bremazocine and naloxone

bremazocine has been researched along with naloxone in 81 studies

Research

Studies (81)

TimeframeStudies, this research(%)All Research%
pre-199044 (54.32)18.7374
1990's27 (33.33)18.2507
2000's9 (11.11)29.6817
2010's1 (1.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Pinnock, RD1
Bianchi, G1
Negus, SS; Picker, MJ; Powell, KR1
Borsodi, A; Lajtha, A; Zawilska, J1
Christensen, JD; Fjalland, B1
Deviche, P; Lowry, CA; Moore, FL2
Hammer, RP1
Doty, P; Dykstra, LA; Mattox, SR; Negus, SS; Picker, MJ1
Heijna, MH; Hogenboom, F; Mulder, AH; Padt, M; Portoghese, PS; Schoffelmeer, AN1
Dissanayake, VU; Hill, RG; Hughes, J; Hunter, JC1
Baraldi, M; Zanoli, P1
Gyires, K1
Ahmed, MS; Cavinato, AG; Maulik, D; Zhou, DH1
Kobylyansky, AG; Nesterenko, PN; Pivovarov, AS; Yarygin, KN1
Kobylyansky, AG1
Makimura, M; Murakoshi, Y1
Huidobro-Toro, JP; Roblero, J; Salas, SP; Ureta, H1
Christensen, JD; Fjalland, B; Grell, S1
Dykstra, LA; Picker, MJ1
Bourgoin, S; Gallissot, MC; Gozlan, H; Hamon, M; Menard, F; Vergé, D1
Deviche, P; Moore, FL1
La Regina, A; Petrillo, P; Sbacchi, M; Tavani, A1
Bolger, GT; Marcus, KA; Skolnick, P; Thibou, R; Weissman, BA1
Frey, HH1
Millan, MJ; Morris, BJ1
Herz, A; Millan, MJ; Morris, BJ1
Barlow, JJ; Carroll, JA; Costello, GF; Main, BG; Shaw, JS1
Di Chiara, G; Imperato, A1
Frances, B; Meunier, JC; Moisand, C1
Ensinger, HA1
Hayes, A; Kelly, A1
Grace, M; Kneip, J; Levine, AS; Morley, JE; Shearman, GT; Zeugner, H1
Hayes, AG; Stewart, BR1
Barber, DJ; Cooper, SJ; Jackson, A; Moores, WR1
Starr, MS1
Conway, S; Koenig, JI; Krulich, L; Mayfield, MA; McCann, SM1
Shearman, GT; Stenfors, C1
Leander, JD3
Bakalkin, GIa; Pivovarov, AS; Romanenko, OK1
Dykstra, LA; Heise, JW; Picker, M1
Itzhak, Y; Simon, EJ1
Bakalkin, GIa; Bespalova, ZhD; Iakovleva, TV; Korobov, KP; Vinogradov, VA1
Huidobro-Toro, JP; Parada, S1
Corbett, AD; Gillan, MG; Kosterlitz, HW; McKnight, AT; Paterson, SJ; Robson, LE1
Fuller, RW; Leander, JD1
Akil, H; Khachaturian, H; Lewis, ME; Watson, SJ1
Akkerman, AM; Bakel, HC; Büscher, H; Hill, RC; Maurer, R; Petcher, TJ; Römer, D; Welle, HB1
Kattau, RW; Leander, JD; Rathbun, RC1
Code, RA; Tang, AH1
Flórez, J; Pazos, A; Tristán, C1
Gambino, MC; Petrillo, P; Tavani, A1
Chaillet, P; Costentin, J; Marçais-Collado, H1
Markó, M; Römer, D1
Amico, MC; Morrone, LA; Romanelli, L; Valeri, P1
Agmo, A; Contreras, JL; Paredes, RG1
Boersma, CJ; Pool, CW; Van Heerikhuize, JJ; Van Leeuwen, FW1
Howells, RD; Jin, J; Shahrestanifar, M; Wang, WW1
Cook, CD; Morgan, D; Negus, SS; Picker, MJ1
Kaputlu, I; Oğütman, C; Sadan, G1
Angel, F; Chevalier, E; Dahl, SG; Friese, N; Junien, JL; Pascaud, X; Riviere, PJ1
Fowler, CJ; Tiger, G1
Adams, DJ; Trequattrini, C1
Gioannini, TL; Hiller, JM; Onoprishvili, I; Simon, EJ1
Bakalkin, G; Derjabin, V; Hauser, KF; Nazarevskaja, G; Reznikov, K; Trunova, Y1
Ananthanarayanan, VS; Zhorov, BS1
Cheong, YP; Cho, KP; Kim, CJ; Kim, JK; Kim, KW; Kwun, J; Woo, RS1
Akil, H; Bonner, G; Meng, F1
Bandari, P; Chaturvedi, K; Chinen, N; Christoffers, KH; Dondio, G; Howells, RD; Jiang, X; Raveglia, LF; Ronzoni, S1
Chen, C; de Riel, JK; Huang, P; Javitch, JA; Li, J; Liu-Chen, LY; Xu, W1
Kuzmin, A; Ogren, SO; Sandin, J; Terenius, L1
Cancela, LM; del Rosario Capriles, N1
Ansonoff, M; Borsodi, A; Clarke, S; Czyzyk, T; Hill, R; Hsu, MS; Kitchen, I; Larsson, K; Nilsson, L; Nitsche, JF; Pintar, JE; Toth, G1
Azzi, M; Bouvier, M; deLéan, A; Piñeyro, G; Schiller, PW1
Dasher, WE; Klein, P; Nelson, WL1
Klein, P; Nelson, WL1
Klein, P; Nelson, WL; Olsen, LD; Simon, EJ; Yao, YH1
Klein, P; Nelson, WL; Simon, EJ; Yao, YH1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1

