bunazosin and prazosin

bunazosin has been researched along with prazosin in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19909 (31.03)18.7374
1990's16 (55.17)18.2507
2000's3 (10.34)29.6817
2010's0 (0.00)24.3611
2020's1 (3.45)2.80

Authors

AuthorsStudies
Pedretti, A; Testa, B; Villa, L; Vistoli, G1
Lombardo, F; Obach, RS; Waters, NJ1
Bansal, R; Malhotra, A1
Kondo, S; Morita, T1
Hayashi, Y; Ikeda, K; Ohnishi, H; Watanabe, K2
Baba, S; Kinami, J; Mano, F; Maruyama, K; Nagatomo, T; Tsuchihashi, H1
Kinami, J; Maruyama, K; Nagatomo, T; Tsuchihashi, H1
Kato, Y; Kawabe, K; Kimura, R; Maruyama, M; Matsuoka, Y; Suzuki, M; Yamada, S1
Kobayashi, S1
Akimoto, Y; Fujiwara, M; Kurahashi, K; Sono, K1
Nagatomo, T; Tsuchihashi, H1
Kanaide, H; Miwa-Nishimura, N; Nakamura, M; Nishimura, J1
Akima, M; Imagawa, J; Sakai, K1
Mikami, H; Ogihara, T1
Fujioka, M; Ibengwe, JK; Ishikawa, S; Komori, K; Nagao, T; Suzuki, H1
Shoji, T1
Fujimoto, S; Kida, O; Morotomi, Y; Tanaka, K1
Ludvig, N; Vizi, ES1
Anderton, JL; Gill, M; Notghi, A1
Kono, M; Morita, S; Rubsamen, R1
Asano, M; Inagaki, O; Sudoh, K; Takenaka, T; Tanaka, H1
Rieckert, H1
Hirawa, N; Numabe, A; Takada, S; Uehara, Y; Yagi, S1
Inagaki, O; Sudoh, K; Takenaka, T1
Ishii, M; Umemura, S; Yasuda, G1
Suzuki, H1
Endo, T; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Satoh, Y; Suzuguchi, T1
Nagano, M; Osada, Y; Yamaguchi, T1

Reviews

2 review(s) available for bunazosin and prazosin

ArticleYear
Therapeutic progression of quinazolines as targeted chemotherapeutic agents.
    European journal of medicinal chemistry, 2021, Feb-05, Volume: 211

    Topics: Animals; Antineoplastic Agents; Cell Proliferation; Enzyme Inhibitors; Humans; Molecular Structure; Neoplasms; Quinazolines

2021
Treatment of benign prostatic hyperplasia and hypertension in elderly hypertensive patients.
    British journal of urology, 1998, Volume: 81 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Aged; Female; Humans; Hypertension; Male; Multicenter Studies as Topic; Prazosin; Product Surveillance, Postmarketing; Prostatic Hyperplasia; Quinazolines; Randomized Controlled Trials as Topic

1998

Trials

3 trial(s) available for bunazosin and prazosin

ArticleYear
Renal haemodynamic effects of bunazosin retard and prazosin in mild to moderately hypertensive patients with normal or moderately impaired renal function.
    Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association, 1994, Volume: 9, Issue:6

    Topics: Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Blood Pressure; Female; Glomerular Filtration Rate; Humans; Hypertension; Male; Middle Aged; Prazosin; Quinazolines; Renal Insufficiency; Renal Plasma Flow, Effective

1994
Orthostatic hypotension: how to avoid it during antihypertensive therapy.
    American journal of hypertension, 1996, Volume: 9, Issue:11

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Antihypertensive Agents; Blood Pressure; Double-Blind Method; Humans; Hypertension; Hypotension, Orthostatic; Middle Aged; Plethysmography; Posture; Prazosin; Quinazolines; Regional Blood Flow; Vascular Resistance

1996
Characterization of bunazosin-sensitive alpha1-adrenoceptors in human renal medulla.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Double-Blind Method; Female; Humans; In Vitro Techniques; Kidney Function Tests; Kidney Medulla; Male; Middle Aged; Prazosin; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha-1

1997

Other Studies

24 other study(ies) available for bunazosin and prazosin

ArticleYear
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
[Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1992, Volume: 83, Issue:3

    Topics: Adenoma; Adrenergic alpha-Antagonists; Aged; Humans; Male; Piperazines; Prazosin; Prostatic Hyperplasia; Prostatic Neoplasms; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha

1992
[Effect of moxisylyte on the lower urinary tracts (1). Effect on the isolated rabbit urethra and bladder].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Moxisylyte; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Prazosin; Quinazolines; Rabbits; Urethra; Urinary Bladder

1991
[Effect of moxisylyte on the lower urinary tracts (2). Effect on the urethra in anesthetized dogs].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Moxisylyte; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phenylephrine; Prazosin; Quinazolines; Urethra; Yohimbine

1991
Comparison of alpha 1-adrenoceptors between rat brain and spleen.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Dibenzylchlorethamine; Kinetics; Male; Phenoxybenzamine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Spleen

1991
Binding characteristics of alpha 1-adrenoceptors in bovine prostate using a radioligand binding assay.
    Journal of pharmacobio-dynamics, 1991, Volume: 14, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Cattle; Kinetics; Male; Membranes; Phentolamine; Prazosin; Prostate; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium

1991
[3H]bunazosin, a novel selective radioligand of alpha 1 adrenoceptors in human prostates.
    The Journal of urology, 1991, Volume: 146, Issue:3

