Page last updated: 2024-09-02

bretazenil and l 663581

bretazenil has been researched along with l 663581 in 3 studies

Compound Research Comparison

Studies
(bretazenil)
Trials
(bretazenil)
Recent Studies (post-2010)
(bretazenil)
Studies
(l 663581)
Trials
(l 663581)
Recent Studies (post-2010) (l 663581)
1018141200

Protein Interaction Comparison

ProteinTaxonomybretazenil (IC50)l 663581 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0036
GABA theta subunitRattus norvegicus (Norway rat)0.0036
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0036

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1
Bristow, LJ; Cook, GP; Guscott, MR1

Other Studies

3 other study(ies) available for bretazenil and l 663581

ArticleYear
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995
Contextual fear conditioning and baseline startle responses in the rat fear-potentiated startle test: a comparison of benzodiazepine/gamma-aminobutyric acid-A receptor agonists.
    Behavioural pharmacology, 2000, Volume: 11, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Avoidance Learning; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Conditioning, Operant; Electric Stimulation; Fear; GABA Modulators; Male; Rats; Rats, Sprague-Dawley; Reflex, Startle

2000