bunazosin has been researched along with quinazolines in 225 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 83 (36.89) | 18.7374 |
1990's | 110 (48.89) | 18.2507 |
2000's | 31 (13.78) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (0.44) | 2.80 |
Authors | Studies |
---|---|
Amano, M; Kanamori, T; Kinoshita, M; Shichiri, G; Takahashi, M | 1 |
Kimura, H; Kusaba, T; Nagasawa, K; Otsuka, T; Sakata, T; Tada, Y; Tsuda, Y | 1 |
Atarashi, K; Matsuoka, H; Sugimoto, T; Takagi, M | 1 |
Gotoh, S; Hiraga, S; Hosoda, K; Kakehi, R; Kaneoya, F; Kojima, S; Mizuo, T; Satoh, T; Tanizawa, A; Yokokawa, M | 1 |
Hirakawa, S; Imai, Y; Ito, H; Kakami, M; Koshiji, M; Minatoguchi, S; Watanabe, H | 1 |
Baba, T; Ishizaki, T; Murabayashi, S; Tomiyama, T | 1 |
Evans, RG; Hayes, IP; Ludbrook, J | 1 |
Kono, K; Masuda, T; Nakamura, Y; Oyama, M; Shimizu, T; Takahashi, M; Takeda, K; Yagi, S | 1 |
García-Sáinz, JA; González-Espinosa, C; Romero-Avila, MT; Torres-Márquez, ME | 1 |
Kawai, C; Matsumori, A; Okada, I; Tominaga, M; Yamada, T | 1 |
Arakawa, K; Hidaka, K; Matsunaga, A; Sasaki, J | 1 |
Asakura, Y; Harano, Y; Hirose, J; Kageyama, A; Omae, T; Sato, A; Suzuki, M | 1 |
Kondo, S; Morita, T | 1 |
Asano, H; Fujita, T; Hirabayashi, S; Kato, N; Kinukawa, T; Ohshima, S; Ono, Y | 1 |
Abiko, Y; Ichihara, K; Nasa, Y; Yoshida, R | 1 |
Kondo, M; Nakanishi, T; Nishimura, M; Takahashi, H; Yoshida, T; Yoshimura, M | 1 |
Hosoda, S; Kaneko, N; Kawagoe, Y; Kimata, S; Kimura, H; Konno, K; Miki, N; Nagashima, H; Sumiyoshi, T | 1 |
Hattori, K; Kobayashi, Y; Shimoura, K; Shinozuka, K | 1 |
Hori, M; Inoue, M; Iwai, K; Iwakura, K; Kagiya, T; Kamada, T; Kitabatake, A; Uchida, S; Watanabe, Y; Yoshida, H | 1 |
Haneda, N; Hayashi, Y; Inoue, M; Kishida, K; Mori, C; Ozasa, H; Watanabe, K | 1 |
Hayashi, Y; Ikeda, K; Ohnishi, H; Watanabe, K | 2 |
Fujioka, S; Kawamoto, T; Keno, Y; Kobatake, T; Matsuzawa, Y; Tarui, S; Tokunaga, K; Watanabe, Y; Yoshida, H | 1 |
Smith, SE; Trew, DR; Wright, LA | 1 |
Kusunoki, T; Kuwayama, Y; Manabe, R; Shimizu, Y; Sun, N; Takagi, T; Tanaka, M; Yamamoto, R | 1 |
Sugiyama, T | 1 |
Iwai, T; Nagano, M; Nakamura, I; Ohkubo, T; Takeda, N; Tanamura, A | 1 |
Hikida, M; Kinoshita, M; Kuwayama, Y; Nishimura, K; Shirasawa, E | 1 |
Baba, S; Kinami, J; Mano, F; Maruyama, K; Nagatomo, T; Tsuchihashi, H | 1 |
Araie, M; Azuma, I; Nakajima, M; Oshika, T; Sugiyama, T | 1 |
Yamashita, Y | 1 |
Kinami, J; Maruyama, K; Nagatomo, T; Tsuchihashi, H | 1 |
Chiba, S; Skrbic, R | 1 |
Hashimoto, T; Kaguchi, Y; Kuriyama, S; Nakamura, K; Sakai, O; Tokutome, G; Tomonari, H | 1 |
Hasegawa, J; Hisatome, I; Kotake, H; Mashiba, H; Matsuoka, S; Noguchi, N | 1 |
Baba, T; Murabayashi, S; Takebe, K; Tomiyama, T | 1 |
Kaneko, S; Koyanagi, T; Kumamoto, Y; Maru, A; Nishizawa, O; Orikasa, S; Togashi, M; Tsuchida, S; Tsukamoto, T; Yachiku, S | 1 |
Kato, Y; Kawabe, K; Kimura, R; Maruyama, M; Matsuoka, Y; Suzuki, M; Yamada, S | 1 |
Kobayashi, S | 1 |
Chiba, S; Matsuura, M; Zenda, H | 1 |
Haneda, T; Obata, H; Tanaka, H | 1 |
Baba, T; Takebe, K; Tomiyama, T | 1 |
Esato, K; Katoh, T; Miyamoto, M; Mori, F | 1 |
Abiko, Y; Ichihara, K; Yoshida, R | 1 |
Chiba, S; Haniuda, M | 2 |
Hirabayashi, M; Ikegaki, I; Matsusawa, M; Nakanishi, T; Nishimura, M; Takahashi, H; Yoshimura, M | 1 |
Araie, M; Oshika, T | 1 |
Aso, Y; Honma, Y; Koyanagi, T; Maru, A; Miyake, K; Orikasa, S; Shimazaki, J; Soma, F; Togashi, M; Yasuda, K | 1 |
Araki, T; Chigusa, I; Kato, T; Kawamura, J; Morisita, H; Nakano, S; Saito, K; Sugimura, Y; Tajima, K; Tochigi, H | 1 |
Inukai, T; Ishii, A; Iwashita, A; Kobayashi, I; Kobayashi, S; Kobayashi, T; Shimomura, Y; Yamaguchi, T; Yamaguchi, Y | 1 |
Chiba, S; Tsukada, M | 3 |
Doi, T; Hasegawa, J; Hisatome, I; Kotake, H; Mashiba, H; Noguchi, N; Sawaguchi, M | 1 |
Fujiwara, H; Ishida, M; Kawai, C; Kawamura, A; Kida, M; Takemura, G; Tanaka, M; Uegaito, T | 1 |
Hasegawa, J; Kotake, H; Kurata, Y; Mashiba, H; Ogino, K; Ohtahara, A; Saitoh, M | 1 |
Ozawa, T; Sugiyama, S | 1 |
Kondo, A; Mitsuya, H; Otani, T; Takita, T | 1 |
Chiba, S; Nakane, T | 1 |
Aso, Y; Ishibashi, A; Koshiba, K; Kumamoto, Y; Nishizawa, O; Ogawa, A; Tomita, Y; Tsuchida, S; Tsukamoto, T; Yokoyama, E | 1 |
Aoyama, T; Furuya, S; Honma, A; Kumamoto, Y; Miyamoto, S; Takagi, Y; Takatsuka, K; Tamiya, T; Tsukamoto, T; Yokoyama, E | 1 |
Araie, M; Sugiura, Y | 2 |
Akimoto, Y; Fujiwara, M; Kurahashi, K; Sono, K | 1 |
Chiba, S; Haniuda, M; Itoh, N | 1 |
Katayama, E; Mitsui, T; Mizukawa, K; Ogawa, N; Ogura, T; Ota, Z; Takatori, K; Yamamoto, I | 1 |
Hasegawa, K; Inoue, S; Kawahara, Y; Nezuo, S; Sawayama, T; Tadaoka, S | 1 |
Fujioka, M; Ibengwe, JK; Komori, K; Nagao, T; Suzuki, H; Zhang, GL | 1 |
Nagatomo, T; Tsuchihashi, H | 1 |
Fukuta, S; Itagaki, T; Kusukawa, R; Toma, Y; Umemoto, S; Yamakawa, K; Yoshinaga, T | 1 |
Kanaide, H; Miwa-Nishimura, N; Nakamura, M; Nishimura, J | 1 |
Dan, Y; Fukui, K; Hirata, Y; Ishii, M; Matsuoka, H; Sugimoto, T | 1 |
Akima, M; Imagawa, J; Sakai, K | 1 |
Hirawa, N; Numabe, A; Takada, S; Uehara, Y; Yagi, S | 2 |
Mikami, H; Ogihara, T | 1 |
Hasegawa, A; Hatori, M; Murata, K; Nakano, A; Suzuki, T; Tamura, M | 2 |
Geshi, E; Hiroshige, J; Katagiri, T; Konno, N; Mochizuki, M; Umetsu, K | 1 |
Asada, S; Hirayama, A; Komamura, K; Lee, JM; Matsumura, Y; Mishima, M; Nishida, K; Ohara, T; Okazaki, Y; Yamamoto, K | 1 |
Fujii, T; Inoue, S; Nagai, K; Nakagawa, H | 1 |
Hasegawa, K; Inoue, S; Kakumae, S; Kawahara, Y; Nakamura, T; Nakao, M; Nezuo, S; Sawayama, T; Tadaoka, S | 1 |
Ebihara, A; Fujimura, A; Kumagai, Y; Nakashima, H; Oribe, H; Shitoh, T; Sugimoto, K | 1 |
Kaneko, M; Kimura, S; Shoumura, K | 1 |
Arakawa, K; Koga, S; Sasaki, J; Uzawa, H | 1 |
Matsumoto, M; Minami, M; Saito, H; Togashi, H; Yoshioka, M | 1 |
Haginaka, T; Katsumi, T; Murayama, K; Nakamura, T; Sakai, A; Tazika, E | 1 |
Matsui, Y; Nakai, M; Yamamoto, J | 1 |
Kato, T; Miyamoto, Y; Nakasone, J; Noguchi, K; Sakanashi, M; Takeo, S | 1 |
Hashimoto, J; Mitsuya, H; Miyake, K; Takaba, H; Yamamoto, M | 1 |
Ozawa, T; Sugiyama, S; Takamura, T | 1 |
Itoh, T; Kimoto, Y; Nozaki, M | 1 |
Ishibashi, Y; Kato, A; Miyake, Y | 1 |
Chiba, S; Ohkubo, H | 1 |
Chiba, S; Sinanović, O | 2 |
Ikegaki, I; Matsuzawa, M; Okabayashi, H; Suga, K; Takahashi, H; Yoshimura, M | 1 |
Orimo, H; Ouchi, Y; Watanabe, M | 1 |
Ikegaya, T; Kobayashi, A; Nishiyama, T; Yamazaki, N | 1 |
Hanaki, Y; Ozawa, T; Saito, H; Sugiyama, S | 1 |
Kuroiwa, A; Nakashima, Y; Sugano, M; Tasaki, H; Yashiro, A | 1 |
Iwata, S; Kato, A | 3 |
Azuma, T; Higa, S; Kishimoto, S; Mizuno, R; Sakoda, S; Suzuki, T; Tsujino, S; Watanabe, Y; Yoshida, H | 1 |
Matsumoto, M; Minematsu, R; Miyake, K; Takeo, S; Tanonaka, K | 1 |
Goto, K; Ishikawa, T; Kimura, S; Masaki, T; Yanagisawa, M | 1 |
Hasegawa, J; Hirai, S; Kotake, H; Mashiba, H; Saitoh, M | 1 |
Harada, T; Iida, H; Sone, T; Tanahashi, T; Tanaka, S; Tsukahara, I | 1 |
Kunieda, T; Naito, M; Nakanishi, N; Obayashi, Y; Okubo, S; Yoshioka, T | 1 |
Katayama, E; Mitsui, T; Mizukawa, K; Ogawa, N; Ogura, T; Ota, Z; Takatori, K | 1 |
Hashimoto, T; Kaguchi, Y; Kimura, M; Kuriyama, S; Miyahara, T; Nakamura, K; Tamai, K; Tamura, H | 1 |
Fujioka, M; Ibengwe, JK; Ishikawa, S; Komori, K; Nagao, T; Suzuki, H | 1 |
Ishikawa, Y; Kaneko, Y; Shindo, T; Toya, Y; Uchino, K; Umemura, S; Yasuda, G | 1 |
Ohno, M; Oishi, S; Sasaki, M; Sato, T; Umeda, T | 1 |
Ajioka, M; Nagai, S; Ozawa, T; Sugiyama, S; Takamura, T | 1 |
Chiba, S; Katsuyama, Y; Tada, A; Tsukada, M; Zenda, H | 1 |
