bu 224 and benzofurans

bu 224 has been researched along with benzofurans in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (10.53)18.2507
2000's6 (31.58)29.6817
2010's11 (57.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Danbury, TC; Hudson, AL; Kestin, SC; Ruban, B; Waterman-Pearson, AE1
Gouch, RE; Hudson, AL; Luscombe, S; Nutt, DJ; Tyacke, RJ1
Hudson, AL; Nutt, DJ; Robinson, ES; Tyacke, RJ1
Hudson, AL; Nutt, DJ; Paterson, LM; Tyacke, RJ1
Handley, SL; MacInnes, N1
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES1
Hayashi, Y; Itoh, I; Iwasaki, M; Kagawa, K; Kamibayashi, T; Mashimo, T; Takada, K; Yamatodani, A1
Bour, S; Carpéné, C; Duro, P; Garcia-Barrado, MJ; Iglesias-Osma, MC; Marti, L; Moratinos, J; Pastor, MF; Prévot, D; Valet, P; Visentin, V1
Li, JX; Winter, JC; Zhang, Y1
Li, JX; Peng, BW; Thorn, DA; Winter, JC; Zhang, Y1
An, XF; Li, JX; Winter, JC; Zhang, Y1
Ali, I; Andurkar, SV; Bhalla, S; Gulati, A; Lee, H1
Chen, MF; Cheng, JT; Chiu, NH; Chou, MT; Chung, HH; Mar, GY1
Cheng, JT; Chung, HH; Hsu, CT; Ku, PM; Lee, WJ; Yang, TT1
He, X; Li, JX; Min, JW; Peng, BW; Zhang, Y1
He, XH; Li, JX; Qiu, Y; Zhang, Y1
García-Sevilla, JA; Keller, B2
Jia, S; Li, JX; Qiu, Y; Thorn, DA; Zhang, Y1

Other Studies

19 other study(ies) available for bu 224 and benzofurans

ArticleYear
Imidazoline (I2) binding sites in chicken brain.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Amiloride; Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Chickens; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug; Tritium

1999
Endogenous indoleamines demonstrate moderate affinity for I2 binding sites.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Agmatine; Animals; Benzofurans; Binding Sites; Binding, Competitive; Biogenic Monoamines; Brain; Cell Membrane; Female; Histamine; Imidazoles; Imidazoline Receptors; Isatin; Kinetics; Male; Rabbits; Rats; Rats, Wistar; Receptors, Drug; Serotonin; Tritium; Tryptamines; Tryptophan

1999
Distribution of [(3)H]BU224, a selective imidazoline I(2) binding site ligand, in rat brain.
    European journal of pharmacology, 2002, Aug-16, Volume: 450, Issue:1

    Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kinetics; Ligands; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Drug

2002
Relationship between imidazoline(2) sites and monoamine oxidase.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Animals; Benzofurans; Brain; Cell Membrane; Clorgyline; Imidazoles; Imidazoline Receptors; Ligands; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Radioligand Assay; Rats; Receptors, Drug; Selegiline

2003
Autoradiographic localisation of [3H]2-BFI imidazoline I2 binding sites in mouse brain.
    European journal of pharmacology, 2005, Jun-01, Volume: 516, Issue:2

    Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Male; Mice; Mice, Inbred C57BL; Midline Thalamic Nuclei; Nucleus Accumbens; Radioligand Assay; Raphe Nuclei; Tritium

2005
Characterisation of imidazoline I2 binding sites in pig brain.
    European journal of pharmacology, 2005, Sep-05, Volume: 519, Issue:1-2

    Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium

2005
Identification of the central imidazoline receptor subtype involved in modulation of halothane-epinephrine arrhythmias in rats.
    Anesthesia and analgesia, 2005, Volume: 101, Issue:6

    Topics: Animals; Arrhythmias, Cardiac; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Epinephrine; Halothane; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug

2005
The imidazoline I2-site ligands BU 224 and 2-BFI inhibit MAO-A and MAO-B activities, hydrogen peroxide production, and lipolysis in rodent and human adipocytes.
    European journal of pharmacology, 2006, Dec-15, Volume: 552, Issue:1-3

    Topics: Adipocytes; Adipose Tissue; Amine Oxidase (Copper-Containing); Animals; Benzofurans; Binding Sites; Blood Platelets; Cells, Cultured; Dose-Response Relationship, Drug; Glucose; Humans; Hydrogen Peroxide; Imidazoles; Imidazolines; Lipolysis; Liver; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Rabbits; Rats; Rats, Wistar; Rats, Zucker

