bunazosin and quinazolines

bunazosin has been researched along with quinazolines in 225 studies

Research

Studies (225)

TimeframeStudies, this research(%)All Research%
pre-199083 (36.89)18.7374
1990's110 (48.89)18.2507
2000's31 (13.78)29.6817
2010's0 (0.00)24.3611
2020's1 (0.44)2.80

Authors

AuthorsStudies
Amano, M; Kanamori, T; Kinoshita, M; Shichiri, G; Takahashi, M1
Kimura, H; Kusaba, T; Nagasawa, K; Otsuka, T; Sakata, T; Tada, Y; Tsuda, Y1
Atarashi, K; Matsuoka, H; Sugimoto, T; Takagi, M1
Gotoh, S; Hiraga, S; Hosoda, K; Kakehi, R; Kaneoya, F; Kojima, S; Mizuo, T; Satoh, T; Tanizawa, A; Yokokawa, M1
Hirakawa, S; Imai, Y; Ito, H; Kakami, M; Koshiji, M; Minatoguchi, S; Watanabe, H1
Baba, T; Ishizaki, T; Murabayashi, S; Tomiyama, T1
Evans, RG; Hayes, IP; Ludbrook, J1
Kono, K; Masuda, T; Nakamura, Y; Oyama, M; Shimizu, T; Takahashi, M; Takeda, K; Yagi, S1
García-Sáinz, JA; González-Espinosa, C; Romero-Avila, MT; Torres-Márquez, ME1
Kawai, C; Matsumori, A; Okada, I; Tominaga, M; Yamada, T1
Arakawa, K; Hidaka, K; Matsunaga, A; Sasaki, J1
Asakura, Y; Harano, Y; Hirose, J; Kageyama, A; Omae, T; Sato, A; Suzuki, M1
Kondo, S; Morita, T1
Asano, H; Fujita, T; Hirabayashi, S; Kato, N; Kinukawa, T; Ohshima, S; Ono, Y1
Abiko, Y; Ichihara, K; Nasa, Y; Yoshida, R1
Kondo, M; Nakanishi, T; Nishimura, M; Takahashi, H; Yoshida, T; Yoshimura, M1
Hosoda, S; Kaneko, N; Kawagoe, Y; Kimata, S; Kimura, H; Konno, K; Miki, N; Nagashima, H; Sumiyoshi, T1
Hattori, K; Kobayashi, Y; Shimoura, K; Shinozuka, K1
Hori, M; Inoue, M; Iwai, K; Iwakura, K; Kagiya, T; Kamada, T; Kitabatake, A; Uchida, S; Watanabe, Y; Yoshida, H1
Haneda, N; Hayashi, Y; Inoue, M; Kishida, K; Mori, C; Ozasa, H; Watanabe, K1
Hayashi, Y; Ikeda, K; Ohnishi, H; Watanabe, K2
Fujioka, S; Kawamoto, T; Keno, Y; Kobatake, T; Matsuzawa, Y; Tarui, S; Tokunaga, K; Watanabe, Y; Yoshida, H1
Smith, SE; Trew, DR; Wright, LA1
Kusunoki, T; Kuwayama, Y; Manabe, R; Shimizu, Y; Sun, N; Takagi, T; Tanaka, M; Yamamoto, R1
Sugiyama, T1
Iwai, T; Nagano, M; Nakamura, I; Ohkubo, T; Takeda, N; Tanamura, A1
Hikida, M; Kinoshita, M; Kuwayama, Y; Nishimura, K; Shirasawa, E1
Baba, S; Kinami, J; Mano, F; Maruyama, K; Nagatomo, T; Tsuchihashi, H1
Araie, M; Azuma, I; Nakajima, M; Oshika, T; Sugiyama, T1
Yamashita, Y1
Kinami, J; Maruyama, K; Nagatomo, T; Tsuchihashi, H1
Chiba, S; Skrbic, R1
Hashimoto, T; Kaguchi, Y; Kuriyama, S; Nakamura, K; Sakai, O; Tokutome, G; Tomonari, H1
Hasegawa, J; Hisatome, I; Kotake, H; Mashiba, H; Matsuoka, S; Noguchi, N1
Baba, T; Murabayashi, S; Takebe, K; Tomiyama, T1
Kaneko, S; Koyanagi, T; Kumamoto, Y; Maru, A; Nishizawa, O; Orikasa, S; Togashi, M; Tsuchida, S; Tsukamoto, T; Yachiku, S1
Kato, Y; Kawabe, K; Kimura, R; Maruyama, M; Matsuoka, Y; Suzuki, M; Yamada, S1
Kobayashi, S1
Chiba, S; Matsuura, M; Zenda, H1
Haneda, T; Obata, H; Tanaka, H1
Baba, T; Takebe, K; Tomiyama, T1
Esato, K; Katoh, T; Miyamoto, M; Mori, F1
Abiko, Y; Ichihara, K; Yoshida, R1
Chiba, S; Haniuda, M2
Hirabayashi, M; Ikegaki, I; Matsusawa, M; Nakanishi, T; Nishimura, M; Takahashi, H; Yoshimura, M1
Araie, M; Oshika, T1
Aso, Y; Honma, Y; Koyanagi, T; Maru, A; Miyake, K; Orikasa, S; Shimazaki, J; Soma, F; Togashi, M; Yasuda, K1
Araki, T; Chigusa, I; Kato, T; Kawamura, J; Morisita, H; Nakano, S; Saito, K; Sugimura, Y; Tajima, K; Tochigi, H1
Inukai, T; Ishii, A; Iwashita, A; Kobayashi, I; Kobayashi, S; Kobayashi, T; Shimomura, Y; Yamaguchi, T; Yamaguchi, Y1
Chiba, S; Tsukada, M3
Doi, T; Hasegawa, J; Hisatome, I; Kotake, H; Mashiba, H; Noguchi, N; Sawaguchi, M1
Fujiwara, H; Ishida, M; Kawai, C; Kawamura, A; Kida, M; Takemura, G; Tanaka, M; Uegaito, T1
Hasegawa, J; Kotake, H; Kurata, Y; Mashiba, H; Ogino, K; Ohtahara, A; Saitoh, M1
Ozawa, T; Sugiyama, S1
Kondo, A; Mitsuya, H; Otani, T; Takita, T1
Chiba, S; Nakane, T1
Aso, Y; Ishibashi, A; Koshiba, K; Kumamoto, Y; Nishizawa, O; Ogawa, A; Tomita, Y; Tsuchida, S; Tsukamoto, T; Yokoyama, E1
Aoyama, T; Furuya, S; Honma, A; Kumamoto, Y; Miyamoto, S; Takagi, Y; Takatsuka, K; Tamiya, T; Tsukamoto, T; Yokoyama, E1
Araie, M; Sugiura, Y2
Akimoto, Y; Fujiwara, M; Kurahashi, K; Sono, K1
Chiba, S; Haniuda, M; Itoh, N1
Katayama, E; Mitsui, T; Mizukawa, K; Ogawa, N; Ogura, T; Ota, Z; Takatori, K; Yamamoto, I1
Hasegawa, K; Inoue, S; Kawahara, Y; Nezuo, S; Sawayama, T; Tadaoka, S1
Fujioka, M; Ibengwe, JK; Komori, K; Nagao, T; Suzuki, H; Zhang, GL1
Nagatomo, T; Tsuchihashi, H1
Fukuta, S; Itagaki, T; Kusukawa, R; Toma, Y; Umemoto, S; Yamakawa, K; Yoshinaga, T1
Kanaide, H; Miwa-Nishimura, N; Nakamura, M; Nishimura, J1
Dan, Y; Fukui, K; Hirata, Y; Ishii, M; Matsuoka, H; Sugimoto, T1
Akima, M; Imagawa, J; Sakai, K1
Hirawa, N; Numabe, A; Takada, S; Uehara, Y; Yagi, S2
Mikami, H; Ogihara, T1
Hasegawa, A; Hatori, M; Murata, K; Nakano, A; Suzuki, T; Tamura, M2
Geshi, E; Hiroshige, J; Katagiri, T; Konno, N; Mochizuki, M; Umetsu, K1
Asada, S; Hirayama, A; Komamura, K; Lee, JM; Matsumura, Y; Mishima, M; Nishida, K; Ohara, T; Okazaki, Y; Yamamoto, K1
Fujii, T; Inoue, S; Nagai, K; Nakagawa, H1
Hasegawa, K; Inoue, S; Kakumae, S; Kawahara, Y; Nakamura, T; Nakao, M; Nezuo, S; Sawayama, T; Tadaoka, S1
Ebihara, A; Fujimura, A; Kumagai, Y; Nakashima, H; Oribe, H; Shitoh, T; Sugimoto, K1
Kaneko, M; Kimura, S; Shoumura, K1
Arakawa, K; Koga, S; Sasaki, J; Uzawa, H1
Matsumoto, M; Minami, M; Saito, H; Togashi, H; Yoshioka, M1
Haginaka, T; Katsumi, T; Murayama, K; Nakamura, T; Sakai, A; Tazika, E1
Matsui, Y; Nakai, M; Yamamoto, J1
Kato, T; Miyamoto, Y; Nakasone, J; Noguchi, K; Sakanashi, M; Takeo, S1
Hashimoto, J; Mitsuya, H; Miyake, K; Takaba, H; Yamamoto, M1
Ozawa, T; Sugiyama, S; Takamura, T1
Itoh, T; Kimoto, Y; Nozaki, M1
Ishibashi, Y; Kato, A; Miyake, Y1
Chiba, S; Ohkubo, H1
Chiba, S; Sinanović, O2
Ikegaki, I; Matsuzawa, M; Okabayashi, H; Suga, K; Takahashi, H; Yoshimura, M1
Orimo, H; Ouchi, Y; Watanabe, M1
Ikegaya, T; Kobayashi, A; Nishiyama, T; Yamazaki, N1
Hanaki, Y; Ozawa, T; Saito, H; Sugiyama, S1
Kuroiwa, A; Nakashima, Y; Sugano, M; Tasaki, H; Yashiro, A1
Iwata, S; Kato, A3
Azuma, T; Higa, S; Kishimoto, S; Mizuno, R; Sakoda, S; Suzuki, T; Tsujino, S; Watanabe, Y; Yoshida, H1
Matsumoto, M; Minematsu, R; Miyake, K; Takeo, S; Tanonaka, K1
Goto, K; Ishikawa, T; Kimura, S; Masaki, T; Yanagisawa, M1
Hasegawa, J; Hirai, S; Kotake, H; Mashiba, H; Saitoh, M1
Harada, T; Iida, H; Sone, T; Tanahashi, T; Tanaka, S; Tsukahara, I1
Kunieda, T; Naito, M; Nakanishi, N; Obayashi, Y; Okubo, S; Yoshioka, T1
Katayama, E; Mitsui, T; Mizukawa, K; Ogawa, N; Ogura, T; Ota, Z; Takatori, K1
Hashimoto, T; Kaguchi, Y; Kimura, M; Kuriyama, S; Miyahara, T; Nakamura, K; Tamai, K; Tamura, H1
Fujioka, M; Ibengwe, JK; Ishikawa, S; Komori, K; Nagao, T; Suzuki, H1
Ishikawa, Y; Kaneko, Y; Shindo, T; Toya, Y; Uchino, K; Umemura, S; Yasuda, G1
Ohno, M; Oishi, S; Sasaki, M; Sato, T; Umeda, T1
Ajioka, M; Nagai, S; Ozawa, T; Sugiyama, S; Takamura, T1
Chiba, S; Katsuyama, Y; Tada, A; Tsukada, M; Zenda, H1
Ebina, K; Fukuda, T; Nakamura, H; Nishizawa, O; Noto, H; Suzuki, K; Tsuchida, S1
Kakuta, Y; Kodera, T; Konishi, T; Koyama, T; Makino, K; Morimoto, Y; Nagano, K; Nakano, T; Takezawa, H; Umino, M1
Hirogami, M; Minami, M; Morii, K; Nomura, A; Saito, H; Saito, I; Sano, M; Tochihara, M; Togashi, H; Yoshioka, M1
Ishihara, Y; Kitamura, S; Kosaka, K; Yotsumoto, H1
Fujino, S; Hoshi, K1
Daiku, Y; Igarashi, T; Shoji, T1
Abe, I; Kawasaki, T; Kawazoe, N; Nakamuta, S; Omae, T; Ueno, M; Uezono, K1
Chiba, S; Furukawa, Y; Watanabe, H1
Shoji, T1
Fujimoto, S; Kida, O; Morotomi, Y; Tanaka, K1
Hata, F; Ishida, H; Kagawa, K; Kondo, E; Kondo, S1
Hattori, Y; Kanno, M1
Ludvig, N; Vizi, ES1
Fujimoto, T; Nakajima, S; Ohishi, M; Shiba, K; Takagi, O; Tsuya, Y; Uenishi, H1
Bando, S; Kakutani, A; Minezono, K; Mori, H; Noda, T; Shinomiya, H1
Itoh, K; Kohya, T; Minami, S; Nishijima, H; Tsujinaga, H; Yasuda, H1
Amagai, T; Fuse, T; Hirano, D; Kawazoe, K; Kitamura, K; Kiyotaki, S; Takimoto, Y1
Fujita, T; Kinoshita, K; Takahashi, T; Yamato, C1
Hamada, M; Kawanami, C; Konishi, T; Morimoto, Y; Nakai, K; Nakano, T; Noda, E; Takezawa, H; Yamamori, M1
Hattori, K; Kunitomo, M; Shimoura, K; Shinozuka, K1
Ishida, Y; Kawabe, K; Kurimoto, S; Moriyama, N; Nakamura, T; Orikasa, E1
Hirayama, T; Kikuchi, K; Morita, K; Ogawa, Y; Onodera, S; Takeda, A; Takenaka, T; Tobise, K1
Hibi, H; Miyake, K; Yamamoto, M4
Kitada, M; Mori, H; Takahashi, K; Tanabe, T; Usui, K1
Chiba, S; Vhora, S1
Gotoh, E; Ishii, M; Minamisawa, K; Minamisawa, M; Shionoiri, H; Sugimoto, K; Takasaki, I; Takizawa, T; Ueda, S1
Handa, S; Kitada, M; Mori, H; Takahashi, K; Tanabe, T; Yoshioka, K1
Kato, M; Kinugawa, T; Kitamura, H; Kotake, H; Mashiba, H; Matsumoto, T; Miyakoda, H; Noguchi, N; Ogino, K; Osaki, S1
Azuma, I1
De Luca, N; Fontana, D; Lamenza, F; Marchegiano, R; Sarno, D; Tozzi, N1
Azuma, I; Moriya, S; Oku, H; Shimizu, K; Sugiyama, T1
Kirsten, R; Weidinger, G1
Chiba, S; Nakane, T; Ren, LM1
Harder, S; Thürmann, P1
Inoue, M; Mori, C; Tanaka, O; Watanabe, K1
Aihara, M; Araie, M; Kaburaki, T; Shirato, S1
Anderton, JL; Gill, M; Notghi, A1
Galbiati, I; Gazzaniga, A; Gianesello, V; Soldati, L; Virno, M1
Kuwayama, Y; Matsugi, T; Nishimura, K; Shirasawa, E; Sun, N1
Chiba, S; Fujiwara, T1
Nagatomo, T; Shibata, A; Shimada, K; Tsuchihashi, H; Wakabayashi, H; Watanabe, K1
Kawamura, K; Kubota, J; Nishimura, H; Oka, T; Okabe, M; Ueyama, M1
Kono, M; Morita, S; Rubsamen, R1
Iwai, M; Shimazu, T1
Adachi, K; Hidaka, T; Muraishi, A; Okamoto, T; Seki, Y; Toshima, H1
Asano, M; Inagaki, O; Sudoh, K; Takenaka, T; Tanaka, H1
Fukuda, N; Izumi, Y; Kanmatsuse, K; Kubo, A; Matsuoka, M; Nakayama, T; Soma, M; Watanabe, Y1
Gatzka, C; Langenfeld, M; Schmieder, RE; Schobel, HP1
Weidinger, G1
Rieckert, H1
Herrmann, W; Schmitz, G; Stumpe, KO; Weidinger, G1
Eriksson, JW; Foley, K; Jansson, PA; Lithell, H1
Bönner, G; Chrosch, R; Schmieder, R; Weidinger, G1
Assmann, I; Bräutigam, M; Krönig, B; Langenfeld, MR; Schmieder, RE; Weidinger, G1
Inagaki, O; Sudoh, K; Takenaka, T1
Nasa, Y; Takeo, S; Yabe, K1
Rabl, W; Standl, E; Stemplinger, J; Stiegler, H; Weichenhain, B; Ziegler, AG1
Hara, Y; Harano, Y; Kanazawa, A; Nishioheda, Y; Ryomoto, K; Shinozaki, K; Suzuki, M; Tsushima, M1
Ishii, M; Umemura, S; Yasuda, G1
Arai, M; Fujiwara, H; Fujiwara, T; Kariya, T; Koshiji, M; Minatoguchi, S; Ohno, T; Uno, Y; Yamashita, K1
Asakura, Y; Ebihara, Y; Hasegawa, H; Nakamura, Y; Shinmura, K; Suganuma, Y; Tani, M1
Handa, S; Iwamoto, T; Kusuzaki, S; Takigawa, O; Tanabe, T; Usui, K; Yoshitake, M1
Suzuki, H1
Araie, M; Nagahara, M; Tamaki, Y; Tomidokoro, A; Tomita, K1
Meyer, U; Schmidt, J1
Camras, CB; Toris, CB; Wang, YL; Yablonski, ME; Zhan, GL1
Egashira, K; Ichiki, T; Katoh, M; Takeshita, A; Usui, M1
Fukuda, N; Hu, WY; Izumi, Y; Kanmatsuse, K; Soma, M1
Endo, T; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Satoh, Y; Suzuguchi, T1
Handa, S; Mori, H; Shinozaki, Y; Tanabe, T; Usui, K1
Koike, Y; Mineshita, S; Mizoguchi, H; Nomura, Y1
Mochizuki, Y; Oishi, M; Takasu, T1
Aikawa, M; Deguchi, Y; Handa, S; Tanabe, T; Yoshioka, K1
Akaike, T; Egashira, K; Funakoshi, H; Huang, P; Kandabashi, T; Miyata, K; Okamoto, S; Shimokawa, H; Takeshita, A; Yogo, K1
Araie, M; Koide, T; Mizuno, K; Yoshimura, M1
Endo, T; Hamaue, N; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Parvez, H1
Higaki, J; Kamide, K; Moriguchi, K; Nagai, M; Ogihara, T; Ohishi, M; Okamura, A; Rakugi, H; Satoh, N; Tuck, ML1
Kunitomo, M; Mizuno, H; Nakamura, K; Shinozuka, K1
Maehara, K; Maruyama, Y; Sakabe, A; Yaoita, H1
Kawai, T; Koshimizu, T; Nasa, Y; Oshikawa, S; Shinoura, H; Sunada, S; Takeo, S; Tanoue, A; Tsujimoto, G1
Iizuka, Y; Kashiwagi, K; Tsukahara, S1
Goto, W; Ikeda, T; Oku, H; Okuno, T; Sugiyama, T2
Akaishi, T; Hara, H; Kuwayama, Y; Matsugi, T; Miyawaki, N; Shimazaki, A1
Kobayashi, H; Kobayashi, K; Okinami, S1
Araie, M; Goto, W; Hara, H; Ichikawa, M; Tanaka, E1
Kawakami, S; Kawazu, K; Kitahara, T; Nakamura, J; Nakashima, M; Nishida, K; Sakanaka, K; Sasaki, H; Tomonari, M1
Akaishi, T; Hara, H; Ishida, N; Kashiwagi, K; Matsugi, T; Takagi, Y1
Araie, M; Asai, Y; Hara, H; Ichikawa, M; Ishii, K; Okada, Y1
Baba, K; Fujiwara, H; Kariya, T; Kawai, T; Minatoguchi, S; Takahashi, M; Takemura, G; Uno, Y; Zhang, C1
Araie, M; Hara, H; Ichikawa, M; Oku, H; Shimazawa, M1
Maehara, K; Maruyama, Y; Oikawa, Y; Saito, T; Tamagawa, K; Yaoita, H1
Nagano, M; Osada, Y; Yamaguchi, T1
Fujita, Y; Inamura, M; Koyama, T; Miyoshi, T; Ohashi, Y; Ohki, K; Okamoto, S; Oshika, T; Sakabe, I; Takahashi, K; Yasuma, T1
Ihara, S; Kawana, M; Sakai, R; Shimamoto, K; Watanabe, H1
Higashide, T; Sugiyama, K; Wakabayashi, T1
Narioka, J; Ohashi, Y1
Ji-Fei, T; Jia-Feng, L; Jiang-Hua, R; Li-Sha, G; Peng, C; Peng-Lin, Y; Yue-Chun, L; Zhan-Qiu, Y1
Chen, WP; Lee, AS; Su, MJ1
Goseki, T; Ishikawa, H; Nemoto, N; Nishimoto, H; Patil, PN; Shimizu, K; Uga, S1
Higuchi, S; Kawazu, K; Kitahara, T; Nakamura, J; Nakashima, M; Nishida, K; Sakanaka, K; Sasaki, H; Tomonari, M1
Levin, IaI; Strygin, KN1
Parati, G; Pengo, MF; Steier, J1

