bucladesine has been researched along with rolipram in 65 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 11 (16.92) | 18.7374 |
1990's | 26 (40.00) | 18.2507 |
2000's | 22 (33.85) | 29.6817 |
2010's | 6 (9.23) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Ainz, LF; Carou, M; Gáldiz, B; Gandarias, JM; Gil-Rodrigo, CE; Gómez, R; Vallejo, A | 1 |
Correa-Sales, C; Maze, M; Nacif-Coelho, C; Reid, K | 1 |
Conti, M; Swinnen, JV; Tsikalas, KE | 1 |
Rapoport, RM | 1 |
Mulder, AH; Schoffelmeer, AN; Wierenga, EA | 1 |
Donaldson, J; Hall, IP; Hill, SJ | 1 |
Lohse, MJ; Puurunen, J; Schwabe, U | 1 |
Bhalla, VK; Guo, YS; Singh, P; Thompson, JC | 1 |
Hara, K; Ikoma, Y; Kimura, K; Mizokawa, T; Oshino, N; Ueki, S; Yamamoto, T | 1 |
Meisburger, JG; Ortmann, R | 1 |
Astrachan, DI; Astrachan, E; Davis, M; Kehne, JH; Tallman, JF | 1 |
Löschmann, PA; Wachtel, H | 1 |
Wachtel, H | 1 |
Fredholm, BB; Jondal, M; Lanefelt, F; Ullberg, M | 1 |
Mulder, AH; Schoffelmeer, AN; Wemer, J | 1 |
Hamacher, L; Jin, SL; Lenhard, JM; McConnell, RT; Verghese, MW | 1 |
Dent, G; Liebig, S; Magnussen, H; Rabe, KF; Schudt, C; Tenor, H | 1 |
Barnette, MS; Burman, M; Christensen, SB; Cieslinski, LB; Grous, M; Torphy, TJ | 1 |
Furdon, PJ; Gooding, RC; McConnell, RT; Stimpson, SA; Strickland, AB; Taylor, JD; Verghese, MW; Yarnall, DP | 1 |
Brett, J; Karakurum, M; Liao, H; Morris, S; Nowygrod, R; Oz, M; Pinsky, D; Platt, J; Sciacca, R; Van Lookeren Campagne, M | 1 |
Ormandy, GC | 1 |
Alves, AC; Cordeiro, RS; Cruz, HN; Diaz, BL; Lagente, V; Martins, MA; Pires, AL; Serra, MF | 1 |
Ichimaru, Y; Imanishi, T; Kato, S; Miyashiro, M; Sawa, A; Ueki, S; Yamamoto, T | 1 |
Chini, CC; Chini, EN; Dousa, TP; Grande, JP | 1 |
Berends, C; de Monchy, JG; Dijkhuizen, B; Dubois, AE; Gerritsen, J; Kauffman, HF | 1 |
Agematsu, K; Hu, B; Komiyama, A; Nakazawa, T; Yasui, K | 1 |
Kobayashi, J; Kurita, C; Nagai, H; Nagao, T; Nakao, T; Tanaka, H; Usami, E; Watanabe, S; Yamazaki, F; Yoshimura, T | 1 |
Inagaki, N; Kobayashi, J; Nagai, H; Nagao, T; Nakao, T; Tanaka, H; Usami, E; Watanabe, S; Yamazaki, F; Yoshimura, T | 1 |
Anderson, R; Feldman, C; Goolam Mahomed, A; Ramafi, G; Theron, AJ | 1 |
Capasso, F; Izzo, AA; Mascolo, N | 1 |
Benjamin, AR; Stephens, RH; Walters, DV | 1 |
Kim, DH; Lerner, A | 1 |
Bertin, B; Boichot, E; Germain, N; Lagente, V; Legendre, A; Martin, B; Payne, A | 1 |
Boichot, E; Escofier, N; Germain, N; Lagente, V; Martins, MA; Silva, PM | 1 |
Beleta, J; Giménez-Arnau, AM; Giménez-Camarasa, JM; Palacios, JM; Ryder, H; Santamaria, LF; Torres, R | 1 |
Dinter, H; Martin, R; McFarland, HF; Muraro, PA; Pette, DF; Pette, M | 1 |
Kitamura, K; Matsumoto, M; Oka, K; Oku, A; Sugiura, M; Taguchi, I | 1 |
Dent, G; Djukanović, R; Hidi, R; Holgate, ST; Liu, E; Schudt, C; Timmermans, S | 1 |
Jankovic, V; Maksimovic, D; Samardzic, T; Stosic-Grujicic, S; Trajkovic, V | 1 |
Bodstein, M; Gaspar Elsas, MI; Joseph, D; Lintomen, L; Maximiano, ES; Vargaftig, BB; Xavier Elsas, P | 1 |
Campos-Toimil, M; Droy-Lefaix, MT; Lugnier, C; Takeda, K | 1 |
Anderson, R; Cole, PJ; Feldman, C; Ramafi, G; Taylor, GW; Theron, AJ; Wilson, R | 1 |
Beshay, E; Croze, F; Prud'homme, GJ | 1 |
Botana, LM; de la Rosa, LA; Vieytes, MR; Vilariño, N | 1 |
Belleguic, C; Boichot, E; Corbel, M; Germain, N; Lagente, V | 1 |
Anderson, R; Steel, HC | 1 |
Bobalova, J; Mutafova-Yambolieva, VN; Smyth, L | 1 |
Ahmed, S; Brennan, FM; Feldmann, M; Field, S; Foey, AD; Jain, A; Williams, R | 1 |
Barreto, EO; Carvalho, VF; Cordeiro, RS; E Silva, PM; Lagente, V; Lugnier, C; Martins, MA | 1 |
Bates, ML; Berrocal, YA; Bunge, MB; Filbin, MT; Marcillo, AE; Pearse, DD; Pereira, FC | 1 |
Kelly, J; Strada, SJ; Thompson, WJ; Vemavarapu, L; Zhu, B | 1 |
Allen, JM; Bertrand, C; Jacob, C; Lagente, V; Szilagyi, C | 1 |
