM; Jamal, Q; Khan, NH; Shah, A; Sutherland, C; Wahid, S1
Aguado-Martinez, A; Arranz-Solís, D; Balmer, V; Hemphill, A; Hostettler, I; Manser, V; Müller, J; Ortega-Mora, L; Ritler, D; Winzer, P1
Ajroud, K; BenAbderrazak, S; Chaouch, M; Darghouth, MA; Mhadhbi, M1
Aguado-Martínez, A; Haynes, RK; Hemphill, A; Manser, V; Müller, J; Wong, HN1
Hillerton, JE; McDougall, S; Pegram, D1
Bartolomé, A; Checa, R; Gálvez, R; González-Fraga, JL; Marino, V; Miró, G; Montoya, A; Ortega, N1
Aguado-Martínez, A; Barrett, LK; Choi, R; Ferre, I; Hemphill, A; Hulverson, MA; Maly, DJ; McCloskey, MC; Moreno-Gonzalo, J; Müller, J; Ojo, KK; Ortega-Mora, LM; Van Voorhis, W1
Abd El-Aty, AM; Chang, BJ; Cho, SH; Jeong, JH; Kim, JS; Kim, SK; Park, JA; Shim, JH; Shin, HC; Shin, SC; Wang, Y; Zhang, D1
Choudhury, S; Gupta, KK; Shanker, D; Singh, SK; Srivastava, M; Sudan, V1
Bolás-Fernández, F; Dea-Ayuela, MA; Lalatsa, A; Mauger, M; Serrano, DR; Smith, L1
Hemphill, A; Manser, V; Müller, J1
D'Ascoli, L; Dick, L; Hemphill, A; Hizem, A; Lundström-Stadelmann, B; Ritler, D; Rufener, R; Wells, TNC1
Abdo Abubaker, H; Amin Alnour, S; Chatanga, E; Katakura, K; Mosssad, E; Nakao, R; Salim, B1
Awino, E; Nene, V; Nyagwange, J; Pelle, R; Svitek, N; Tijhaar, E1
Marsolier, J; Medjkane, S; Perichon, M; Weitzman, JB1
Guan, G; Hassan, MA; Liu, J; Luo, J; Mukhtar, MU; Rashid, M; Rashid, MI; Wang, X; Yin, H; Zhao, S1
Bou-Chacra, N; Cotrim, PC; de Araújo, GLB; Fotaki, N; Löbenberg, R; Monteiro, LM1
Bishop, RP; Dolan, RB; Dolan, TT; Odongo, DO; Sayer, PD; Skilton, RA1
Chaudhari, PR; Devarajan, PV; Maithania, HV; Mohanty, BS; Samad, A1
Gedye, K; Lawrence, KE; Pomroy, WE1
Chatanga, E; Jannot, G; Mossaad, E; Nakao, R; Salim, B; Weitzman, JB1
Adewusi, O; Adriana de Jesus, J; Auxiliadora Dea-Ayuela, M; Bolas-Fernandez, F; Dalastra Laurenti, M; Felipe Domingues Passero, L; Lalatsa, A; Serrano, DR; Statts, L1
Lehto, VP; Mondal, S; Näkki, S; Närvänen, A; Nissinen, T; Rantanen, J; Riikonen, J; Thapa, R1
Barbosa, EJ; Bou-Chacra, NA; de Araujo Eliodoro, RH; de Araujo, GLB; de Freitas, VLT; Fotaki, N; Kanashiro, E; Löbenberg, R; Monteiro, LM; Rocha, M; Sato, PK1
Dan, XG; Guan, GQ; Li, X; Liu, JL; Zhao, HX1

Reviews

1 review(s) available for buparvaquone and naphthoquinones

ArticleYear
Drug delivery systems for the topical treatment of cutaneous leishmaniasis.
    Expert opinion on drug delivery, 2012, Volume: 9, Issue:9

    Topics: Administration, Cutaneous; Aminoquinolines; Amphotericin B; Animals; Antiprotozoal Agents; Drug Delivery Systems; Humans; Imiquimod; Leishmaniasis, Cutaneous; Naphthoquinones; Paromomycin; Phosphorylcholine; Skin Absorption

2012

Trials

5 trial(s) available for buparvaquone and naphthoquinones

ArticleYear
A clinical trial of buparvaquone in the treatment of East Coast fever.
    The Veterinary record, 1992, Jun-13, Volume: 130, Issue:24

    Topics: Anaplasmosis; Animals; Antiprotozoal Agents; Cattle; Injections, Intramuscular; Kenya; Naphthoquinones; Theileria parva; Theileriasis

1992
Stage-specific activity in vitro on the Theileria infection process of serum from calves treated prophylactically with buparvaquone.
    Veterinary parasitology, 1998, Dec-31, Volume: 80, Issue:2

    Topics: Animals; Antiprotozoal Agents; Biological Assay; Cattle; Cell Line; Naphthoquinones; Theileria annulata; Theileria parva; Theileriasis; Time Factors

1998
In-vivo therapeutic efficacy trial with artemisinin derivative, buparvaquone and imidocarb dipropionate against Babesia equi infection in donkeys.
    The Journal of veterinary medical science, 2003, Volume: 65, Issue:11

    Topics: Animals; Antiprotozoal Agents; Artemisinins; Babesiosis; Blood Cell Count; Drug Therapy, Combination; Equidae; Imidocarb; India; Naphthoquinones; Sesquiterpenes; Splenectomy

2003
Clinical efficacy and plasma concentrations of two formulations of buparvaquone in cattle infected with East Coast fever (Theileria parva infection).
    Research in veterinary science, 2006, Volume: 81, Issue:1

    Topics: Animals; Antiprotozoal Agents; Area Under Curve; Cattle; Cattle Diseases; Male; Naphthoquinones; Theileriasis

2006
Clinical, haematological and therapeutic studies on tropical theileriosis in water buffaloes (Bubalus bubalis) in Egypt.
    Veterinary parasitology, 2007, May-31, Volume: 146, Issue:3-4

    Topics: Animals; Antiprotozoal Agents; Buffaloes; Cattle; Cattle Diseases; Egypt; Naphthoquinones; Theileriasis

2007

Other Studies

94 other study(ies) available for buparvaquone and naphthoquinones

ArticleYear
Effect of buparvaquone on the expression of interleukin 2 receptors in Theileria annulata-infected cells.
    Parasitology research, 1992, Volume: 78, Issue:4