Ebina, K; Fukuda, T; Nakamura, H; Nishizawa, O; Noto, H; Suzuki, K; Tsuchida, S | 1 |
Kakuta, Y; Kodera, T; Konishi, T; Koyama, T; Makino, K; Morimoto, Y; Nagano, K; Nakano, T; Takezawa, H; Umino, M | 1 |
Hirogami, M; Minami, M; Morii, K; Nomura, A; Saito, H; Saito, I; Sano, M; Tochihara, M; Togashi, H; Yoshioka, M | 1 |
Ishihara, Y; Kitamura, S; Kosaka, K; Yotsumoto, H | 1 |
Fujino, S; Hoshi, K | 1 |
Daiku, Y; Igarashi, T; Shoji, T | 1 |
Abe, I; Kawasaki, T; Kawazoe, N; Nakamuta, S; Omae, T; Ueno, M; Uezono, K | 1 |
Chiba, S; Furukawa, Y; Watanabe, H | 1 |
Shoji, T | 1 |
Fujimoto, S; Kida, O; Morotomi, Y; Tanaka, K | 1 |
Hata, F; Ishida, H; Kagawa, K; Kondo, E; Kondo, S | 1 |
Hattori, Y; Kanno, M | 1 |
Ludvig, N; Vizi, ES | 1 |
Fujimoto, T; Nakajima, S; Ohishi, M; Shiba, K; Takagi, O; Tsuya, Y; Uenishi, H | 1 |
Bando, S; Kakutani, A; Minezono, K; Mori, H; Noda, T; Shinomiya, H | 1 |
Itoh, K; Kohya, T; Minami, S; Nishijima, H; Tsujinaga, H; Yasuda, H | 1 |
Amagai, T; Fuse, T; Hirano, D; Kawazoe, K; Kitamura, K; Kiyotaki, S; Takimoto, Y | 1 |
Fujita, T; Kinoshita, K; Takahashi, T; Yamato, C | 1 |
Hamada, M; Kawanami, C; Konishi, T; Morimoto, Y; Nakai, K; Nakano, T; Noda, E; Takezawa, H; Yamamori, M | 1 |
Hattori, K; Kunitomo, M; Shimoura, K; Shinozuka, K | 1 |
Ishida, Y; Kawabe, K; Kurimoto, S; Moriyama, N; Nakamura, T; Orikasa, E | 1 |
Hirayama, T; Kikuchi, K; Morita, K; Ogawa, Y; Onodera, S; Takeda, A; Takenaka, T; Tobise, K | 1 |
Hibi, H; Miyake, K; Yamamoto, M | 4 |
Kitada, M; Mori, H; Takahashi, K; Tanabe, T; Usui, K | 1 |
Chiba, S; Vhora, S | 1 |
Gotoh, E; Ishii, M; Minamisawa, K; Minamisawa, M; Shionoiri, H; Sugimoto, K; Takasaki, I; Takizawa, T; Ueda, S | 1 |
Handa, S; Kitada, M; Mori, H; Takahashi, K; Tanabe, T; Yoshioka, K | 1 |
Kato, M; Kinugawa, T; Kitamura, H; Kotake, H; Mashiba, H; Matsumoto, T; Miyakoda, H; Noguchi, N; Ogino, K; Osaki, S | 1 |
Azuma, I | 1 |
De Luca, N; Fontana, D; Lamenza, F; Marchegiano, R; Sarno, D; Tozzi, N | 1 |
Azuma, I; Moriya, S; Oku, H; Shimizu, K; Sugiyama, T | 1 |
Kirsten, R; Weidinger, G | 1 |
Chiba, S; Nakane, T; Ren, LM | 1 |
Harder, S; Thürmann, P | 1 |
Inoue, M; Mori, C; Tanaka, O; Watanabe, K | 1 |
Aihara, M; Araie, M; Kaburaki, T; Shirato, S | 1 |
Anderton, JL; Gill, M; Notghi, A | 1 |
Galbiati, I; Gazzaniga, A; Gianesello, V; Soldati, L; Virno, M | 1 |
Kuwayama, Y; Matsugi, T; Nishimura, K; Shirasawa, E; Sun, N | 1 |
Chiba, S; Fujiwara, T | 1 |
Nagatomo, T; Shibata, A; Shimada, K; Tsuchihashi, H; Wakabayashi, H; Watanabe, K | 1 |
Kawamura, K; Kubota, J; Nishimura, H; Oka, T; Okabe, M; Ueyama, M | 1 |
Kono, M; Morita, S; Rubsamen, R | 1 |
Iwai, M; Shimazu, T | 1 |
Adachi, K; Hidaka, T; Muraishi, A; Okamoto, T; Seki, Y; Toshima, H | 1 |
Asano, M; Inagaki, O; Sudoh, K; Takenaka, T; Tanaka, H | 1 |
Fukuda, N; Izumi, Y; Kanmatsuse, K; Kubo, A; Matsuoka, M; Nakayama, T; Soma, M; Watanabe, Y | 1 |
Gatzka, C; Langenfeld, M; Schmieder, RE; Schobel, HP | 1 |
Weidinger, G | 1 |
Rieckert, H | 1 |
Herrmann, W; Schmitz, G; Stumpe, KO; Weidinger, G | 1 |
Eriksson, JW; Foley, K; Jansson, PA; Lithell, H | 1 |
Bönner, G; Chrosch, R; Schmieder, R; Weidinger, G | 1 |
Assmann, I; Bräutigam, M; Krönig, B; Langenfeld, MR; Schmieder, RE; Weidinger, G | 1 |
Inagaki, O; Sudoh, K; Takenaka, T | 1 |
Nasa, Y; Takeo, S; Yabe, K | 1 |
Rabl, W; Standl, E; Stemplinger, J; Stiegler, H; Weichenhain, B; Ziegler, AG | 1 |
Hara, Y; Harano, Y; Kanazawa, A; Nishioheda, Y; Ryomoto, K; Shinozaki, K; Suzuki, M; Tsushima, M | 1 |
Ishii, M; Umemura, S; Yasuda, G | 1 |
Arai, M; Fujiwara, H; Fujiwara, T; Kariya, T; Koshiji, M; Minatoguchi, S; Ohno, T; Uno, Y; Yamashita, K | 1 |
Asakura, Y; Ebihara, Y; Hasegawa, H; Nakamura, Y; Shinmura, K; Suganuma, Y; Tani, M | 1 |
Handa, S; Iwamoto, T; Kusuzaki, S; Takigawa, O; Tanabe, T; Usui, K; Yoshitake, M | 1 |
Suzuki, H | 1 |
Araie, M; Nagahara, M; Tamaki, Y; Tomidokoro, A; Tomita, K | 1 |
Meyer, U; Schmidt, J | 1 |
Camras, CB; Toris, CB; Wang, YL; Yablonski, ME; Zhan, GL | 1 |
Egashira, K; Ichiki, T; Katoh, M; Takeshita, A; Usui, M | 1 |
Fukuda, N; Hu, WY; Izumi, Y; Kanmatsuse, K; Soma, M | 1 |
Endo, T; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Satoh, Y; Suzuguchi, T | 1 |
Handa, S; Mori, H; Shinozaki, Y; Tanabe, T; Usui, K | 1 |
Koike, Y; Mineshita, S; Mizoguchi, H; Nomura, Y | 1 |
Mochizuki, Y; Oishi, M; Takasu, T | 1 |
Aikawa, M; Deguchi, Y; Handa, S; Tanabe, T; Yoshioka, K | 1 |
Akaike, T; Egashira, K; Funakoshi, H; Huang, P; Kandabashi, T; Miyata, K; Okamoto, S; Shimokawa, H; Takeshita, A; Yogo, K | 1 |
Araie, M; Koide, T; Mizuno, K; Yoshimura, M | 1 |
Endo, T; Hamaue, N; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Parvez, H | 1 |
Higaki, J; Kamide, K; Moriguchi, K; Nagai, M; Ogihara, T; Ohishi, M; Okamura, A; Rakugi, H; Satoh, N; Tuck, ML | 1 |
Kunitomo, M; Mizuno, H; Nakamura, K; Shinozuka, K | 1 |
Maehara, K; Maruyama, Y; Sakabe, A; Yaoita, H | 1 |
Kawai, T; Koshimizu, T; Nasa, Y; Oshikawa, S; Shinoura, H; Sunada, S; Takeo, S; Tanoue, A; Tsujimoto, G | 1 |
Iizuka, Y; Kashiwagi, K; Tsukahara, S | 1 |
Goto, W; Ikeda, T; Oku, H; Okuno, T; Sugiyama, T | 2 |
Akaishi, T; Hara, H; Kuwayama, Y; Matsugi, T; Miyawaki, N; Shimazaki, A | 1 |
Kobayashi, H; Kobayashi, K; Okinami, S | 1 |
Araie, M; Goto, W; Hara, H; Ichikawa, M; Tanaka, E | 1 |
Kawakami, S; Kawazu, K; Kitahara, T; Nakamura, J; Nakashima, M; Nishida, K; Sakanaka, K; Sasaki, H; Tomonari, M | 1 |
Akaishi, T; Hara, H; Ishida, N; Kashiwagi, K; Matsugi, T; Takagi, Y | 1 |
Araie, M; Asai, Y; Hara, H; Ichikawa, M; Ishii, K; Okada, Y | 1 |
Baba, K; Fujiwara, H; Kariya, T; Kawai, T; Minatoguchi, S; Takahashi, M; Takemura, G; Uno, Y; Zhang, C | 1 |
Araie, M; Hara, H; Ichikawa, M; Oku, H; Shimazawa, M | 1 |
Maehara, K; Maruyama, Y; Oikawa, Y; Saito, T; Tamagawa, K; Yaoita, H | 1 |
Nagano, M; Osada, Y; Yamaguchi, T | 1 |
Fujita, Y; Inamura, M; Koyama, T; Miyoshi, T; Ohashi, Y; Ohki, K; Okamoto, S; Oshika, T; Sakabe, I; Takahashi, K; Yasuma, T | 1 |
Ihara, S; Kawana, M; Sakai, R; Shimamoto, K; Watanabe, H | 1 |
Higashide, T; Sugiyama, K; Wakabayashi, T | 1 |
Narioka, J; Ohashi, Y | 1 |
Ji-Fei, T; Jia-Feng, L; Jiang-Hua, R; Li-Sha, G; Peng, C; Peng-Lin, Y; Yue-Chun, L; Zhan-Qiu, Y | 1 |
Chen, WP; Lee, AS; Su, MJ | 1 |
Goseki, T; Ishikawa, H; Nemoto, N; Nishimoto, H; Patil, PN; Shimizu, K; Uga, S | 1 |
Higuchi, S; Kawazu, K; Kitahara, T; Nakamura, J; Nakashima, M; Nishida, K; Sakanaka, K; Sasaki, H; Tomonari, M | 1 |
Levin, IaI; Strygin, KN | 1 |
Parati, G; Pengo, MF; Steier, J | 1 |
6 review(s) available for bunazosin and quinazolines
Article | Year |
---|---|
Periodic fluctuation of blood pressure and its management in a patient with pheochromocytoma. Case report and review of the literature.
Topics: Adrenal Gland Neoplasms; Antihypertensive Agents; Blood Pressure; Catecholamines; Ethanolamines; Humans; Hypertension; Male; Middle Aged; Periodicity; Pheochromocytoma; Quinazolines | 1988 |
[Progress in medical treatment for glaucoma].
Topics: Adrenergic alpha-Antagonists; Choroid; Dinoprost; Endothelins; Glaucoma; Humans; Intraocular Pressure; Ophthalmic Solutions; Quinazolines; Regional Blood Flow | 1993 |
Pharmacokinetic and pharmacodynamic properties and therapeutic use of bunazosin in hypertension. A review.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Humans; Hypertension; Quinazolines | 1995 |
Treatment of benign prostatic hyperplasia and hypertension in elderly hypertensive patients.
