Page last updated: 2024-08-25

brl 46470 and granisetron

brl 46470 has been researched along with granisetron in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blaney, FE; Edge, C; Phippen, RW1
Blackshaw, LA; Dent, J; Nisyrios, V1
Sanger, GJ; Wardle, KA1
Blackburn, TP; Grahame-Smith, DG; Leslie, RA; Newberry, NR; Sprosen, TS; Watkins, CJ1
Barber, PC; Barnes, NM; Bentley, KR; Blackburn, TP; Ge, J; Hope, AG; Lambert, JJ; Peters, JA; Steward, LJ1

Other Studies

5 other study(ies) available for brl 46470 and granisetron

ArticleYear
Molecular surface comparison. 2. Similarity of electrostatic vector fields in drug design.
    Journal of molecular graphics, 1995, Volume: 13, Issue:3

    Topics: Anti-Anxiety Agents; Benzamides; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Drug Design; Electricity; GABA-A Receptor Agonists; Granisetron; Indoles; Isomerism; Molecular Conformation; Ondansetron; Pharmaceutical Preparations; Protein Binding; Pyrazoles; Pyridazines; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship; Surface Properties; Triazolam; Tropisetron

1995
Responses of ferret lower esophageal sphincter to 5-hydroxytryptamine: pathways and receptor subtypes.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Animals; Atropine; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Esophagus; Female; Ferrets; Granisetron; Guanethidine; Indoles; Ketanserin; Male; Muscle, Smooth; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Splanchnic Nerves; Time Factors; Vagotomy; Vagus Nerve

1995
Constipation evoked by 5-HT3-receptor antagonism: evidence for heterogeneous efficacy among different antagonists in guinea-pigs.
    The Journal of pharmacy and pharmacology, 1994, Volume: 46, Issue:8

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Clonidine; Colon; Constipation; Defecation; Drug Interactions; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Injections, Intraperitoneal; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Serotonin Antagonists; Tropisetron

1994
BRL 46470 potently antagonizes neural responses activated by 5-HT3 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:8

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electrophysiology; Glioma; Granisetron; In Vitro Techniques; Indoles; Kinetics; Male; Neuroblastoma; Neurons; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Tropisetron; Tubocurarine; Tumor Cells, Cultured; Vagus Nerve

1993
Evidence that the atypical 5-HT3 receptor ligand, [3H]-BRL46470, labels additional 5-HT3 binding sites compared to [3H]-granisetron.
    British journal of pharmacology, 1995, Volume: 116, Issue:2

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Female; Granisetron; Hippocampus; Indoles; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Time Factors

1995