Page last updated: 2024-09-03

brl 44408 and wb 4101

brl 44408 has been researched along with wb 4101 in 6 studies

Compound Research Comparison

Studies
(brl 44408)
Trials
(brl 44408)
Recent Studies (post-2010)
(brl 44408)
Studies
(wb 4101)
Trials
(wb 4101)
Recent Studies (post-2010) (wb 4101)
82016477134

Protein Interaction Comparison

ProteinTaxonomybrl 44408 (IC50)wb 4101 (IC50)
Alpha-1A adrenergic receptorHomo sapiens (human)0.001

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (66.67)18.2507
2000's1 (16.67)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Neubig, RR; Porter, AC; Uhlén, S1
Alberts, P1
Bencsics, A; Elenkov, IJ; Vizi, ES1
Dóda, M1
Centurión, D; Görnemann, T; Jähnichen, S; Kleuser, B; Pertz, HH; Villalón, CM; von Wenckstern, H1
Centurión, D; Hofmann, RA; Jantschak, F; Pertz, HH; Popp, AM; Villalón, CM1

Other Studies

6 other study(ies) available for brl 44408 and wb 4101

ArticleYear
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2

1994
Presynaptic alpha 2A-adrenoceptors regulate the 3H-noradrenaline secretion in the guinea-pig urethra.
    Pharmacology & toxicology, 1995, Volume: 77, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Dibenzazepines; Dioxanes; Dose-Response Relationship, Drug; Guinea Pigs; Imidazoles; Indoles; Isoindoles; Linear Models; Male; Norepinephrine; Rats; Receptors, Adrenergic, alpha-2; Structure-Activity Relationship; Tritium; Urethra

1995
alpha 2-, alpha 2A-, alpha 2B/2C-Adrenoceptor subtype antagonists prevent lipopolysaccharide-induced fever response in rabbits.
    Brain research, 1995, Dec-24, Volume: 705, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Body Temperature; Dioxanes; Fever; Imidazoles; Indoles; Injections, Intravenous; Isoindoles; Isoquinolines; Lipopolysaccharides; Male; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-2; Skin Physiological Phenomena

1995
Role of different subtypes of adrenoceptors in pressor responses to catecholamines released from sympathetic nerve endings.
    Brain research bulletin, 1997, Volume: 42, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Berberine; Blood Pressure; Cats; Dimethylphenylpiperazinium Iodide; Dioxanes; Female; Ganglionic Stimulants; Imidazoles; Indoles; Isoindoles; Male; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Sympathetic Nervous System

1997
Characterization of the postjunctional alpha 2C-adrenoceptor mediating vasoconstriction to UK14304 in porcine pulmonary veins.
    British journal of pharmacology, 2007, Volume: 151, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Gene Expression; Imidazoles; In Vitro Techniques; Indoles; Isoindoles; Isoquinolines; Neuromuscular Junction; Norepinephrine; Piperazines; Prazosin; Pulmonary Veins; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Vasoconstriction; Yohimbine

2007
Postjunctional α2C-adrenoceptors mediate vasoconstriction in rat tail artery: influence of precontraction and temperature on vasoreactivity.
    Naunyn-Schmiedeberg's archives of pharmacology, 2010, Volume: 382, Issue:5-6

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Brimonidine Tartrate; Dioxanes; Imidazoles; In Vitro Techniques; Isoindoles; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Piperazines; Prazosin; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Serotonin; Tail; Temperature; Vasoconstriction; Yohimbine

2010