Kyoi, T; Noda, K; Oka, M; Ukai, Y | 1 |
Bengtsson, T; Evans, BA; Nevzorova, J; Summers, RJ | 1 |
Bergamaschi, A; Corsi, M; Garnier, MJ | 1 |
Bobalova, J; Mutafova-Yambolieva, VN | 1 |
Bolton, S; Butt, AM | 1 |
Campos-Toimil, M; Keravis, T; Lugnier, C; Orallo, F; Takeda, K | 1 |
Chamoto, K; Fukuda, Y; Goto, M; Hayashi, Y; Inoue, H; Kadoshima-Yamaoka, K; Miura, K; Murafuji, H; Murakawa, M; Nagahira, K; Nakatsuka, T; Nishimura, T; Tanaka, Y | 1 |
Abe, K; Fujita, M; Hong, J; Innis, RB; Inoue, O; Itoh, T; Pike, VW | 1 |
Avni, D; Meijler, MM; Philosoph, A; Zor, T | 1 |
Flanagan, LA; Sharp, KG; Steward, O; Yee, KM | 1 |
Butchbach, ME; Cook, DJ; Dhurjati, P; Mack, SG | 1 |
Harada, T; Inoue, A; Matsuoka, K; Ochiai, H; Ohnishi, M; Ohsugi, Y; Takeo, S; Urasaki, T | 1 |
65 other study(ies) available for bucladesine and rolipram
Article | Year |
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Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
[Specific inhibition by ATP of histamine-stimulated acid secretion in the gastric glands of the rabbit].
Topics: Adenosine Triphosphate; Animals; Bucladesine; Carbachol; Depression, Chemical; Female; Gastric Acid; Gastric Mucosa; Histamine; Histamine Antagonists; Indomethacin; Male; Prostaglandins; Pyrrolidinones; Rabbits; Rolipram; Secretory Rate; Theophylline | 1992 |
Inhibition of adenylate cyclase in the locus coeruleus mediates the hypnotic response to an alpha 2 agonist in the rat.
Topics: Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Animals; Bucladesine; Hypnotics and Sedatives; Imidazoles; Locus Coeruleus; Male; Medetomidine; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram | 1992 |
Properties and hormonal regulation of two structurally related cAMP phosphodiesterases from the rat Sertoli cell.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Amino Acid Sequence; Animals; Blotting, Northern; Blotting, Western; Bucladesine; DNA; Follicle Stimulating Hormone; Hormones; Male; Molecular Sequence Data; Nucleic Acid Hybridization; Precipitin Tests; Pyrrolidinones; Rats; Recombinant Proteins; RNA, Messenger; Rolipram; Sequence Homology, Nucleic Acid; Sertoli Cells; Transcription, Genetic | 1991 |
Inhibitory effects of cyclic AMP-elevating agents on norepinephrine-induced phosphatidylinositide hydrolysis and contraction in rat aorta.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Aorta, Thoracic; Arachidonic Acid; Arachidonic Acids; Bucladesine; Cyclic AMP; Hydrolysis; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phosphatidylglycerols; Phosphatidylinositols; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Inbred Strains; Rolipram | 1991 |
Role of adenylate cyclase in presynaptic alpha 2-adrenoceptor- and mu-opioid receptor-mediated inhibition of [3H]noradrenaline release from rat brain cortex slices.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Bucladesine; Cadmium; Calcimycin; Cerebral Cortex; Clonidine; Colforsin; Cyclic AMP; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Morphine; Norepinephrine; Phentolamine; Pyrrolidinones; Rats; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu; Rolipram | 1986 |
Inhibition of histamine-stimulated inositol phospholipid hydrolysis by agents which increase cyclic AMP levels in bovine tracheal smooth muscle.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Albuterol; Animals; Bucladesine; Cattle; Colforsin; Cyclic AMP; Histamine; Histamine Antagonists; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Muscle, Smooth; Phosphodiesterase Inhibitors; Pyrrolidinones; Rolipram; Sugar Phosphates; Trachea; Vasoactive Intestinal Peptide | 1989 |
Interactions between intracellular cyclic AMP and agonist-induced inositol phospholipid breakdown in isolated gastric mucosal cells of the rat.