    Topics: Adrenergic alpha-Antagonists; Cell Membrane; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Tritium

1991
[Characterization and localization of alpha 1-adrenoceptors in human prostate--with special reference to the zonal difference in receptor distribution].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1991, Volume: 82, Issue:8

    Topics: Autoradiography; Binding Sites; Humans; Male; Prazosin; Prostate; Prostatic Hyperplasia; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha; Urinary Bladder Neoplasms

1991
Effects of specific alpha-adrenoceptive agents on extraneuronal uptake (uptake2) of isoproterenol in perfused rat heart.
    Life sciences, 1989, Volume: 44, Issue:14

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Guanabenz; Isoproterenol; Male; Methoxamine; Myocardium; Neurons; Phenylephrine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Sulfonamides; Tropolone

1989
Alpha-blocking potencies of antihypertensive agents (prazosin, terazosin, bunazosin, SGB-1534 and ketanserin) having with quinazoline or quinazolinedione as assessed by radioligand binding assay methods in rat brain.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brain; Cell Membrane; Clonidine; Dihydroalprenolol; Ketanserin; Male; Prazosin; Quinazolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1989
Selective blockade of alpha 1-adrenoceptors of porcine vascular smooth muscle cells by bunazosin.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; In Vitro Techniques; Membranes; Microsomes; Muscle, Smooth, Vascular; Muscles; Prazosin; Quinazolines; Swine; Yohimbine

1989
In vivo experiments for the evaluation of alpha 1-adrenoceptor antagonistic effects of SGB-1534 on canine urethra.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Dose-Response Relationship, Drug; Female; Hypogastric Plexus; Phenylephrine; Prazosin; Quinazolines; Urethra

1989
[Clinical application of adrenoceptor blockers in the treatment of hypertension].
    Nihon rinsho. Japanese journal of clinical medicine, 1989, Volume: 47, Issue:9

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Carbazoles; Carvedilol; Humans; Hypertension; Labetalol; Prazosin; Propanolamines; Quinazolines

1989
Effects of bunazosin on electrical responses of smooth muscle cells of the guinea-pig mesenteric artery and vein to perivascular nerve stimulation and to noradrenaline.
    General pharmacology, 1987, Volume: 18, Issue:2

    Topics: Animals; Electric Stimulation; Evoked Potentials; Female; Guinea Pigs; Male; Membrane Potentials; Mesenteric Arteries; Mesenteric Veins; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Yohimbine

1987
Comparison of pre- and postsynaptic alpha-adrenoceptor blocking effects of E-643 in the isolated vas deferens of the rat.
    Japanese journal of pharmacology, 1981, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens

1981
[Effects of quinazoline derivatives (E-643 and prazosin) on blood pressure, pulse and renin-angiotensin system in two cases of pheochromocytoma (author's transl)].
    Nihon Jinzo Gakkai shi, 1981, Volume: 23, Issue:8

    Topics: Adolescent; Adrenal Gland Neoplasms; Adrenergic alpha-Antagonists; Adult; Blood Pressure; Humans; Male; Pheochromocytoma; Prazosin; Pulse; Quinazolines; Renin-Angiotensin System

1981
(-)-Amidephrine, a selective agonist for alpha 1-adrenoceptors.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Electric Stimulation; Ethanolamines; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Quinazolines; Rats; Vas Deferens

1983
Effects of alpha-adrenergic blockade on regional myocardial function in canine ischemic myocardium during beta-adrenergic blockade.
    Journal of cardiothoracic and vascular anesthesia, 1995, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Coronary Circulation; Dogs; Female; Hemodynamics; Male; Myocardial Contraction; Myocardial Ischemia; Myocardium; Prazosin; Propranolol; Prospective Studies; Quinazolines; Random Allocation; Yohimbine

1995
Effect of tamsulosin, a novel alpha 1-adrenoceptor antagonist, on urethral pressure profile in anaesthetized dogs.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Captopril; Dogs; Dose-Response Relationship, Drug; Male; Nicardipine; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin

1996
Thromboxane inhibition potentiates antihypertensive effects of alpha 1 adrenoceptor antagonists in the rat.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aorta; Blood Pressure; Body Weight; Cells, Cultured; Drug Synergism; Eicosanoids; Ethanolamines; Kidney; Methacrylates; Muscle, Smooth, Vascular; Prazosin; Quinazolines; Rats; Rats, Inbred SHR; Sodium; Thromboxane-A Synthase; Thromboxanes

1997
Effect of alpha 1-adrenoceptor antagonists on urinary bladder function in urethane-anesthetized rats.
    General pharmacology, 1997, Volume: 28, Issue:4

    Topics: Adrenergic alpha-Antagonists; Anesthetics; Animals; Flavoxate; Male; Parasympatholytics; Prazosin; Quinazolines; Rats; Rats, Wistar; Sulfonamides; Tamsulosin; Urethane; Urinary Bladder

1997
[Signal transduction of serotonin release from enterochromaffin cells in mouse ileal crypts].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1998, Volume: 112 Suppl 1

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Clonidine; Enterochromaffin Cells; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Norepinephrine; Phosphodiesterase Inhibitors; Prazosin; Pyrrolidinones; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Rolipram; Serotonin; Signal Transduction; Yohimbine

1998
Effects of different alpha-1 adrenoceptor blockers on proximal urethral function using in vivo isovolumetric pressure changes.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2005, Volume: 41, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Male; Phenylephrine; Prazosin; Quinazolines; Rabbits; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urethra

2005