Reviews

6 review(s) available for bunazosin and quinazolines

ArticleYear
Periodic fluctuation of blood pressure and its management in a patient with pheochromocytoma. Case report and review of the literature.
    Japanese heart journal, 1988, Volume: 29, Issue:3

    Topics: Adrenal Gland Neoplasms; Antihypertensive Agents; Blood Pressure; Catecholamines; Ethanolamines; Humans; Hypertension; Male; Middle Aged; Periodicity; Pheochromocytoma; Quinazolines

1988
[Progress in medical treatment for glaucoma].
    Nippon Ganka Gakkai zasshi, 1993, Volume: 97, Issue:12

    Topics: Adrenergic alpha-Antagonists; Choroid; Dinoprost; Endothelins; Glaucoma; Humans; Intraocular Pressure; Ophthalmic Solutions; Quinazolines; Regional Blood Flow

1993
Pharmacokinetic and pharmacodynamic properties and therapeutic use of bunazosin in hypertension. A review.
    Arzneimittel-Forschung, 1995, Volume: 45, Issue:11

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Humans; Hypertension; Quinazolines

1995
Treatment of benign prostatic hyperplasia and hypertension in elderly hypertensive patients.
    British journal of urology, 1998, Volume: 81 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Aged; Female; Humans; Hypertension; Male; Multicenter Studies as Topic; Prazosin; Product Surveillance, Postmarketing; Prostatic Hyperplasia; Quinazolines; Randomized Controlled Trials as Topic

1998
Bunazosin, a selective alpha1-adrenoceptor antagonist, as an anti-glaucoma drug: effects on ocular circulation and retinal neuronal damage.
    Cardiovascular drug reviews, 2005,Spring, Volume: 23, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Eye; Glaucoma; Humans; Neurons; Optic Nerve; Quinazolines; Receptors, Adrenergic, alpha-1; Retina; Retinal Vessels

2005
The ANDANTE Project: A Worldwide Individual Data Meta-Analysis of the Effect of Sleep Apnea Treatment on Blood Pressure.
    Archivos de bronconeumologia, 2021, Volume: 57, Issue:11

    Topics: Blood Pressure; Continuous Positive Airway Pressure; Humans; Quinazolines; Sleep Apnea Syndromes

2021

Trials

32 trial(s) available for bunazosin and quinazolines

ArticleYear
Acute effect of an alpha 1-adrenoceptor antagonist on urinary sodium excretion, plasma atrial natriuretic peptide, arginine vasopressin, and the renin-aldosterone system in healthy subjects.
    European journal of clinical pharmacology, 1992, Volume: 43, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adult; Arginine Vasopressin; Atrial Natriuretic Factor; Enalapril; Humans; Male; Premedication; Quinazolines; Renin-Angiotensin System; Sodium

1992
[The evaluation of the effects of bunazosin hydrochloride in the treatment of prostatic hyperplasia].
    Hinyokika kiyo. Acta urologica Japonica, 1992, Volume: 38, Issue:5

    Topics: Adrenergic alpha-Antagonists; Aged; Drug Administration Schedule; Humans; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Urination

1992
Ocular responses in healthy subjects to topical bunazosin 0.3%--an alpha 1-adrenoceptor antagonist.
    The British journal of ophthalmology, 1991, Volume: 75, Issue:7

    Topics: Adrenergic alpha-Antagonists; Adult; Double-Blind Method; Eye; Eyelids; Female; Humans; Intraocular Pressure; Male; Middle Aged; Ophthalmic Solutions; Pupil; Quinazolines

1991
[The effect of bunazosin hydrochloride on intraocular pressure and aqueous humor dynamics in human].
    Nippon Ganka Gakkai zasshi, 1991, Volume: 95, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Female; Humans; Intraocular Pressure; Male; Quinazolines

1991
Effect of bunazosin hydrochloride on intraocular pressure and aqueous humor dynamics in normotensive human eyes.
    Archives of ophthalmology (Chicago, Ill. : 1960), 1991, Volume: 109, Issue:11

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Capillary Permeability; Dosage Forms; Dose-Response Relationship, Drug; Eye Proteins; Humans; Intraocular Pressure; Middle Aged; Quinazolines

1991
Renal effects of bunazosin, a new alpha 1-adrenoceptor blocker, in patients with mild-to-moderate essential hypertension.
    Journal of cardiovascular pharmacology, 1990, Volume: 15, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Female; Glomerular Filtration Rate; Hemodynamics; Humans; Hypertension; Kidney; Male; Middle Aged; Osmotic Pressure; Quinazolines; Renal Circulation; Vascular Resistance

1990
[A double-blind trial on the effect of bunazosin hydrochloride for the symptoms of benign prostatic hypertrophy].
    Hinyokika kiyo. Acta urologica Japonica, 1990, Volume: 36, Issue:10

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Alanine; Chi-Square Distribution; Double-Blind Method; Drug Combinations; Glutamates; Glycine; Humans; Japan; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Urination; Urination Disorders