Topics: Animals; Bucladesine; Carbachol; Cimetidine; Colforsin; Cyclic AMP; Dibutyryl Cyclic GMP; Enzyme Activation; Histamine; In Vitro Techniques; Inositol Phosphates; Male; Parietal Cells, Gastric; Phorbol Esters; Phosphodiesterase Inhibitors; Protein Kinase C; Pyrrolidinones; Rats; Rats, Inbred Strains; Rolipram; Sugar Phosphates | 1987 |
Effect of cyclic nucleotides on bombesin-evoked gastrin release from isolated perfused rat stomach.
Topics: Animals; Bombesin; Bucladesine; Carrier Proteins; Cyclic AMP; Cyclic GMP; Dibutyryl Cyclic GMP; Gastric Mucosa; Gastrins; Intracellular Signaling Peptides and Proteins; Male; Nucleotides, Cyclic; Perfusion; Protein Kinase Inhibitors; Pyrrolidinones; Rats; Rolipram | 1988 |
The effect of a selective phosphodiesterase inhibitor, rolipram, on muricide in olfactory bulbectomized rats.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Bucladesine; Male; Mice; Neurotransmitter Agents; Olfactory Bulb; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Inbred Strains; Rolipram | 1988 |
Rolipram forms a potent discriminative stimulus in drug discrimination experiments in rats.
Topics: Animals; Behavior, Animal; Brain; Bucladesine; Conditioning, Operant; Cues; Dibutyryl Cyclic GMP; Discrimination Learning; Generalization, Psychological; Pyrrolidinones; Rats; Rolipram | 1986 |
The role of spinal cord cyclic AMP in the acoustic startle response in rats.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bucladesine; Colforsin; Injections, Spinal; Pyrrolidinones; Rats; Rats, Inbred Strains; Reflex, Startle; Rolipram | 1986 |
Effects of forskolin and cyclic nucleotides in animal models predictive of antidepressant activity: interactions with rolipram.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; alpha-Methyltyrosine; Animals; Antidepressive Agents; Body Temperature; Bucladesine; Colforsin; Dibutyryl Cyclic GMP; Fenclonine; Male; Methyltyrosines; Mice; Motor Activity; Nucleotides, Cyclic; Pyrrolidinones; Reserpine; Rolipram | 1986 |
Characteristic behavioural alterations in rats induced by rolipram and other selective adenosine cyclic 3', 5'-monophosphate phosphodiesterase inhibitors.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Behavior, Animal; Body Temperature; Bucladesine; Imidazoles; Male; Motor Activity; Pyrimidines; Pyrrolidinones; Rats; Rats, Inbred Strains; Rolipram | 1982 |
Inhibition of human NK cell cytotoxicity by induction of cyclic AMP depends on impaired target cell recognition.
Topics: Alprostadil; Bucladesine; Cyclic AMP; Cytotoxicity, Immunologic; Humans; Interferons; Killer Cells, Natural; Lymphocytes; Prostaglandins E; Pyrrolidinones; Rolipram | 1983 |
Effects of cyclic AMP analogues and phosphodiesterase inhibitors on K+-induced [3H]noradrenaline release from rat brain slices and on its presynaptic alpha-adrenergic modulation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bucladesine; Cerebral Cortex; Cyclic AMP; Male; Norepinephrine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Potassium; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Rolipram; Sodium Fluoride; Synapses | 1982 |
Regulation of distinct cyclic AMP-specific phosphodiesterase (phosphodiesterase type 4) isozymes in human monocytic cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Base Sequence; Bucladesine; Cells, Cultured; Cytosol; Gene Expression Regulation, Enzymologic; Humans; Isoenzymes; Kinetics; Lipopolysaccharides; Molecular Sequence Data; Monocytes; Oligodeoxyribonucleotides; Pyrrolidinones; RNA, Messenger; Rolipram | 1995 |
Phosphodiesterase isozymes modulating inherent tone in human airways: identification and characterization.