    Topics: Animals; Cattle; Cells, Cultured; Gene Expression Regulation; Humans; Interleukin-2; Lymphocyte Activation; Lymphocytes; Naphthoquinones; Receptors, Interleukin-2; Recombinant Proteins; RNA, Messenger; Theileria annulata

1992
Further evaluation of the use of buparvaquone in the infection and treatment method of immunizing cattle against Theileria parva derived from African buffalo (Syncerus caffer).
    Veterinary parasitology, 1992, Volume: 43, Issue:1-2

    Topics: Animals; Antibodies, Protozoan; Antiprotozoal Agents; Buffaloes; Cattle; Evaluation Studies as Topic; Immunization; Naphthoquinones; Oxytetracycline; Theileria parva; Theileriasis

1992
Efficacy of buparvaquone as a therapeutic and clearing agent of Babesia equi of European origin in horses.
    American journal of veterinary research, 1992, Volume: 53, Issue:8

    Topics: Acute Disease; Animals; Antibodies, Protozoan; Antiprotozoal Agents; Babesia; Babesiosis; Carrier State; Complement Fixation Tests; Female; Fluorescent Antibody Technique; Horse Diseases; Horses; Injections, Intravenous; Male; Naphthoquinones; Splenectomy

1992
Integrated strategy to control East Coast fever.
    The Veterinary record, 1991, Nov-23, Volume: 129, Issue:21

    Topics: Animals; Antiprotozoal Agents; Cattle; Immunization; Naphthoquinones; Theileriasis; Tick Control

1991
Lymphocytes infected with Theileria parva require both cell-cell contact and growth factor to proliferate.
    European journal of immunology, 1991, Volume: 21, Issue:1

    Topics: Animals; Apicomplexa; Cattle; Cell Adhesion; Cell Communication; Cell Division; Growth Substances; In Vitro Techniques; Interleukin-2; Lymphocytes; Lymphokines; Naphthoquinones; Theileriasis

1991
Activity of buparvaquone against Theileria cervi in white-tailed deer.
    Veterinary parasitology, 1991, Volume: 38, Issue:1

    Topics: Animals; Antiprotozoal Agents; Apicomplexa; Cells, Cultured; Chloroquine; Deer; Erythrocytes; Hypoxanthine; Hypoxanthines; Imidocarb; Naphthoquinones; Theileriasis

1991
Epidemiological observations on theileriosis following field immunisation using infection and treatment.
    Tropical animal health and production, 1991, Volume: 23, Issue:2

    Topics: Animals; Antibodies, Protozoan; Antiprotozoal Agents; Apicomplexa; Arachnid Vectors; Carrier State; Cattle; Disease Reservoirs; Female; Fluorescent Antibody Technique; Immunization; Male; Naphthoquinones; Nymph; Oxytetracycline; Pregnancy; Pregnancy Complications, Infectious; Theileriasis; Ticks

1991
Chemotherapeutic value of parvaquone and buparvaquone against Theileria annulata infection of cattle.
    Research in veterinary science, 1991, Volume: 50, Issue:2

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Cattle; Iran; Naphthoquinones; Theileriasis

1991
Treatment of experimentally induced cytauxzoonosis in cats with parvaquone and buparvaquone.
    Veterinary parasitology, 1990, Volume: 35, Issue:1-2

    Topics: Animals; Antiprotozoal Agents; Apicomplexa; Cat Diseases; Cats; Female; Male; Naphthoquinones; Protozoan Infections; Protozoan Infections, Animal

1990
Elimination of Theileria buffeli infections from cattle by concurrent treatment with buparvaquone and primaquine phosphate.
    Tropical animal health and production, 1990, Volume: 22, Issue:2

    Topics: Animals; Antibodies, Protozoan; Antiprotozoal Agents; Apicomplexa; Cattle; Drug Therapy, Combination; Naphthoquinones; Primaquine; Random Allocation; Theileriasis

1990
Buparvaquone but not cyclosporin A prevents Theileria annulata-infected bovine lymphoblastoid cells from stimulating uninfected lymphocytes.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1990, Volume: 41, Issue:2

    Topics: Animals; Antiprotozoal Agents; Apicomplexa; Cattle; Cells, Cultured; Cyclosporins; Host-Parasite Interactions; Lymphocyte Activation; Lymphocytes; Naphthoquinones; Theileriasis

1990
Treatment of bovine tropical theileriosis with buparvaquone.
    Tropical animal health and production, 1990, Volume: 22, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cattle; Injections, Intramuscular; Male; Naphthoquinones; Theileriasis

1990
Chemoimmunoprophylaxis against bovine tropical theileriosis in young calves: a comparison between buparvaquone and long-acting oxytetracycline.
    Research in veterinary science, 1990, Volume: 49, Issue:1

    Topics: Animals; Cattle; Naphthoquinones; Oxytetracycline; Random Allocation; Theileriasis; Ticks

1990
Effect of treatment of chronic theileriosis with buparvaquone on milk yields.
    Tropical animal health and production, 1989, Volume: 21, Issue:4

    Topics: Animals; Antiprotozoal Agents; Body Temperature; Cattle; Female; Lactation; Naphthoquinones; Pregnancy; Random Allocation; Theileriasis

1989
Evaluations of buparvaquone as a treatment for equine babesiosis (Babesia equi).
    American journal of veterinary research, 1989, Volume: 50, Issue:5

    Topics: Animals; Antiprotozoal Agents; Babesiosis; Carrier State; Horse Diseases; Horses; Male; Naphthoquinones; Splenectomy; Time Factors

1989
Prophylactic efficacy of buparvaquone in experimentally induced Theileria annulata infection in calves.
    Veterinary parasitology, 1989, Volume: 33, Issue:3-4

    Topics: Animals; Antiprotozoal Agents; Cattle; Male; Naphthoquinones; Random Allocation; Theileriasis

1989
Parvaquone and buparvaquone: HPLC analysis and comparative pharmacokinetics in cattle.
    Acta tropica, 1988, Volume: 45, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cattle; Chromatography, High Pressure Liquid; Naphthoquinones

1988
Immunization of cattle using varying infective doses of Theileria parva lawrencei sporozoites derived from an African buffalo (Syncerus caffer) and treatment with buparvaquone.
    Parasitology, 1988, Volume: 96 ( Pt 2)

