Page last updated: 2024-09-02

bretazenil and abecarnil

bretazenil has been researched along with abecarnil in 8 studies

Compound Research Comparison

Studies
(bretazenil)
Trials
(bretazenil)
Recent Studies (post-2010)
(bretazenil)
Studies
(abecarnil)
Trials
(abecarnil)
Recent Studies (post-2010) (abecarnil)
10181496122

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (75.00)18.2507
2000's2 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Haefely, W; Martin, JR; Schoch, P1
Hönack, D; Löscher, W; Rundfeldt, C; Wlaź, P1
Mehta, AK; Shank, RP1
Drescher, U; Knoflach, F; Malherbe, P; Mohler, H; Scheurer, L1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1
Griebel, G; Perrault, G; Sanger, DJ1
Basile, AS; Lippa, AS; Skolnick, P1

Reviews

2 review(s) available for bretazenil and abecarnil

ArticleYear
Novel anxiolytics that act as partial agonists at benzodiazepine receptors.
    Trends in pharmacological sciences, 1990, Volume: 11, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Clonazepam; Humans; Imidazoles; Pyridines; Receptors, GABA-A

1990
Anxioselective anxiolytics: can less be more?
    European journal of pharmacology, 2004, Oct-01, Volume: 500, Issue:1-3

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepinones; Carbolines; Clinical Trials as Topic; Fluorobenzenes; GABA-A Receptor Agonists; Humans; Indoles; Pyrroles; Quinolones; Triazoles

2004

Other Studies

6 other study(ies) available for bretazenil and abecarnil

ArticleYear
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Anticonvulsant tolerance and withdrawal characteristics of benzodiazepine receptor ligands in different seizure models in mice. Comparison of diazepam, bretazenil and abecarnil.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Carbolines; Diazepam; Disease Models, Animal; Drug Tolerance; Male; Mice; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome

1995
Interaction of abecarnil, bretazenil, and RO 19-8022 with diazepam-sensitive and -insensitive benzodiazepine sites in the rat cerebellum and cerebral cortex.
    Life sciences, 1995, Volume: 57, Issue:24

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Diazepam; Male; Pyrrolidines; Quinolizines; Rats; Rats, Wistar; Receptors, GABA-A

1995
Full and partial agonism displayed by benzodiazepine receptor ligands at recombinant gamma-aminobutyric acidA receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Benzodiazepinones; Carbolines; Cells, Cultured; DNA; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Imidazoles; Kinetics; Ligands; Macromolecular Substances; Pyrimidines; Receptors, GABA-A; Recombinant Proteins; Sensitivity and Specificity; Substrate Specificity; Transfection

1993
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995
Study of the modulatory activity of BZ (omega) receptor ligands on defensive behaviors in mice: evaluation of the importance of intrinsic efficacy and receptor subtype selectivity.
    Progress in neuro-psychopharmacology & biological psychiatry, 1999, Volume: 23, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Diazepam; Escape Reaction; Male; Mice; Motor Activity; Rats; Receptors, GABA-A

1999