Topics: Adrenergic alpha-Antagonists; Aged; Female; Humans; Hypertension; Male; Multicenter Studies as Topic; Prazosin; Product Surveillance, Postmarketing; Prostatic Hyperplasia; Quinazolines; Randomized Controlled Trials as Topic | 1998 |
Bunazosin, a selective alpha1-adrenoceptor antagonist, as an anti-glaucoma drug: effects on ocular circulation and retinal neuronal damage.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Eye; Glaucoma; Humans; Neurons; Optic Nerve; Quinazolines; Receptors, Adrenergic, alpha-1; Retina; Retinal Vessels | 2005 |
The ANDANTE Project: A Worldwide Individual Data Meta-Analysis of the Effect of Sleep Apnea Treatment on Blood Pressure.
Topics: Blood Pressure; Continuous Positive Airway Pressure; Humans; Quinazolines; Sleep Apnea Syndromes | 2021 |
32 trial(s) available for bunazosin and quinazolines
Article | Year |
---|---|
Acute effect of an alpha 1-adrenoceptor antagonist on urinary sodium excretion, plasma atrial natriuretic peptide, arginine vasopressin, and the renin-aldosterone system in healthy subjects.
Topics: Adrenergic alpha-Antagonists; Adult; Arginine Vasopressin; Atrial Natriuretic Factor; Enalapril; Humans; Male; Premedication; Quinazolines; Renin-Angiotensin System; Sodium | 1992 |
[The evaluation of the effects of bunazosin hydrochloride in the treatment of prostatic hyperplasia].
Topics: Adrenergic alpha-Antagonists; Aged; Drug Administration Schedule; Humans; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Urination | 1992 |
Ocular responses in healthy subjects to topical bunazosin 0.3%--an alpha 1-adrenoceptor antagonist.
Topics: Adrenergic alpha-Antagonists; Adult; Double-Blind Method; Eye; Eyelids; Female; Humans; Intraocular Pressure; Male; Middle Aged; Ophthalmic Solutions; Pupil; Quinazolines | 1991 |
[The effect of bunazosin hydrochloride on intraocular pressure and aqueous humor dynamics in human].
Topics: Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Female; Humans; Intraocular Pressure; Male; Quinazolines | 1991 |
Effect of bunazosin hydrochloride on intraocular pressure and aqueous humor dynamics in normotensive human eyes.
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Capillary Permeability; Dosage Forms; Dose-Response Relationship, Drug; Eye Proteins; Humans; Intraocular Pressure; Middle Aged; Quinazolines | 1991 |
Renal effects of bunazosin, a new alpha 1-adrenoceptor blocker, in patients with mild-to-moderate essential hypertension.
Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Female; Glomerular Filtration Rate; Hemodynamics; Humans; Hypertension; Kidney; Male; Middle Aged; Osmotic Pressure; Quinazolines; Renal Circulation; Vascular Resistance | 1990 |
[A double-blind trial on the effect of bunazosin hydrochloride for the symptoms of benign prostatic hypertrophy].
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Alanine; Chi-Square Distribution; Double-Blind Method; Drug Combinations; Glutamates; Glycine; Humans; Japan; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Urination; Urination Disorders | 1990 |
Enhancement by an ACE inhibitor of first-dose hypotension caused by an alpha 1-blocker.
Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Cholinesterase Inhibitors; Drug Synergism; Enalapril; Humans; Quinazolines | 1990 |
[Clinical evaluation of bunazosin hydrochloride for the treatment of voiding disturbances due to neurogenic bladder--a double-blind study].
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Bethanechol; Bethanechol Compounds; Chi-Square Distribution; Double-Blind Method; Female; Humans; Japan; Male; Middle Aged; Quinazolines; Urinary Bladder, Neurogenic; Urination; Urination Disorders | 1990 |
[Clinical study of bunazosin hydrochloride, an alpha 1-adrenergic blocker, in benign prostatic obstruction and neurogenic bladder dysfunction].
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Evaluation; Humans; Male; Middle Aged; Prostatic Diseases; Prostatic Hyperplasia; Quinazolines; Urinary Bladder, Neurogenic; Urination; Urination Disorders | 1987 |
[A double-blind trial on the effect of alpha-adrenergic blocker (bunazosin hydrochloride) in the symptomatic treatment of prostatism].
Topics: Adrenergic alpha-Antagonists; Aged; Clinical Trials as Topic; Double-Blind Method; Humans; Male; Middle Aged; Prostatic Hyperplasia; Quinazolines; Sympathetic Nervous System; Urination; Urination Disorders | 1987 |
[Clinical efficacy of oxendolene (antiandrogen) and bunazosin hydrochloride (alpha-adrenergic blocker) in the treatment of prostatism--comparative study of oxendolone, bunazocin hydrochloride and their combination].
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Androgen Antagonists; Drug Evaluation; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Nandrolone; Prostatic Hyperplasia; Quinazolines; Urinary Bladder Neck Obstruction; Urination | 1987 |
Chronopharmacological study of bunazosin hydrochloride in healthy subjects.
Topics: Adrenergic alpha-Antagonists; Adult; Blood Pressure; Drug Evaluation; Fingers; Humans; Male; Quinazolines; Regional Blood Flow; Skin; Time Factors | 1989 |
Comparative effects of bunazosin and propranolol on serum lipids and apolipoproteins in patients with essential hypertension.
Topics: Apolipoproteins; Blood Pressure; Female; Humans; Hypertension; Lipids; Lipoproteins; Male; Middle Aged; Multicenter Studies as Topic; Propranolol; Pulse; Quinazolines | 1989 |
[A double blind clinical trial of the alpha-adrenergic blocker, Ea-0643 tablet, in the treatment of neurogenic bladder].
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Male; Middle Aged; Quinazolines; Tablets; Urinary Bladder, Neurogenic | 1985 |
Comparison of the effectiveness of placebo and alpha-blocker therapy for the treatment of idiopathic oligozoospermia.
Topics: Adrenergic alpha-Antagonists; Adult; Double-Blind Method; Female; Humans; Infertility, Male; Male; Oligospermia; Placebos; Pregnancy; Quinazolines; Sperm Count; Sperm Motility | 1995 |
Pharmacokinetics and pharmacodynamics of the alpha 1-adrenergic antagonist bunazosin retard in hypertensives.
Topics: Adrenergic alpha-1 Receptor Antagonists; Blood Pressure; Delayed-Action Preparations; Female; Half-Life; Humans; Hypertension; Kidney Diseases; Male; Middle Aged; Pulse; Quinazolines | 1994 |
[Dose-response study of bunazosin in the treatment of light-to-moderate arterial hypertension].
Topics: Adrenergic alpha-Antagonists; Adult; Dose-Response Relationship, Drug; Drug Evaluation; Female; Humans; Hypertension; Male; Quinazolines | 1993 |
[Treatment of essential hypertension with the alpha-1 antagonist bunazosin retard. A multicenter, double-blind, placebo-controlled study].
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Blood Pressure; Delayed-Action Preparations; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Posture; Quinazolines | 1994 |
Concentration/effect relationship of bunazosin, a selective alpha 1-adrenoceptor antagonist in hypertensive patients after single and multiple oral doses.
Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Delayed-Action Preparations; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Quinazolines | 1994 |
Renal haemodynamic effects of bunazosin retard and prazosin in mild to moderately hypertensive patients with normal or moderately impaired renal function.
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Female; Glomerular Filtration Rate; Humans; Hypertension; Male; Middle Aged; Prazosin; Quinazolines; Renal Insufficiency; Renal Plasma Flow, Effective | 1994 |
Treatment and post-treatment effects of alpha- versus beta-receptor blockers on left ventricular structure and function in essential hypertension.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Double-Blind Method; Female; Heart Ventricles; Hemodynamics; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Metoprolol; Middle Aged; Quinazolines; Ventricular Function, Left | 1996 |
Orthostatic hypotension: how to avoid it during antihypertensive therapy.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Antihypertensive Agents; Blood Pressure; Double-Blind Method; Humans; Hypertension; Hypotension, Orthostatic; Middle Aged; Plethysmography; Posture; Prazosin; Quinazolines; Regional Blood Flow; Vascular Resistance | 1996 |
Effects of bunazosin and atenolol on serum lipids and apolipoproteins in a randomised trial.
Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Apolipoproteins; Atenolol; Double-Blind Method; Female; Humans; Hypertension; Lipids; Male; Middle Aged; Quinazolines; Treatment Outcome | 1996 |
Insulin sensitivity following treatment with the alpha 1-blocker bunazosin retard and the beta 1-blocker atenolol in hypertensive non-insulin-dependent diabetes mellitus patients.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Aged; Atenolol; Blood Glucose; Blood Pressure; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Double-Blind Method; Female; Humans; Hypertension; Insulin; Male; Middle Aged; Quinazolines | 1996 |
Effect of bunazosin and atenolol on glucose metabolism in obese, nondiabetic patients with primary hypertension.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Antihypertensive Agents; Atenolol; Blood Glucose; Double-Blind Method; Female; Glucose; Glucose Tolerance Test; Humans; Hypertension; Insulin; Lipids; Male; Middle Aged; Obesity; Quinazolines | 1997 |
Antihypertensive efficacy and orthostatic tolerance of bunazosin vs nitrendipine: a multicentre double-blind randomized controlled study.
Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Double-Blind Method; Humans; Hypertension; Lower Body Negative Pressure; Nitrendipine; Quinazolines | 1996 |
Characterization of bunazosin-sensitive alpha1-adrenoceptors in human renal medulla.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Double-Blind Method; Female; Humans; In Vitro Techniques; Kidney Function Tests; Kidney Medulla; Male; Middle Aged; Prazosin; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha-1 | 1997 |
Effects of topical adrenergic agents on tissue circulation in rabbit and human optic nerve head evaluated with laser speckle tissue circulation analyzer.
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Animals; Betaxolol; Blood Circulation; Blood Flow Velocity; Blood Pressure; Carteolol; Double-Blind Method; Hemorheology; Humans; Intraocular Pressure; Ophthalmic Solutions; Optic Disk; Propanolamines; Quinazolines; Rabbits | 1997 |
Pharmacokinetics and pharmacodynamics of bunazosin in patients with renal insufficiency.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Area Under Curve; Dose-Response Relationship, Drug; Female; Half-Life; Hemodynamics; Humans; Male; Middle Aged; Quinazolines; Renal Insufficiency; Time Factors | 1999 |
Efficacy of bunazosin hydrochloride 0.01% as adjunctive therapy of latanoprost or timolol.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aged; Drug Administration Schedule; Drug Therapy, Combination; Female; Glaucoma, Open-Angle; Humans; Intraocular Pressure; Latanoprost; Male; Middle Aged; Prostaglandins F, Synthetic; Pupil; Quinazolines; Timolol | 2004 |
An alpha1-receptor blocker reduces plasma leptin levels in hypertensive patients with obesity and hyperleptinemia.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Body Mass Index; Delayed-Action Preparations; Fatty Acids, Nonesterified; Female; Heart Rate; Humans; Hypertension; Insulin Resistance; Leptin; Male; Middle Aged; Obesity; Quinazolines; Receptors, Leptin; Treatment Outcome | 2006 |
187 other study(ies) available for bunazosin and quinazolines
Article | Year |
---|---|
Increased uncoupling of beta-, beta 1- and beta 2-adrenoceptor to myocardial contraction in failing human myocardium.
Topics: Adult; Aged; Binding, Competitive; Dobutamine; Down-Regulation; Female; Heart Failure; Humans; Iodocyanopindolol; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Pindolol; Quinazolines; Receptors, Adrenergic, beta; Terbutaline | 1992 |
Case report: nifedipine-rifampicin interaction attenuates the effect on blood pressure in a patient with essential hypertension.
Topics: Adrenergic alpha-Antagonists; Aged; Blood Pressure; Drug Interactions; Ethambutol; Female; Humans; Hypertension; Isoniazid; Nicardipine; Nifedipine; Propranolol; Quinazolines; Rifampin | 1992 |
A biphasic effect of noradrenaline on renin release from rat juxtaglomerular cells in vitro is mediated by alpha 1- and beta-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Juxtaglomerular Apparatus; Norepinephrine; Perfusion; Propranolol; Quinazolines; Rats; Renin; Yohimbine | 1992 |
[Usefulness and safety of bunazosin hydrochloride in neurogenic bladder after prolonged administration].
