Page last updated: 2024-09-03

brl 35135 and isoproterenol

brl 35135 has been researched along with isoproterenol in 10 studies

Compound Research Comparison

Studies
(brl 35135)
Trials
(brl 35135)
Recent Studies (post-2010)
(brl 35135)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
383130,7808032,640

Protein Interaction Comparison

ProteinTaxonomybrl 35135 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (90.00)18.2507
2000's1 (10.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Holloway, BR; Howe, R; Rao, BS; Stribling, D1
Carlisle, HJ; Stock, MJ3
Ilyés, I; Stock, M; Yahata, T1
Ilyés, I; Stock, MJ1
Carlisle, HJ; Dubuc, PU; Stock, MJ1
Nakamura, S; Nishimura, M; Shirahase, H; Takahashi, H; Yoshida, T; Yoshimura, M1
Barber, A; Cobo, MT; Díez-Sampedro, A; Martínez, JA; Pérez, M1
Obels, PP; van den Thillart, GE; Vianen, GJ; Zaagsma, J1

Other Studies

10 other study(ies) available for brl 35135 and isoproterenol

ArticleYear
Selective beta 3-adrenergic agonists of brown adipose tissue and thermogenesis. 1. [4-[2-[(2-Hydroxy-3-phenoxypropyl)amino]ethoxy]phenoxy]acetates.
    Journal of medicinal chemistry, 1992, May-15, Volume: 35, Issue:10

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Body Temperature Regulation; Oxygen; Phenoxyacetates; Rats; Rats, Zucker; Stereoisomerism; Structure-Activity Relationship

1992
Potentiation of thermoregulatory responses to isoproterenol by beta-adrenergic antagonists.
    The American journal of physiology, 1992, Volume: 263, Issue:4 Pt 2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Behavior, Animal; Body Temperature; Body Temperature Regulation; Drug Synergism; Female; Fever; Heart Rate; Isoproterenol; Phenethylamines; Propanolamines; Rats; Rats, Sprague-Dawley; Rats, Zucker

1992
Brown adipose tissue cell respiration in hypo- and hyperthyroidism after stimulation with selective and non selective beta-adrenergic agonists.
    Acta biologica Hungarica, 1991, Volume: 42, Issue:4

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Body Temperature Regulation; Hyperthyroidism; Hypothyroidism; In Vitro Techniques; Isoproterenol; Male; Oxygen Consumption; Phenethylamines; Rats; Rats, Sprague-Dawley

1991
Thermogenic responses to selective and nonselective beta-adrenerg agonists in hypothyroidism of Sprague-Dawley rats.
    Acta physiologica Hungarica, 1991, Volume: 78, Issue:4

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Animals; Body Weight; Disease Models, Animal; Guanosine Diphosphate; Hypothyroidism; Isoproterenol; Male; Methimazole; Oxygen Consumption; Phenethylamines; Rats; Rats, Sprague-Dawley; Thermoreceptors; Thyroidectomy

1991
Effects of beta-adrenoceptor agonists and antagonists on thermoregulation in the cold in lean and obese Zucker rats.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:4

    Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Cold Temperature; Female; Isoproterenol; Phenethylamines; Propanolamines; Propranolol; Rats; Rats, Zucker; Receptors, Adrenergic, beta-2

1993
Thermoregulatory responses to beta-adrenergic agonists at low ambient temperatures in the rat.
    Experimental physiology, 1993, Volume: 78, Issue:6

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Animals; Body Temperature Regulation; Cold Temperature; Isoproterenol; Male; Models, Biological; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1993
Heterogenous activity of BRL 35135, a beta 3-adrenoceptor agonist, in thermogenesis and increased blood flow in brown adipose tissue in anaesthetized rats.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:7

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Anesthesia; Animals; Blood Pressure; Body Temperature Regulation; Dose-Response Relationship, Drug; Heart Rate; Isoproterenol; Male; Phenethylamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Regional Blood Flow

1994
Thermoregulatory effects of beta adrenoceptors: effects of selective agonists and the interaction of antagonists with isoproterenol and BRL-35135 in the cold.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Body Temperature; Body Temperature Regulation; Cold Temperature; Drug Interactions; Isoproterenol; Metabolism; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Temperature

1993
Effect of different beta-adrenergic agonists on the intestinal absorption of galactose and phenylalanine.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:8

    Topics: Adrenergic beta-Agonists; Albuterol; Animals; Benzyl Alcohols; Galactose; In Vitro Techniques; Intestinal Absorption; Isoproterenol; Jejunum; Male; Metaproterenol; Phenethylamines; Phenoxyacetates; Phenoxypropanolamines; Phenylalanine; Rats; Rats, Wistar

1998
Beta-adrenoceptors mediate inhibition of lipolysis in adipocytes of tilapia (Oreochromis mossambicus).
    American journal of physiology. Endocrinology and metabolism, 2002, Volume: 282, Issue:2

    Topics: Adipocytes; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Glucose; Cells, Cultured; Fatty Acids, Nonesterified; Female; Hypoxia; Isoproterenol; Lactic Acid; Lipolysis; Male; Neurotransmitter Agents; Norepinephrine; Phenethylamines; Phentolamine; Receptors, Adrenergic, beta; Tilapia; Timolol

2002