Topics: 1-Methyl-3-isobutylxanthine; 2',3'-Cyclic-Nucleotide Phosphodiesterases; Adult; Aged; Bucladesine; Colforsin; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Female; Forced Expiratory Volume; Humans; In Vitro Techniques; Isoenzymes; Lung; Lung Neoplasms; Male; Middle Aged; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Nitroprusside; Purinones; Pyrazines; Pyridazines; Pyrrolidinones; Rolipram; Vital Capacity | 1993 |
Inhibitors of phosphodiesterase IV (PDE IV) increase acid secretion in rabbit isolated gastric glands: correlation between function and interaction with a high-affinity rolipram binding site.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Aminopyrine; Animals; Binding Sites; Bucladesine; Cyclic Nucleotide Phosphodiesterases, Type 4; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; Rabbits; Rolipram | 1995 |
Differential regulation of human monocyte-derived TNF alpha and IL-1 beta by type IV cAMP-phosphodiesterase (cAMP-PDE) inhibitors.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Alprostadil; Base Sequence; Bucladesine; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; DNA Primers; Gene Expression; Humans; In Vitro Techniques; Indomethacin; Interleukin-1; Molecular Sequence Data; Monocytes; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; RNA, Messenger; Rolipram; Tumor Necrosis Factor-alpha | 1995 |
Restoration of the cAMP second messenger pathway enhances cardiac preservation for transplantation in a heterotopic rat model.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenylyl Cyclases; Animals; Bucladesine; Cattle; Cell Hypoxia; Cyclic AMP; Heart Transplantation; Indoles; Male; Muscle, Smooth, Vascular; Myocardium; Neutrophils; Organ Preservation; Oxindoles; Perfusion; Peroxidase; Pyridazines; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram; Second Messenger Systems; Thionucleotides; Transplantation, Heterotopic; Transplantation, Homologous | 1993 |
Increased cyclic AMP reduces 5-HT1D receptor-mediated inhibition of [3H]5-hydroxytryptamine release from guinea-pig cortical slices.
Topics: Animals; Bucladesine; Cerebral Cortex; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Indoles; Phosphodiesterase Inhibitors; Potassium; Pyrrolidinones; Receptors, Serotonin; Rolipram; Serotonin; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan | 1993 |
Selective inhibition of phosphodiesterase type IV suppresses the chemotactic responsiveness of rat eosinophils in vitro.
Topics: Adrenergic beta-Agonists; Animals; Bucladesine; Chemotaxis, Leukocyte; Colforsin; Cyclic AMP; Eosinophils; Isoenzymes; Leukotriene B4; Phosphodiesterase Inhibitors; Platelet Activating Factor; Platelet Aggregation; Pyrrolidinones; Rats; Rats, Wistar; Rolipram | 1996 |
Ameliorating effects of rolipram on experimentally induced impairments of learning and memory in rodents.
Topics: Animals; Avoidance Learning; Brain Ischemia; Bucladesine; Cyclic AMP; Electroshock; Learning; Male; Memory; Mice; Motor Activity; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Wistar; Rolipram; Scopolamine | 1997 |
Compartmentalization of cAMP signaling in mesangial cells by phosphodiesterase isozymes PDE3 and PDE4. Regulation of superoxidation and mitogenesis.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Bucladesine; Cell Compartmentation; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Glomerular Mesangium; Kinetics; Mitosis; NADPH Oxidases; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; Quinolones; Rats; Rolipram; Signal Transduction; Superoxides; Xanthines | 1997 |
Inhibition of PAF-induced expression of CD11b and shedding of L-selectin on human neutrophils and eosinophils by the type IV selective PDE inhibitor, rolipram.
Topics: Bucladesine; CD11 Antigens; Dinoprostone; Eosinophils; Flow Cytometry; Humans; Isoproterenol; L-Selectin; Neutrophils; Phosphodiesterase Inhibitors; Platelet Activating Factor; Pyrrolidinones; Rolipram | 1997 |
Theophylline accelerates human granulocyte apoptosis not via phosphodiesterase inhibition.
Topics: 1-Methyl-3-isobutylxanthine; Anti-Inflammatory Agents, Non-Steroidal; Apoptosis; Bucladesine; Cell Survival; Cyclic AMP; Dose-Response Relationship, Drug; fas Receptor; Granulocyte-Macrophage Colony-Stimulating Factor; Granulocytes; Humans; Interleukin-5; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Proto-Oncogene Proteins c-bcl-2; Pyrrolidinones; Rolipram; Theophylline | 1997 |
Effects of cAMP-phosphodiesterase isozyme inhibitor on cytokine production by lipopolysaccharide-stimulated human peripheral blood mononuclear cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Aminophylline; Bucladesine; Cytokines; Humans; In Vitro Techniques; Interleukin-1; Interleukin-8; Isoenzymes; Leukocytes, Mononuclear; Lipopolysaccharides; Milrinone; Naphthyridines; Phosphodiesterase Inhibitors; Purinones; Pyridones; Pyrrolidinones; Rolipram; Terbutaline; Tumor Necrosis Factor-alpha | 1997 |
Modulation of Th1- and Th2-like cytokine production from mitogen-stimulated human peripheral blood mononuclear cells by phosphodiesterase inhibitors.