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Drug Evaluation; Female; Humans; Male; Middle Aged; Quinazolines; Safety; Time Factors; Urinary Bladder, Neurogenic | 1992 |
A comparison of guanfacine, bunazosin, atenolol and nadolol on blood pressure and plasma noradrenaline responses to cold pressor testing.
Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Atenolol; Blood Pressure; Cold Temperature; Guanfacine; Humans; Hypertension; Nadolol; Norepinephrine; Quinazolines; Receptors, Adrenergic; Stress, Physiological | 1992 |
Effects of alpha-adrenoceptor antagonists and clonidine on the haemodynamic response to acute hypovolaemia in conscious rabbits.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Drug Interactions; Heart Rate; Hemorrhage; Injections, Intravenous; Pharmaceutical Vehicles; Plasma Volume; Quinazolines; Rabbits; Yohimbine | 1992 |
Effect of alpha 1-adrenoceptor blockade on the left ventricular force-length relationship in dogs.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Myocardial Contraction; Quinazolines; Regression Analysis; Ventricular Function, Left | 1992 |
Characterization of rat white fat cell alpha 1B-adrenoceptors.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Animals; Blotting, Northern; Epinephrine; Iodine Radioisotopes; Kinetics; Male; Membranes; Phenethylamines; Phosphatidylinositols; Propranolol; Quinazolines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; RNA, Messenger; Stimulation, Chemical; Tetralones; Tritium | 1992 |
The effect of alpha 1-blocker, bunazosin on a murine model of congestive heart failure induced by viral myocarditis.
Topics: Adrenergic alpha-Antagonists; Animals; Disease Models, Animal; Encephalomyocarditis virus; Enterovirus Infections; Heart Failure; Male; Mice; Mice, Inbred BALB C; Myocarditis; Myocardium; Quinazolines | 1992 |
Bunazosin enhances receptor-mediated endocytosis of low-density lipoproteins.
Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Endocytosis; Humans; Iodine Radioisotopes; Lipoproteins, LDL; Quinazolines; Receptors, LDL; Swine; Tumor Cells, Cultured | 1992 |
Insulin insensitivity in nonobese, nondiabetic essential hypertension and its improvement by an alpha 1-blocker (bunazosin).
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Apoproteins; Blood Glucose; Blood Pressure; Catecholamines; Diabetes Mellitus; Female; Glucose Tolerance Test; Humans; Hypertension; Insulin; Insulin Resistance; Lipids; Male; Middle Aged; Obesity; Quinazolines; Sodium | 1992 |
[Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].
Topics: Adenoma; Adrenergic alpha-Antagonists; Aged; Humans; Male; Piperazines; Prazosin; Prostatic Hyperplasia; Prostatic Neoplasms; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha | 1992 |
Positive inotropic and negative chronotropic effects of (-)-cis-diltiazem in rat isolated atria.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Atenolol; Calcium; Diltiazem; Endothelium, Vascular; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Potassium Chloride; Quinazolines; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil | 1992 |
Beta-3 adrenergic agonist, BRL-26830A, and alpha/beta blocker, arotinolol, markedly increase regional blood flow in the brown adipose tissue in anesthetized rats.
Topics: Adipose Tissue, Brown; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Cardiac Output; Ethanolamines; Male; Propanolamines; Quinazolines; Rats; Rats, Wistar; Regional Blood Flow; Vascular Resistance | 1992 |
[The acute and chronic effects of bunazosin on exercise capacity estimated by the anaerobic threshold in patients with chronic congestive heart failure].
Topics: Adult; Aged; Anaerobic Threshold; Chronic Disease; Exercise Test; Exercise Tolerance; Female; Heart Failure; Humans; Male; Middle Aged; Quinazolines | 1992 |
Role of nitric oxide from the endothelium on the neurogenic contractile responses of rabbit pulmonary artery.
Topics: Animals; Arginine; Chromatography, High Pressure Liquid; Electric Stimulation; Electrochemistry; Endothelium, Vascular; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; Norepinephrine; Pulmonary Artery; Quinazolines; Rabbits; Sympathetic Nervous System; Tetrodotoxin | 1992 |
Role of increased alpha 1-adrenergic activity in cardiomyopathic Syrian hamster.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channels; Cardiomegaly; Cardiomyopathies; Cricetinae; Dose-Response Relationship, Drug; Heart; Hydrolysis; Mesocricetus; Myocardium; Norepinephrine; Organ Size; Phosphatidylinositols; Quinazolines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Signal Transduction | 1991 |
Chronic alpha 1 blockade in a patient with Eisenmenger syndrome.
Topics: Adolescent; Adrenergic alpha-Antagonists; Eisenmenger Complex; Humans; Male; Quinazolines | 1991 |
[Effect of moxisylyte on the lower urinary tracts (1). Effect on the isolated rabbit urethra and bladder].
Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Moxisylyte; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Prazosin; Quinazolines; Rabbits; Urethra; Urinary Bladder | 1991 |
[Effect of moxisylyte on the lower urinary tracts (2). Effect on the urethra in anesthetized dogs].
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Moxisylyte; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phenylephrine; Prazosin; Quinazolines; Urethra; Yohimbine | 1991 |
Age-related changes in adrenergic alpha 1, alpha 2, and beta receptors of rat white fat cell membranes: an analysis using [3H]bunazosin as a novel ligand for the alpha 1 adrenoceptor.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aging; Animals; Binding Sites; Cell Membrane; Epididymis; Kinetics; Male; Obesity; Propanolamines; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1991 |
[Effects of topically applied bunazosin hydrochloride on choroidal capillary blood flow and intraocular pressure of rabbit eye].
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Capillaries; Choroid; Intraocular Pressure; Propranolol; Quinazolines; Rabbits; Regional Blood Flow | 1991 |
Effects of long term treatment with an alpha 1 adrenoceptor blocker on cardiac hypertrophy, contractility, and myosin isoenzymes in spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Heart; Hypertension; Male; Myocardial Contraction; Myocardium; Myosins; Organ Size; Quinazolines; Rats; Rats, Inbred SHR; Time Factors | 1991 |
[Ocular hypotensive effects of topically applied bunazosin, an alpha 1-adrenoceptor blocker, in rabbits and cats].
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Cats; Intraocular Pressure; Male; Quinazolines; Rabbits | 1991 |
Comparison of alpha 1-adrenoceptors between rat brain and spleen.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Dibenzylchlorethamine; Kinetics; Male; Phenoxybenzamine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spleen | 1991 |
[Fundamental and clinical studies on alpha 1-blocker therapy for idiopathic male infertility].
Topics: Administration, Oral; Adrenergic alpha-Antagonists; Humans; Infertility, Male; Male; Prostate; Quinazolines; Sperm Motility; Testis; Vas Deferens | 1991 |
Binding characteristics of alpha 1-adrenoceptors in bovine prostate using a radioligand binding assay.
Topics: Adrenergic alpha-Antagonists; Animals; Cattle; Kinetics; Male; Membranes; Phentolamine; Prazosin; Prostate; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium | 1991 |
Pharmacological features of vascular responses of isolated dog and monkey lingual arteries to vasoactive substances.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Macaca; Male; Norepinephrine; Perfusion; Potassium Chloride; Quinazolines; Tongue; Vasoconstrictor Agents | 1991 |
Differential effects of antihypertensive agents on proliferation of vascular smooth muscle cells from spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Cell Division; Cells, Cultured; Hypertension; Male; Muscle, Smooth, Vascular; Nifedipine; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY | 1991 |
Bunazosin, an alpha-adrenoceptor antagonist, blocks calcium current in guinea-pig ventricular myocytes.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Guinea Pigs; Heart; Heart Ventricles; Quinazolines | 1991 |
[3H]bunazosin, a novel selective radioligand of alpha 1 adrenoceptors in human prostates.
Topics: Adrenergic alpha-Antagonists; Cell Membrane; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium | 1991 |
[Characterization and localization of alpha 1-adrenoceptors in human prostate--with special reference to the zonal difference in receptor distribution].
Topics: Autoradiography; Binding Sites; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Urinary Bladder Neoplasms | 1991 |
Pharmacologic analysis of 7-O-ethyl-fangchinoline-induced vasodilation properties in isolated perfused common carotid arteries of Wistar Kyoto rats and spontaneously hypertensive rats.
Topics: Alkaloids; Animals; Atropine; Benzylisoquinolines; Carotid Arteries; Diltiazem; In Vitro Techniques; Isoproterenol; Male; Phenylephrine; Propranolol; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Vasoconstriction; Vasodilation; Vasodilator Agents | 1991 |
Effects of regression of left ventricular hypertrophy following atenolol or bunazosin therapy on ischemic cardiac function and myocardial metabolism in spontaneously hypertensive rats.
Topics: Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Atenolol; Blood Pressure; Cardiomegaly; Coronary Circulation; Coronary Disease; Lactates; Lactic Acid; Male; Myocardium; Phosphocreatine; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Remission Induction | 1991 |
Effect of combined dopamine and bunazosin on the ischemic heart after occlusion of the coronary artery.
Topics: Adrenergic alpha-Antagonists; Animals; Arterial Occlusive Diseases; Cardiac Output, Low; Coronary Circulation; Coronary Disease; Dogs; Dopamine; Drug Evaluation, Preclinical; Drug Therapy, Combination; Hemodynamics; Infusions, Intravenous; Myocardium; Oxygen Consumption; Quinazolines | 1990 |
Effects of bunazosin, a selective alpha 1-adrenergic blocking agent, on myocardial energy metabolism in ischemic dog heart.
Topics: Adenine Nucleotides; Adrenergic alpha-Antagonists; Animals; Carbohydrate Metabolism; Coronary Disease; Dogs; Electrocardiography; Energy Metabolism; Female; Heart; Hemodynamics; Hexosephosphates; In Vitro Techniques; Lactates; Male; Myocardium; Phosphocreatine; Pyruvates; Quinazolines | 1990 |
Perfusion-time dependent enhancements of guanabenz- and KCl-induced vasoconstrictions in isolated and perfused dog pulmonary veins.
Topics: Adrenergic alpha-Antagonists; Animals; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Guanabenz; Imidazoles; Male; Potassium Chloride; Pulmonary Veins; Quinazolines; Receptors, Adrenergic, alpha; Time Factors; Vasoconstriction | 1990 |
Intracerebroventricular injections of endothelin increase arterial pressure in conscious rats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Brain; Endothelins; Guanidines; Injections, Intraventricular; Male; Niacinamide; Nicardipine; Nicorandil; Pinacidil; Quinazolines; Rats; Rats, Inbred Strains; Vasodilator Agents | 1990 |
[Changes in intraocular pressure and aqueous humor dynamics of normal human eyes after topical application of bunazosin hydrochloride].
Topics: Adrenergic alpha-Antagonists; Adult; Aqueous Humor; Depression, Chemical; Eye Proteins; Humans; Intraocular Pressure; Male; Middle Aged; Ophthalmic Solutions; Quinazolines | 1990 |
[Efficacy of combination of Ea-0643 (bunazosin hydrochloride) and bethanechol chloride in patients with neurogenic bladder].
Topics: Adrenergic alpha-Antagonists; Aged; Bethanechol; Bethanechol Compounds; Drug Evaluation; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Parasympathomimetics; Quinazolines; Urinary Bladder, Neurogenic | 1990 |
Parasympathetic nervous system in patients with Graves' disease determined by R-R interval variations on electrocardiogram.
Topics: Adrenergic alpha-Antagonists; Adult; Electrocardiography; Female; Graves Disease; Humans; Male; Metoprolol; Parasympathetic Nervous System; Propranolol; Quinazolines; Receptors, Adrenergic, beta | 1990 |
Predominant acetylcholine-induced vasoconstriction in isolated, perfused simian facial veins.
