Page last updated: 2024-09-02

bretazenil and midazolam

bretazenil has been researched along with midazolam in 10 studies

Compound Research Comparison

Studies
(bretazenil)
Trials
(bretazenil)
Recent Studies (post-2010)
(bretazenil)
Studies
(midazolam)
Trials
(midazolam)
Recent Studies (post-2010) (midazolam)
1018149,8343,1913,301

Protein Interaction Comparison

ProteinTaxonomybretazenil (IC50)midazolam (IC50)
Cytochrome P450 3A4Homo sapiens (human)2.7427

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's7 (70.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Danhof, M; Kuck, MT; Mandema, JW1
Järbe, TU; Rijnders, HJ; Slangen, JL1
Cooper, SJ; Yerbury, RE1
Ator, NA; Sannerud, CA1
Acri, JB; Witkin, JM; Wong, G1
Acri, JB; Barrett, JE; Gleeson, S; Witkin, JM1
Członkowska, A; Nazar, M; Płaźnik, A; Siemiatkowski, M; Sienkiewicz-Jarosz, H1
Bergman, J; Paronis, CA1
Danhof, M; Tuk, B; van Gool, T1
France, CP; McMahon, LR1

Other Studies

10 other study(ies) available for bretazenil and midazolam

ArticleYear
In vivo modeling of the pharmacodynamic interaction between benzodiazepines which differ in intrinsic efficacy.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:1

    Topics: Animals; Azepines; Benzodiazepinones; Drug Interactions; Electroencephalography; Infusions, Intravenous; Male; Midazolam; Rats; Rats, Inbred Strains

1992
The pentylenetetrazole-cue antagonist actions of bretazenil (Ro 16-6028) as compared to midazolam.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:1

    Topics: Animals; Benzodiazepinones; Cues; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Psychological; Male; Midazolam; Pentylenetetrazole; Rats; Rats, Inbred Strains

1991
The benzodiazepine partial agonists, Ro16-6028 and Ro17-1812, increase palatable food consumption in nondeprived rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:4

    Topics: Animals; Benzodiazepinones; Drug Interactions; Eating; Male; Midazolam; Motor Activity; Rats; Receptors, GABA-A

1987
Drug discrimination analysis of midazolam under a three-lever procedure. II: Differential effects of benzodiazepine receptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Midazolam; Pyridines; Rats; Rats, Sprague-Dawley; Zolpidem

1995
Stereospecific transduction of behavioral effects via diazepam-insensitive GABAA receptors.
    European journal of pharmacology, 1995, May-24, Volume: 278, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Columbidae; Diazepam; Discrimination Learning; Flumazenil; GABA Modulators; Imidazoles; Male; Midazolam; Oxadiazoles; Radioligand Assay; Receptors, GABA-A; Sensitivity and Specificity; Stereoisomerism

1995
Blockade of behavioral effects of bretazenil by flumazenil and ZK 93,426 in pigeons.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 56, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Carbolines; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Male; Midazolam; Punishment; Receptors, GABA

1997
The role of the hippocampus and 5-HT/GABA interaction in the central effects of benzodiazepine receptor ligands.
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:5-6

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Brain; Conflict, Psychological; Dentate Gyrus; Dopamine; Drinking Behavior; Electroshock; Exploratory Behavior; Fenclonine; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Hydroxyindoleacetic Acid; Male; Microinjections; Midazolam; Motor Activity; Norepinephrine; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Serotonin; Zolpidem

1999
Apparent pA2 values of benzodiazepine antagonists and partial agonists in monkeys.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Carbolines; Dose-Response Relationship, Drug; Electroshock; Feeding Behavior; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Kinetics; Male; Midazolam; Receptors, GABA-A; Reinforcement Schedule; Saimiri

1999
Mechanism-based pharmacodynamic modeling of the interaction of midazolam, bretazenil, and zolpidem with ethanol.
    Journal of pharmacokinetics and pharmacodynamics, 2002, Volume: 29, Issue:3

    Topics: Animals; Benzodiazepinones; Drug Interactions; Electroencephalography; Ethanol; Male; Midazolam; Models, Biological; Protein Binding; Pyridines; Rats; Rats, Wistar; Zolpidem

2002
Differential behavioral effects of low efficacy positive GABAA modulators in combination with benzodiazepines and a neuroactive steroid in rhesus monkeys.
    British journal of pharmacology, 2006, Volume: 147, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; GABA Modulators; Macaca mulatta; Midazolam; Pregnanediones; Receptors, GABA-A; Triazoles

2006