1990
Enhancement by an ACE inhibitor of first-dose hypotension caused by an alpha 1-blocker.
    The New England journal of medicine, 1990, Apr-26, Volume: 322, Issue:17

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Cholinesterase Inhibitors; Drug Synergism; Enalapril; Humans; Quinazolines

1990
[Clinical evaluation of bunazosin hydrochloride for the treatment of voiding disturbances due to neurogenic bladder--a double-blind study].
    Hinyokika kiyo. Acta urologica Japonica, 1990, Volume: 36, Issue:10

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Bethanechol; Bethanechol Compounds; Chi-Square Distribution; Double-Blind Method; Female; Humans; Japan; Male; Middle Aged; Quinazolines; Urinary Bladder, Neurogenic; Urination; Urination Disorders

1990
[Clinical study of bunazosin hydrochloride, an alpha 1-adrenergic blocker, in benign prostatic obstruction and neurogenic bladder dysfunction].
    Hinyokika kiyo. Acta urologica Japonica, 1987, Volume: 33, Issue:9

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Evaluation; Humans; Male; Middle Aged; Prostatic Diseases; Prostatic Hyperplasia; Quinazolines; Urinary Bladder, Neurogenic; Urination; Urination Disorders

1987
[A double-blind trial on the effect of alpha-adrenergic blocker (bunazosin hydrochloride) in the symptomatic treatment of prostatism].
    Hinyokika kiyo. Acta urologica Japonica, 1987, Volume: 33, Issue:10

    Topics: Adrenergic alpha-Antagonists; Aged; Clinical Trials as Topic; Double-Blind Method; Humans; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Sympathetic Nervous System; Urination; Urination Disorders

1987
[Clinical efficacy of oxendolene (antiandrogen) and bunazosin hydrochloride (alpha-adrenergic blocker) in the treatment of prostatism--comparative study of oxendolone, bunazocin hydrochloride and their combination].
    Hinyokika kiyo. Acta urologica Japonica, 1987, Volume: 33, Issue:11

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Androgen Antagonists; Drug Evaluation; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nandrolone; Prostatic Hyperplasia; Quinazolines; Urinary Bladder Neck Obstruction; Urination

1987
Chronopharmacological study of bunazosin hydrochloride in healthy subjects.
    International journal of clinical pharmacology research, 1989, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Drug Evaluation; Fingers; Humans; Male; Quinazolines; Regional Blood Flow; Skin; Time Factors

1989
Comparative effects of bunazosin and propranolol on serum lipids and apolipoproteins in patients with essential hypertension.
    International journal of clinical pharmacology, therapy, and toxicology, 1989, Volume: 27, Issue:8

    Topics: Apolipoproteins; Blood Pressure; Female; Humans; Hypertension; Lipids; Lipoproteins; Male; Middle Aged; Multicenter Studies as Topic; Propranolol; Pulse; Quinazolines

1989
[A double blind clinical trial of the alpha-adrenergic blocker, Ea-0643 tablet, in the treatment of neurogenic bladder].
    Hinyokika kiyo. Acta urologica Japonica, 1985, Volume: 31, Issue:10

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Male; Middle Aged; Quinazolines; Tablets; Urinary Bladder, Neurogenic

1985
Comparison of the effectiveness of placebo and alpha-blocker therapy for the treatment of idiopathic oligozoospermia.
    Fertility and sterility, 1995, Volume: 63, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Double-Blind Method; Female; Humans; Infertility, Male; Male; Oligospermia; Placebos; Pregnancy; Quinazolines; Sperm Count; Sperm Motility

1995
Pharmacokinetics and pharmacodynamics of the alpha 1-adrenergic antagonist bunazosin retard in hypertensives.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:11

    Topics: Adrenergic alpha-1 Receptor Antagonists; Blood Pressure; Delayed-Action Preparations; Female; Half-Life; Humans; Hypertension; Kidney Diseases; Male; Middle Aged; Pulse; Quinazolines

1994
[Dose-response study of bunazosin in the treatment of light-to-moderate arterial hypertension].
    Minerva cardioangiologica, 1993, Volume: 41, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adult; Dose-Response Relationship, Drug; Drug Evaluation; Female; Humans; Hypertension; Male; Quinazolines

1993
[Treatment of essential hypertension with the alpha-1 antagonist bunazosin retard. A multicenter, double-blind, placebo-controlled study].
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Blood Pressure; Delayed-Action Preparations; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Posture; Quinazolines

1994
Concentration/effect relationship of bunazosin, a selective alpha 1-adrenoceptor antagonist in hypertensive patients after single and multiple oral doses.
    International journal of clinical pharmacology and therapeutics, 1994, Volume: 32, Issue:1

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Delayed-Action Preparations; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Quinazolines

1994
Renal haemodynamic effects of bunazosin retard and prazosin in mild to moderately hypertensive patients with normal or moderately impaired renal function.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 1994, Volume: 9, Issue:6

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Female; Glomerular Filtration Rate; Humans; Hypertension; Male; Middle Aged; Prazosin; Quinazolines; Renal Insufficiency; Renal Plasma Flow, Effective

1994
Treatment and post-treatment effects of alpha- versus beta-receptor blockers on left ventricular structure and function in essential hypertension.
    American heart journal, 1996, Volume: 132, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Double-Blind Method; Female; Heart Ventricles; Hemodynamics; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Metoprolol; Middle Aged; Quinazolines; Ventricular Function, Left

1996
Orthostatic hypotension: how to avoid it during antihypertensive therapy.
    American journal of hypertension, 1996, Volume: 9, Issue:11

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Antihypertensive Agents; Blood Pressure; Double-Blind Method; Humans; Hypertension; Hypotension, Orthostatic; Middle Aged; Plethysmography; Posture; Prazosin; Quinazolines; Regional Blood Flow; Vascular Resistance

1996
Effects of bunazosin and atenolol on serum lipids and apolipoproteins in a randomised trial.
    Blood pressure, 1996, Volume: 5, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Apolipoproteins; Atenolol; Double-Blind Method; Female; Humans; Hypertension; Lipids; Male; Middle Aged; Quinazolines; Treatment Outcome

1996
Insulin sensitivity following treatment with the alpha 1-blocker bunazosin retard and the beta 1-blocker atenolol in hypertensive non-insulin-dependent diabetes mellitus patients.
    Journal of hypertension, 1996, Volume: 14, Issue:12

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Aged; Atenolol; Blood Glucose; Blood Pressure; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Double-Blind Method; Female; Humans; Hypertension; Insulin; Male; Middle Aged; Quinazolines

1996
Effect of bunazosin and atenolol on glucose metabolism in obese, nondiabetic patients with primary hypertension.
    Cardiovascular drugs and therapy, 1997, Volume: 11, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Antihypertensive Agents; Atenolol; Blood Glucose; Double-Blind Method; Female; Glucose; Glucose Tolerance Test; Humans; Hypertension; Insulin; Lipids; Male; Middle Aged; Obesity; Quinazolines

1997
Antihypertensive efficacy and orthostatic tolerance of bunazosin vs nitrendipine: a multicentre double-blind randomized controlled study.
    Journal of human hypertension, 1996, Volume: 10, Issue:12

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Double-Blind Method; Humans; Hypertension; Lower Body Negative Pressure; Nitrendipine; Quinazolines

1996
Characterization of bunazosin-sensitive alpha1-adrenoceptors in human renal medulla.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Double-Blind Method; Female; Humans; In Vitro Techniques; Kidney Function Tests; Kidney Medulla; Male; Middle Aged; Prazosin; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha-1

1997
Effects of topical adrenergic agents on tissue circulation in rabbit and human optic nerve head evaluated with laser speckle tissue circulation analyzer.
    Survey of ophthalmology, 1997, Volume: 42 Suppl 1

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Animals; Betaxolol; Blood Circulation; Blood Flow Velocity; Blood Pressure; Carteolol; Double-Blind Method; Hemorheology; Humans; Intraocular Pressure; Ophthalmic Solutions; Optic Disk; Propanolamines; Quinazolines; Rabbits

1997
Pharmacokinetics and pharmacodynamics of bunazosin in patients with renal insufficiency.
    American journal of therapeutics, 1999, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Area Under Curve; Dose-Response Relationship, Drug; Female; Half-Life; Hemodynamics; Humans; Male; Middle Aged; Quinazolines; Renal Insufficiency; Time Factors

1999
Efficacy of bunazosin hydrochloride 0.01% as adjunctive therapy of latanoprost or timolol.
    Journal of glaucoma, 2004, Volume: 13, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aged; Drug Administration Schedule; Drug Therapy, Combination; Female; Glaucoma, Open-Angle; Humans; Intraocular Pressure; Latanoprost; Male; Middle Aged; Prostaglandins F, Synthetic; Pupil; Quinazolines; Timolol

2004
An alpha1-receptor blocker reduces plasma leptin levels in hypertensive patients with obesity and hyperleptinemia.
    Hypertension research : official journal of the Japanese Society of Hypertension, 2006, Volume: 29, Issue:10

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Body Mass Index; Delayed-Action Preparations; Fatty Acids, Nonesterified; Female; Heart Rate; Humans; Hypertension; Insulin Resistance; Leptin; Male; Middle Aged; Obesity; Quinazolines; Receptors, Leptin; Treatment Outcome

2006

Other Studies

187 other study(ies) available for bunazosin and quinazolines

ArticleYear
Increased uncoupling of beta-, beta 1- and beta 2-adrenoceptor to myocardial contraction in failing human myocardium.
    Japanese circulation journal, 1992, Volume: 56, Issue:7

    Topics: Adult; Aged; Binding, Competitive; Dobutamine; Down-Regulation; Female; Heart Failure; Humans; Iodocyanopindolol; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Pindolol; Quinazolines; Receptors, Adrenergic, beta; Terbutaline

1992
Case report: nifedipine-rifampicin interaction attenuates the effect on blood pressure in a patient with essential hypertension.
    The American journal of the medical sciences, 1992, Volume: 303, Issue:1

    Topics: Adrenergic alpha-Antagonists; Aged; Blood Pressure; Drug Interactions; Ethambutol; Female; Humans; Hypertension; Isoniazid; Nicardipine; Nifedipine; Propranolol; Quinazolines; Rifampin

1992
A biphasic effect of noradrenaline on renin release from rat juxtaglomerular cells in vitro is mediated by alpha 1- and beta-adrenoceptors.
    The Journal of endocrinology, 1992, Volume: 132, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Juxtaglomerular Apparatus; Norepinephrine; Perfusion; Propranolol; Quinazolines; Rats; Renin; Yohimbine

1992
[Usefulness and safety of bunazosin hydrochloride in neurogenic bladder after prolonged administration].
    Hinyokika kiyo. Acta urologica Japonica, 1992, Volume: 38, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Drug Evaluation; Female; Humans; Male; Middle Aged; Quinazolines; Safety; Time Factors; Urinary Bladder, Neurogenic

1992
A comparison of guanfacine, bunazosin, atenolol and nadolol on blood pressure and plasma noradrenaline responses to cold pressor testing.
    Clinical and experimental pharmacology & physiology, 1992, Volume: 19, Issue:7

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Atenolol; Blood Pressure; Cold Temperature; Guanfacine; Humans; Hypertension; Nadolol; Norepinephrine; Quinazolines; Receptors, Adrenergic; Stress, Physiological

1992
Effects of alpha-adrenoceptor antagonists and clonidine on the haemodynamic response to acute hypovolaemia in conscious rabbits.
    European journal of pharmacology, 1992, Jun-05, Volume: 216, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Drug Interactions; Heart Rate; Hemorrhage; Injections, Intravenous; Pharmaceutical Vehicles; Plasma Volume; Quinazolines; Rabbits; Yohimbine

1992
Effect of alpha 1-adrenoceptor blockade on the left ventricular force-length relationship in dogs.
    Japanese circulation journal, 1992, Volume: 56, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Myocardial Contraction; Quinazolines; Regression Analysis; Ventricular Function, Left

1992
Characterization of rat white fat cell alpha 1B-adrenoceptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Animals; Blotting, Northern; Epinephrine; Iodine Radioisotopes; Kinetics; Male; Membranes; Phenethylamines; Phosphatidylinositols; Propranolol; Quinazolines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; RNA, Messenger; Stimulation, Chemical; Tetralones; Tritium

1992
The effect of alpha 1-blocker, bunazosin on a murine model of congestive heart failure induced by viral myocarditis.
    Japanese circulation journal, 1992, Volume: 56, Issue:11

    Topics: Adrenergic alpha-Antagonists; Animals; Disease Models, Animal; Encephalomyocarditis virus; Enterovirus Infections; Heart Failure; Male; Mice; Mice, Inbred BALB C; Myocarditis; Myocardium; Quinazolines

1992
Bunazosin enhances receptor-mediated endocytosis of low-density lipoproteins.
    Artery, 1992, Volume: 19, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Endocytosis; Humans; Iodine Radioisotopes; Lipoproteins, LDL; Quinazolines; Receptors, LDL; Swine; Tumor Cells, Cultured

1992
Insulin insensitivity in nonobese, nondiabetic essential hypertension and its improvement by an alpha 1-blocker (bunazosin).
    American journal of hypertension, 1992, Volume: 5, Issue:12 Pt 1