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Blood Pressure; Diltiazem; Face; Female; In Vitro Techniques; Macaca; Male; Muscle, Smooth, Vascular; Parasympatholytics; Physostigmine; Piperidines; Pirenzepine; Potassium Chloride; Quinazolines; Receptors, Muscarinic; Saponins; Vasoconstriction; Veins | 1990 |
Bunazosin induces use-dependent slowing of conduction in guinea-pig ventricular myocardium.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Guinea Pigs; Heart Conduction System; In Vitro Techniques; Kinetics; Membrane Potentials; Papillary Muscles; Quinazolines | 1990 |
Protective effects of nipradilol, isosorbide dinitrate, and bunazosin on coronary artery constriction induced by intracoronary injection of acetylcholine in pigs.
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Coronary Angiography; Coronary Vessels; Dose-Response Relationship, Drug; Isosorbide Dinitrate; Propanolamines; Quinazolines; Vasoconstriction | 1990 |
Inhibition of Ca2+ inward current in rabbit sinoatrial node by bunazosin, an alpha-adrenoceptor antagonist.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Quinazolines; Rabbits; Sinoatrial Node | 1987 |
Biochemical basis for reperfusion arrhythmias.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Coronary Circulation; Coronary Disease; Dogs; Female; Ion Channels; Male; Mitochondria, Heart; Myocardium; Phospholipases; Quinazolines | 1987 |
Postjunctional alpha-adrenoceptor subtypes in isolated and perfused canine epicardial coronary arteries.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Coronary Vessels; Dogs; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Quinazolines; Receptors, Adrenergic, alpha; Vasoconstriction; Vasodilation; Xylazine | 1987 |
Effects of intraocular pressure change on movement of FITC-dextran across vitreous-aqueous interface.
Topics: Adrenergic alpha-Antagonists; Animals; Anterior Chamber; Aqueous Humor; Dextrans; Female; Fluorescein-5-isothiocyanate; Fluoresceins; Fluorometry; Intraocular Pressure; Male; Quinazolines; Rabbits; Vitreous Body | 1989 |
Effects of specific alpha-adrenoceptive agents on extraneuronal uptake (uptake2) of isoproterenol in perfused rat heart.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Guanabenz; Isoproterenol; Male; Methoxamine; Myocardium; Neurons; Phenylephrine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Sulfonamides; Tropolone | 1989 |
Time-dependent enhancement of xylazine-induced, alpha-2 adrenoceptor-mediated vasoconstriction in isolated and perfused canine pulmonary veins.
Topics: Adrenergic alpha-Agonists; Animals; Dogs; Endothelium, Vascular; Female; Imidazoles; In Vitro Techniques; Male; Perfusion; Pulmonary Veins; Quinazolines; Receptors, Adrenergic, alpha; Saponins; Thiazines; Time Factors; Vasoconstriction; Xylazine | 1989 |
Localization of alpha 1-adrenoceptor in the rat kidney: in vitro autoradiography using [3H]-bunazosin.
Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; In Vitro Techniques; Kidney; Kidney Cortex; Kidney Medulla; Male; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1989 |
[Acute and chronic effects of bunazosin in patients with congestive heart failure].
Topics: Adrenergic alpha-Antagonists; Atrial Natriuretic Factor; Chronic Disease; Exercise Test; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines | 1989 |
Bunazosin, an alpha 1-adrenoceptor blocker, differentially releases co-transmitters in dog mesenteric vessels.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Dogs; In Vitro Techniques; Mesenteric Arteries; Mesenteric Veins; Methoxyhydroxyphenylglycol; Muscle, Smooth, Vascular; Neurotransmitter Agents; Norepinephrine; Phentolamine; Quinazolines; Yohimbine | 1989 |
Alpha-blocking potencies of antihypertensive agents (prazosin, terazosin, bunazosin, SGB-1534 and ketanserin) having with quinazoline or quinazolinedione as assessed by radioligand binding assay methods in rat brain.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brain; Cell Membrane; Clonidine; Dihydroalprenolol; Ketanserin; Male; Prazosin; Quinazolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1989 |
Hemodynamic benefits of long-term bunazosin (alpha-1 blocker) therapy in rats with myocardial infarction and heart failure.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiac Output, Low; Chronic Disease; Female; Heart Ventricles; Hemodynamics; Myocardial Infarction; Quinazolines; Rats; Rats, Inbred Strains; Vascular Resistance; Weight Gain | 1989 |
Selective blockade of alpha 1-adrenoceptors of porcine vascular smooth muscle cells by bunazosin.
Topics: Adrenergic alpha-Antagonists; Animals; In Vitro Techniques; Membranes; Microsomes; Muscle, Smooth, Vascular; Muscles; Prazosin; Quinazolines; Swine; Yohimbine | 1989 |
Renal and hormonal effects of alpha 1-adrenoceptor blockade by bunazosin in essential hypertension.
Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Atrial Natriuretic Factor; Blood Pressure; Creatinine; Glomerular Filtration Rate; Humans; Hypertension; Kidney; Norepinephrine; Quinazolines; Regional Blood Flow; Vascular Resistance | 1989 |
In vivo experiments for the evaluation of alpha 1-adrenoceptor antagonistic effects of SGB-1534 on canine urethra.
Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Dose-Response Relationship, Drug; Female; Hypogastric Plexus; Phenylephrine; Prazosin; Quinazolines; Urethra | 1989 |
[Roles of vascular and renal thromboxanes in the antihypertensive effects of alpha 1 adrenoceptor antagonists].
Topics: Adrenergic alpha-Antagonists; Animals; Blood Vessels; Hypertension; Kidney; Male; Methacrylates; Quinazolines; Rats; Rats, Inbred SHR; Thromboxane A2; Thromboxane-A Synthase | 1989 |
[Clinical application of adrenoceptor blockers in the treatment of hypertension].
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Carbazoles; Carvedilol; Humans; Hypertension; Labetalol; Prazosin; Propanolamines; Quinazolines | 1989 |
[Exercise testing of the chronic effects of bunazosin hydrochloride on dilated cardiomyopathy].
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Cardiomyopathy, Dilated; Drug Evaluation; Exercise Test; Female; Hemodynamics; Humans; Male; Middle Aged; Quinazolines | 1989 |
Protection of acute ischemic myocardial injury by pharmacological intervention.
Topics: Adenosine Triphosphatases; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium-Transporting ATPases; Coenzymes; Coronary Disease; Diltiazem; Dogs; Myocardium; Niacinamide; Nicorandil; Quinazolines; Sarcoplasmic Reticulum; Ubiquinone; Vasodilator Agents | 1989 |
[Acute effects of oral bunazosin-hydrochloride in acute heart failure].
Topics: Acute Disease; Administration, Oral; Adrenergic alpha-Antagonists; Aged; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines | 1989 |
Involvement of adrenergic mechanism in hyperglycemia due to SCN stimulation.
Topics: Adrenergic alpha-Antagonists; Animals; Autonomic Nervous System; Electric Stimulation; Female; Glucagon; Hexamethonium; Hexamethonium Compounds; Hyperglycemia; Insulin; Propranolol; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Suprachiasmatic Nucleus; Yohimbine | 1989 |
[The effect of bunazosin vs captopril on hemodynamic and neurohumoral parameters in patients with congestive heart failure].
Topics: Adrenergic alpha-Antagonists; Aldosterone; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Atrial Natriuretic Factor; Captopril; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines; Renin | 1989 |
Exercise testing of the chronic effects of bunazosin hydrochloride on dilated cardiomyopathy.
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Cardiomyopathy, Dilated; Echocardiography; Electrocardiography; Exercise Test; Female; Hemodynamics; Humans; Male; Middle Aged; Quinazolines | 1989 |
Properties of the pupillary dilation produced by the humoral factor in the pupillary reflex dilation: an experimental study in the cat.
Topics: Animals; Atropine; Biological Factors; Cats; Electric Stimulation; Iris; Phenoxybenzamine; Propranolol; Quinazolines; Reflex, Pupillary; Sciatic Nerve; Yohimbine | 1989 |
Effect of bunazosin on cardiac sympathetic nerve activity in anesthetized rats.
Topics: Anesthesia; Animals; Blood Pressure; Heart Conduction System; Heart Rate; Kidney; Male; Nervous System; Nervous System Physiological Phenomena; Quinazolines; Rats; Rats, Inbred Strains; Sympathetic Nervous System | 1989 |
Perfusion-time-dependent appearance of blocking effect of diltiazem on norepinephrine-induced vasoconstriction in isolated, perfused dog pulmonary veins.
Topics: Animals; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Perfusion; Propranolol; Pulmonary Veins; Quinazolines; Time Factors; Vasoconstriction | 1989 |
Acute systemic and regional hemodynamic effects of alpha 1-adrenoceptor blockade in conscious spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Consciousness; Dose-Response Relationship, Drug; Hemodynamics; Hypertension; Male; Quinazolines; Rats; Rats, Inbred SHR; Regional Blood Flow | 1986 |
Acute effects of bunazosin on aortic, vertebral, coronary and renal blood flows of anesthetized dogs.
Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Aorta; Coronary Circulation; Dogs; Female; Male; Quinazolines; Regional Blood Flow; Renal Circulation; Time Factors; Vascular Resistance; Vertebral Artery; Yohimbine | 1986 |
Successful treatment of oligospermic and azoospermic men with alpha 1-blocker and beta-stimulator: new treatment for idiopathic male infertility.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Ethanolamines; Female; Humans; Infertility, Male; Male; Oligospermia; Pregnancy; Procaterol; Quinazolines; Sperm Count; Sperm Motility; Time Factors | 1986 |
Effects of bunazosin and propranolol on ventricular arrhythmias in dogs with hypokalemia.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dogs; Female; Heart Ventricles; Hypokalemia; Male; Mitochondria, Heart; Potassium; Propranolol; Quinazolines; Sodium | 1987 |
Actions of the alpha-1 adrenoceptor blocker bunazosin on the norepinephrine-induced contraction of smooth muscles in the rabbit proximal urethra.
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Calcium; Dose-Response Relationship, Drug; Guanethidine; Microelectrodes; Muscle Contraction; Muscle, Smooth; Norepinephrine; Potassium; Propranolol; Quinazolines; Rabbits; Urethra | 1987 |
Effect of egg yolk lecithin on transdermal delivery of bunazosin hydrochloride.
Topics: Adjuvants, Pharmaceutic; Administration, Cutaneous; Adrenergic alpha-Antagonists; Animals; Egg Yolk; In Vitro Techniques; Male; Mice; Mice, Hairless; Phosphatidylcholines; Quinazolines; Rabbits; Skin Absorption | 1987 |
Pharmacological analysis of vasoconstriction of isolated canine ophthalmic and ciliary arteries to alpha-adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Ciliary Body; Diltiazem; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Nitroprusside; Ophthalmic Artery; Quinazolines; Vasoconstriction | 1987 |
Potentiating effect of tyramine on acetaldehyde-induced vasoconstriction in isolated dog mesenteric arteries.
Topics: Acetaldehyde; Adrenergic alpha-Antagonists; Animals; Dogs; In Vitro Techniques; Mesenteric Arteries; Norepinephrine; Quinazolines; Tachyphylaxis; Tyramine; Vasoconstriction | 1987 |
Pharmacological analysis of 5-HT-induced vasoconstriction in isolated, perfused dog skeletal muscle arteries.
Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Cold Temperature; Diltiazem; Dogs; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Quinazolines; Serotonin; Vasoconstriction | 1987 |
Sympatholytic effects of the intravenously injected alpha 1-adrenergic blocker, bunazosin, in anaesthetized rats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Denervation; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Phentolamine; Phenylephrine; Pressoreceptors; Quinazolines; Rats; Rats, Inbred Strains; Sympathetic Nervous System | 1987 |
Alpha-blocker, bunazosinhydrochloride decreases cytosolic Ca++ of cultured rat aortic smooth muscle cells.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Calcium; Cells, Cultured; Cytosol; Kinetics; Muscle, Smooth, Vascular; Phenylephrine; Quinazolines; Rats; Rats, Inbred Strains | 1988 |
Role of alpha 1-adrenergic receptors and the effect of bunazosin on the histopathology of cardiomyopathic Syrian hamsters of strain BIO 14.6.
