Page last updated: 2024-09-02

bretazenil and alphaxalone

bretazenil has been researched along with alphaxalone in 2 studies

Compound Research Comparison

Studies
(bretazenil)
Trials
(bretazenil)
Recent Studies (post-2010)
(bretazenil)
Studies
(alphaxalone)
Trials
(alphaxalone)
Recent Studies (post-2010) (alphaxalone)
101814559157314

Protein Interaction Comparison

ProteinTaxonomybretazenil (IC50)alphaxalone (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.4805
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)0.538
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.4805
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)0.538
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.538
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.538
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.4805
GABA theta subunitRattus norvegicus (Norway rat)0.4805
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.4805

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cagetti, E; Liang, J; Olsen, RW; Spigelman, I1
France, CP; McMahon, LR1

Other Studies

2 other study(ies) available for bretazenil and alphaxalone

ArticleYear
Withdrawal from chronic intermittent ethanol treatment changes subunit composition, reduces synaptic function, and decreases behavioral responses to positive allosteric modulators of GABAA receptors.
    Molecular pharmacology, 2003, Volume: 63, Issue:1

    Topics: Affinity Labels; Alcoholism; Allosteric Regulation; Anesthetics; Animals; Anxiety; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Diazepam; Electrophysiology; Ethanol; GABA Modulators; Hippocampus; Hypnosis; Immunoblotting; Kinetics; Male; Maze Learning; Neurons; Pregnanediones; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; Sleep

2003
Differential behavioral effects of low efficacy positive GABAA modulators in combination with benzodiazepines and a neuroactive steroid in rhesus monkeys.
    British journal of pharmacology, 2006, Volume: 147, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Fluorobenzenes; GABA Modulators; Macaca mulatta; Midazolam; Pregnanediones; Receptors, GABA-A; Triazoles

2006