bretazenil has been researched along with abecarnil in 8 studies
Studies (bretazenil) | Trials (bretazenil) | Recent Studies (post-2010) (bretazenil) | Studies (abecarnil) | Trials (abecarnil) | Recent Studies (post-2010) (abecarnil) |
---|---|---|---|---|---|
101 | 8 | 14 | 96 | 12 | 2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (75.00) | 18.2507 |
2000's | 2 (25.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Haefely, W; Martin, JR; Schoch, P | 1 |
Hönack, D; Löscher, W; Rundfeldt, C; Wlaź, P | 1 |
Mehta, AK; Shank, RP | 1 |
Drescher, U; Knoflach, F; Malherbe, P; Mohler, H; Scheurer, L | 1 |
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ | 1 |
Griebel, G; Perrault, G; Sanger, DJ | 1 |
Basile, AS; Lippa, AS; Skolnick, P | 1 |
2 review(s) available for bretazenil and abecarnil
Article | Year |
---|---|
Novel anxiolytics that act as partial agonists at benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Clonazepam; Humans; Imidazoles; Pyridines; Receptors, GABA-A | 1990 |
Anxioselective anxiolytics: can less be more?
Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepinones; Carbolines; Clinical Trials as Topic; Fluorobenzenes; GABA-A Receptor Agonists; Humans; Indoles; Pyrroles; Quinolones; Triazoles | 2004 |
6 other study(ies) available for bretazenil and abecarnil
Article | Year |
---|---|
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Anticonvulsant tolerance and withdrawal characteristics of benzodiazepine receptor ligands in different seizure models in mice. Comparison of diazepam, bretazenil and abecarnil.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Carbolines; Diazepam; Disease Models, Animal; Drug Tolerance; Male; Mice; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome | 1995 |
Interaction of abecarnil, bretazenil, and RO 19-8022 with diazepam-sensitive and -insensitive benzodiazepine sites in the rat cerebellum and cerebral cortex.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Diazepam; Male; Pyrrolidines; Quinolizines; Rats; Rats, Wistar; Receptors, GABA-A | 1995 |
Full and partial agonism displayed by benzodiazepine receptor ligands at recombinant gamma-aminobutyric acidA receptor subtypes.
Topics: Benzodiazepinones; Carbolines; Cells, Cultured; DNA; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Imidazoles; Kinetics; Ligands; Macromolecular Substances; Pyrimidines; Receptors, GABA-A; Recombinant Proteins; Sensitivity and Specificity; Substrate Specificity; Transfection | 1993 |
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem | 1995 |
Study of the modulatory activity of BZ (omega) receptor ligands on defensive behaviors in mice: evaluation of the importance of intrinsic efficacy and receptor subtype selectivity.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Diazepam; Escape Reaction; Male; Mice; Motor Activity; Rats; Receptors, GABA-A | 1999 |