Topics: Adrenergic alpha-Antagonists; Animals; Cardiomyopathies; Cricetinae; Female; Male; Mesocricetus; Myocardium; Quinazolines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1988 |
Effect of the alpha 1-blocker bunazosin on reperfusion-induced mitochondrial dysfunction in canine hearts.
Topics: Adrenergic alpha-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dogs; Female; In Vitro Techniques; Male; Mitochondria, Heart; Oxygen Consumption; Perfusion; Phospholipases; Quinazolines | 1988 |
Effects of a new alpha 1-blocker, bunazosin hydrochloride, on plasma lipid components in hypertensive patients with hypercholesterolemia.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Apolipoproteins; Blood Pressure; Cholesterol; Female; Humans; Hypercholesterolemia; Hypertension; Lipids; Lipoproteins; Male; Middle Aged; Quinazolines; Triglycerides | 1987 |
In vitro study on corneal permeability to bunazosin.
Topics: Adrenergic alpha-Antagonists; Animals; Caprylates; Cornea; Decanoic Acids; In Vitro Techniques; Octanols; Permeability; Quinazolines; Rabbits; Water | 1988 |
The aortic alpha 1-adrenergic receptor in familial amyloidotic polyneuropathy.
Topics: Adrenergic alpha-Antagonists; Amyloidosis; Aorta; Female; Humans; Male; Middle Aged; Peripheral Nervous System Diseases; Quinazolines; Receptors, Adrenergic, alpha | 1988 |
Cardioprotective action of alpha-blocking agents, phentolamine and bunazosin, on hypoxic and reoxygenated myocardium.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Energy Metabolism; Heart; Hypoxia; Male; Myocardial Contraction; Myocardium; Oxygen; Phentolamine; Quinazolines; Rabbits | 1988 |
Corneal permeability to bunazosin in rabbits.
Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Cornea; Male; Permeability; Quinazolines; Rabbits | 1988 |
Studies on improved corneal permeability to bunazosin.
Topics: Adrenergic alpha-Antagonists; Animals; Caprylates; Chromatography, High Pressure Liquid; Cornea; Hydrogen-Ion Concentration; In Vitro Techniques; Permeability; Protein Binding; Quinazolines; Rabbits | 1988 |
Positive inotropic action of novel vasoconstrictor peptide endothelin on guinea pig atria.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Atenolol; Atrial Function; Calcium; Cimetidine; Diphenhydramine; Endothelins; Guinea Pigs; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Methysergide; Myocardial Contraction; Nicardipine; Peptides; Potassium; Quinazolines; Reference Values | 1988 |
[The effect of bunazosin hydrochloride on the intraocular pressure and the aqueous humor dynamics of the rabbit eye].
Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Female; Intraocular Pressure; Quinazolines; Rabbits | 1988 |
Antiarrhythmic effects of alpha-adrenoceptor antagonists in guinea pig ventricular myocardium.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Guinea Pigs; Heart; In Vitro Techniques; Quinazolines; Receptors, Adrenergic, beta; Strophanthidin | 1988 |
[The effect of bunazosin on hypertension during anesthesia; effectiveness of nasal instillation].
Topics: Administration, Intranasal; Adrenergic alpha-Antagonists; Anesthesia, General; Female; Humans; Hypertension; Male; Middle Aged; Quinazolines | 1988 |
Effects of selective alpha 1-adrenoceptor blockade in dogs with hypoxic pulmonary vasoconstriction.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Gas Analysis; Dogs; Hemodynamics; Hypertension, Pulmonary; Hypoxia; Pulmonary Circulation; Quinazolines; Vasoconstriction | 1988 |
Possible mechanism of acetaldehyde-induced noradrenaline release from sympathetic nerve terminals in isolated blood vessels.
Topics: Acetaldehyde; Adrenergic alpha-Antagonists; Animals; Dogs; Hydrocortisone; In Vitro Techniques; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Quinazolines; Sympathetic Nervous System; Tachyphylaxis; Tyramine; Vasoconstriction | 1988 |
Properties of [3H]bunazosin binding in rat kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Cations; Hot Temperature; Kidney; Kidney Cortex; Kinetics; Male; Membranes; Quinazolines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Subcellular Fractions; Tissue Distribution; Tritium | 1988 |
The effects of vasoactive agents on the proliferation of vascular smooth muscle cells grown in vitro.
Topics: Amiloride; Animals; Captopril; Cell Division; Cells, Cultured; Chlorpromazine; In Vitro Techniques; Labetalol; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Nifedipine; Norepinephrine; Propranolol; Quinazolines; Rats; Sulfonamides | 1988 |
Effects of bunazosin on electrical responses of smooth muscle cells of the guinea-pig mesenteric artery and vein to perivascular nerve stimulation and to noradrenaline.
Topics: Animals; Electric Stimulation; Evoked Potentials; Female; Guinea Pigs; Male; Membrane Potentials; Mesenteric Arteries; Mesenteric Veins; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Yohimbine | 1987 |
Existence of renal alpha 1- and alpha 2-adrenoceptors in the human kidney: radioligand binding study in membranes from the human renal cortex and medulla.
Topics: Humans; Kidney; Kidney Cortex; Kidney Medulla; Membranes; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
Mechanism of myocardial injury in dogs with hypokalaemia.
Topics: Animals; Calcium; Cardiomyopathies; Coronary Circulation; Creatine Kinase; Dogs; Epinephrine; Female; Hypokalemia; Male; Mitochondria, Heart; Myocardium; Quinazolines | 1988 |
Different antagonistic effects of bunazosin and ketanserin on the norepinephrine-induced vasoconstriction in isolated, perfused canine and simian skeletal muscle arteries.
Topics: Animals; Arteries; Dogs; Female; In Vitro Techniques; Ketanserin; Macaca; Male; Muscles; Norepinephrine; Quinazolines; Regional Blood Flow; Vasoconstriction | 1988 |
Vasoconstrictor effects of endogenous digitalis-like factors extracted from urine of hypertensive patients.
Topics: Animals; Arteries; Blood Proteins; Cardenolides; Digoxin; Dogs; Ear, External; Epinephrine; Humans; Hypertension; In Vitro Techniques; Mesenteric Arteries; Ouabain; Phentolamine; Potassium Chloride; Quinazolines; Saponins; Vasoconstrictor Agents; Verapamil | 1987 |
[Effect of bunazosin on lower urinary tract function in the decerebrated dog].
Topics: Animals; Decerebrate State; Dogs; Electric Stimulation; Electromyography; Pons; Quinazolines; Urethra; Urinary Bladder | 1987 |
[Effects of oral bunazosin hydrochloride on hemodynamic and metabolic responses to exercise (ergometer, 25W, 5 min) in patients with severe congestive heart failure].
Topics: Aged; Exercise Test; Female; Heart Failure; Hemodynamics; Humans; Male; Metabolism; Middle Aged; Quinazolines | 1987 |
[Effects of new antihypertensive agent, 2-[4-(n-butyryl)-homopiperazine-1-ul]-4-amino-6, 7-dimethoxy-quinazoline (E-643), on blood pressure, urinary sodium excretion and urinary norepinephrine excretion rate in stroke-prone, spontaneously hypertensive rat
Topics: Animals; Antihypertensive Agents; Blood Pressure; Body Weight; Catecholamines; Cerebrovascular Disorders; Eating; Heart Rate; Humans; Hypertension; Kidney; Male; Natriuresis; Norepinephrine; Potassium; Quinazolines; Rats; Rats, Inbred SHR | 1985 |
The potentiating effect of an alpha-adrenergic blocking agent (E-643) on the action of bronchodilators.
Topics: Adrenergic alpha-Antagonists; Animals; Bronchodilator Agents; Cyclic AMP; Cyclic GMP; Drug Synergism; Epinephrine; Guinea Pigs; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Prostaglandins E; Quinazolines; Trachea | 1980 |
Effects of alpha blockers on blood pressure and on the Ca-contracture of cat aortic strips.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Blood Pressure; Calcium; Cats; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Phentolamine; Quinazolines; Regional Blood Flow | 1980 |
alpha-Adrenoceptor blocking properties of a new antihypertensive agent, 2-[4-(n-butyryl)-homopiperazine-1-yl]-4-amino-6,7-dimethoxyquinazoline (E-643).
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Barium; Blood Pressure; Calcium; Dose-Response Relationship, Drug; Epinephrine; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Phentolamine; Potassium; Quinazolines; Rabbits; Rats; Vasoconstriction | 1980 |
Antihypertensive effect of E-643, a new alpha-adrenergic blocking agent.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aldosterone; Blood Pressure; Chemical Phenomena; Chemistry; Dopamine beta-Hydroxylase; Epinephrine; Female; Humans; Male; Middle Aged; Norepinephrine; Posture; Pulse; Quinazolines; Renin | 1981 |
Chronotropic and inotropic effects of 3 kinds of alpha-adrenergic blockers on the isolated dog atria.
Topics: Adrenergic alpha-Antagonists; Animals; Atropine; Dogs; Female; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Phenoxybenzamine; Phentolamine; Propranolol; Quinazolines | 1981 |
Comparison of pre- and postsynaptic alpha-adrenoceptor blocking effects of E-643 in the isolated vas deferens of the rat.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens | 1981 |
[Effects of quinazoline derivatives (E-643 and prazosin) on blood pressure, pulse and renin-angiotensin system in two cases of pheochromocytoma (author's transl)].
Topics: Adolescent; Adrenal Gland Neoplasms; Adrenergic alpha-Antagonists; Adult; Blood Pressure; Humans; Male; Pheochromocytoma; Prazosin; Pulse; Quinazolines; Renin-Angiotensin System | 1981 |
Characteristics of [3H]E-643-binding to alpha adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Binding Sites; Binding, Competitive; Brain; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Protein Binding; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Temperature; Tritium | 1982 |
Effect of E-643 on alpha-adrenoceptor-mediated inotropic responses to phenylephrine in the left atria of guinea pigs.
Topics: Adrenergic alpha-Antagonists; Animals; Guinea Pigs; Heart Atria; In Vitro Techniques; Myocardial Contraction; Phenylephrine; Quinazolines; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Sotalol; Stimulation, Chemical | 1982 |
(-)-Amidephrine, a selective agonist for alpha 1-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Animals; Electric Stimulation; Ethanolamines; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Quinazolines; Rats; Vas Deferens | 1983 |
[Effects and site of action of alpha-receptor blocker in bronchial asthma].
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Asthma; Dinoprost; Female; Humans; Male; Metaproterenol; Middle Aged; Prostaglandins F; Quinazolines | 1983 |
[Effects of E-643 on the regional myocardial function and hemodynamics in experimental acute coronary artery occlusion].
Topics: Adrenergic alpha-Antagonists; Animals; Coronary Disease; Dogs; Hemodynamics; Myocardial Contraction; Quinazolines | 1983 |
[Acute effect of a new alpha 1-receptor blocking drug, E-643, on severe congestive heart failure--pharmacokinetic and hemodynamic studies].
Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Drug Evaluation; Female; Heart Failure; Hemodynamics; Humans; Kinetics; Male; Middle Aged; Quinazolines | 1983 |
[Clinical effect of new alpha-adrenergic blocker on micturition disturbance of neurogenic bladder and lower urinary tract obstruction].
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Female; Humans; Male; Middle Aged; Quinazolines; Urethral Obstruction; Urinary Bladder, Neurogenic; Urodynamics | 1983 |
The metabolic fate of 4-amino-2-(4-butanoyl-hexahydro-1H-1, 4-diazepin-1-yl)-6,7-dimethoxy-quinazoline HCl.
Topics: Adult; Animals; Bile; Enterohepatic Circulation; Feces; Female; Humans; In Vitro Techniques; Intestinal Absorption; Male; Microsomes, Liver; Quinazolines; Rabbits; Rats; Rats, Inbred Strains; Tissue Distribution | 1982 |
[Acute effects of a new antihypertensive quinazoline derivative, E-643 in severe heart failure--hemodynamics, plasma catecholamine levels and blood gas data (author's transl)].