2006
Morphine-induced antinociception in the rat: supra-additive interactions with imidazoline I₂ receptor ligands.
    European journal of pharmacology, 2011, Nov-01, Volume: 669, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Agmatine; Analgesics; Analgesics, Opioid; Animals; Benzofurans; Disease Models, Animal; Drug Synergism; Idazoxan; Imidazoles; Imidazoline Receptors; Ligands; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Saline Solution, Hypertonic; Yohimbine

2011
Effects of imidazoline I₂ receptor ligands on morphine- and tramadol-induced antinociception in rats.
    European journal of pharmacology, 2011, Nov-30, Volume: 670, Issue:2-3

    Topics: Agmatine; Analgesics; Animals; Behavior, Animal; Benzofurans; Dose-Response Relationship, Drug; Drug Interactions; Imidazoles; Imidazoline Receptors; Ligands; Morphine; Rats; Rats, Sprague-Dawley; Tramadol

2011
Effects of imidazoline I(2) receptor agonists and morphine on schedule-controlled responding in rats.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 101, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Benzofurans; Conditioning, Operant; Drug Interactions; Imidazoles; Imidazoline Receptors; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Reinforcement Schedule

2012
Potentiation of oxycodone antinociception in mice by agmatine and BMS182874 via an imidazoline I2 receptor-mediated mechanism.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 103, Issue:3

    Topics: Agmatine; Analgesics, Opioid; Animals; Benzofurans; Dansyl Compounds; Drug Synergism; Imidazoles; Imidazoline Receptors; Male; Mice; Oxycodone; Pain Measurement

2013
Changes of imidazoline receptors in spontaneously hypertensive rats.
    International journal of experimental pathology, 2013, Volume: 94, Issue:1

    Topics: Agmatine; Animals; Antihypertensive Agents; Aorta, Thoracic; Benzofurans; Blood Pressure; Blotting, Western; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; Hypertension; Imidazoles; Imidazoline Receptors; KATP Channels; Male; Potassium Channel Blockers; Protein Kinase Inhibitors; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Up-Regulation; Vasodilation; Vasodilator Agents

2013
Mediation of AMP kinase in the increase of glucose uptake in L6 cells induced by activation of imidazoline I-2 receptors.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2013, Volume: 45, Issue:5

    Topics: Adenylate Kinase; Aminoimidazole Carboxamide; Animals; Benzofurans; Cell Line; Glucose; Imidazoles; Imidazoline Receptors; Metformin; Muscle Cells; Phosphorylation; Rats; Ribonucleotides

2013
Gender difference in epileptogenic effects of 2-BFI and BU224 in mice.
    European journal of pharmacology, 2013, Oct-15, Volume: 718, Issue:1-3

    Topics: Animals; Benzofurans; Female; Imidazoles; Imidazoline Receptors; Male; Mice; Mice, Inbred C57BL; Seizures; Sex Characteristics

2013
Discriminative stimulus effects of the novel imidazoline I₂ receptor ligand CR4056 in rats.
    Scientific reports, 2014, Oct-13, Volume: 4

    Topics: Animals; Benzofurans; Imidazoles; Imidazoline Receptors; Imidazolines; Male; Methadone; Morphine; Quinazolines; Rats

2014
Immunodetection and subcellular distribution of imidazoline receptor proteins with three antibodies in mouse and human brains: Effects of treatments with I1- and I2-imidazoline drugs.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:9

    Topics: Adult; Animals; Antibodies; Benzofurans; Binding Sites; Brain; Cell Membrane; Cytosol; Female; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Male; Mice; Styrenes; Up-Regulation

2015
Antinociceptive effects of imidazoline I2 receptor agonists in the formalin test in rats.
    Behavioural pharmacology, 2016, Volume: 27, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Benzofurans; Disease Models, Animal; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Injections, Intraperitoneal; Injections, Intraventricular; Locomotion; Male; Pain; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Time Factors

2016
Inhibitory effects of imidazoline receptor ligands on basal and kainic acid-induced neurotoxic signalling in mice.
    Journal of psychopharmacology (Oxford, England), 2016, Volume: 30, Issue:9

    Topics: Animals; Benzofurans; Cerebral Cortex; Cyclin-Dependent Kinase 5; Glutamic Acid; Hippocampus; Idazoxan; Imidazoles; Imidazoline Receptors; Kainic Acid; Ligands; Male; Mice; Neurodegenerative Diseases; Neuroprotective Agents; Styrenes; Time Factors

2016