    Topics: Animals; Antiprotozoal Agents; Apicomplexa; Buffaloes; Carrier State; Cattle; Dose-Response Relationship, Immunologic; Immunization; Naphthoquinones; Oxytetracycline; Theileriasis; Thelazioidea

1988
Treatment of experimentally induced Theileria annulata infection in cross-bred calves with buparvaquone.
    Veterinary parasitology, 1988, Volume: 27, Issue:3-4

    Topics: Acute Disease; Animals; Antiprotozoal Agents; Body Temperature; Cattle; Erythrocytes; Hematocrit; Hemoglobins; Injections, Intramuscular; Lymph Nodes; Naphthoquinones; Random Allocation; Theileriasis; Ticks

1988
Chemoimmunoprophylaxis with buparvaquone against theileriosis in calves.
    The Veterinary record, 1987, Apr-11, Volume: 120, Issue:15

    Topics: Animals; Antiprotozoal Agents; Cattle; Naphthoquinones; Theileriasis

1987
Antitheilerial activity of BW720C (buparvaquone): a comparison with parvaquone.
    Research in veterinary science, 1985, Volume: 39, Issue:1

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Apicomplexa; Cattle; Chemical Phenomena; Chemistry; Kenya; Naphthoquinones; Species Specificity; Theileriasis

1985
Efficacy of Butalex in field cases of bovine theileriosis--short communication.
    Acta veterinaria Hungarica, 1993, Volume: 41, Issue:3-4

    Topics: Animals; Antiprotozoal Agents; Cattle; Female; Male; Naphthoquinones; Theileriasis; Treatment Outcome

1993
Treatment of theileriosis in crossbred cattle in the Punjab.
    Tropical animal health and production, 1993, Volume: 25, Issue:2

    Topics: Age Factors; Animals; Antiprotozoal Agents; Cattle; India; Naphthoquinones; Oxytetracycline; Protozoan Vaccines; Theileria; Theileriasis; Vaccination

1993
The efficacy of two electron transport inhibitors (720C80 and 993C76) on murine strongyloidiasis: a comparison with albendazole.
    International journal for parasitology, 1993, Volume: 23, Issue:6

    Topics: Albendazole; Animals; Antiprotozoal Agents; Female; Naphthoquinones; Rats; Rats, Sprague-Dawley; Strongyloidiasis

1993
Chemotherapeutic trials with four drugs in crossbred calves experimentally infected with Theileria annulata.
    Research in veterinary science, 1993, Volume: 54, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cattle; Male; Naphthoquinones; Oxytetracycline; Quinazolines; Quinazolinones; Theileria annulata; Theileriasis

1993
The Bo-RBC-SCID mouse model for evaluating the efficacy of anti-theilerial drugs.
    International journal for parasitology, 1993, Volume: 23, Issue:1

    Topics: Aminoquinolines; Animals; Antiprotozoal Agents; Cattle; Diminazene; Drug Evaluation, Preclinical; Erythrocyte Transfusion; Female; Mice; Mice, SCID; Models, Biological; Naphthoquinones; Theileria

1993
A mild Theileria parva parasite with potential for immunisation against East Coast fever.
    Veterinary parasitology, 1996, Volume: 61, Issue:1-2

    Topics: Animals; Antiprotozoal Agents; Cattle; Immunization; Naphthoquinones; Protozoan Vaccines; Theileria parva; Theileriasis; Time Factors

1996
Macrophage-parasite relationship in theileriosis. Reversible phenotypic and functional dedifferentiation of macrophages infected with Theileria annulata.
    Journal of leukocyte biology, 1997, Volume: 61, Issue:4

    Topics: Animals; Antigens, Surface; Antiprotozoal Agents; Cattle; Cell Differentiation; Cell Line, Transformed; Down-Regulation; Female; Flow Cytometry; Host-Parasite Interactions; Lipopolysaccharides; Macrophages; Naphthoquinones; Phenotype; Sensitivity and Specificity; Theileria annulata; Theileriasis

1997
Jun NH2-terminal kinase is constitutively activated in T cells transformed by the intracellular parasite Theileria parva.
    Proceedings of the National Academy of Sciences of the United States of America, 1997, May-13, Volume: 94, Issue:10

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antiprotozoal Agents; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Enzyme Activation; Enzyme Inhibitors; Humans; Immunosuppressive Agents; Indoles; JNK Mitogen-Activated Protein Kinases; Kinetics; Lymph Nodes; Lymphocyte Activation; Maleimides; Mitogen-Activated Protein Kinase 9; Mitogen-Activated Protein Kinases; Naphthoquinones; Polyenes; Protein Kinase C; Protein Kinases; Receptor-CD3 Complex, Antigen, T-Cell; Sirolimus; T-Lymphocytes; Tacrolimus; Theileria parva

1997
Theileria-mediated constitutive expression of the casein kinase II-alpha subunit in bovine lymphoblastoid cells.
    Parasitology research, 1997, Volume: 83, Issue:6

    Topics: Animals; Antiprotozoal Agents; Casein Kinase II; Cattle; Cell Division; Cell Line; Concanavalin A; Dichlororibofuranosylbenzimidazole; DNA; Gene Expression Regulation; Lymphocytes; Mitogens; Naphthoquinones; Nucleic Acid Synthesis Inhibitors; Protein Serine-Threonine Kinases; RNA, Messenger; Theileria annulata; Theileria parva; Ticks

1997
Failure of buparvaquone (Butalex) in the treatment of canine visceral leishmaniosis.
    Veterinary parasitology, 1998, Volume: 77, Issue:1

    Topics: Animals; Antiprotozoal Agents; Dog Diseases; Dogs; Female; Injections, Intramuscular; Leishmaniasis, Visceral; Male; Naphthoquinones

1998
Theileria annulata: carrier state and immunity.
    Annals of the New York Academy of Sciences, 1998, Jun-29, Volume: 849

    Topics: Animals; Antibodies, Protozoan; Antibody Formation; Antigens, Protozoan; Antigens, Surface; Antiprotozoal Agents; Carrier State; Cattle; Cell Line; Enzyme-Linked Immunosorbent Assay; Fluorescent Antibody Technique, Indirect; Life Cycle Stages; Male; Naphthoquinones; Polymerase Chain Reaction; RNA, Protozoan; RNA, Ribosomal; Sensitivity and Specificity; Theileria annulata; Theileriasis; Ticks