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Apoproteins; Blood Glucose; Blood Pressure; Catecholamines; Diabetes Mellitus; Female; Glucose Tolerance Test; Humans; Hypertension; Insulin; Insulin Resistance; Lipids; Male; Middle Aged; Obesity; Quinazolines; Sodium

1992
[Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1992, Volume: 83, Issue:3

    Topics: Adenoma; Adrenergic alpha-Antagonists; Aged; Humans; Male; Piperazines; Prazosin; Prostatic Hyperplasia; Prostatic Neoplasms; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha

1992
Positive inotropic and negative chronotropic effects of (-)-cis-diltiazem in rat isolated atria.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Atenolol; Calcium; Diltiazem; Endothelium, Vascular; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Potassium Chloride; Quinazolines; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil

1992
Beta-3 adrenergic agonist, BRL-26830A, and alpha/beta blocker, arotinolol, markedly increase regional blood flow in the brown adipose tissue in anesthetized rats.
    Japanese circulation journal, 1992, Volume: 56, Issue:9

    Topics: Adipose Tissue, Brown; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Cardiac Output; Ethanolamines; Male; Propanolamines; Quinazolines; Rats; Rats, Wistar; Regional Blood Flow; Vascular Resistance

1992
[The acute and chronic effects of bunazosin on exercise capacity estimated by the anaerobic threshold in patients with chronic congestive heart failure].
    Kokyu to junkan. Respiration & circulation, 1992, Volume: 40, Issue:11

    Topics: Adult; Aged; Anaerobic Threshold; Chronic Disease; Exercise Test; Exercise Tolerance; Female; Heart Failure; Humans; Male; Middle Aged; Quinazolines

1992
Role of nitric oxide from the endothelium on the neurogenic contractile responses of rabbit pulmonary artery.
    European journal of pharmacology, 1992, Nov-03, Volume: 222, Issue:1

    Topics: Animals; Arginine; Chromatography, High Pressure Liquid; Electric Stimulation; Electrochemistry; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; Norepinephrine; Pulmonary Artery; Quinazolines; Rabbits; Sympathetic Nervous System; Tetrodotoxin

1992
Role of increased alpha 1-adrenergic activity in cardiomyopathic Syrian hamster.
    The American journal of physiology, 1991, Volume: 260, Issue:1 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channels; Cardiomegaly; Cardiomyopathies; Cricetinae; Dose-Response Relationship, Drug; Heart; Hydrolysis; Mesocricetus; Myocardium; Norepinephrine; Organ Size; Phosphatidylinositols; Quinazolines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Signal Transduction

1991
Chronic alpha 1 blockade in a patient with Eisenmenger syndrome.
    Pediatric cardiology, 1991, Volume: 12, Issue:1

    Topics: Adolescent; Adrenergic alpha-Antagonists; Eisenmenger Complex; Humans; Male; Quinazolines

1991
[Effect of moxisylyte on the lower urinary tracts (1). Effect on the isolated rabbit urethra and bladder].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Moxisylyte; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Prazosin; Quinazolines; Rabbits; Urethra; Urinary Bladder

1991
[Effect of moxisylyte on the lower urinary tracts (2). Effect on the urethra in anesthetized dogs].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Moxisylyte; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phenylephrine; Prazosin; Quinazolines; Urethra; Yohimbine

1991
Age-related changes in adrenergic alpha 1, alpha 2, and beta receptors of rat white fat cell membranes: an analysis using [3H]bunazosin as a novel ligand for the alpha 1 adrenoceptor.
    Journal of lipid research, 1991, Volume: 32, Issue:2

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aging; Animals; Binding Sites; Cell Membrane; Epididymis; Kinetics; Male; Obesity; Propanolamines; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1991
[Effects of topically applied bunazosin hydrochloride on choroidal capillary blood flow and intraocular pressure of rabbit eye].
    Nippon Ganka Gakkai zasshi, 1991, Volume: 95, Issue:5

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Capillaries; Choroid; Intraocular Pressure; Propranolol; Quinazolines; Rabbits; Regional Blood Flow

1991
Effects of long term treatment with an alpha 1 adrenoceptor blocker on cardiac hypertrophy, contractility, and myosin isoenzymes in spontaneously hypertensive rats.
    Cardiovascular research, 1991, Volume: 25, Issue:7

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Heart; Hypertension; Male; Myocardial Contraction; Myocardium; Myosins; Organ Size; Quinazolines; Rats; Rats, Inbred SHR; Time Factors

1991
[Ocular hypotensive effects of topically applied bunazosin, an alpha 1-adrenoceptor blocker, in rabbits and cats].
    Nippon Ganka Gakkai zasshi, 1991, Volume: 95, Issue:8

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Cats; Intraocular Pressure; Male; Quinazolines; Rabbits

1991
Comparison of alpha 1-adrenoceptors between rat brain and spleen.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Dibenzylchlorethamine; Kinetics; Male; Phenoxybenzamine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spleen

1991
[Fundamental and clinical studies on alpha 1-blocker therapy for idiopathic male infertility].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1991, Volume: 82, Issue:11

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Humans; Infertility, Male; Male; Prostate; Quinazolines; Sperm Motility; Testis; Vas Deferens

1991
Binding characteristics of alpha 1-adrenoceptors in bovine prostate using a radioligand binding assay.
    Journal of pharmacobio-dynamics, 1991, Volume: 14, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Cattle; Kinetics; Male; Membranes; Phentolamine; Prazosin; Prostate; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium

1991
Pharmacological features of vascular responses of isolated dog and monkey lingual arteries to vasoactive substances.
    Japanese journal of pharmacology, 1991, Volume: 57, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Macaca; Male; Norepinephrine; Perfusion; Potassium Chloride; Quinazolines; Tongue; Vasoconstrictor Agents

1991
Differential effects of antihypertensive agents on proliferation of vascular smooth muscle cells from spontaneously hypertensive rats.
    Japanese heart journal, 1991, Volume: 32, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Cell Division; Cells, Cultured; Hypertension; Male; Muscle, Smooth, Vascular; Nifedipine; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY

1991
Bunazosin, an alpha-adrenoceptor antagonist, blocks calcium current in guinea-pig ventricular myocytes.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1991, Volume: 100, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Guinea Pigs; Heart; Heart Ventricles; Quinazolines

1991
[3H]bunazosin, a novel selective radioligand of alpha 1 adrenoceptors in human prostates.
    The Journal of urology, 1991, Volume: 146, Issue:3

    Topics: Adrenergic alpha-Antagonists; Cell Membrane; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium

1991
[Characterization and localization of alpha 1-adrenoceptors in human prostate--with special reference to the zonal difference in receptor distribution].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1991, Volume: 82, Issue:8

    Topics: Autoradiography; Binding Sites; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Urinary Bladder Neoplasms

1991
Pharmacologic analysis of 7-O-ethyl-fangchinoline-induced vasodilation properties in isolated perfused common carotid arteries of Wistar Kyoto rats and spontaneously hypertensive rats.
    Chemical & pharmaceutical bulletin, 1991, Volume: 39, Issue:10

    Topics: Alkaloids; Animals; Atropine; Benzylisoquinolines; Carotid Arteries; Diltiazem; In Vitro Techniques; Isoproterenol; Male; Phenylephrine; Propranolol; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Vasoconstriction; Vasodilation; Vasodilator Agents

1991
Effects of regression of left ventricular hypertrophy following atenolol or bunazosin therapy on ischemic cardiac function and myocardial metabolism in spontaneously hypertensive rats.
    Japanese circulation journal, 1991, Volume: 55, Issue:12

    Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Atenolol; Blood Pressure; Cardiomegaly; Coronary Circulation; Coronary Disease; Lactates; Lactic Acid; Male; Myocardium; Phosphocreatine; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Remission Induction

1991
Effect of combined dopamine and bunazosin on the ischemic heart after occlusion of the coronary artery.
    The Japanese journal of surgery, 1990, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Arterial Occlusive Diseases; Cardiac Output, Low; Coronary Circulation; Coronary Disease; Dogs; Dopamine; Drug Evaluation, Preclinical; Drug Therapy, Combination; Hemodynamics; Infusions, Intravenous; Myocardium; Oxygen Consumption; Quinazolines

1990
Effects of bunazosin, a selective alpha 1-adrenergic blocking agent, on myocardial energy metabolism in ischemic dog heart.
    Japanese journal of pharmacology, 1990, Volume: 53, Issue:4

    Topics: Adenine Nucleotides; Adrenergic alpha-Antagonists; Animals; Carbohydrate Metabolism; Coronary Disease; Dogs; Electrocardiography; Energy Metabolism; Female; Heart; Hemodynamics; Hexosephosphates; In Vitro Techniques; Lactates; Male; Myocardium; Phosphocreatine; Pyruvates; Quinazolines

1990
Perfusion-time dependent enhancements of guanabenz- and KCl-induced vasoconstrictions in isolated and perfused dog pulmonary veins.
    Heart and vessels, 1990, Volume: 5, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Guanabenz; Imidazoles; Male; Potassium Chloride; Pulmonary Veins; Quinazolines; Receptors, Adrenergic, alpha; Time Factors; Vasoconstriction

1990
Intracerebroventricular injections of endothelin increase arterial pressure in conscious rats.
    Japanese circulation journal, 1990, Volume: 54, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Brain; Endothelins; Guanidines; Injections, Intraventricular; Male; Niacinamide; Nicardipine; Nicorandil; Pinacidil; Quinazolines; Rats; Rats, Inbred Strains; Vasodilator Agents

1990
[Changes in intraocular pressure and aqueous humor dynamics of normal human eyes after topical application of bunazosin hydrochloride].
    Nippon Ganka Gakkai zasshi, 1990, Volume: 94, Issue:8

    Topics: Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Depression, Chemical; Eye Proteins; Humans; Intraocular Pressure; Male; Middle Aged; Ophthalmic Solutions; Quinazolines

1990
[Efficacy of combination of Ea-0643 (bunazosin hydrochloride) and bethanechol chloride in patients with neurogenic bladder].
    Hinyokika kiyo. Acta urologica Japonica, 1990, Volume: 36, Issue:11

    Topics: Adrenergic alpha-Antagonists; Aged; Bethanechol; Bethanechol Compounds; Drug Evaluation; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Parasympathomimetics; Quinazolines; Urinary Bladder, Neurogenic

1990
Parasympathetic nervous system in patients with Graves' disease determined by R-R interval variations on electrocardiogram.
    Experimental and clinical endocrinology, 1990, Volume: 96, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adult; Electrocardiography; Female; Graves Disease; Humans; Male; Metoprolol; Parasympathetic Nervous System; Propranolol; Quinazolines; Receptors, Adrenergic, beta

1990
Predominant acetylcholine-induced vasoconstriction in isolated, perfused simian facial veins.
    European journal of pharmacology, 1990, Dec-04, Volume: 191, Issue:3

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Blood Pressure; Diltiazem; Face; Female; In Vitro Techniques; Macaca; Male; Muscle, Smooth, Vascular; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Potassium Chloride; Quinazolines; Receptors, Muscarinic; Saponins; Vasoconstriction; Veins

1990
Bunazosin induces use-dependent slowing of conduction in guinea-pig ventricular myocardium.
    European journal of pharmacology, 1990, Dec-04, Volume: 191, Issue:3

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Guinea Pigs; Heart Conduction System; In Vitro Techniques; Kinetics; Membrane Potentials; Papillary Muscles; Quinazolines

1990
Protective effects of nipradilol, isosorbide dinitrate, and bunazosin on coronary artery constriction induced by intracoronary injection of acetylcholine in pigs.
    Cardiovascular research, 1990, Volume: 24, Issue:12

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Coronary Angiography; Coronary Vessels; Dose-Response Relationship, Drug; Isosorbide Dinitrate; Propanolamines; Quinazolines; Vasoconstriction

1990
Inhibition of Ca2+ inward current in rabbit sinoatrial node by bunazosin, an alpha-adrenoceptor antagonist.
    European journal of pharmacology, 1987, Apr-07, Volume: 136, Issue:1

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Quinazolines; Rabbits; Sinoatrial Node

1987
Biochemical basis for reperfusion arrhythmias.
    Journal of molecular and cellular cardiology, 1987, Volume: 19 Suppl 5

    Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Coronary Circulation; Coronary Disease; Dogs; Female; Ion Channels; Male; Mitochondria, Heart; Myocardium; Phospholipases; Quinazolines

1987
Postjunctional alpha-adrenoceptor subtypes in isolated and perfused canine epicardial coronary arteries.
    Journal of cardiovascular pharmacology, 1987, Volume: 10, Issue:6

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Coronary Vessels; Dogs; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Quinazolines; Receptors, Adrenergic, alpha; Vasoconstriction; Vasodilation; Xylazine

1987
Effects of intraocular pressure change on movement of FITC-dextran across vitreous-aqueous interface.
    Japanese journal of ophthalmology, 1989, Volume: 33, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Anterior Chamber; Aqueous Humor; Dextrans; Female; Fluorescein-5-isothiocyanate; Fluoresceins; Fluorometry; Intraocular Pressure; Male; Quinazolines; Rabbits; Vitreous Body