Topics: Adrenergic beta-Agonists; Bucladesine; Humans; In Vitro Techniques; Interferon-gamma; Interleukins; Leukocytes, Mononuclear; Milrinone; Mitogens; Phosphodiesterase Inhibitors; Pyridones; Pyrrolidinones; Rolipram; Th1 Cells; Th2 Cells; Theophylline | 1998 |
Effect of rolipram and dibutyryl cyclic AMP on resequestration of cytosolic calcium in FMLP-activated human neutrophils.
Topics: Adrenergic beta-Agonists; Adult; Albuterol; Bucladesine; Calcium; Calcium Radioisotopes; Cytosol; Fluorescent Dyes; Fura-2; Humans; In Vitro Techniques; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphodiesterase Inhibitors; Pyrrolidinones; Rolipram; Superoxides; Theophylline | 1998 |
Effect of selective phosphodiesterase inhibitors on synaptic transmission in the guinea-pig ileum.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bucladesine; Electric Stimulation; Enteric Nervous System; Guinea Pigs; Ileum; In Vitro Techniques; Male; Motor Neurons; Phosphodiesterase Inhibitors; Pyrrolidinones; Rolipram; Synaptic Transmission | 1998 |
The regulation of lung liquid absorption by endogenous cAMP in postnatal sheep lungs perfused in situ.
Topics: Absorption; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Bucladesine; Cyclic AMP; Lung; Osmotic Pressure; Perfusion; Phosphodiesterase Inhibitors; Purinergic Antagonists; Pyrrolidinones; Rolipram; Sheep; Sotalol; Theophylline | 1998 |
Type 4 cyclic adenosine monophosphate phosphodiesterase as a therapeutic target in chronic lymphocytic leukemia.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Antibodies, Anti-Idiotypic; Antigens, CD19; Antineoplastic Agents; Apoptosis; B-Lymphocytes; Bucladesine; Calcium; Calmodulin; Cells, Cultured; Colforsin; Cyclic AMP; DNA, Complementary; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Humans; Interleukin-2; Isoenzymes; Leukemia, Lymphocytic, Chronic, B-Cell; Leukocytes, Mononuclear; Phosphodiesterase Inhibitors; Polymerase Chain Reaction; Pyrrolidinones; RNA, Messenger; Rolipram; Tumor Cells, Cultured; Tumor Stem Cell Assay; Vinca Alkaloids | 1998 |
Selective phosphodiesterase inhibitors modulate the activity of alveolar macrophages from sensitized guinea-pigs.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Allergens; Animals; Arachidonic Acid; Bronchoalveolar Lavage Fluid; Bucladesine; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Isoenzymes; Macrophages, Alveolar; Male; Milrinone; Ovalbumin; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrrolidinones; Respiratory Hypersensitivity; Rolipram | 1998 |
Effects of interleukin-10 and modulators of cyclic AMP formation on endotoxin-induced inflammation in rat lung.
Topics: Administration, Inhalation; Adrenergic beta-Agonists; Albuterol; Animals; Bronchoalveolar Lavage Fluid; Bucladesine; Cell Count; Cyclic AMP; Dose-Response Relationship, Drug; Endotoxins; Free Radical Scavengers; Inflammation; Interleukin-10; Lipopolysaccharides; Luminescent Measurements; Luminol; Lung; Male; Neutrophils; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Wistar; Rolipram; Salmeterol Xinafoate; Superoxide Dismutase; Theophylline; Tumor Necrosis Factor-alpha; Zymosan | 1999 |
Rolipram inhibits staphylococcal enterotoxin B-mediated induction of the human skin-homing receptor on T lymphocytes.
Topics: Animals; Antigens, Differentiation, T-Lymphocyte; Antigens, Neoplasm; Bucladesine; CD3 Complex; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Enterotoxins; Flow Cytometry; Humans; Interleukin-12; Lymphocyte Activation; Membrane Glycoproteins; Mice; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Receptors, Lymphocyte Homing; Rolipram; Skin; T-Lymphocytes | 1999 |
Differential effects of phosphodiesterase type 4-specific inhibition on human autoreactive myelin-specific T cell clones.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Antibodies; Autoantigens; Bucladesine; Cell Division; Clone Cells; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Flow Cytometry; Humans; Interleukin-10; Interleukin-2; Lymphotoxin-alpha; Multiple Sclerosis; Myelin Proteins; Myelin Sheath; Oligonucleotide Probes; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptors, Interleukin-2; RNA, Messenger; Rolipram; T-Lymphocytes; Tumor Necrosis Factor-alpha | 1999 |
Protection by a cyclic AMP-specific phosphodiesterase inhibitor, rolipram, and dibutyryl cyclic AMP against Propionibacterium acnes and lipopolysaccharide-induced mouse hepatitis.