1998
Chemoprophylaxis of Theileria annulata and Theileria parva infections of calves with buparvaquone.
    Veterinary parasitology, 1998, Jul-17, Volume: 78, Issue:1

    Topics: Animals; Antibodies, Protozoan; Antiprotozoal Agents; Cattle; Fluorescent Antibody Technique, Indirect; Naphthoquinones; Parasitemia; Theileria annulata; Theileria parva; Theileriasis

1998
Modulation of enzymatic activity of Src-family kinases in bovine T cells transformed by Theileria parva.
    Parasitology, 1998, Volume: 117 ( Pt 2)

    Topics: Animals; Antiprotozoal Agents; Cattle; Cell Line, Transformed; Herpesvirus 2, Saimiriine; Humans; Jurkat Cells; Naphthoquinones; Phosphorylation; Precipitin Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; src-Family Kinases; T-Lymphocytes; Theileria parva; Tyrosine

1998
Susceptibility to tropical theileriosis of calves born to dams immunized with Theileria annulata (Hisar) cell culture vaccine.
    Tropical animal health and production, 1998, Volume: 30, Issue:6

    Topics: Animals; Animals, Newborn; Antibodies, Protozoan; Antigens, Protozoan; Antiprotozoal Agents; Arachnid Vectors; Body Temperature; Cattle; Disease Susceptibility; Female; Fluorescent Antibody Technique, Indirect; Hematocrit; Hemoglobins; Immunity, Maternally-Acquired; India; Naphthoquinones; Protozoan Vaccines; Theileria annulata; Theileriasis; Ticks; Vaccination

1998
Therapeutic effects of some antihaematozoal drugs against Haemoproteus columbae in domestic pigeons.
    DTW. Deutsche tierarztliche Wochenschrift, 1999, Volume: 106, Issue:2

    Topics: Animals; Animals, Domestic; Antiprotozoal Agents; Bird Diseases; Coccidiosis; Columbidae; Diminazene; Haemosporida; Naphthoquinones; Quinolinium Compounds

1999
The effect of buparvaquone treatment on the levels of some antioxidant vitamins, lipid peroxidation and glutathione peroxidase in cattle with theileriosis.
    Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B, 1999, Volume: 46, Issue:4

    Topics: Animals; Antiprotozoal Agents; beta Carotene; Cattle; Cattle Diseases; Erythrocytes; Glutathione; Glutathione Peroxidase; Lipid Peroxidation; Naphthoquinones; Reference Values; Theileriasis; Vitamin A; Vitamin E; Vitamins

1999
Treatment of East Coast fever: a comparison of parvaquone and buparvaquone.
    Veterinary parasitology, 1999, Volume: 87, Issue:1

    Topics: Administration, Topical; Animals; Antimalarials; Biopsy; Cattle; Female; Fever; Injections, Intramuscular; Insecticides; Kenya; Male; Naphthoquinones; Nitriles; Parasitemia; Pyrethrins; Random Allocation; Theileriasis; Tick Infestations

1999
Screening of five drugs for efficacy against Babesia felis in experimentally infected cats.
    Journal of the South African Veterinary Association, 2000, Volume: 71, Issue:1

    Topics: Animals; Anti-Infective Agents; Antiprotozoal Agents; Babesiosis; Cat Diseases; Cats; Drug Combinations; Enrofloxacin; Fluoroquinolones; Hematocrit; Naphthoquinones; Parasitemia; Primaquine; Quinolones; Rifampin; Sulfadiazine; Trimethoprim

2000
In vivo monitoring of intracellular ATP levels in Leishmania donovani promastigotes as a rapid method to screen drugs targeting bioenergetic metabolism.
    Antimicrobial agents and chemotherapy, 2001, Volume: 45, Issue:4

    Topics: Adenosine Triphosphate; Animals; Antiprotozoal Agents; Cell Division; Cell Line; Dose-Response Relationship, Drug; Energy Metabolism; Firefly Luciferin; Kinetics; Leishmania donovani; Luciferases; Luminescent Measurements; Membrane Potentials; Mitochondria; Naphthoquinones; Parasitic Sensitivity Tests; Transfection

2001
Production and characterisation of mucoadhesive nanosuspensions for the formulation of bupravaquone.
    International journal of pharmaceutics, 2001, Feb-19, Volume: 214, Issue:1-2

    Topics: Animals; Antiprotozoal Agents; Chemistry, Pharmaceutical; Chitin; Chitosan; Cryptosporidium parvum; Drug Delivery Systems; Drug Stability; Gels; Naphthoquinones; Particle Size; Suspensions

2001
Buparvaquone mucoadhesive nanosuspension: preparation, optimisation and long-term stability.
    International journal of pharmaceutics, 2002, Apr-26, Volume: 237, Issue:1-2

    Topics: Adhesives; Antiprotozoal Agents; Drug Stability; Hydrogels; Microscopy, Electron; Nanotechnology; Naphthoquinones; Particle Size; Technology, Pharmaceutical

2002
Constitutive exclusion of Csk from Hck-positive membrane microdomains permits Src kinase-dependent proliferation of Theileria-transformed B lymphocytes.
    Blood, 2003, Mar-01, Volume: 101, Issue:5

    Topics: Animals; Antiprotozoal Agents; B-Lymphocytes; Cattle; Cell Division; Cell Transformation, Neoplastic; CSK Tyrosine-Protein Kinase; Enzyme Activation; Enzyme Inhibitors; Lymphocyte Activation; Membrane Microdomains; Membrane Proteins; Naphthoquinones; Phenotype; Phosphatidylinositol 3-Kinases; Phosphoproteins; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-hck; Pyrimidines; Signal Transduction; src-Family Kinases; Theileria parva; Transcription Factor AP-1

2003
Hijacking of host cell IKK signalosomes by the transforming parasite Theileria.
    Science (New York, N.Y.), 2002, Nov-01, Volume: 298, Issue:5595

    Topics: Active Transport, Cell Nucleus; Animals; Antiprotozoal Agents; Apoptosis; Cattle; Cell Cycle; Cell Division; Cell Line, Transformed; Cell Nucleus; Down-Regulation; I-kappa B Kinase; I-kappa B Proteins; Leukocytes; Microscopy, Confocal; Naphthoquinones; NF-kappa B; Phosphorylation; Protein Serine-Threonine Kinases; Signal Transduction; Theileria