1989
Effects of specific alpha-adrenoceptive agents on extraneuronal uptake (uptake2) of isoproterenol in perfused rat heart.
    Life sciences, 1989, Volume: 44, Issue:14

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Guanabenz; Isoproterenol; Male; Methoxamine; Myocardium; Neurons; Phenylephrine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Sulfonamides; Tropolone

1989
Time-dependent enhancement of xylazine-induced, alpha-2 adrenoceptor-mediated vasoconstriction in isolated and perfused canine pulmonary veins.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Dogs; Endothelium, Vascular; Female; Imidazoles; In Vitro Techniques; Male; Perfusion; Pulmonary Veins; Quinazolines; Receptors, Adrenergic, alpha; Saponins; Thiazines; Time Factors; Vasoconstriction; Xylazine

1989
Localization of alpha 1-adrenoceptor in the rat kidney: in vitro autoradiography using [3H]-bunazosin.
    Research communications in chemical pathology and pharmacology, 1989, Volume: 64, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; In Vitro Techniques; Kidney; Kidney Cortex; Kidney Medulla; Male; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1989
[Acute and chronic effects of bunazosin in patients with congestive heart failure].
    Kokyu to junkan. Respiration & circulation, 1989, Volume: 37, Issue:5

    Topics: Adrenergic alpha-Antagonists; Atrial Natriuretic Factor; Chronic Disease; Exercise Test; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines

1989
Bunazosin, an alpha 1-adrenoceptor blocker, differentially releases co-transmitters in dog mesenteric vessels.
    European journal of pharmacology, 1989, May-02, Volume: 164, Issue:1

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Dogs; In Vitro Techniques; Mesenteric Arteries; Mesenteric Veins; Methoxyhydroxyphenylglycol; Muscle, Smooth, Vascular; Neurotransmitter Agents; Norepinephrine; Phentolamine; Quinazolines; Yohimbine

1989
Alpha-blocking potencies of antihypertensive agents (prazosin, terazosin, bunazosin, SGB-1534 and ketanserin) having with quinazoline or quinazolinedione as assessed by radioligand binding assay methods in rat brain.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brain; Cell Membrane; Clonidine; Dihydroalprenolol; Ketanserin; Male; Prazosin; Quinazolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1989
Hemodynamic benefits of long-term bunazosin (alpha-1 blocker) therapy in rats with myocardial infarction and heart failure.
    Japanese circulation journal, 1989, Volume: 53, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiac Output, Low; Chronic Disease; Female; Heart Ventricles; Hemodynamics; Myocardial Infarction; Quinazolines; Rats; Rats, Inbred Strains; Vascular Resistance; Weight Gain

1989
Selective blockade of alpha 1-adrenoceptors of porcine vascular smooth muscle cells by bunazosin.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; In Vitro Techniques; Membranes; Microsomes; Muscle, Smooth, Vascular; Muscles; Prazosin; Quinazolines; Swine; Yohimbine

1989
Renal and hormonal effects of alpha 1-adrenoceptor blockade by bunazosin in essential hypertension.
    European journal of clinical pharmacology, 1989, Volume: 36, Issue:6

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Atrial Natriuretic Factor; Blood Pressure; Creatinine; Glomerular Filtration Rate; Humans; Hypertension; Kidney; Norepinephrine; Quinazolines; Regional Blood Flow; Vascular Resistance

1989
In vivo experiments for the evaluation of alpha 1-adrenoceptor antagonistic effects of SGB-1534 on canine urethra.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Dose-Response Relationship, Drug; Female; Hypogastric Plexus; Phenylephrine; Prazosin; Quinazolines; Urethra

1989
[Roles of vascular and renal thromboxanes in the antihypertensive effects of alpha 1 adrenoceptor antagonists].
    Nihon Jinzo Gakkai shi, 1989, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Vessels; Hypertension; Kidney; Male; Methacrylates; Quinazolines; Rats; Rats, Inbred SHR; Thromboxane A2; Thromboxane-A Synthase

1989
[Clinical application of adrenoceptor blockers in the treatment of hypertension].
    Nihon rinsho. Japanese journal of clinical medicine, 1989, Volume: 47, Issue:9

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Carbazoles; Carvedilol; Humans; Hypertension; Labetalol; Prazosin; Propanolamines; Quinazolines

1989
[Exercise testing of the chronic effects of bunazosin hydrochloride on dilated cardiomyopathy].
    Kokyu to junkan. Respiration & circulation, 1989, Volume: 37, Issue:10

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Cardiomyopathy, Dilated; Drug Evaluation; Exercise Test; Female; Hemodynamics; Humans; Male; Middle Aged; Quinazolines

1989
Protection of acute ischemic myocardial injury by pharmacological intervention.
    Japanese circulation journal, 1989, Volume: 53, Issue:9

    Topics: Adenosine Triphosphatases; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium-Transporting ATPases; Coenzymes; Coronary Disease; Diltiazem; Dogs; Myocardium; Niacinamide; Nicorandil; Quinazolines; Sarcoplasmic Reticulum; Ubiquinone; Vasodilator Agents

1989
[Acute effects of oral bunazosin-hydrochloride in acute heart failure].
    Kokyu to junkan. Respiration & circulation, 1989, Volume: 37, Issue:11

    Topics: Acute Disease; Administration, Oral; Adrenergic alpha-Antagonists; Aged; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines

1989
Involvement of adrenergic mechanism in hyperglycemia due to SCN stimulation.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1989, Volume: 21, Issue:12

    Topics: Adrenergic alpha-Antagonists; Animals; Autonomic Nervous System; Electric Stimulation; Female; Glucagon; Hexamethonium; Hexamethonium Compounds; Hyperglycemia; Insulin; Propranolol; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Suprachiasmatic Nucleus; Yohimbine

1989
[The effect of bunazosin vs captopril on hemodynamic and neurohumoral parameters in patients with congestive heart failure].
    Kokyu to junkan. Respiration & circulation, 1989, Volume: 37, Issue:12

    Topics: Adrenergic alpha-Antagonists; Aldosterone; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Atrial Natriuretic Factor; Captopril; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines; Renin

1989
Exercise testing of the chronic effects of bunazosin hydrochloride on dilated cardiomyopathy.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:12

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Cardiomyopathy, Dilated; Echocardiography; Electrocardiography; Exercise Test; Female; Hemodynamics; Humans; Male; Middle Aged; Quinazolines

1989
Properties of the pupillary dilation produced by the humoral factor in the pupillary reflex dilation: an experimental study in the cat.
    Japanese journal of ophthalmology, 1989, Volume: 33, Issue:4

    Topics: Animals; Atropine; Biological Factors; Cats; Electric Stimulation; Iris; Phenoxybenzamine; Propranolol; Quinazolines; Reflex, Pupillary; Sciatic Nerve; Yohimbine

1989
Effect of bunazosin on cardiac sympathetic nerve activity in anesthetized rats.
    Clinical and experimental hypertension. Part A, Theory and practice, 1989, Volume: 11, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Heart Conduction System; Heart Rate; Kidney; Male; Nervous System; Nervous System Physiological Phenomena; Quinazolines; Rats; Rats, Inbred Strains; Sympathetic Nervous System

1989
Perfusion-time-dependent appearance of blocking effect of diltiazem on norepinephrine-induced vasoconstriction in isolated, perfused dog pulmonary veins.
    Japanese journal of pharmacology, 1989, Volume: 49, Issue:1

    Topics: Animals; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Perfusion; Propranolol; Pulmonary Veins; Quinazolines; Time Factors; Vasoconstriction

1989
Acute systemic and regional hemodynamic effects of alpha 1-adrenoceptor blockade in conscious spontaneously hypertensive rats.
    Clinical and experimental hypertension. Part A, Theory and practice, 1986, Volume: 8, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Consciousness; Dose-Response Relationship, Drug; Hemodynamics; Hypertension; Male; Quinazolines; Rats; Rats, Inbred SHR; Regional Blood Flow

1986
Acute effects of bunazosin on aortic, vertebral, coronary and renal blood flows of anesthetized dogs.
    Arzneimittel-Forschung, 1986, Volume: 36, Issue:8

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Aorta; Coronary Circulation; Dogs; Female; Male; Quinazolines; Regional Blood Flow; Renal Circulation; Time Factors; Vascular Resistance; Vertebral Artery; Yohimbine

1986
Successful treatment of oligospermic and azoospermic men with alpha 1-blocker and beta-stimulator: new treatment for idiopathic male infertility.
    Fertility and sterility, 1986, Volume: 46, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Ethanolamines; Female; Humans; Infertility, Male; Male; Oligospermia; Pregnancy; Procaterol; Quinazolines; Sperm Count; Sperm Motility; Time Factors

1986
Effects of bunazosin and propranolol on ventricular arrhythmias in dogs with hypokalemia.
    Journal of electrocardiology, 1987, Volume: 20, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dogs; Female; Heart Ventricles; Hypokalemia; Male; Mitochondria, Heart; Potassium; Propranolol; Quinazolines; Sodium

1987
Actions of the alpha-1 adrenoceptor blocker bunazosin on the norepinephrine-induced contraction of smooth muscles in the rabbit proximal urethra.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Calcium; Dose-Response Relationship, Drug; Guanethidine; Microelectrodes; Muscle Contraction; Muscle, Smooth; Norepinephrine; Potassium; Propranolol; Quinazolines; Rabbits; Urethra

1987
Effect of egg yolk lecithin on transdermal delivery of bunazosin hydrochloride.
    The Journal of pharmacy and pharmacology, 1987, Volume: 39, Issue:5

    Topics: Adjuvants, Pharmaceutic; Administration, Cutaneous; Adrenergic alpha-Antagonists; Animals; Egg Yolk; In Vitro Techniques; Male; Mice; Mice, Hairless; Phosphatidylcholines; Quinazolines; Rabbits; Skin Absorption

1987
Pharmacological analysis of vasoconstriction of isolated canine ophthalmic and ciliary arteries to alpha-adrenoceptor agonists.
    Experimental eye research, 1987, Volume: 45, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Ciliary Body; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Nitroprusside; Ophthalmic Artery; Quinazolines; Vasoconstriction

1987
Potentiating effect of tyramine on acetaldehyde-induced vasoconstriction in isolated dog mesenteric arteries.
    Japanese journal of pharmacology, 1987, Volume: 44, Issue:3

    Topics: Acetaldehyde; Adrenergic alpha-Antagonists; Animals; Dogs; In Vitro Techniques; Mesenteric Arteries; Norepinephrine; Quinazolines; Tachyphylaxis; Tyramine; Vasoconstriction

1987
Pharmacological analysis of 5-HT-induced vasoconstriction in isolated, perfused dog skeletal muscle arteries.
    European journal of pharmacology, 1987, Nov-17, Volume: 143, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Cold Temperature; Diltiazem; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Quinazolines; Serotonin; Vasoconstriction

1987
Sympatholytic effects of the intravenously injected alpha 1-adrenergic blocker, bunazosin, in anaesthetized rats.
    Journal of hypertension, 1987, Volume: 5, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Denervation; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Phentolamine; Phenylephrine; Pressoreceptors; Quinazolines; Rats; Rats, Inbred Strains; Sympathetic Nervous System

1987
Alpha-blocker, bunazosinhydrochloride decreases cytosolic Ca++ of cultured rat aortic smooth muscle cells.
    Biochemical and biophysical research communications, 1988, Feb-15, Volume: 150, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Calcium; Cells, Cultured; Cytosol; Kinetics; Muscle, Smooth, Vascular; Phenylephrine; Quinazolines; Rats; Rats, Inbred Strains

1988
Role of alpha 1-adrenergic receptors and the effect of bunazosin on the histopathology of cardiomyopathic Syrian hamsters of strain BIO 14.6.
    Japanese circulation journal, 1988, Volume: 52, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Cardiomyopathies; Cricetinae; Female; Male; Mesocricetus; Myocardium; Quinazolines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1988
Effect of the alpha 1-blocker bunazosin on reperfusion-induced mitochondrial dysfunction in canine hearts.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dogs; Female; In Vitro Techniques; Male; Mitochondria, Heart; Oxygen Consumption; Perfusion; Phospholipases; Quinazolines

1988
Effects of a new alpha 1-blocker, bunazosin hydrochloride, on plasma lipid components in hypertensive patients with hypercholesterolemia.
    Clinical therapeutics, 1987, Volume: 10, Issue:1

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Apolipoproteins; Blood Pressure; Cholesterol; Female; Humans; Hypercholesterolemia; Hypertension; Lipids; Lipoproteins; Male; Middle Aged; Quinazolines; Triglycerides

1987
In vitro study on corneal permeability to bunazosin.
    Journal of pharmacobio-dynamics, 1988, Volume: 11, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Caprylates; Cornea; Decanoic Acids; In Vitro Techniques; Octanols; Permeability; Quinazolines; Rabbits; Water

1988
The aortic alpha 1-adrenergic receptor in familial amyloidotic polyneuropathy.
    Journal of neural transmission, 1988, Volume: 73, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amyloidosis; Aorta; Female; Humans; Male; Middle Aged; Peripheral Nervous System Diseases; Quinazolines; Receptors, Adrenergic, alpha

1988
Cardioprotective action of alpha-blocking agents, phentolamine and bunazosin, on hypoxic and reoxygenated myocardium.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:2

