bretazenil has been researched along with midazolam in 10 studies
Studies (bretazenil) | Trials (bretazenil) | Recent Studies (post-2010) (bretazenil) | Studies (midazolam) | Trials (midazolam) | Recent Studies (post-2010) (midazolam) |
---|---|---|---|---|---|
101 | 8 | 14 | 9,834 | 3,191 | 3,301 |
Protein | Taxonomy | bretazenil (IC50) | midazolam (IC50) |
---|---|---|---|
Cytochrome P450 3A4 | Homo sapiens (human) | 2.7427 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (10.00) | 18.7374 |
1990's | 7 (70.00) | 18.2507 |
2000's | 2 (20.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Danhof, M; Kuck, MT; Mandema, JW | 1 |
Järbe, TU; Rijnders, HJ; Slangen, JL | 1 |
Cooper, SJ; Yerbury, RE | 1 |
Ator, NA; Sannerud, CA | 1 |
Acri, JB; Witkin, JM; Wong, G | 1 |
Acri, JB; Barrett, JE; Gleeson, S; Witkin, JM | 1 |
Członkowska, A; Nazar, M; Płaźnik, A; Siemiatkowski, M; Sienkiewicz-Jarosz, H | 1 |
Bergman, J; Paronis, CA | 1 |
Danhof, M; Tuk, B; van Gool, T | 1 |
France, CP; McMahon, LR | 1 |
10 other study(ies) available for bretazenil and midazolam
Article | Year |
---|---|
In vivo modeling of the pharmacodynamic interaction between benzodiazepines which differ in intrinsic efficacy.
Topics: Animals; Azepines; Benzodiazepinones; Drug Interactions; Electroencephalography; Infusions, Intravenous; Male; Midazolam; Rats; Rats, Inbred Strains | 1992 |
The pentylenetetrazole-cue antagonist actions of bretazenil (Ro 16-6028) as compared to midazolam.
Topics: Animals; Benzodiazepinones; Cues; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Psychological; Male; Midazolam; Pentylenetetrazole; Rats; Rats, Inbred Strains | 1991 |
The benzodiazepine partial agonists, Ro16-6028 and Ro17-1812, increase palatable food consumption in nondeprived rats.
Topics: Animals; Benzodiazepinones; Drug Interactions; Eating; Male; Midazolam; Motor Activity; Rats; Receptors, GABA-A | 1987 |
Drug discrimination analysis of midazolam under a three-lever procedure. II: Differential effects of benzodiazepine receptor agonists.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Midazolam; Pyridines; Rats; Rats, Sprague-Dawley; Zolpidem | 1995 |
Stereospecific transduction of behavioral effects via diazepam-insensitive GABAA receptors.
Topics: Animals; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Columbidae; Diazepam; Discrimination Learning; Flumazenil; GABA Modulators; Imidazoles; Male; Midazolam; Oxadiazoles; Radioligand Assay; Receptors, GABA-A; Sensitivity and Specificity; Stereoisomerism | 1995 |
Blockade of behavioral effects of bretazenil by flumazenil and ZK 93,426 in pigeons.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Carbolines; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Male; Midazolam; Punishment; Receptors, GABA | 1997 |
The role of the hippocampus and 5-HT/GABA interaction in the central effects of benzodiazepine receptor ligands.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Brain; Conflict, Psychological; Dentate Gyrus; Dopamine; Drinking Behavior; Electroshock; Exploratory Behavior; Fenclonine; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Hydroxyindoleacetic Acid; Male; Microinjections; Midazolam; Motor Activity; Norepinephrine; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Serotonin; Zolpidem | 1999 |
Apparent pA2 values of benzodiazepine antagonists and partial agonists in monkeys.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Carbolines; Dose-Response Relationship, Drug; Electroshock; Feeding Behavior; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Kinetics; Male; Midazolam; Receptors, GABA-A; Reinforcement Schedule; Saimiri | 1999 |
Mechanism-based pharmacodynamic modeling of the interaction of midazolam, bretazenil, and zolpidem with ethanol.
Topics: Animals; Benzodiazepinones; Drug Interactions; Electroencephalography; Ethanol; Male; Midazolam; Models, Biological; Protein Binding; Pyridines; Rats; Rats, Wistar; Zolpidem | 2002 |
Differential behavioral effects of low efficacy positive GABAA modulators in combination with benzodiazepines and a neuroactive steroid in rhesus monkeys.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; GABA Modulators; Macaca mulatta; Midazolam; Pregnanediones; Receptors, GABA-A; Triazoles | 2006 |