2002
Transition metal complexes of buparvaquone as potent new antimalarial agents. 1. Synthesis, X-ray crystal-structures, electrochemistry and antimalarial activity against Plasmodium falciparum.
    Journal of inorganic biochemistry, 2003, Jul-01, Volume: 95, Issue:4

    Topics: Animals; Antimalarials; Crystallography, X-Ray; Electrochemistry; Metals; Models, Molecular; Naphthoquinones; Oxidation-Reduction; Plasmodium falciparum; Spectrophotometry, Infrared

2003
Theileria parva-transformed T cells show enhanced resistance to Fas/Fas ligand-induced apoptosis.
    Journal of immunology (Baltimore, Md. : 1950), 2003, Aug-01, Volume: 171, Issue:3

    Topics: Animals; Antiprotozoal Agents; Apoptosis; Carrier Proteins; CASP8 and FADD-Like Apoptosis Regulating Protein; Caspases; Cattle; Cell Line, Transformed; Enzyme Activation; Fas Ligand Protein; fas Receptor; Homeostasis; Host-Parasite Interactions; Immunity, Innate; Inhibitor of Apoptosis Proteins; Intracellular Signaling Peptides and Proteins; Ligands; Membrane Glycoproteins; Naphthoquinones; Protein Biosynthesis; Proteins; T-Lymphocyte Subsets; Theileria parva; Up-Regulation; X-Linked Inhibitor of Apoptosis Protein

2003
Apoptosis of Theileria-infected lymphocytes induced upon parasite death involves activation of caspases 9 and 3.
    Biochimie, 2003, Volume: 85, Issue:8

    Topics: Amino Acid Chloromethyl Ketones; Animals; Antiprotozoal Agents; Apoptosis; Caspase 3; Caspase 9; Caspase Inhibitors; Caspases; Cattle; Cell Death; Cysteine Proteinase Inhibitors; Enzyme Activation; Naphthoquinones; Poly(ADP-ribose) Polymerases; T-Lymphocytes; Theileria parva; Theileriasis

2003
Synthesis, in vitro evaluation, and antileishmanial activity of water-soluble prodrugs of buparvaquone.
    Journal of medicinal chemistry, 2004, Jan-01, Volume: 47, Issue:1

    Topics: Administration, Oral; Administration, Topical; Alkaline Phosphatase; Animals; Antiprotozoal Agents; Cricetinae; Female; Humans; Hydrolysis; In Vitro Techniques; Leishmania; Leishmaniasis, Cutaneous; Leishmaniasis, Visceral; Macrophages, Peritoneal; Mice; Naphthoquinones; Organophosphates; Permeability; Prodrugs; Skin; Solubility; Water

2004
Cerebral theileriosis in a Holstein calf.
    The Veterinary record, 2004, Apr-24, Volume: 154, Issue:17

    Topics: Animals; Anti-Bacterial Agents; Antiprotozoal Agents; Brain Diseases; Cattle; Cattle Diseases; Erythrocytes; Injections, Intramuscular; Male; Naphthoquinones; Oxytetracycline; Polymerase Chain Reaction; Theileria; Theileriasis; Treatment Outcome

2004
Synthesis and antileishmanial activity of novel buparvaquone oxime derivatives.
    Bioorganic & medicinal chemistry, 2004, Jul-01, Volume: 12, Issue:13

    Topics: Animals; Antiprotozoal Agents; Leishmania donovani; Leishmaniasis, Visceral; Macrophages; Magnetic Resonance Spectroscopy; Microsomes, Liver; Molecular Structure; Naphthoquinones; Oximes; Rats; Rats, Wistar

2004
The effect of dexamethasone and promethazine in combination with buparvaquone in the management of East Coast fever.
    The Onderstepoort journal of veterinary research, 2004, Volume: 71, Issue:2

    Topics: Animals; Antiprotozoal Agents; Cattle; Cattle Diseases; Dexamethasone; Drug Therapy, Combination; Glucocorticoids; Histamine H1 Antagonists; Male; Naphthoquinones; Promethazine; Pulmonary Edema; Random Allocation; Theileria; Theileriasis; Treatment Outcome

2004
Design, synthesis and in vitro evaluation of novel water-soluble prodrugs of buparvaquone.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2004, Volume: 23, Issue:2

    Topics: Alkaline Phosphatase; Antiprotozoal Agents; Buffers; Drug Design; Hydrolysis; Indicators and Reagents; Lipids; Magnetic Resonance Spectroscopy; Naphthoquinones; Prodrugs; Solubility

2004
Evaluation of buparvaquone (BUTA-Kel KELA, Belgium) as a treatment of East Coast fever in cattle, in the peri-urban of Dar Es Salaam city, Tanzania.
    Veterinary parasitology, 2006, Jun-30, Volume: 139, Issue:1-3

    Topics: Animals; Antiprotozoal Agents; Cattle; Cattle Diseases; Female; Male; Naphthoquinones; Tanzania; Theileria parva; Theileriasis; Treatment Outcome

2006
Development and validation of RP-HPLC-UV method for simultaneous determination of buparvaquone, atenolol, propranolol, quinidine and verapamil: a tool for the standardization of rat in situ intestinal permeability studies.
    Journal of pharmaceutical and biomedical analysis, 2007, Mar-12, Volume: 43, Issue:4

    Topics: Animals; Antiprotozoal Agents; Atenolol; Buffers; Chromatography, High Pressure Liquid; Drug Stability; Hydrogen-Ion Concentration; Intestinal Mucosa; Male; Molecular Structure; Naphthoquinones; Perfusion; Permeability; Propranolol; Quinidine; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Spectrophotometry, Ultraviolet; Verapamil

2007
Topical buparvaquone formulations for the treatment of cutaneous leishmaniasis.
    The Journal of pharmacy and pharmacology, 2007, Volume: 59, Issue:1

    Topics: Administration, Cutaneous; Animals; Antiprotozoal Agents; Chemistry, Pharmaceutical; Ethanol; Female; Humans; In Vitro Techniques; Leishmaniasis, Cutaneous; Melanins; Mice; Mice, Inbred BALB C; Myristates; Naphthoquinones; Organophosphates; Polyethylene Glycols; Prodrugs; Propylene Glycol; Skin; Skin Absorption