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Energy Metabolism; Heart; Hypoxia; Male; Myocardial Contraction; Myocardium; Oxygen; Phentolamine; Quinazolines; Rabbits

1988
Corneal permeability to bunazosin in rabbits.
    Journal of pharmacobio-dynamics, 1988, Volume: 11, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Cornea; Male; Permeability; Quinazolines; Rabbits

1988
Studies on improved corneal permeability to bunazosin.
    Journal of pharmacobio-dynamics, 1988, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Caprylates; Chromatography, High Pressure Liquid; Cornea; Hydrogen-Ion Concentration; In Vitro Techniques; Permeability; Protein Binding; Quinazolines; Rabbits

1988
Positive inotropic action of novel vasoconstrictor peptide endothelin on guinea pig atria.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Atenolol; Atrial Function; Calcium; Cimetidine; Diphenhydramine; Endothelins; Guinea Pigs; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Methysergide; Myocardial Contraction; Nicardipine; Peptides; Potassium; Quinazolines; Reference Values

1988
[The effect of bunazosin hydrochloride on the intraocular pressure and the aqueous humor dynamics of the rabbit eye].
    Nippon Ganka Gakkai zasshi, 1988, Volume: 92, Issue:7

    Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Female; Intraocular Pressure; Quinazolines; Rabbits

1988
Antiarrhythmic effects of alpha-adrenoceptor antagonists in guinea pig ventricular myocardium.
    Journal of the American College of Cardiology, 1988, Volume: 12, Issue:6

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Guinea Pigs; Heart; In Vitro Techniques; Quinazolines; Receptors, Adrenergic, beta; Strophanthidin

1988
[The effect of bunazosin on hypertension during anesthesia; effectiveness of nasal instillation].
    Masui. The Japanese journal of anesthesiology, 1988, Volume: 37, Issue:10

    Topics: Administration, Intranasal; Adrenergic alpha-Antagonists; Anesthesia, General; Female; Humans; Hypertension; Male; Middle Aged; Quinazolines

1988
Effects of selective alpha 1-adrenoceptor blockade in dogs with hypoxic pulmonary vasoconstriction.
    Japanese circulation journal, 1988, Volume: 52, Issue:10

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Gas Analysis; Dogs; Hemodynamics; Hypertension, Pulmonary; Hypoxia; Pulmonary Circulation; Quinazolines; Vasoconstriction

1988
Possible mechanism of acetaldehyde-induced noradrenaline release from sympathetic nerve terminals in isolated blood vessels.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Acetaldehyde; Adrenergic alpha-Antagonists; Animals; Dogs; Hydrocortisone; In Vitro Techniques; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Quinazolines; Sympathetic Nervous System; Tachyphylaxis; Tyramine; Vasoconstriction

1988
Properties of [3H]bunazosin binding in rat kidney.
    Clinical therapeutics, 1988, Volume: 10, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Cations; Hot Temperature; Kidney; Kidney Cortex; Kinetics; Male; Membranes; Quinazolines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Subcellular Fractions; Tissue Distribution; Tritium

1988
The effects of vasoactive agents on the proliferation of vascular smooth muscle cells grown in vitro.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:4

    Topics: Amiloride; Animals; Captopril; Cell Division; Cells, Cultured; Chlorpromazine; In Vitro Techniques; Labetalol; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Nifedipine; Norepinephrine; Propranolol; Quinazolines; Rats; Sulfonamides

1988
Effects of bunazosin on electrical responses of smooth muscle cells of the guinea-pig mesenteric artery and vein to perivascular nerve stimulation and to noradrenaline.
    General pharmacology, 1987, Volume: 18, Issue:2

    Topics: Animals; Electric Stimulation; Evoked Potentials; Female; Guinea Pigs; Male; Membrane Potentials; Mesenteric Arteries; Mesenteric Veins; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Yohimbine

1987
Existence of renal alpha 1- and alpha 2-adrenoceptors in the human kidney: radioligand binding study in membranes from the human renal cortex and medulla.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1986, Volume: 4, Issue:6

    Topics: Humans; Kidney; Kidney Cortex; Kidney Medulla; Membranes; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1986
Mechanism of myocardial injury in dogs with hypokalaemia.
    Cardiovascular research, 1988, Volume: 22, Issue:4

    Topics: Animals; Calcium; Cardiomyopathies; Coronary Circulation; Creatine Kinase; Dogs; Epinephrine; Female; Hypokalemia; Male; Mitochondria, Heart; Myocardium; Quinazolines

1988
Different antagonistic effects of bunazosin and ketanserin on the norepinephrine-induced vasoconstriction in isolated, perfused canine and simian skeletal muscle arteries.
    Japanese journal of pharmacology, 1988, Volume: 46, Issue:2

    Topics: Animals; Arteries; Dogs; Female; In Vitro Techniques; Ketanserin; Macaca; Male; Muscles; Norepinephrine; Quinazolines; Regional Blood Flow; Vasoconstriction

1988
Vasoconstrictor effects of endogenous digitalis-like factors extracted from urine of hypertensive patients.
    Heart and vessels, 1987, Volume: 3, Issue:3

    Topics: Animals; Arteries; Blood Proteins; Cardenolides; Digoxin; Dogs; Ear, External; Epinephrine; Humans; Hypertension; In Vitro Techniques; Mesenteric Arteries; Ouabain; Phentolamine; Potassium Chloride; Quinazolines; Saponins; Vasoconstrictor Agents; Verapamil

1987
[Effect of bunazosin on lower urinary tract function in the decerebrated dog].
    Hinyokika kiyo. Acta urologica Japonica, 1987, Volume: 33, Issue:11

    Topics: Animals; Decerebrate State; Dogs; Electric Stimulation; Electromyography; Pons; Quinazolines; Urethra; Urinary Bladder

1987
[Effects of oral bunazosin hydrochloride on hemodynamic and metabolic responses to exercise (ergometer, 25W, 5 min) in patients with severe congestive heart failure].
    Kokyu to junkan. Respiration & circulation, 1987, Volume: 35, Issue:2

    Topics: Aged; Exercise Test; Female; Heart Failure; Hemodynamics; Humans; Male; Metabolism; Middle Aged; Quinazolines

1987
[Effects of new antihypertensive agent, 2-[4-(n-butyryl)-homopiperazine-1-ul]-4-amino-6, 7-dimethoxy-quinazoline (E-643), on blood pressure, urinary sodium excretion and urinary norepinephrine excretion rate in stroke-prone, spontaneously hypertensive rat
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1985, Volume: 60, Issue:4

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Body Weight; Catecholamines; Cerebrovascular Disorders; Eating; Heart Rate; Humans; Hypertension; Kidney; Male; Natriuresis; Norepinephrine; Potassium; Quinazolines; Rats; Rats, Inbred SHR

1985
The potentiating effect of an alpha-adrenergic blocking agent (E-643) on the action of bronchodilators.
    Arzneimittel-Forschung, 1980, Volume: 30, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Bronchodilator Agents; Cyclic AMP; Cyclic GMP; Drug Synergism; Epinephrine; Guinea Pigs; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Prostaglandins E; Quinazolines; Trachea

1980
Effects of alpha blockers on blood pressure and on the Ca-contracture of cat aortic strips.
    Japanese journal of pharmacology, 1980, Volume: 30, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Blood Pressure; Calcium; Cats; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Phentolamine; Quinazolines; Regional Blood Flow

1980
alpha-Adrenoceptor blocking properties of a new antihypertensive agent, 2-[4-(n-butyryl)-homopiperazine-1-yl]-4-amino-6,7-dimethoxyquinazoline (E-643).
    Japanese journal of pharmacology, 1980, Volume: 30, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Barium; Blood Pressure; Calcium; Dose-Response Relationship, Drug; Epinephrine; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Phentolamine; Potassium; Quinazolines; Rabbits; Rats; Vasoconstriction

1980
Antihypertensive effect of E-643, a new alpha-adrenergic blocking agent.
    European journal of clinical pharmacology, 1981, Volume: 20, Issue:6

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aldosterone; Blood Pressure; Chemical Phenomena; Chemistry; Dopamine beta-Hydroxylase; Epinephrine; Female; Humans; Male; Middle Aged; Norepinephrine; Posture; Pulse; Quinazolines; Renin

1981
Chronotropic and inotropic effects of 3 kinds of alpha-adrenergic blockers on the isolated dog atria.
    Japanese heart journal, 1981, Volume: 22, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Atropine; Dogs; Female; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Phenoxybenzamine; Phentolamine; Propranolol; Quinazolines

1981
Comparison of pre- and postsynaptic alpha-adrenoceptor blocking effects of E-643 in the isolated vas deferens of the rat.
    Japanese journal of pharmacology, 1981, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens

1981
[Effects of quinazoline derivatives (E-643 and prazosin) on blood pressure, pulse and renin-angiotensin system in two cases of pheochromocytoma (author's transl)].
    Nihon Jinzo Gakkai shi, 1981, Volume: 23, Issue:8

    Topics: Adolescent; Adrenal Gland Neoplasms; Adrenergic alpha-Antagonists; Adult; Blood Pressure; Humans; Male; Pheochromocytoma; Prazosin; Pulse; Quinazolines; Renin-Angiotensin System

1981
Characteristics of [3H]E-643-binding to alpha adrenoceptors.
    Japanese journal of pharmacology, 1982, Volume: 32, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Binding Sites; Binding, Competitive; Brain; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Protein Binding; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Temperature; Tritium

1982
Effect of E-643 on alpha-adrenoceptor-mediated inotropic responses to phenylephrine in the left atria of guinea pigs.
    Japanese journal of pharmacology, 1982, Volume: 32, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Guinea Pigs; Heart Atria; In Vitro Techniques; Myocardial Contraction; Phenylephrine; Quinazolines; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Sotalol; Stimulation, Chemical

1982
(-)-Amidephrine, a selective agonist for alpha 1-adrenoceptors.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Electric Stimulation; Ethanolamines; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Quinazolines; Rats; Vas Deferens

1983
[Effects and site of action of alpha-receptor blocker in bronchial asthma].
    Nihon Kyobu Shikkan Gakkai zasshi, 1983, Volume: 21, Issue:5

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Asthma; Dinoprost; Female; Humans; Male; Metaproterenol; Middle Aged; Prostaglandins F; Quinazolines

1983
[Effects of E-643 on the regional myocardial function and hemodynamics in experimental acute coronary artery occlusion].
    Kokyu to junkan. Respiration & circulation, 1983, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Coronary Disease; Dogs; Hemodynamics; Myocardial Contraction; Quinazolines

1983
[Acute effect of a new alpha 1-receptor blocking drug, E-643, on severe congestive heart failure--pharmacokinetic and hemodynamic studies].
    Kokyu to junkan. Respiration & circulation, 1983, Volume: 31, Issue:10

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Drug Evaluation; Female; Heart Failure; Hemodynamics; Humans; Kinetics; Male; Middle Aged; Quinazolines

1983
[Clinical effect of new alpha-adrenergic blocker on micturition disturbance of neurogenic bladder and lower urinary tract obstruction].
    Hinyokika kiyo. Acta urologica Japonica, 1983, Volume: 29, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Female; Humans; Male; Middle Aged; Quinazolines; Urethral Obstruction; Urinary Bladder, Neurogenic; Urodynamics

1983
The metabolic fate of 4-amino-2-(4-butanoyl-hexahydro-1H-1, 4-diazepin-1-yl)-6,7-dimethoxy-quinazoline HCl.
    Xenobiotica; the fate of foreign compounds in biological systems, 1982, Volume: 12, Issue:9

    Topics: Adult; Animals; Bile; Enterohepatic Circulation; Feces; Female; Humans; In Vitro Techniques; Intestinal Absorption; Male; Microsomes, Liver; Quinazolines; Rabbits; Rats; Rats, Inbred Strains; Tissue Distribution

1982
[Acute effects of a new antihypertensive quinazoline derivative, E-643 in severe heart failure--hemodynamics, plasma catecholamine levels and blood gas data (author's transl)].
    Kokyu to junkan. Respiration & circulation, 1981, Volume: 29, Issue:7

    Topics: Adult; Aged; Catecholamines; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines

1981
Participation of endogenous noradrenaline in the release of ATP by high potassium in the rat caudal artery.
    Japanese journal of pharmacology, 1995, Volume: 68, Issue:1

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Arteries; In Vitro Techniques; Male; Norepinephrine; Potassium; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha

1995
Effect of bunazosin, alpha 1-adrenoceptor blocker, on multidirectional contractile response and localization of bunazosin binding sites in human hypertrophied prostate.
    General pharmacology, 1995, Volume: 26, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Autoradiography; Binding Sites; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prostate; Prostatic Hyperplasia; Quinazolines; Receptors, Adrenergic, alpha-1

1995
Comparison of 5-hydroxytryptamine-induced contraction of rat pulmonary artery to that of aorta in vitro.
    Japanese circulation journal, 1995, Volume: 59, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Ketanserin; Male; Pindolol; Pulmonary Artery; Quinazolines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Ritanserin; Serotonin; Vasoconstriction

1995
Effects of alpha-blocker on sperm concentration, motility, intraluminal pressure and fluid movement in the rat cauda epididymis.
    The Journal of urology, 1995, Volume: 154, Issue:2 Pt 1

