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brexanolone and tetrahydrodeoxycorticosterone

brexanolone has been researched along with tetrahydrodeoxycorticosterone in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (37.50)18.2507
2000's4 (50.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blinn, JR; Morrow, AL; Paul, SM; Purdy, RH1
Anderson, A; Boyd, AC; Byford, A; Campbell, AC; Gemmell, DK; Hamilton, NM; Hill, DR; Hill-Venning, C; Lambert, JJ; Maidment, MS; Marshall, RJ; May, V; Peters, JA; Rees, DC; Stevenson, D; Sundaram, H1
Combs, DW; Dubinsky, B; Jacobs, K; Rybczynski, PJ; Shank, RP1
Benz, A; Coleman, M; Covey, DF; de La Cruz, MA; Evers, AS; Han, M; Hu, Y; Kumar, AS; Meadows, ES; Mennerick, S; Nathan, D; Tonnies, A; Zorumski, CF1
Anderson, A; Boyd, AC; Clark, JK; Fielding, L; Gemmell, DK; Hamilton, NM; Maidment, MS; May, V; McGuire, R; McPhail, P; Sansbury, FH; Sundaram, H; Taylor, R1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Dawson, M; Fairweather, EE; Hamilton, NM; Hamilton, NS; Hitchin, JR; James, DI; Jones, SD; Jordan, AM; Lyons, AJ; Ogilvie, DJ; Small, HF; Thomson, GJ; Waddell, ID1

Other Studies

8 other study(ies) available for brexanolone and tetrahydrodeoxycorticosterone

ArticleYear
Synthesis, metabolism, and pharmacological activity of 3 alpha-hydroxy steroids which potentiate GABA-receptor-mediated chloride ion uptake in rat cerebral cortical synaptoneurosomes.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Acetates; Animals; Cerebral Cortex; Chlorides; Desoxycorticosterone; Drug Synergism; Isomerism; Male; Molecular Conformation; Muscimol; Pregnanes; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes

1990
Anesthetic activity of novel water-soluble 2 beta-morpholinyl steroids and their modulatory effects at GABAA receptors.
    Journal of medicinal chemistry, 1997, May-23, Volume: 40, Issue:11

    Topics: Anesthesia; Anesthetics; Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Membrane; Chromaffin System; Electric Conductivity; Electrophysiology; Male; Mice; Molecular Structure; Morpholines; Pregnanediones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Solubility; Structure-Activity Relationship; Water

1997
gamma-Aminobutyrate-A receptor modulation by 3-aryl-1-(arylsulfonyl)- 1,4,5,6-tetrahydropyridazines.
    Journal of medicinal chemistry, 1999, Jul-01, Volume: 42, Issue:13

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain Stem; Cerebellum; Cerebral Cortex; GABA Agonists; GABA-A Receptor Agonists; In Vitro Techniques; Male; Mice; Motor Activity; Pentylenetetrazole; Pyridazines; Radioligand Assay; Rats; Rats, Wistar; Seizures; Structure-Activity Relationship

1999
Neurosteroid analogues. 8. Structure-activity studies of N-acylated 17a-aza-D-homosteroid analogues of the anesthetic steroids (3alpha, 5alpha)- and (3alpha,5beta)-3-hydroxypregnan-20-one.
    Journal of medicinal chemistry, 2000, Aug-24, Volume: 43, Issue:17

    Topics: Anesthetics; Animals; Binding, Competitive; Brain; Crystallography, X-Ray; Electrophysiology; Homosteroids; In Vitro Techniques; Molecular Conformation; Oocytes; Pregnanes; Rats; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2000
Conformationally constrained anesthetic steroids that modulate GABA(A) receptors.
    Journal of medicinal chemistry, 2000, Nov-02, Volume: 43, Issue:22

    Topics: Androstanols; Anesthetics; Animals; Brain; GABA Modulators; Hydrogen Bonding; In Vitro Techniques; Injections, Intravenous; Mice; Models, Molecular; Radioligand Assay; Rats; Receptors, GABA-A; Structure-Activity Relationship

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Novel steroid inhibitors of glucose 6-phosphate dehydrogenase.
    Journal of medicinal chemistry, 2012, May-10, Volume: 55, Issue:9

    Topics: Antineoplastic Agents; Cell Survival; Enzyme Inhibitors; Glucosephosphate Dehydrogenase; HEK293 Cells; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mass Spectrometry; Pregnanes; Structure-Activity Relationship

2012