Topics: Animals; Bucladesine; Hepatitis, Animal; Lipopolysaccharides; Male; Mice; Mice, Inbred BALB C; Phosphodiesterase Inhibitors; Propionibacterium acnes; Pyrrolidinones; Rolipram; Tumor Necrosis Factor-alpha | 1999 |
Phosphodiesterase and cyclic adenosine monophosphate-dependent inhibition of T-lymphocyte chemotaxis.
Topics: Albuterol; Asthma; Bucladesine; Chemotaxis, Leukocyte; Colforsin; Cyclic AMP; Humans; Interleukin-8; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Platelet Activating Factor; Rolipram; T-Lymphocytes; Theophylline | 2000 |
Differential regulation of nitric oxide production by increase of intracellular cAMP in murine primary fibroblasts and L929 fibrosarcoma cell line.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bucladesine; Catalysis; Cells, Cultured; Cyclic AMP; Fibroblasts; Fibrosarcoma; Interferon-gamma; Intracellular Fluid; Mice; Mice, Inbred CBA; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Phosphodiesterase Inhibitors; Rolipram; Tumor Cells, Cultured | 2000 |
Murine myeloid progenitor responses to GM-CSF and eosinophil precursor responses to IL-5 represent distinct targets for downmodulation by prostaglandin E(2).
Topics: Animals; Bone Marrow Cells; Bucladesine; Cell Differentiation; Cells, Cultured; Colforsin; Colony-Forming Units Assay; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Eosinophils; Female; Granulocyte-Macrophage Colony-Stimulating Factor; Hematopoietic Stem Cells; Interleukin-5; Male; Mice; Mice, Inbred BALB C; Mice, Inbred CBA; Mice, Inbred Strains; Prostaglandin D2; Rolipram | 2000 |
Inhibition of type 4 phosphodiesterase by rolipram and Ginkgo biloba extract (EGb 761) decreases agonist-induced rises in internal calcium in human endothelial cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Antioxidants; Biological Transport; Bucladesine; Calcium; Cells, Cultured; Cyclic Nucleotide Phosphodiesterases, Type 4; Endothelium, Vascular; Flavonoids; Ginkgo biloba; Humans; Phosphodiesterase Inhibitors; Plant Extracts; Rolipram | 2000 |
CGS 21680, dibutyryl cyclic AMP and rolipram attenuate the pro-inflammatory interactions of the Pseudomonas aeruginosa -derived pigment, 1-hydroxyphenazine, with human neutrophils.
Topics: Adenosine; Antihypertensive Agents; Bucladesine; Calcium; Calcium Channels; Dose-Response Relationship, Drug; Homeostasis; Humans; Neutrophils; Phenazines; Phenethylamines; Phosphodiesterase Inhibitors; Pseudomonas aeruginosa; Rolipram | 2000 |
The phosphodiesterase inhibitors pentoxifylline and rolipram suppress macrophage activation and nitric oxide production in vitro and in vivo.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Autoimmune Diseases; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Diabetes Mellitus, Type 1; Dibutyryl Cyclic GMP; Disease Models, Animal; Drug Evaluation, Preclinical; Enterotoxins; Enzyme Induction; Female; Interferon-gamma; Interleukin-12; Lipopolysaccharides; Macrophage Activation; Macrophages, Peritoneal; Mice; Mice, Inbred NOD; Nitric Oxide; Nitric Oxide Synthase; Nitrites; Pentoxifylline; Phosphodiesterase Inhibitors; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Rolipram; Tumor Necrosis Factor-alpha | 2001 |
Modulation of thapsigargin-induced calcium mobilisation by cyclic AMP-elevating agents in human lymphocytes is insensitive to the action of the protein kinase A inhibitor H-89.