    Topics: Adrenergic alpha-Antagonists; Animals; Body Fluids; Epididymis; Male; Organ Size; Pressure; Quinazolines; Rats; Rats, Sprague-Dawley; Seminiferous Tubules; Sperm Count; Sperm Motility; Testis

1995
Effects of bunazosin, a selective alpha 1-blocking agent, and propranolol used alone and in combination on canine ventricular refractoriness and its dispersion during myocardial ischemia.
    Journal of cardiovascular pharmacology, 1993, Volume: 21, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Coronary Circulation; Dogs; Drug Therapy, Combination; Electrocardiography; Injections, Intravenous; Myocardial Ischemia; Propranolol; Quinazolines

1993
Functional 5-HT receptor subtypes in the isolated canine common carotid artery.
    Heart and vessels, 1994, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Carotid Artery, Common; Diltiazem; Dogs; Female; Ketanserin; Male; Methysergide; Norepinephrine; Potassium Chloride; Quinazolines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spiperone; Vasoconstriction

1994
Effects of sympathetic stimulation, with and without previous alpha 1 and beta adrenoceptor blockade, on refractoriness dispersion in canine heart.
    Cardiovascular research, 1994, Volume: 28, Issue:12

    Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Electrophysiology; Heart; Myocardial Ischemia; Propranolol; Quinazolines; Stimulation, Chemical; Sympathetic Nervous System

1994
Acute hemodynamic effects of bunazosin in congestive heart failure--differing responses according to degree of cardiac dysfunction.
    General pharmacology, 1993, Volume: 24, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Female; Heart; Heart Failure; Heart Rate; Hemodynamics; Humans; Male; Middle Aged; Pulmonary Wedge Pressure; Quinazolines; Stroke Volume; Vascular Resistance

1993
[Evaluation of bunazosin hydrochloride with a model of ocular circulation disturbance induced by endothelin-1].
    Nippon Ganka Gakkai zasshi, 1994, Volume: 98, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Endothelins; Optic Disk; Quinazolines; Rabbits; Regional Blood Flow; Retinal Artery

1994
Characteristics of the responses of isolated and perfused canine splenic arteries to vasoactive substances and to periarterially electrical stimulation.
    Japanese journal of pharmacology, 1994, Volume: 64, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dogs; Electric Stimulation; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Quinazolines; Splenic Artery; Vasoconstriction; Vasoconstrictor Agents

1994
The effect of bunazosin on monocrotaline-induced pulmonary hypertension in rats.
    Acta paediatrica Japonica : Overseas edition, 1994, Volume: 36, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Hemodynamics; Hypertension, Pulmonary; Monocrotaline; Quinazolines; Rats; Rats, Sprague-Dawley

1994
[Effects of long-term application of bunazosin hydrochloride eye drops on the aqueous flow rate and blood-aqueous barrier permiability in rabbit eyes].
    Nippon Ganka Gakkai zasshi, 1994, Volume: 98, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Blood; Intraocular Pressure; Ophthalmic Solutions; Permeability; Quinazolines; Rabbits

1994
Ocular pharmacokinetics and pharmacodynamics in rabbits of ibopamine, a new mydriatic agent.
    Experimental eye research, 1993, Volume: 56, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Aqueous Humor; Deoxyepinephrine; Dose-Response Relationship, Drug; Female; Male; Moxisylyte; Mydriatics; Pupil; Quinazolines; Rabbits; Reserpine; Swine; Time Factors

1993
Selective suppression by bunazosin of alpha-adrenergic agonist evoked elevation of intraocular pressure in sympathectomized rabbit eyes.
    Investigative ophthalmology & visual science, 1993, Volume: 34, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Ganglia, Sympathetic; Ganglionectomy; Intraocular Pressure; Male; Norepinephrine; Ocular Hypotension; Ophthalmic Solutions; Phenylephrine; Pupil; Quinazolines; Rabbits; Receptors, Adrenergic, alpha

1993
Vascular responsiveness of rabbit common carotid, renal and femoral arteries to alpha-adrenoceptor agonists.
    Japanese journal of pharmacology, 1993, Volume: 61, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dinoprost; Dose-Response Relationship, Drug; Drug Interactions; Female; Femoral Artery; In Vitro Techniques; Male; Phenylephrine; Quinazolines; Rabbits; Renal Artery; Vasoconstriction

1993
Alterations of binding characteristics of alpha 1-,beta 1-adrenoceptors and Ca2+ binding sites in the myocardium of spontaneously hypertensive rats (SHR) by chronically administered bunazosin, atenolol, ketanserin and verapamil.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Atenolol; Binding Sites; Blood Pressure; Calcium Channels; Heart; In Vitro Techniques; Ketanserin; Kinetics; Myocardium; Norepinephrine; Quinazolines; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Verapamil

1993
Long-term alpha 1 blockade does not reverse cardiac hypertrophy in spontaneously hypertensive rats.
    Japanese circulation journal, 1993, Volume: 57, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Hemodynamics; Hypertension; Hypertrophy, Left Ventricular; Male; Norepinephrine; Quinazolines; Rats; Rats, Inbred SHR; Renin

1993
Effects of alpha-adrenergic blockade on regional myocardial function in canine ischemic myocardium during beta-adrenergic blockade.
    Journal of cardiothoracic and vascular anesthesia, 1995, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Coronary Circulation; Dogs; Female; Hemodynamics; Male; Myocardial Contraction; Myocardial Ischemia; Myocardium; Prazosin; Propranolol; Prospective Studies; Quinazolines; Random Allocation; Yohimbine

1995
Exaggeration of acute liver damage by hepatic sympathetic nerves and circulating catecholamines in perfused liver of rats treated with D-galactosamine.
    Hepatology (Baltimore, Md.), 1996, Volume: 23, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Analysis of Variance; Animals; Aspartate Aminotransferases; Calcium; Electric Stimulation; Galactosamine; Isoproterenol; L-Lactate Dehydrogenase; Liver; Male; Norepinephrine; Perfusion; Phenylephrine; Quinazolines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Sympathomimetics

1996
Effects of alpha-blocker on daily testicular sperm production and sperm concentration, motility, intraluminal pressure and fluid movement in the rat epididymis.
    The Tohoku journal of experimental medicine, 1995, Volume: 177, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Biological Transport; Body Fluids; Epididymis; Male; Organ Size; Pressure; Quinazolines; Rats; Rats, Sprague-Dawley; Seminiferous Tubules; Sperm Count; Sperm Motility; Spermatogenesis; Testis

1995
Induction of DNA breaks in cardiac myoblast cells by norepinephrine.
    Biochemistry and molecular biology international, 1996, Volume: 38, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Calcium Channel Blockers; Captopril; DNA; DNA Damage; DNA, Single-Stranded; Heart; Hydrogen Peroxide; Myocardium; Norepinephrine; Propranolol; Quinazolines; Rats; Stimulation, Chemical; Verapamil

1996
Effect of alpha-blockers on epididymal sperm concentration, motility and testicular productivity in the rat.
    Hinyokika kiyo. Acta urologica Japonica, 1996, Volume: 42, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Epididymis; Male; Quinazolines; Rats; Rats, Sprague-Dawley; Sperm Count; Sperm Motility; Spermatogenesis; Testis

1996
Effect of tamsulosin, a novel alpha 1-adrenoceptor antagonist, on urethral pressure profile in anaesthetized dogs.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Captopril; Dogs; Dose-Response Relationship, Drug; Male; Nicardipine; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin

1996
Prevention of cardiac hypertrophy by a sub-antihypertensive dose of the alpha 1-adrenergic antagonist bunazosin in Dahl salt-sensitive rats.
    Hypertension research : official journal of the Japanese Society of Hypertension, 1996, Volume: 19, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiomegaly; Hypertension; Male; Quinazolines; Rats; Sodium Chloride

1996
Thromboxane inhibition potentiates antihypertensive effects of alpha 1 adrenoceptor antagonists in the rat.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aorta; Blood Pressure; Body Weight; Cells, Cultured; Drug Synergism; Eicosanoids; Ethanolamines; Kidney; Methacrylates; Muscle, Smooth, Vascular; Prazosin; Quinazolines; Rats; Rats, Inbred SHR; Sodium; Thromboxane-A Synthase; Thromboxanes

1997
Effect of alpha 1-adrenoceptor antagonists on urinary bladder function in urethane-anesthetized rats.
    General pharmacology, 1997, Volume: 28, Issue:4

    Topics: Adrenergic alpha-Antagonists; Anesthetics; Animals; Flavoxate; Male; Parasympatholytics; Prazosin; Quinazolines; Rats; Rats, Wistar; Sulfonamides; Tamsulosin; Urethane; Urinary Bladder

1997
Beta-adrenoceptor stimulation-mediated preconditioning-like cardioprotection in perfused rat hearts.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Creatine Kinase; Heart; Heart Rate; Isoproterenol; Male; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion; Myocardial Reperfusion Injury; Myocardium; Norepinephrine; Phenylephrine; Quinazolines; Random Allocation; Rats; Rats, Sprague-Dawley; Timolol; Ventricular Function, Left

1997
[Alström syndrome--a rare disease of diabetic association].
    Medizinische Klinik (Munich, Germany : 1983), 1997, Mar-15, Volume: 92, Issue:3

    Topics: Adult; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diagnosis, Differential; DNA Mutational Analysis; Humans; Male; Obesity; Optic Atrophy; Quinazolines; Retinitis Pigmentosa; Second Messenger Systems; Syndrome

1997
Clinical impact of insulin resistance syndrome in cardiovascular diseases and its therapeutic approach.
    Hypertension research : official journal of the Japanese Society of Hypertension, 1996, Volume: 19 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Amlodipine; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Calcium Channel Blockers; Cardiovascular Diseases; Cilazapril; Humans; Insulin Resistance; Middle Aged; Quinazolines

1996
Infarct size-reducing effect of ischemic preconditioning is related to alpha1b-adrenoceptors but not to alpha1a-adrenoceptors in rabbits.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Ischemic Preconditioning, Myocardial; Male; Phenoxybenzamine; Piperazines; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1

1997
Effects of alpha 1-adrenoreceptor subtype blockade on ischemia-reperfusion injury.
    Japanese circulation journal, 1997, Volume: 61, Issue:11

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Clonidine; Dioxanes; Energy Metabolism; In Vitro Techniques; Male; Myocardial Reperfusion Injury; Quinazolines; Rats; Rats, Sprague-Dawley

1997
Differences in refractory-period response of canine subendocardium and subepicardium to bunazosin, an alpha1-adrenoceptor antagonist, and propranolol during myocardial ischemia.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Dogs; Endocardium; Heart Ventricles; Myocardial Ischemia; Pericardium; Propranolol; Quinazolines; Receptors, Adrenergic, alpha-1; Refractory Period, Electrophysiological; Tachycardia, Ventricular; Ventricular Fibrillation; Ventricular Function

1997
[Alpha-1 blockers for therapy of essential hypertension. 2 clinical studies with bunazosin].
    Fortschritte der Medizin, 1998, May-20, Volume: 116, Issue:14

    Topics: Adrenergic alpha-Antagonists; Blood Pressure; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Hypertension; Quinazolines; Treatment Outcome

1998
Bunazosin reduces intraocular pressure in rabbits by increasing uveoscleral outflow.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 1998, Volume: 14, Issue:3

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aqueous Humor; Cyclooxygenase Inhibitors; Fluorophotometry; Flurbiprofen; Indomethacin; Intraocular Pressure; Quinazolines; Rabbits; Sclera; Tonometry, Ocular; Uvea

1998
Regulation of angiotensin II receptor expression by nitric oxide in rat adrenal gland.
    Hypertension (Dallas, Tex. : 1979), 1998, Volume: 32, Issue:3

    Topics: Adrenal Glands; Adrenergic alpha-Antagonists; Aldosterone; Animals; Blotting, Northern; Body Weight; DNA, Complementary; Enzyme Inhibitors; Gene Expression Regulation; Hemodynamics; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptidyl-Dipeptidase A; Quinazolines; Rats; Rats, Wistar; Receptors, Angiotensin; Renin; RNA, Messenger

1998
Bunazosin hydrochloride inhibits exaggerated growth of vascular smooth muscle cells from spontaneously hypertensive rats by suppressing the response to growth factors.
    Journal of cardiovascular pharmacology, 1998, Volume: 32, Issue:6

    Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Antihypertensive Agents; Cell Division; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Epidermal Growth Factor; Growth Inhibitors; Muscle, Smooth, Vascular; Platelet-Derived Growth Factor; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; RNA, Messenger

1998
[Signal transduction of serotonin release from enterochromaffin cells in mouse ileal crypts].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1998, Volume: 112 Suppl 1

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Clonidine; Enterochromaffin Cells; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Norepinephrine; Phosphodiesterase Inhibitors; Prazosin; Pyrrolidinones; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Rolipram; Serotonin; Signal Transduction; Yohimbine

1998
Disproportional response between refractory period and blood flow to alpha 1- and beta-adrenoceptor blockade in canine ischemic myocardium.
    Cardiovascular drugs and therapy, 1998, Volume: 12, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Coronary Circulation; Dogs; Electrocardiography; Endocardium; Heart; Myocardial Ischemia; Pericardium; Propranolol; Quinazolines; Refractory Period, Electrophysiological; Tachycardia, Ventricular; Ventricular Fibrillation

