Page last updated: 2024-09-03

brl 44408 and buspirone

brl 44408 has been researched along with buspirone in 1 studies

Compound Research Comparison

Studies
(brl 44408)
Trials
(brl 44408)
Recent Studies (post-2010)
(brl 44408)
Studies
(buspirone)
Trials
(buspirone)
Recent Studies (post-2010) (buspirone)
820162,096351382

Protein Interaction Comparison

ProteinTaxonomybrl 44408 (IC50)buspirone (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.025
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)1.75
Angiotensin-converting enzyme Homo sapiens (human)0.024
D(2) dopamine receptorHomo sapiens (human)0.323
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)2.125
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)4.16
DRattus norvegicus (Norway rat)0.12
D(3) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0266
D(2) dopamine receptorBos taurus (cattle)4
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)4.16
Alpha-1D adrenergic receptorHomo sapiens (human)1.077
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.286
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.016
D(4) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)2.125
D(3) dopamine receptorHomo sapiens (human)0.044
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.75
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)4.16
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2055
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.9811
Alpha-2A adrenergic receptorBos taurus (cattle)0.025
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.7
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.2666
Lysosomal alpha-glucosidaseBos taurus (cattle)0.03

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lodge, NJ; Myers, RA; Plym, MJ; Signor, LJ1

Other Studies

1 other study(ies) available for brl 44408 and buspirone

ArticleYear
1-(2-pyrimidinyl)-piperazine, a buspirone metabolite, modulates bladder function in the anesthetized rat.
    Neurourology and urodynamics, 2004, Volume: 23, Issue:7

    Topics: Acetic Acid; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; ATP-Binding Cassette Transporters; Benzhydryl Compounds; Buspirone; Cresols; Cromakalim; Dose-Response Relationship, Drug; Female; Imidazoles; Indoles; Isoindoles; KATP Channels; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Phenylpropanolamine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tolterodine Tartrate; Urinary Bladder; Urodynamics; Yohimbine

2004