Topics: Adenosine Triphosphatases; Bucladesine; Calcium; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Humans; Isoquinolines; Lymphocytes; Microscopy, Fluorescence; Milrinone; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Rolipram; Sulfonamides; Thapsigargin; Time Factors | 2001 |
Effects of PDE4 inhibitors on lipopolysaccharide-induced priming of superoxide anion production from human mononuclear cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Benzamides; Bucladesine; Cells, Cultured; Cyclic Nucleotide Phosphodiesterases, Type 4; Humans; Interleukin-10; Leukocytes, Mononuclear; Lipopolysaccharides; N-Formylmethionine Leucyl-Phenylalanine; Phosphodiesterase Inhibitors; Pyridines; Rolipram; Superoxides; Time Factors | 2001 |
Dissociation of the PAF-receptor from NADPH oxidase and adenylate cyclase in human neutrophils results in accelerated influx and delayed clearance of cytosolic calcium.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Adenylyl Cyclases; Bucladesine; Calcium; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cytosol; Homeostasis; Humans; In Vitro Techniques; Leukocyte Elastase; Luminescent Measurements; Membrane Potentials; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophil Activation; Neutrophils; Phenethylamines; Phosphodiesterase Inhibitors; Platelet Activating Factor; Platelet Membrane Glycoproteins; Purinergic P1 Receptor Agonists; Radioimmunoassay; Receptor, Adenosine A2A; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Rolipram; Spectrometry, Fluorescence; Superoxides | 2002 |
Involvement of cyclic AMP-mediated pathway in neural release of noradrenaline in canine isolated mesenteric artery and vein.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Animals; Autonomic Nervous System; Bucladesine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dogs; Edetic Acid; Electric Stimulation; Isoproterenol; Mesenteric Arteries; Mesenteric Veins; Milrinone; Norepinephrine; Phosphodiesterase Inhibitors; Propranolol; Rolipram; Second Messenger Systems | 2003 |
Impact of VIP and cAMP on the regulation of TNF-alpha and IL-10 production: implications for rheumatoid arthritis.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Arthritis, Rheumatoid; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Gene Expression Regulation; Humans; Interferon-gamma; Interleukin-10; Ionomycin; Lipopolysaccharides; Macrophages; Monocytes; Phosphodiesterase Inhibitors; Protein Kinase C; Rolipram; Synovial Membrane; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Vasoactive Intestinal Peptide | 2003 |
Increased levels of cyclic adenosine monophosphate contribute to the hyporesponsiveness of mast cells in alloxan diabetes.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Antigens; Bradykinin; Bucladesine; Cell Degranulation; Cell Separation; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Diabetes Mellitus, Experimental; Dinitrophenols; Dose-Response Relationship, Drug; Immunoglobulin E; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Phosphodiesterase Inhibitors; Pleura; Rats; Rolipram; Stimulation, Chemical | 2004 |
cAMP and Schwann cells promote axonal growth and functional recovery after spinal cord injury.
Topics: Animals; Axons; Brain Stem; Bucladesine; Cell Transplantation; Cyclic AMP; Female; Interleukin-1; Motor Activity; Nerve Regeneration; Rats; Rats, Inbred F344; Recovery of Function; Rolipram; Schwann Cells; Second Messenger Systems; Serotonin; Spinal Cord Injuries; Tumor Necrosis Factor-alpha | 2004 |
Activation and induction of cyclic AMP phosphodiesterase (PDE4) in rat pulmonary microvascular endothelial cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Bucladesine; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Endothelium, Vascular; Enzyme Activation; Immunohistochemistry; Lung; Phosphodiesterase Inhibitors; Phosphorylation; Rats; RNA, Messenger; Rolipram | 2004 |
Role of PDE4 in superoxide anion generation through p44/42MAPK regulation: a cAMP and a PKA-independent mechanism.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Bronchoalveolar Lavage Fluid; Bucladesine; CREB-Binding Protein; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Flavonoids; Gene Expression Regulation, Enzymologic; Imidazoles; Lipopolysaccharides; Macrophages; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nitriles; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-raf; Pyridines; Rats; Rats, Wistar; Reactive Oxygen Species; Rolipram; Superoxides; Trans-Activators | 2004 |
Irsogladine, an anti-ulcer drug, suppresses superoxide production by inhibiting phosphodiesterase type 4 in human neutrophils.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Adult; Anti-Ulcer Agents; Bucladesine; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 1; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Gastric Mucosa; Humans; Isoenzymes; Isoquinolines; Neutrophils; Rolipram; Sulfonamides; Superoxides; Triazines | 2004 |
Multiple signalling pathways involved in beta2-adrenoceptor-mediated glucose uptake in rat skeletal muscle cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Bucladesine; Cell Line; Cholera Toxin; Chromones; Colforsin; Cyclic AMP; Dideoxyadenosine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanolamines; Glucose; Isoproterenol; Morpholines; Muscle, Skeletal; Phosphatidylinositol 3-Kinases; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Rats; Receptors, Adrenergic, beta-2; Rolipram; Signal Transduction | 2006 |
Synergistic effects of cAMP-dependent signalling pathways and IL-1 on IL-6 production by H19-7/IGF-IR neuronal cells.