1998
Bunazosin. Andante, Detantol, E 1015, E 643, EA 0643.
    Drugs in R&D, 1999, Volume: 2, Issue:6

    Topics: Adrenergic alpha-Antagonists; Aged; Antihypertensive Agents; Area Under Curve; Clinical Trials as Topic; Humans; Hypertension; Male; Prostatic Hyperplasia; Quinazolines

1999
Effects of bunazosin hydrochloride sustained-release formulation on cerebral circulation.
    International angiology : a journal of the International Union of Angiology, 2000, Volume: 19, Issue:1

    Topics: Acetazolamide; Adrenergic alpha-Antagonists; Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Flow Velocity; Caudate Nucleus; Cerebral Infarction; Cerebrovascular Circulation; Delayed-Action Preparations; Diuretics; Enalapril; Female; Humans; Injections, Intravenous; Male; Occipital Lobe; Parietal Lobe; Quinazolines; Tomography, X-Ray Computed

2000
Attenuation of KATP channel-opener induced shortening of repolarization time by alpha 1-adrenoceptor antagonist during ischemia in canine heart.
    Cardiovascular drugs and therapy, 2000, Volume: 14, Issue:3

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; ATP-Binding Cassette Transporters; Benzopyrans; Blood Pressure; Dogs; Electrocardiography; Electrophysiology; Heart; In Vitro Techniques; KATP Channels; Myocardial Reperfusion Injury; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinazolines

2000
Different vasculoprotective roles of NO synthase isoforms in vascular lesion formation in mice.
    Arteriosclerosis, thrombosis, and vascular biology, 2000, Volume: 20, Issue:11

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aspirin; Carotid Arteries; Female; Fibrinolytic Agents; Isoenzymes; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neovascularization, Pathologic; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Quinazolines; Tunica Intima

2000
Neuroprotective effect and intraocular penetration of nipradilol, a beta-blocker with nitric oxide donative action.
    Investigative ophthalmology & visual science, 2001, Volume: 42, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood-Retinal Barrier; Cell Count; Dose-Response Relationship, Drug; Drug Combinations; Male; N-Methylaspartate; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Propanolamines; Quinazolines; Rabbits; Rats; Rats, Sprague-Dawley; Retina; Retinal Artery; Timolol; Vasoconstriction

2001
Noradrenaline stimulates 5-hydroxytryptamine release from mouse ileal tissues via alpha(2)-adrenoceptors.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Ileum; In Vitro Techniques; Male; Methoxamine; Mice; Mice, Inbred ICR; Norepinephrine; Pertussis Toxin; Phenylephrine; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha-2; Serotonin; Virulence Factors, Bordetella; Yohimbine

2001
The renin-angiotensin and adrenergic nervous system in cardiac hypertrophy in fructose-fed rats.
    American journal of hypertension, 2002, Volume: 15, Issue:1 Pt 1

    Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Antihypertensive Agents; Blood Glucose; Blood Pressure; Catecholamines; Diet; Fructose; Glucose Tolerance Test; Heart Rate; Hydralazine; Hyperinsulinism; Hypertrophy, Left Ventricular; Imidazoles; Insulin; Male; Myocardium; Olmesartan Medoxomil; Organ Size; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Renin-Angiotensin System; Sympathetic Nervous System; Tetrazoles

2002
Purinergic modulation of vascular sympathetic neurotransmission.
    Japanese journal of pharmacology, 2002, Volume: 88, Issue:1

    Topics: Adenosine Triphosphate; Animals; Arteries; Electrophysiology; Norepinephrine; Purines; Quinazolines; Rats; Receptors, Purinergic; Synaptic Transmission; Tail; Vasomotor System

2002
Different effects of carvedilol, metoprolol, and propranolol on left ventricular remodeling after coronary stenosis or after permanent coronary occlusion in rats.
    Circulation, 2002, Feb-26, Volume: 105, Issue:8

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Carbazoles; Cardiac Catheterization; Carvedilol; Coronary Disease; Coronary Stenosis; Disease Models, Animal; Dose-Response Relationship, Drug; Echocardiography; Hemodynamics; Male; Metoprolol; Norepinephrine; Propanolamines; Propranolol; Quinazolines; Rats; Rats, Sprague-Dawley; Severity of Illness Index; Stroke Volume; Survival Rate; Thiobarbituric Acid Reactive Substances; Ventricular Function, Left; Ventricular Remodeling

2002
The alpha(1D)-adrenergic receptor directly regulates arterial blood pressure via vasoconstriction.
    The Journal of clinical investigation, 2002, Volume: 109, Issue:6

    Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Aorta; Arteries; Blood Pressure; Cardiovascular System; Female; Gene Targeting; In Vitro Techniques; Male; Mice; Mice, Knockout; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Piperazines; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Serotonin; Tissue Extracts; Vasoconstriction; Vasoconstrictor Agents; Vasopressins

2002
Neuroprotective effects of nipradilol on purified cultured retinal ganglion cells.
    Journal of glaucoma, 2002, Volume: 11, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antihypertensive Agents; Cell Separation; Cell Survival; Cells, Cultured; Culture Media, Serum-Free; Cyclic N-Oxides; Dose-Response Relationship, Drug; Flow Cytometry; Imidazoles; Neuroprotective Agents; Nitric Oxide; Propanolamines; Quinazolines; Rats; Rats, Sprague-Dawley; Retinal Ganglion Cells; Timolol

2002
Amelioration by topical bunazosin hydrochloride of the impairment in ocular blood flow caused by nitric oxide synthase inhibition in rabbits.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2003, Volume: 19, Issue:1

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Evoked Potentials, Visual; Fundus Oculi; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Optic Disk; Quinazolines; Rabbits; Reaction Time; Regional Blood Flow; Vision, Ocular

2003
[Effects of ocular hypotensive agents on the circadian rhythm in intraocular pressure in rabbits as measured by telemetry].
    Nippon Ganka Gakkai zasshi, 2003, Volume: 107, Issue:9

    Topics: Animals; Circadian Rhythm; Intraocular Pressure; Male; Quinazolines; Rabbits; Sulfonamides; Telemetry; Thiophenes; Timolol

2003
Bunazosin hydrochloride reduces glutamate-induced neurotoxicity in rat primary retinal cultures.
    Brain research, 2004, Apr-02, Volume: 1003, Issue:1-2

    Topics: Animals; Brain; Cell Death; Cells, Cultured; Dose-Response Relationship, Drug; Female; Glutamic Acid; Pregnancy; Protein Binding; Quinazolines; Rats; Rats, Wistar; Retina

2004
Ocular pharmacokinetic/ pharmacodynamic modeling for bunazosin after instillation into rabbits.
    Pharmaceutical research, 2004, Volume: 21, Issue:5

    Topics: Adrenergic alpha-Antagonists; Algorithms; Animals; Aqueous Humor; Eye; Injections; Intraocular Pressure; Male; Models, Biological; Quinazolines; Rabbits; Tears

2004
Effects of bunazosin hydrochloride on ciliary muscle constriction and matrix metalloproteinase activities.
    Journal of glaucoma, 2004, Volume: 13, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aqueous Humor; Cattle; Cells, Cultured; Ciliary Body; Drug Combinations; Intraocular Pressure; Isometric Contraction; Latanoprost; Macaca fascicularis; Male; Matrix Metalloproteinases; Muscle Relaxation; Muscle, Smooth; Phenylephrine; Prostaglandins F, Synthetic; Quinazolines; Trabecular Meshwork

2004
Effects of topically instilled bunazosin, an alpha1-adrenoceptor antagonist, on constrictions induced by phenylephrine and ET-1 in rabbit retinal arteries.
    Investigative ophthalmology & visual science, 2004, Volume: 45, Issue:11

    Topics: Administration, Topical; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Combinations; Endothelin-1; Ganglionectomy; Injections; Male; Phenylephrine; Quinazolines; Rabbits; Receptors, Endothelin; Retinal Artery; Superior Cervical Ganglion; Vasoconstriction; Vasoconstrictor Agents; Vitreous Body

2004
Alpha1-receptor or adenosine A1-receptor dependent pathway alone is not sufficient but summation of these pathways is required to achieve an ischaemic preconditioning effect in rabbits.
    Clinical and experimental pharmacology & physiology, 2005, Volume: 32, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Enzyme Inhibitors; Heart Rate; Ischemic Preconditioning, Myocardial; Male; Myocardial Infarction; Protein Kinase C; Quinazolines; Rabbits; Receptor, Adenosine A1; Receptors, Adrenergic, alpha-1; Staurosporine; Theophylline; Tyramine; Vasodilator Agents

2005
Amelioration of endothelin-1-induced optic nerve head ischemia by topical bunazosin.
    Current eye research, 2005, Volume: 30, Issue:2

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Endothelin-1; Evoked Potentials, Visual; Injections; Intraocular Pressure; Ischemia; Optic Disk; Quinazolines; Rabbits; Regional Blood Flow; Retina; Vitreous Body

2005
Alterations of alpha-adrenergic modulations of coronary microvascular tone in dogs with heart failure.
    Journal of cardiac failure, 2005, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Flow Velocity; Cineangiography; Coronary Angiography; Coronary Circulation; Coronary Vessels; Disease Models, Animal; Dogs; Enzyme Inhibitors; Female; Heart Failure; Injections, Intra-Arterial; Male; Microcirculation; NG-Nitroarginine Methyl Ester; Propranolol; Quinazolines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vascular Resistance; Vasodilation; Yohimbine

2005
Effects of different alpha-1 adrenoceptor blockers on proximal urethral function using in vivo isovolumetric pressure changes.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2005, Volume: 41, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Male; Phenylephrine; Prazosin; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urethra

2005
Incidence of intraoperative floppy iris syndrome in patients on either systemic or topical alpha(1)-adrenoceptor antagonist.
    American journal of ophthalmology, 2007, Volume: 143, Issue:1

    Topics: Administration, Topical; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Cataract Extraction; Female; Humans; Incidence; Intraoperative Complications; Iris Diseases; Male; Naphthalenes; Piperazines; Prospective Studies; Prostatic Hyperplasia; Pupil; Quinazolines; Sulfonamides; Syndrome; Tamsulosin

2007
[Case of pigmentary glaucoma treated with medical therapy, laser treatment, and trabeculotomy].
    Nippon Ganka Gakkai zasshi, 2007, Volume: 111, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Argon; Glaucoma, Open-Angle; Humans; Intraocular Pressure; Iris; Laser Therapy; Male; Ophthalmic Solutions; Quinazolines; Sulfonamides; Thiophenes; Trabeculectomy; Treatment Outcome

2007
Effects of adrenergic and cholinergic antagonists on diameter of nasolacrimal drainage system.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 2007, Volume: 245, Issue:12

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Female; Humans; Infusions, Parenteral; Male; Middle Aged; Muscarinic Antagonists; Nasolacrimal Duct; Quinazolines; Radiography; Sympathetic Nervous System; Tropicamide

2007
Protective effects of carvedilol in murine model with the coxsackievirus B3-induced viral myocarditis.
    Journal of cardiovascular pharmacology, 2008, Volume: 51, Issue:1

    Topics: Acute Disease; Adrenergic beta-Antagonists; Animals; Anti-Inflammatory Agents; Antioxidants; Carbazoles; Cardiotonic Agents; Carvedilol; Coxsackievirus Infections; Disease Models, Animal; Enterovirus B, Human; Interleukins; Male; Malondialdehyde; Metoprolol; Mice; Mice, Inbred BALB C; Myocarditis; Propanolamines; Quinazolines; Superoxide Dismutase; Up-Regulation

2008
Comparison of the cardiac electrophysiological effects between doxazosin and bunazosin.
    Journal of biomedical science, 2008, Volume: 15, Issue:4

    Topics: Animals; Arrhythmias, Cardiac; Cardiac Electrophysiology; Doxazosin; Drug-Related Side Effects and Adverse Reactions; Heart; In Vitro Techniques; Ion Channels; Quinazolines; Rats

2008
Possible mechanism of intraoperative floppy iris syndrome: a clinicopathological study.
    The British journal of ophthalmology, 2008, Volume: 92, Issue:8

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Antihypertensive Agents; Female; Glaucoma; Humans; Iris Diseases; Male; Quinazolines; Syndrome

2008
Ocular pharmacokinetic/pharmacodynamic modeling for multiple anti-glaucoma drugs.
    Biological & pharmaceutical bulletin, 2008, Volume: 31, Issue:8

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Algorithms; Animals; Aqueous Humor; Drug Combinations; Glaucoma; Intraocular Pressure; Male; Models, Statistical; Ocular Hypertension; Ophthalmic Solutions; Quinazolines; Rabbits; Telemetry; Timolol

2008
[The use of andante in the therapy of insomnia].
    Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova, 2009, Volume: 109, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adult; Dose-Response Relationship, Drug; Female; Follow-Up Studies; Humans; Male; Middle Aged; Polysomnography; Quinazolines; Sleep; Sleep Initiation and Maintenance Disorders; Surveys and Questionnaires; Treatment Outcome

2009