Topics: Adult; Aged; Catecholamines; Female; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Quinazolines | 1981 |
Participation of endogenous noradrenaline in the release of ATP by high potassium in the rat caudal artery.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Arteries; In Vitro Techniques; Male; Norepinephrine; Potassium; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha | 1995 |
Effect of bunazosin, alpha 1-adrenoceptor blocker, on multidirectional contractile response and localization of bunazosin binding sites in human hypertrophied prostate.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Autoradiography; Binding Sites; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prostate; Prostatic Hyperplasia; Quinazolines; Receptors, Adrenergic, alpha-1 | 1995 |
Comparison of 5-hydroxytryptamine-induced contraction of rat pulmonary artery to that of aorta in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Ketanserin; Male; Pindolol; Pulmonary Artery; Quinazolines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Ritanserin; Serotonin; Vasoconstriction | 1995 |
Effects of alpha-blocker on sperm concentration, motility, intraluminal pressure and fluid movement in the rat cauda epididymis.
Topics: Adrenergic alpha-Antagonists; Animals; Body Fluids; Epididymis; Male; Organ Size; Pressure; Quinazolines; Rats; Rats, Sprague-Dawley; Seminiferous Tubules; Sperm Count; Sperm Motility; Testis | 1995 |
Effects of bunazosin, a selective alpha 1-blocking agent, and propranolol used alone and in combination on canine ventricular refractoriness and its dispersion during myocardial ischemia.
Topics: Adrenergic alpha-Antagonists; Animals; Coronary Circulation; Dogs; Drug Therapy, Combination; Electrocardiography; Injections, Intravenous; Myocardial Ischemia; Propranolol; Quinazolines | 1993 |
Functional 5-HT receptor subtypes in the isolated canine common carotid artery.
Topics: Adrenergic alpha-Antagonists; Animals; Carotid Artery, Common; Diltiazem; Dogs; Female; Ketanserin; Male; Methysergide; Norepinephrine; Potassium Chloride; Quinazolines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spiperone; Vasoconstriction | 1994 |
Effects of sympathetic stimulation, with and without previous alpha 1 and beta adrenoceptor blockade, on refractoriness dispersion in canine heart.
Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Electrophysiology; Heart; Myocardial Ischemia; Propranolol; Quinazolines; Stimulation, Chemical; Sympathetic Nervous System | 1994 |
Acute hemodynamic effects of bunazosin in congestive heart failure--differing responses according to degree of cardiac dysfunction.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Female; Heart; Heart Failure; Heart Rate; Hemodynamics; Humans; Male; Middle Aged; Pulmonary Wedge Pressure; Quinazolines; Stroke Volume; Vascular Resistance | 1993 |
[Evaluation of bunazosin hydrochloride with a model of ocular circulation disturbance induced by endothelin-1].
Topics: Adrenergic alpha-Antagonists; Animals; Endothelins; Optic Disk; Quinazolines; Rabbits; Regional Blood Flow; Retinal Artery | 1994 |
Characteristics of the responses of isolated and perfused canine splenic arteries to vasoactive substances and to periarterially electrical stimulation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dogs; Electric Stimulation; Female; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Quinazolines; Splenic Artery; Vasoconstriction; Vasoconstrictor Agents | 1994 |
The effect of bunazosin on monocrotaline-induced pulmonary hypertension in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Hemodynamics; Hypertension, Pulmonary; Monocrotaline; Quinazolines; Rats; Rats, Sprague-Dawley | 1994 |
[Effects of long-term application of bunazosin hydrochloride eye drops on the aqueous flow rate and blood-aqueous barrier permiability in rabbit eyes].
Topics: Adrenergic alpha-Antagonists; Animals; Aqueous Humor; Blood; Intraocular Pressure; Ophthalmic Solutions; Permeability; Quinazolines; Rabbits | 1994 |
Ocular pharmacokinetics and pharmacodynamics in rabbits of ibopamine, a new mydriatic agent.
Topics: Adrenergic alpha-Agonists; Animals; Aqueous Humor; Deoxyepinephrine; Dose-Response Relationship, Drug; Female; Male; Moxisylyte; Mydriatics; Pupil; Quinazolines; Rabbits; Reserpine; Swine; Time Factors | 1993 |
Selective suppression by bunazosin of alpha-adrenergic agonist evoked elevation of intraocular pressure in sympathectomized rabbit eyes.
Topics: Adrenergic alpha-Antagonists; Animals; Ganglia, Sympathetic; Ganglionectomy; Intraocular Pressure; Male; Norepinephrine; Ocular Hypotension; Ophthalmic Solutions; Phenylephrine; Pupil; Quinazolines; Rabbits; Receptors, Adrenergic, alpha | 1993 |
Vascular responsiveness of rabbit common carotid, renal and femoral arteries to alpha-adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dinoprost; Dose-Response Relationship, Drug; Drug Interactions; Female; Femoral Artery; In Vitro Techniques; Male; Phenylephrine; Quinazolines; Rabbits; Renal Artery; Vasoconstriction | 1993 |
Alterations of binding characteristics of alpha 1-,beta 1-adrenoceptors and Ca2+ binding sites in the myocardium of spontaneously hypertensive rats (SHR) by chronically administered bunazosin, atenolol, ketanserin and verapamil.
Topics: Adrenergic alpha-Antagonists; Animals; Atenolol; Binding Sites; Blood Pressure; Calcium Channels; Heart; In Vitro Techniques; Ketanserin; Kinetics; Myocardium; Norepinephrine; Quinazolines; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Verapamil | 1993 |
Long-term alpha 1 blockade does not reverse cardiac hypertrophy in spontaneously hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Hemodynamics; Hypertension; Hypertrophy, Left Ventricular; Male; Norepinephrine; Quinazolines; Rats; Rats, Inbred SHR; Renin | 1993 |
Effects of alpha-adrenergic blockade on regional myocardial function in canine ischemic myocardium during beta-adrenergic blockade.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Coronary Circulation; Dogs; Female; Hemodynamics; Male; Myocardial Contraction; Myocardial Ischemia; Myocardium; Prazosin; Propranolol; Prospective Studies; Quinazolines; Random Allocation; Yohimbine | 1995 |
Exaggeration of acute liver damage by hepatic sympathetic nerves and circulating catecholamines in perfused liver of rats treated with D-galactosamine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Analysis of Variance; Animals; Aspartate Aminotransferases; Calcium; Electric Stimulation; Galactosamine; Isoproterenol; L-Lactate Dehydrogenase; Liver; Male; Norepinephrine; Perfusion; Phenylephrine; Quinazolines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Sympathomimetics | 1996 |
Effects of alpha-blocker on daily testicular sperm production and sperm concentration, motility, intraluminal pressure and fluid movement in the rat epididymis.
Topics: Adrenergic alpha-Antagonists; Animals; Biological Transport; Body Fluids; Epididymis; Male; Organ Size; Pressure; Quinazolines; Rats; Rats, Sprague-Dawley; Seminiferous Tubules; Sperm Count; Sperm Motility; Spermatogenesis; Testis | 1995 |
Induction of DNA breaks in cardiac myoblast cells by norepinephrine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Calcium Channel Blockers; Captopril; DNA; DNA Damage; DNA, Single-Stranded; Heart; Hydrogen Peroxide; Myocardium; Norepinephrine; Propranolol; Quinazolines; Rats; Stimulation, Chemical; Verapamil | 1996 |
Effect of alpha-blockers on epididymal sperm concentration, motility and testicular productivity in the rat.
Topics: Adrenergic alpha-Antagonists; Animals; Epididymis; Male; Quinazolines; Rats; Rats, Sprague-Dawley; Sperm Count; Sperm Motility; Spermatogenesis; Testis | 1996 |
Effect of tamsulosin, a novel alpha 1-adrenoceptor antagonist, on urethral pressure profile in anaesthetized dogs.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Captopril; Dogs; Dose-Response Relationship, Drug; Male; Nicardipine; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin | 1996 |
Prevention of cardiac hypertrophy by a sub-antihypertensive dose of the alpha 1-adrenergic antagonist bunazosin in Dahl salt-sensitive rats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiomegaly; Hypertension; Male; Quinazolines; Rats; Sodium Chloride | 1996 |
Thromboxane inhibition potentiates antihypertensive effects of alpha 1 adrenoceptor antagonists in the rat.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aorta; Blood Pressure; Body Weight; Cells, Cultured; Drug Synergism; Eicosanoids; Ethanolamines; Kidney; Methacrylates; Muscle, Smooth, Vascular; Prazosin; Quinazolines; Rats; Rats, Inbred SHR; Sodium; Thromboxane-A Synthase; Thromboxanes | 1997 |
Effect of alpha 1-adrenoceptor antagonists on urinary bladder function in urethane-anesthetized rats.
Topics: Adrenergic alpha-Antagonists; Anesthetics; Animals; Flavoxate; Male; Parasympatholytics; Prazosin; Quinazolines; Rats; Rats, Wistar; Sulfonamides; Tamsulosin; Urethane; Urinary Bladder | 1997 |
Beta-adrenoceptor stimulation-mediated preconditioning-like cardioprotection in perfused rat hearts.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Creatine Kinase; Heart; Heart Rate; Isoproterenol; Male; Myocardial Contraction; Myocardial Ischemia; Myocardial Reperfusion; Myocardial Reperfusion Injury; Myocardium; Norepinephrine; Phenylephrine; Quinazolines; Random Allocation; Rats; Rats, Sprague-Dawley; Timolol; Ventricular Function, Left | 1997 |
[Alström syndrome--a rare disease of diabetic association].
Topics: Adult; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diagnosis, Differential; DNA Mutational Analysis; Humans; Male; Obesity; Optic Atrophy; Quinazolines; Retinitis Pigmentosa; Second Messenger Systems; Syndrome | 1997 |
Clinical impact of insulin resistance syndrome in cardiovascular diseases and its therapeutic approach.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Amlodipine; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Calcium Channel Blockers; Cardiovascular Diseases; Cilazapril; Humans; Insulin Resistance; Middle Aged; Quinazolines | 1996 |
Infarct size-reducing effect of ischemic preconditioning is related to alpha1b-adrenoceptors but not to alpha1a-adrenoceptors in rabbits.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Ischemic Preconditioning, Myocardial; Male; Phenoxybenzamine; Piperazines; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1 | 1997 |
Effects of alpha 1-adrenoreceptor subtype blockade on ischemia-reperfusion injury.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Clonidine; Dioxanes; Energy Metabolism; In Vitro Techniques; Male; Myocardial Reperfusion Injury; Quinazolines; Rats; Rats, Sprague-Dawley | 1997 |
Differences in refractory-period response of canine subendocardium and subepicardium to bunazosin, an alpha1-adrenoceptor antagonist, and propranolol during myocardial ischemia.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Dogs; Endocardium; Heart Ventricles; Myocardial Ischemia; Pericardium; Propranolol; Quinazolines; Receptors, Adrenergic, alpha-1; Refractory Period, Electrophysiological; Tachycardia, Ventricular; Ventricular Fibrillation; Ventricular Function | 1997 |
[Alpha-1 blockers for therapy of essential hypertension. 2 clinical studies with bunazosin].
Topics: Adrenergic alpha-Antagonists; Blood Pressure; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Hypertension; Quinazolines; Treatment Outcome | 1998 |
Bunazosin reduces intraocular pressure in rabbits by increasing uveoscleral outflow.
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aqueous Humor; Cyclooxygenase Inhibitors; Fluorophotometry; Flurbiprofen; Indomethacin; Intraocular Pressure; Quinazolines; Rabbits; Sclera; Tonometry, Ocular; Uvea | 1998 |
Regulation of angiotensin II receptor expression by nitric oxide in rat adrenal gland.
Topics: Adrenal Glands; Adrenergic alpha-Antagonists; Aldosterone; Animals; Blotting, Northern; Body Weight; DNA, Complementary; Enzyme Inhibitors; Gene Expression Regulation; Hemodynamics; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peptidyl-Dipeptidase A; Quinazolines; Rats; Rats, Wistar; Receptors, Angiotensin; Renin; RNA, Messenger | 1998 |
Bunazosin hydrochloride inhibits exaggerated growth of vascular smooth muscle cells from spontaneously hypertensive rats by suppressing the response to growth factors.
Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Antihypertensive Agents; Cell Division; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Epidermal Growth Factor; Growth Inhibitors; Muscle, Smooth, Vascular; Platelet-Derived Growth Factor; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; RNA, Messenger | 1998 |
[Signal transduction of serotonin release from enterochromaffin cells in mouse ileal crypts].