2007
In vivo studies on the antileishmanial activity of buparvaquone and its prodrugs.
    The Journal of antimicrobial chemotherapy, 2007, Volume: 60, Issue:4

    Topics: Animals; Antiprotozoal Agents; Chemistry, Pharmaceutical; Female; Leishmania donovani; Leishmania major; Leishmaniasis, Cutaneous; Leishmaniasis, Visceral; Liver; Mice; Mice, Inbred BALB C; Naphthoquinones; Prodrugs; Skin

2007
Optimization and validation of RP-HPLC-UV method with solid-phase extraction for determination of buparvaquone in human and rabbit plasma: application to pharmacokinetic study.
    Biomedical chromatography : BMC, 2008, Volume: 22, Issue:5

    Topics: Animals; Antiprotozoal Agents; Chromatography, High Pressure Liquid; Humans; Molecular Structure; Naphthoquinones; Rabbits; Reproducibility of Results; Solid Phase Extraction; Spectrophotometry, Ultraviolet

2008
[Therapeutic efficacy of buparvaquone (buparvon) in cattle with theileriosis].
    Turkiye parazitolojii dergisi, 2008, Volume: 32, Issue:4

    Topics: Animals; Antiprotozoal Agents; Cattle; Erythrocytes; Injections, Intramuscular; Naphthoquinones; Theileriasis; Treatment Outcome

2008
The protozoan parasite Theileria annulata alters the differentiation state of the infected macrophage and suppresses musculoaponeurotic fibrosarcoma oncogene (MAF) transcription factors.
    International journal for parasitology, 2009, Volume: 39, Issue:10

    Topics: Animals; Antiprotozoal Agents; Cattle; Cattle Diseases; Cell Dedifferentiation; Cell Differentiation; Host-Parasite Interactions; Macrophages; Maf Transcription Factors; Naphthoquinones; Phenotype; Theileria annulata; Theileriasis

2009
In vitro and in vivo evaluation of self-microemulsifying drug delivery system of buparvaquone.
    Drug development and industrial pharmacy, 2010, Volume: 36, Issue:6

    Topics: Animals; Chemistry, Pharmaceutical; Drug Delivery Systems; Drug Evaluation, Preclinical; Emulsifying Agents; Male; Naphthoquinones; Rabbits

2010
In vivo evidence for the resistance of Theileria annulata to buparvaquone.
    Veterinary parasitology, 2010, May-11, Volume: 169, Issue:3-4

    Topics: Animals; Antiprotozoal Agents; Cattle; Dairying; Disease Outbreaks; Drug Resistance; Hematocrit; Naphthoquinones; Parasitemia; Schizonts; Theileria annulata; Theileriasis; Treatment Failure; Tunisia

2010
Cytoplasmic sequestration of p53 promotes survival in leukocytes transformed by Theileria.
    Oncogene, 2010, May-27, Volume: 29, Issue:21

    Topics: Animals; Antiprotozoal Agents; bcl-2-Associated X Protein; Cattle; Cell Nucleus; Cell Survival; Concanavalin A; DNA, Complementary; Gene Amplification; Kinetics; Leukocytes; Naphthoquinones; Theileria annulata; Theileriasis; Transcription, Genetic; Tumor Suppressor Protein p53

2010
Evaluation and structure-activity relationship study of acute toxicity of naphthoquinones to Photobacterium phosphoreum, Photobacterium T3B.
    Bulletin of environmental contamination and toxicology, 2010, Volume: 85, Issue:2

    Topics: Antiprotozoal Agents; Atovaquone; Microbial Sensitivity Tests; Naphthoquinones; Photobacterium; Structure-Activity Relationship; Toxicity Tests, Acute

2010
Effectiveness of liposomal buparvaquone in an experimental hamster model of Leishmania (L.) infantum chagasi.
    Experimental parasitology, 2012, Volume: 130, Issue:3

    Topics: Animals; Antiprotozoal Agents; Cell Line; Cells, Cultured; Cricetinae; Disease Models, Animal; Humans; Inhibitory Concentration 50; Leishmania infantum; Leishmaniasis, Visceral; Liposomes; Macaca mulatta; Macrophages, Peritoneal; Male; Mesocricetus; Mice; Mice, Inbred BALB C; Naphthoquinones; Phosphatidylserines

2012
Point mutations in the Theileria annulata cytochrome b gene is associated with buparvaquone treatment failure.
    Veterinary parasitology, 2012, Jul-06, Volume: 187, Issue:3-4

    Topics: Animals; Antiprotozoal Agents; Cattle; Cytochromes b; Dairying; Drug Resistance; Female; Gene Expression Regulation; Naphthoquinones; Point Mutation; Theileria annulata; Theileriasis

2012
MDM2 regulates a novel form of incomplete neoplastic transformation of Theileria parva infected lymphocytes.
    Experimental and molecular pathology, 2013, Volume: 94, Issue:1

    Topics: Amino Acid Sequence; Animals; Apoptosis; bcl-2-Associated X Protein; Cattle; Cell Line; Cell Transformation, Neoplastic; Cisplatin; DNA Damage; Enzyme Activation; Lymphocyte Activation; Molecular Sequence Data; Naphthoquinones; NF-kappa B; Protein Isoforms; Proto-Oncogene Proteins c-mdm2; Signal Transduction; T-Lymphocytes; Theileria parva; Tumor Suppressor Protein p53

2013
Theileriosis (Cytauxzoonosis) in Roan antelope (Hippotragus equinus): field exposure to infection and identification of potential vectors.
    The Onderstepoort journal of veterinary research, 2012, Apr-20, Volume: 79, Issue:1

    Topics: Animals; Animals, Wild; Antelopes; Antiprotozoal Agents; DNA, Protozoan; Male; Naphthoquinones; Polymerase Chain Reaction; Rhipicephalus; Salivary Glands; South Africa; Theileria; Theileriasis; Tick Infestations

2012
A Bovine Lymphosarcoma Cell Line Infected with Theileria annulata Exhibits an Irreversible Reconfiguration of Host Cell Gene Expression.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: Animals; Cattle; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Cell Survival; Gene Expression Regulation; Host-Parasite Interactions; Leukocytes; Lymphoma, Non-Hodgkin; Naphthoquinones; Theileria annulata; Transcription, Genetic