Topics: Animals; Bucladesine; Cell Line; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation; Hippocampus; Interleukin-1; Interleukin-6; Neurons; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Rats; Receptors, Interleukin-1; Receptors, Interleukin-6; Receptors, Tumor Necrosis Factor; RNA, Messenger; Rolipram; Signal Transduction | 2006 |
Activation of the adenylyl cyclase/protein kinase A pathway facilitates neural release of beta-nicotinamide adenine dinucleotide in canine mesenteric artery.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Bucladesine; Calcitonin Gene-Related Peptide; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dogs; Electric Stimulation; Enzyme Activation; Female; Imines; In Vitro Techniques; Isoquinolines; Male; Mesenteric Arteries; Milrinone; NAD; Neural Pathways; Phosphodiesterase Inhibitors; Rolipram; Signal Transduction; Vasodilator Agents | 2006 |
Cyclic AMP-mediated regulation of the resting membrane potential in myelin-forming oligodendrocytes in the isolated intact rat optic nerve.
Topics: Age Factors; Animals; Animals, Newborn; Bucladesine; Colforsin; Cyclic AMP; Female; In Vitro Techniques; Male; Membrane Potentials; Myelin Sheath; Oligodendroglia; Optic Nerve; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Rolipram | 2006 |
Short-term or long-term treatments with a phosphodiesterase-4 (PDE4) inhibitor result in opposing agonist-induced Ca(2+) responses in endothelial cells.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Blotting, Northern; Blotting, Western; Bucladesine; Calcium; Calcium Signaling; Cell Line; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cycloheximide; Data Interpretation, Statistical; Endothelial Cells; Fluorescent Dyes; Fura-2; Histamine; Humans; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Protein Synthesis Inhibitors; Rolipram | 2008 |
Effect of phosphodiesterase 7 inhibitor ASB16165 on development and function of cytotoxic T lymphocyte.
Topics: Animals; Bucladesine; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cell Division; Cell Line; Colforsin; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclic Nucleotide Phosphodiesterases, Type 7; Female; Flow Cytometry; Immunosuppressive Agents; Indicators and Reagents; Lymphocyte Culture Test, Mixed; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Phosphodiesterase Inhibitors; Pyrazoles; Rolipram; Spleen; T-Lymphocytes, Cytotoxic; Tacrolimus; Thiophenes | 2009 |
Effects of cAMP-dependent protein kinase activator and inhibitor on in vivo rolipram binding to phosphodiesterase 4 in conscious rats.
Topics: Animals; Brain; Bucladesine; Carbon Radioisotopes; Central Nervous System Agents; Cerebrovascular Circulation; Consciousness; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Male; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Positron-Emission Tomography; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Rolipram; Thionucleotides | 2010 |
The ceramide-1-phosphate analogue PCERA-1 modulates tumour necrosis factor-alpha and interleukin-10 production in macrophages via the cAMP-PKA-CREB pathway in a GTP-dependent manner.
Topics: Adenylyl Cyclases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bucladesine; Calcium Signaling; Cell Line; Cell Membrane; Ceramides; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Enzyme Inhibitors; Genes, Reporter; Guanosine Triphosphate; Imidazoles; Indoles; Interleukin-10; Isoquinolines; Lipopolysaccharides; Macrophages; Mice; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Response Elements; Ribosomal Protein S6 Kinases, 90-kDa; Rolipram; Signal Transduction; Sulfonamides; Transfection; Tumor Necrosis Factor-alpha | 2010 |
A re-assessment of a combinatorial treatment involving Schwann cell transplants and elevation of cyclic AMP on recovery of motor function following thoracic spinal cord injury in rats.
Topics: Animals; Bucladesine; Cell Transplantation; Combined Modality Therapy; Cyclic AMP; Injections, Spinal; Motor Activity; Motor Skills; Rats; Rats, Inbred F344; Recovery of Function; Rolipram; Schwann Cells; Spinal Cord Injuries; Thoracic Vertebrae | 2012 |
Systems biology investigation of cAMP modulation to increase SMN levels for the treatment of spinal muscular atrophy.
Topics: Albuterol; Bucladesine; Colforsin; Cyclic AMP; Epinephrine; Fibroblasts; Fluorescent Antibody Technique; Humans; Models, Biological; Monomeric GTP-Binding Proteins; Muscular Atrophy, Spinal; Promoter Regions, Genetic; Response Elements; Rolipram; Signal Transduction; Survival of Motor Neuron 2 Protein; Systems Biology | 2014 |
Selective enhancement of wnt4 expression by cyclic AMP-associated cooperation between rat central astrocytes and microglia.
Topics: Animals; Animals, Newborn; Astrocytes; Bucladesine; Cell Communication; Coculture Techniques; Corpus Striatum; Cyclic AMP; Gene Expression Regulation; Hippocampus; Injections, Intraperitoneal; Microglia; Phosphodiesterase 4 Inhibitors; Primary Cell Culture; Rats; Rats, Sprague-Dawley; Rats, Wistar; Rolipram; Signal Transduction; Wnt4 Protein | 2015 |