bu 224 has been researched along with benzofurans in 19 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (10.53) | 18.2507 |
2000's | 6 (31.58) | 29.6817 |
2010's | 11 (57.89) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Danbury, TC; Hudson, AL; Kestin, SC; Ruban, B; Waterman-Pearson, AE | 1 |
Gouch, RE; Hudson, AL; Luscombe, S; Nutt, DJ; Tyacke, RJ | 1 |
Hudson, AL; Nutt, DJ; Robinson, ES; Tyacke, RJ | 1 |
Hudson, AL; Nutt, DJ; Paterson, LM; Tyacke, RJ | 1 |
Handley, SL; MacInnes, N | 1 |
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES | 1 |
Hayashi, Y; Itoh, I; Iwasaki, M; Kagawa, K; Kamibayashi, T; Mashimo, T; Takada, K; Yamatodani, A | 1 |
Bour, S; Carpéné, C; Duro, P; Garcia-Barrado, MJ; Iglesias-Osma, MC; Marti, L; Moratinos, J; Pastor, MF; Prévot, D; Valet, P; Visentin, V | 1 |
Li, JX; Winter, JC; Zhang, Y | 1 |
Li, JX; Peng, BW; Thorn, DA; Winter, JC; Zhang, Y | 1 |
An, XF; Li, JX; Winter, JC; Zhang, Y | 1 |
Ali, I; Andurkar, SV; Bhalla, S; Gulati, A; Lee, H | 1 |
Chen, MF; Cheng, JT; Chiu, NH; Chou, MT; Chung, HH; Mar, GY | 1 |
Cheng, JT; Chung, HH; Hsu, CT; Ku, PM; Lee, WJ; Yang, TT | 1 |
He, X; Li, JX; Min, JW; Peng, BW; Zhang, Y | 1 |
He, XH; Li, JX; Qiu, Y; Zhang, Y | 1 |
García-Sevilla, JA; Keller, B | 2 |
Jia, S; Li, JX; Qiu, Y; Thorn, DA; Zhang, Y | 1 |
19 other study(ies) available for bu 224 and benzofurans
Article | Year |
---|---|
Imidazoline (I2) binding sites in chicken brain.
Topics: Agmatine; Amiloride; Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Chickens; Clonidine; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug; Tritium | 1999 |
Endogenous indoleamines demonstrate moderate affinity for I2 binding sites.
Topics: Agmatine; Animals; Benzofurans; Binding Sites; Binding, Competitive; Biogenic Monoamines; Brain; Cell Membrane; Female; Histamine; Imidazoles; Imidazoline Receptors; Isatin; Kinetics; Male; Rabbits; Rats; Rats, Wistar; Receptors, Drug; Serotonin; Tritium; Tryptamines; Tryptophan | 1999 |
Distribution of [(3)H]BU224, a selective imidazoline I(2) binding site ligand, in rat brain.
Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kinetics; Ligands; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Drug | 2002 |
Relationship between imidazoline(2) sites and monoamine oxidase.
Topics: Animals; Benzofurans; Brain; Cell Membrane; Clorgyline; Imidazoles; Imidazoline Receptors; Ligands; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Radioligand Assay; Rats; Receptors, Drug; Selegiline | 2003 |
Autoradiographic localisation of [3H]2-BFI imidazoline I2 binding sites in mouse brain.
Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Idazoxan; Imidazoles; Male; Mice; Mice, Inbred C57BL; Midline Thalamic Nuclei; Nucleus Accumbens; Radioligand Assay; Raphe Nuclei; Tritium | 2005 |
Characterisation of imidazoline I2 binding sites in pig brain.
Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium | 2005 |
Identification of the central imidazoline receptor subtype involved in modulation of halothane-epinephrine arrhythmias in rats.
Topics: Animals; Arrhythmias, Cardiac; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Epinephrine; Halothane; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Rats; Rats, Sprague-Dawley; Receptors, Drug | 2005 |
The imidazoline I2-site ligands BU 224 and 2-BFI inhibit MAO-A and MAO-B activities, hydrogen peroxide production, and lipolysis in rodent and human adipocytes.