2013
Theileria parasites secrete a prolyl isomerase to maintain host leukocyte transformation.
    Nature, 2015, Apr-16, Volume: 520, Issue:7547

    Topics: Animals; Cattle; Cell Line; Cell Transformation, Neoplastic; Drug Resistance; Host-Parasite Interactions; Humans; Leukocytes; Naphthoquinones; NIMA-Interacting Peptidylprolyl Isomerase; Parasites; Peptidylprolyl Isomerase; Protein Stability; Proto-Oncogene Proteins c-jun; Signal Transduction; SKP Cullin F-Box Protein Ligases; Theileria; Transcription Factor AP-1; Ubiquitination; Xenograft Model Antitumor Assays; Zebrafish

2015
In-vitro sensitivity of Pakistani Leishmania tropica field isolate against buparvaquone in comparison to standard anti-leishmanial drugs.
    Experimental parasitology, 2015, Volume: 154

    Topics: Amphotericin B; Antimony Sodium Gluconate; Antiprotozoal Agents; Cell Line, Tumor; Child; Humans; Inhibitory Concentration 50; Leishmania tropica; Leishmaniasis, Cutaneous; Macrophages; Male; Meglumine; Meglumine Antimoniate; Naphthoquinones; Organometallic Compounds; Pakistan; Parasitic Sensitivity Tests

2015
Buparvaquone is active against Neospora caninum in vitro and in experimentally infected mice.
    International journal for parasitology. Drugs and drug resistance, 2015, Volume: 5, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cells, Cultured; Coccidiosis; Female; Fibroblasts; Humans; Mice; Mice, Inbred BALB C; Naphthoquinones; Neospora

2015
Sequence Polymorphism of Cytochrome b Gene in Theileria annulata Tunisian Isolates and Its Association with Buparvaquone Treatment Failure.
    PloS one, 2015, Volume: 10, Issue:6

    Topics: Animals; Antiprotozoal Agents; Cattle; Cytochromes b; Drug Resistance; Naphthoquinones; Point Mutation; Polymorphism, Single Nucleotide; Protozoan Proteins; Theileria annulata; Theileriasis; Treatment Failure

2015
Repurposing of antiparasitic drugs: the hydroxy-naphthoquinone buparvaquone inhibits vertical transmission in the pregnant neosporosis mouse model.
    Veterinary research, 2016, Feb-17, Volume: 47

    Topics: Animals; Antiparasitic Agents; Coccidiosis; Female; Infectious Disease Transmission, Vertical; Male; Mice, Inbred BALB C; Naphthoquinones; Neospora; Pregnancy

2016
Concentrations of buparvaquone in milk and tissue of dairy cows.
    New Zealand veterinary journal, 2016, Volume: 64, Issue:6

    Topics: Animals; Antiprotozoal Agents; Cattle; Female; Injections, Intramuscular; Liver; Milk; Muscle, Skeletal; Naphthoquinones; Theileriasis

2016
Efficacy, safety and tolerance of imidocarb dipropionate versus atovaquone or buparvaquone plus azithromycin used to treat sick dogs naturally infected with the Babesia microti-like piroplasm.
    Parasites & vectors, 2017, Mar-13, Volume: 10, Issue:1

    Topics: Animals; Antiprotozoal Agents; Atovaquone; Azithromycin; Babesia microti; Babesiosis; Dog Diseases; Dogs; Drug Therapy, Combination; Europe; Female; Imidocarb; Male; Naphthoquinones; Parasitemia; Polymerase Chain Reaction

2017
Development of a murine vertical transmission model for Toxoplasma gondii oocyst infection and studies on the efficacy of bumped kinase inhibitor (BKI)-1294 and the naphthoquinone buparvaquone against congenital toxoplasmosis.
    The Journal of antimicrobial chemotherapy, 2017, 08-01, Volume: 72, Issue:8

    Topics: Animals; Antiprotozoal Agents; Disease Models, Animal; Female; Infectious Disease Transmission, Vertical; Male; Mice; Naphthalenes; Naphthoquinones; Piperidines; Pyrazoles; Toxoplasmosis, Animal; Toxoplasmosis, Congenital; Treatment Outcome

2017
Residual detection of buparvaquone, nystatin, and etomidate in animal-derived food products in a single chromatographic run using liquid chromatography-tandem mass spectrometry.
    Food chemistry, 2017, Dec-15, Volume: 237

    Topics: Animals; Chromatography, High Pressure Liquid; Etomidate; Naphthoquinones; Nystatin; Swine; Tandem Mass Spectrometry

2017
Variation in cardiac markers and electrocardiographic alterations in young calves naturally infected with bovine tropical theileriosis.
    Tropical animal health and production, 2018, Volume: 50, Issue:6

    Topics: Animals; Antiprotozoal Agents; Biomarkers; Cattle; Creatine Kinase, MB Form; Electrocardiography; Heart; Naphthoquinones; Theileriasis; Troponin I

2018
Orally Bioavailable and Effective Buparvaquone Lipid-Based Nanomedicines for Visceral Leishmaniasis.
    Molecular pharmaceutics, 2018, 07-02, Volume: 15, Issue:7

    Topics: Administration, Oral; Animals; Antiprotozoal Agents; Biological Availability; Cell Line; Disease Models, Animal; Drug Carriers; Drug Compounding; Drug Liberation; Drug Stability; Emulsions; Excipients; Feasibility Studies; Humans; Leishmania infantum; Leishmaniasis, Visceral; Lipids; Male; Mice; Mice, Inbred BALB C; Nanoparticles; Naphthoquinones; Solubility; Treatment Outcome

2018
In vitro treatment of Besnoitia besnoiti with the naphto-quinone buparvaquone results in marked inhibition of tachyzoite proliferation, mitochondrial alterations and rapid adaptation of tachyzoites to increased drug concentrations.
    Parasitology, 2019, Volume: 146, Issue:1

    Topics: Animals; Antiprotozoal Agents; Cell Line; Chlorocebus aethiops; Drug Resistance; Fibroblasts; Inhibitory Concentration 50; Microscopy, Electron, Transmission; Mitochondria; Naphthoquinones; Sarcocystidae; Vero Cells

2019
Repurposing of an old drug: In vitro and in vivo efficacies of buparvaquone against Echinococcus multilocularis.
    International journal for parasitology. Drugs and drug resistance, 2018, Volume: 8, Issue:3