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Clonidine; Enterochromaffin Cells; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Norepinephrine; Phosphodiesterase Inhibitors; Prazosin; Pyrrolidinones; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Rolipram; Serotonin; Signal Transduction; Yohimbine | 1998 |
Disproportional response between refractory period and blood flow to alpha 1- and beta-adrenoceptor blockade in canine ischemic myocardium.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Coronary Circulation; Dogs; Electrocardiography; Endocardium; Heart; Myocardial Ischemia; Pericardium; Propranolol; Quinazolines; Refractory Period, Electrophysiological; Tachycardia, Ventricular; Ventricular Fibrillation | 1998 |
Bunazosin. Andante, Detantol, E 1015, E 643, EA 0643.
Topics: Adrenergic alpha-Antagonists; Aged; Antihypertensive Agents; Area Under Curve; Clinical Trials as Topic; Humans; Hypertension; Male; Prostatic Hyperplasia; Quinazolines | 1999 |
Effects of bunazosin hydrochloride sustained-release formulation on cerebral circulation.
Topics: Acetazolamide; Adrenergic alpha-Antagonists; Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Flow Velocity; Caudate Nucleus; Cerebral Infarction; Cerebrovascular Circulation; Delayed-Action Preparations; Diuretics; Enalapril; Female; Humans; Injections, Intravenous; Male; Occipital Lobe; Parietal Lobe; Quinazolines; Tomography, X-Ray Computed | 2000 |
Attenuation of KATP channel-opener induced shortening of repolarization time by alpha 1-adrenoceptor antagonist during ischemia in canine heart.
Topics: Action Potentials; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; ATP-Binding Cassette Transporters; Benzopyrans; Blood Pressure; Dogs; Electrocardiography; Electrophysiology; Heart; In Vitro Techniques; KATP Channels; Myocardial Reperfusion Injury; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinazolines | 2000 |
Different vasculoprotective roles of NO synthase isoforms in vascular lesion formation in mice.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aspirin; Carotid Arteries; Female; Fibrinolytic Agents; Isoenzymes; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neovascularization, Pathologic; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Quinazolines; Tunica Intima | 2000 |
Neuroprotective effect and intraocular penetration of nipradilol, a beta-blocker with nitric oxide donative action.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood-Retinal Barrier; Cell Count; Dose-Response Relationship, Drug; Drug Combinations; Male; N-Methylaspartate; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Propanolamines; Quinazolines; Rabbits; Rats; Rats, Sprague-Dawley; Retina; Retinal Artery; Timolol; Vasoconstriction | 2001 |
Noradrenaline stimulates 5-hydroxytryptamine release from mouse ileal tissues via alpha(2)-adrenoceptors.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Ileum; In Vitro Techniques; Male; Methoxamine; Mice; Mice, Inbred ICR; Norepinephrine; Pertussis Toxin; Phenylephrine; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha-2; Serotonin; Virulence Factors, Bordetella; Yohimbine | 2001 |
The renin-angiotensin and adrenergic nervous system in cardiac hypertrophy in fructose-fed rats.
Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Antihypertensive Agents; Blood Glucose; Blood Pressure; Catecholamines; Diet; Fructose; Glucose Tolerance Test; Heart Rate; Hydralazine; Hyperinsulinism; Hypertrophy, Left Ventricular; Imidazoles; Insulin; Male; Myocardium; Olmesartan Medoxomil; Organ Size; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Renin-Angiotensin System; Sympathetic Nervous System; Tetrazoles | 2002 |
Purinergic modulation of vascular sympathetic neurotransmission.
Topics: Adenosine Triphosphate; Animals; Arteries; Electrophysiology; Norepinephrine; Purines; Quinazolines; Rats; Receptors, Purinergic; Synaptic Transmission; Tail; Vasomotor System | 2002 |
Different effects of carvedilol, metoprolol, and propranolol on left ventricular remodeling after coronary stenosis or after permanent coronary occlusion in rats.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Carbazoles; Cardiac Catheterization; Carvedilol; Coronary Disease; Coronary Stenosis; Disease Models, Animal; Dose-Response Relationship, Drug; Echocardiography; Hemodynamics; Male; Metoprolol; Norepinephrine; Propanolamines; Propranolol; Quinazolines; Rats; Rats, Sprague-Dawley; Severity of Illness Index; Stroke Volume; Survival Rate; Thiobarbituric Acid Reactive Substances; Ventricular Function, Left; Ventricular Remodeling | 2002 |
The alpha(1D)-adrenergic receptor directly regulates arterial blood pressure via vasoconstriction.
Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Aorta; Arteries; Blood Pressure; Cardiovascular System; Female; Gene Targeting; In Vitro Techniques; Male; Mice; Mice, Knockout; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Piperazines; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Serotonin; Tissue Extracts; Vasoconstriction; Vasoconstrictor Agents; Vasopressins | 2002 |
Neuroprotective effects of nipradilol on purified cultured retinal ganglion cells.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antihypertensive Agents; Cell Separation; Cell Survival; Cells, Cultured; Culture Media, Serum-Free; Cyclic N-Oxides; Dose-Response Relationship, Drug; Flow Cytometry; Imidazoles; Neuroprotective Agents; Nitric Oxide; Propanolamines; Quinazolines; Rats; Rats, Sprague-Dawley; Retinal Ganglion Cells; Timolol | 2002 |
Amelioration by topical bunazosin hydrochloride of the impairment in ocular blood flow caused by nitric oxide synthase inhibition in rabbits.
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Evoked Potentials, Visual; Fundus Oculi; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Optic Disk; Quinazolines; Rabbits; Reaction Time; Regional Blood Flow; Vision, Ocular | 2003 |
[Effects of ocular hypotensive agents on the circadian rhythm in intraocular pressure in rabbits as measured by telemetry].
Topics: Animals; Circadian Rhythm; Intraocular Pressure; Male; Quinazolines; Rabbits; Sulfonamides; Telemetry; Thiophenes; Timolol | 2003 |
Bunazosin hydrochloride reduces glutamate-induced neurotoxicity in rat primary retinal cultures.
Topics: Animals; Brain; Cell Death; Cells, Cultured; Dose-Response Relationship, Drug; Female; Glutamic Acid; Pregnancy; Protein Binding; Quinazolines; Rats; Rats, Wistar; Retina | 2004 |
Ocular pharmacokinetic/ pharmacodynamic modeling for bunazosin after instillation into rabbits.
Topics: Adrenergic alpha-Antagonists; Algorithms; Animals; Aqueous Humor; Eye; Injections; Intraocular Pressure; Male; Models, Biological; Quinazolines; Rabbits; Tears | 2004 |
Effects of bunazosin hydrochloride on ciliary muscle constriction and matrix metalloproteinase activities.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aqueous Humor; Cattle; Cells, Cultured; Ciliary Body; Drug Combinations; Intraocular Pressure; Isometric Contraction; Latanoprost; Macaca fascicularis; Male; Matrix Metalloproteinases; Muscle Relaxation; Muscle, Smooth; Phenylephrine; Prostaglandins F, Synthetic; Quinazolines; Trabecular Meshwork | 2004 |
Effects of topically instilled bunazosin, an alpha1-adrenoceptor antagonist, on constrictions induced by phenylephrine and ET-1 in rabbit retinal arteries.
Topics: Administration, Topical; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Combinations; Endothelin-1; Ganglionectomy; Injections; Male; Phenylephrine; Quinazolines; Rabbits; Receptors, Endothelin; Retinal Artery; Superior Cervical Ganglion; Vasoconstriction; Vasoconstrictor Agents; Vitreous Body | 2004 |
Alpha1-receptor or adenosine A1-receptor dependent pathway alone is not sufficient but summation of these pathways is required to achieve an ischaemic preconditioning effect in rabbits.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Enzyme Inhibitors; Heart Rate; Ischemic Preconditioning, Myocardial; Male; Myocardial Infarction; Protein Kinase C; Quinazolines; Rabbits; Receptor, Adenosine A1; Receptors, Adrenergic, alpha-1; Staurosporine; Theophylline; Tyramine; Vasodilator Agents | 2005 |
Amelioration of endothelin-1-induced optic nerve head ischemia by topical bunazosin.
Topics: Administration, Topical; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Endothelin-1; Evoked Potentials, Visual; Injections; Intraocular Pressure; Ischemia; Optic Disk; Quinazolines; Rabbits; Regional Blood Flow; Retina; Vitreous Body | 2005 |
Alterations of alpha-adrenergic modulations of coronary microvascular tone in dogs with heart failure.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Flow Velocity; Cineangiography; Coronary Angiography; Coronary Circulation; Coronary Vessels; Disease Models, Animal; Dogs; Enzyme Inhibitors; Female; Heart Failure; Injections, Intra-Arterial; Male; Microcirculation; NG-Nitroarginine Methyl Ester; Propranolol; Quinazolines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vascular Resistance; Vasodilation; Yohimbine | 2005 |
Effects of different alpha-1 adrenoceptor blockers on proximal urethral function using in vivo isovolumetric pressure changes.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Male; Phenylephrine; Prazosin; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urethra | 2005 |
Incidence of intraoperative floppy iris syndrome in patients on either systemic or topical alpha(1)-adrenoceptor antagonist.
Topics: Administration, Topical; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Cataract Extraction; Female; Humans; Incidence; Intraoperative Complications; Iris Diseases; Male; Naphthalenes; Piperazines; Prospective Studies; Prostatic Hyperplasia; Pupil; Quinazolines; Sulfonamides; Syndrome; Tamsulosin | 2007 |
[Case of pigmentary glaucoma treated with medical therapy, laser treatment, and trabeculotomy].
Topics: Adrenergic alpha-Antagonists; Adult; Antihypertensive Agents; Argon; Glaucoma, Open-Angle; Humans; Intraocular Pressure; Iris; Laser Therapy; Male; Ophthalmic Solutions; Quinazolines; Sulfonamides; Thiophenes; Trabeculectomy; Treatment Outcome | 2007 |
Effects of adrenergic and cholinergic antagonists on diameter of nasolacrimal drainage system.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Female; Humans; Infusions, Parenteral; Male; Middle Aged; Muscarinic Antagonists; Nasolacrimal Duct; Quinazolines; Radiography; Sympathetic Nervous System; Tropicamide | 2007 |
Protective effects of carvedilol in murine model with the coxsackievirus B3-induced viral myocarditis.
Topics: Acute Disease; Adrenergic beta-Antagonists; Animals; Anti-Inflammatory Agents; Antioxidants; Carbazoles; Cardiotonic Agents; Carvedilol; Coxsackievirus Infections; Disease Models, Animal; Enterovirus B, Human; Interleukins; Male; Malondialdehyde; Metoprolol; Mice; Mice, Inbred BALB C; Myocarditis; Propanolamines; Quinazolines; Superoxide Dismutase; Up-Regulation | 2008 |
Comparison of the cardiac electrophysiological effects between doxazosin and bunazosin.
Topics: Animals; Arrhythmias, Cardiac; Cardiac Electrophysiology; Doxazosin; Drug-Related Side Effects and Adverse Reactions; Heart; In Vitro Techniques; Ion Channels; Quinazolines; Rats | 2008 |
Possible mechanism of intraoperative floppy iris syndrome: a clinicopathological study.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Antihypertensive Agents; Female; Glaucoma; Humans; Iris Diseases; Male; Quinazolines; Syndrome | 2008 |
Ocular pharmacokinetic/pharmacodynamic modeling for multiple anti-glaucoma drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Algorithms; Animals; Aqueous Humor; Drug Combinations; Glaucoma; Intraocular Pressure; Male; Models, Statistical; Ocular Hypertension; Ophthalmic Solutions; Quinazolines; Rabbits; Telemetry; Timolol | 2008 |
[The use of andante in the therapy of insomnia].
Topics: Adrenergic alpha-Antagonists; Adult; Dose-Response Relationship, Drug; Female; Follow-Up Studies; Humans; Male; Middle Aged; Polysomnography; Quinazolines; Sleep; Sleep Initiation and Maintenance Disorders; Surveys and Questionnaires; Treatment Outcome | 2009 |