Topics: Adipocytes; Adipose Tissue; Amine Oxidase (Copper-Containing); Animals; Benzofurans; Binding Sites; Blood Platelets; Cells, Cultured; Dose-Response Relationship, Drug; Glucose; Humans; Hydrogen Peroxide; Imidazoles; Imidazolines; Lipolysis; Liver; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Rabbits; Rats; Rats, Wistar; Rats, Zucker | 2006 |
Morphine-induced antinociception in the rat: supra-additive interactions with imidazoline I₂ receptor ligands.
Topics: Adrenergic alpha-2 Receptor Antagonists; Agmatine; Analgesics; Analgesics, Opioid; Animals; Benzofurans; Disease Models, Animal; Drug Synergism; Idazoxan; Imidazoles; Imidazoline Receptors; Ligands; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Saline Solution, Hypertonic; Yohimbine | 2011 |
Effects of imidazoline I₂ receptor ligands on morphine- and tramadol-induced antinociception in rats.
Topics: Agmatine; Analgesics; Animals; Behavior, Animal; Benzofurans; Dose-Response Relationship, Drug; Drug Interactions; Imidazoles; Imidazoline Receptors; Ligands; Morphine; Rats; Rats, Sprague-Dawley; Tramadol | 2011 |
Effects of imidazoline I(2) receptor agonists and morphine on schedule-controlled responding in rats.
Topics: Analgesics; Animals; Behavior, Animal; Benzofurans; Conditioning, Operant; Drug Interactions; Imidazoles; Imidazoline Receptors; Male; Morphine; Pain; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Reinforcement Schedule | 2012 |
Potentiation of oxycodone antinociception in mice by agmatine and BMS182874 via an imidazoline I2 receptor-mediated mechanism.
Topics: Agmatine; Analgesics, Opioid; Animals; Benzofurans; Dansyl Compounds; Drug Synergism; Imidazoles; Imidazoline Receptors; Male; Mice; Oxycodone; Pain Measurement | 2013 |
Changes of imidazoline receptors in spontaneously hypertensive rats.
Topics: Agmatine; Animals; Antihypertensive Agents; Aorta, Thoracic; Benzofurans; Blood Pressure; Blotting, Western; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; Hypertension; Imidazoles; Imidazoline Receptors; KATP Channels; Male; Potassium Channel Blockers; Protein Kinase Inhibitors; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Up-Regulation; Vasodilation; Vasodilator Agents | 2013 |
Mediation of AMP kinase in the increase of glucose uptake in L6 cells induced by activation of imidazoline I-2 receptors.
Topics: Adenylate Kinase; Aminoimidazole Carboxamide; Animals; Benzofurans; Cell Line; Glucose; Imidazoles; Imidazoline Receptors; Metformin; Muscle Cells; Phosphorylation; Rats; Ribonucleotides | 2013 |
Gender difference in epileptogenic effects of 2-BFI and BU224 in mice.
Topics: Animals; Benzofurans; Female; Imidazoles; Imidazoline Receptors; Male; Mice; Mice, Inbred C57BL; Seizures; Sex Characteristics | 2013 |
Discriminative stimulus effects of the novel imidazoline I₂ receptor ligand CR4056 in rats.
Topics: Animals; Benzofurans; Imidazoles; Imidazoline Receptors; Imidazolines; Male; Methadone; Morphine; Quinazolines; Rats | 2014 |
Immunodetection and subcellular distribution of imidazoline receptor proteins with three antibodies in mouse and human brains: Effects of treatments with I1- and I2-imidazoline drugs.
Topics: Adult; Animals; Antibodies; Benzofurans; Binding Sites; Brain; Cell Membrane; Cytosol; Female; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Male; Mice; Styrenes; Up-Regulation | 2015 |
Antinociceptive effects of imidazoline I2 receptor agonists in the formalin test in rats.
Topics: Analgesics; Animals; Behavior, Animal; Benzofurans; Disease Models, Animal; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Injections, Intraperitoneal; Injections, Intraventricular; Locomotion; Male; Pain; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Time Factors | 2016 |
Inhibitory effects of imidazoline receptor ligands on basal and kainic acid-induced neurotoxic signalling in mice.
Topics: Animals; Benzofurans; Cerebral Cortex; Cyclin-Dependent Kinase 5; Glutamic Acid; Hippocampus; Idazoxan; Imidazoles; Imidazoline Receptors; Kainic Acid; Ligands; Male; Mice; Neurodegenerative Diseases; Neuroprotective Agents; Styrenes; Time Factors | 2016 |