    Topics: Albendazole; Animals; Anthelmintics; Antiprotozoal Agents; Drug Evaluation, Preclinical; Drug Repositioning; Echinococcosis; Echinococcus multilocularis; Electron Transport Complex III; Glucose-6-Phosphate Isomerase; Inhibitory Concentration 50; Life Cycle Stages; Mice; Microscopy, Electron, Transmission; Naphthoquinones; Parasite Load; Phenyl Ethers; Quinolones

2018
Evidence of multiple point mutations in Theileria annulata cytochrome b gene incriminated in buparvaquone treatment failure.
    Acta tropica, 2019, Volume: 191

    Topics: Animals; Antiprotozoal Agents; Cattle; Cytochromes b; Drug Resistance; Naphthoquinones; Point Mutation; Sudan; Theileria annulata; Theileriasis; Treatment Failure

2019
Leveraging the Medicines for Malaria Venture malaria and pathogen boxes to discover chemical inhibitors of East Coast fever.
    International journal for parasitology. Drugs and drug resistance, 2019, Volume: 9

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Cattle; Cell Line; Cell Proliferation; Dasatinib; Drug Repositioning; High-Throughput Screening Assays; Inhibitory Concentration 50; Leukocytes, Mononuclear; Naphthoquinones; Small Molecule Libraries; Theileria parva; Theileriasis

2019
Secreted parasite Pin1 isomerase stabilizes host PKM2 to reprogram host cell metabolism.
    Communications biology, 2019, Volume: 2

    Topics: Animals; Antiprotozoal Agents; Biological Transport; Carrier Proteins; Cattle; Cell Line, Transformed; Cell Transformation, Neoplastic; Enzyme Inhibitors; Gene Expression Regulation; Glucose; Host-Pathogen Interactions; Hypoxia-Inducible Factor 1, alpha Subunit; Lymphocytes; Membrane Proteins; Metabolic Networks and Pathways; Naphthoquinones; NIMA-Interacting Peptidylprolyl Isomerase; Protozoan Proteins; RNA, Small Interfering; Signal Transduction; Theileria; Thyroid Hormone-Binding Proteins; Thyroid Hormones

2019
Establishment and Expression of Cytokines in a
    Genes, 2019, 04-30, Volume: 10, Issue:5

    Topics: Animals; Antigens; B-Lymphocytes; Cattle; Cytokines; Flow Cytometry; Gene Expression Regulation; Lipopolysaccharides; Macrophages; Naphthoquinones; Single-Cell Analysis; Theileria annulata; Theileriasis

2019
Co-delivery of buparvaquone and polymyxin B in a nanostructured lipid carrier for leishmaniasis treatment.
    Journal of global antimicrobial resistance, 2019, Volume: 18

    Topics: Anti-Bacterial Agents; Biopolymers; Chitosan; Dextrans; Drug Combinations; Drug Delivery Systems; Leishmania infantum; Leishmaniasis; Lipids; Nanostructures; Naphthoquinones; Particle Size; Polymyxin B; Thermogravimetry

2019
THEILERIOSIS IN MOUNTAIN BONGO REPATRIATED TO KENYA: A CLINICAL AND MOLECULAR INVESTIGATION.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2019, Jun-13, Volume: 50, Issue:2

    Topics: Animals; Antelopes; Antiprotozoal Agents; Conservation of Natural Resources; Disease Outbreaks; Female; Kenya; Male; Naphthoquinones; Oxytetracycline; Theileria; Theileriasis

2019
Shape mediated splenotropic delivery of buparvaquone loaded solid lipid nanoparticles.
    Drug delivery and translational research, 2020, Volume: 10, Issue:1

    Topics: Administration, Intravenous; Animals; Chemical Precipitation; Drug Delivery Systems; Female; Lipids; Mice; Microscopy, Electron, Scanning; Nanoparticles; Naphthoquinones; Particle Size; Spleen

2020
A longitudinal study of the effect of Theileria orientalis Ikeda type infection on three New Zealand dairy farms naturally infected at pasture.
    Veterinary parasitology, 2019, Volume: 276

    Topics: Animals; Antiprotozoal Agents; Cattle; Dairying; DNA, Protozoan; Female; Gene Dosage; Hematocrit; Incidence; Lactation; Longitudinal Studies; Naphthoquinones; Prevalence; Prospective Studies; Real-Time Polymerase Chain Reaction; Reproduction; Theileria; Theileriasis

2019
Mutations in the TaPIN1 peptidyl prolyl isomerase gene in Theileria annulata parasites isolated in Sudan.
    International journal for parasitology. Drugs and drug resistance, 2019, Volume: 11

    Topics: Animals; Antiprotozoal Agents; Cattle; Drug Resistance; Naphthoquinones; Peptidylprolyl Isomerase; Phenotype; Point Mutation; Sudan; Theileria annulata; Theileriasis

2019
Topical buparvaquone nano-enabled hydrogels for cutaneous leishmaniasis.
    International journal of pharmaceutics, 2020, Oct-15, Volume: 588

    Topics: Animals; Antiprotozoal Agents; Hydrogels; Leishmaniasis, Cutaneous; Mice; Mice, Inbred BALB C; Naphthoquinones

2020
Biogenic nanoporous silicon carrier improves the efficacy of buparvaquone against resistant visceral leishmaniasis.
    PLoS neglected tropical diseases, 2021, Volume: 15, Issue:6

    Topics: Animals; Antiprotozoal Agents; Drug Carriers; Female; Hordeum; Injections, Intraperitoneal; Leishmania donovani; Leishmaniasis, Visceral; Macrophages; Mice, Inbred BALB C; Nanoparticles; Naphthoquinones; Silicon

2021
Oral administration of buparvaquone nanostructured lipid carrier enables in vivo activity against Leishmania infantum.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2022, Feb-01, Volume: 169

    Topics: Administration, Oral; Antiprotozoal Agents; Leishmania infantum; Lipids; Liposomes; Nanoparticles; Naphthoquinones

2022
Metabolomic profiling of bovine leucocytes transformed by Theileria annulata under BW720c treatment.
    Parasites & vectors, 2022, Oct-05, Volume: 15, Issue:1

    Topics: Animals; Arginine; Carnitine; Cattle; Dimethyl Sulfoxide; Leucine; Naphthoquinones; Theileria; Theileria annulata; Theileriasis

2022