Other Studies

81 other study(ies) available for bremazocine and naloxone

ArticleYear
A highly selective kappa-opioid receptor agonist, CI-977, reduces excitatory synaptic potentials in the rat locus coeruleus in vitro.
    Neuroscience, 1992, Volume: 47, Issue:1

    Topics: Amino Acids; Analgesics; Animals; Benzofurans; Benzomorphans; Bicuculline; Depression, Chemical; Electric Stimulation; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; In Vitro Techniques; Ligands; Locus Coeruleus; Membrane Potentials; Naloxone; Naltrexone; Picrotoxin; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1992
Antidiuretic effect of bremazocine and U-50,488 in rats after alpha 2-adrenoceptor blockade.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Benzomorphans; Dioxanes; Diuresis; Dose-Response Relationship, Drug; Idazoxan; Male; Naloxone; Pyrrolidines; Rats; Rats, Inbred Strains; Yohimbine

1991
Differential cross-tolerance to mu and kappa opioid agonists in morphine-tolerant rats responding under a schedule of food presentation.
    Psychopharmacology, 1991, Volume: 103, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Chlorpromazine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Fentanyl; Food; Male; Methadone; Morphine; Naloxone; Narcotics; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule

1991
Inactivation of kappa opioid receptors by N-ethylmaleimide.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Benzomorphans; Brain; Dihydromorphine; Ethylmaleimide; In Vitro Techniques; Naloxone; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa

1990
Kappa-opioid receptor agonists differentially affect the release of neurohypophysial hormones.
    Pharmacology & toxicology, 1990, Volume: 66, Issue:3

    Topics: Animals; Benzeneacetamides; Benzomorphans; Electric Stimulation; Female; In Vitro Techniques; Naloxone; Nerve Endings; Oxytocin; Pituitary Hormones, Posterior; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vasopressins

1990
Effects of corticotropin-releasing factor (CRF) and opiates on amphibian locomotion.
    Brain research, 1990, Apr-09, Volume: 513, Issue:1

    Topics: Animals; Benzomorphans; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Locomotion; Male; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Salamandridae

1990
Mu-opiate receptor binding in the medial preoptic area is cyclical and sexually dimorphic.
    Brain research, 1990, May-07, Volume: 515, Issue:1-2

    Topics: Animals; Benzomorphans; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estrus; Female; Male; Naloxone; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Sex Characteristics

1990
Discriminative stimulus properties of U50,488 and morphine: effects of training dose on stimulus substitution patterns produced by mu and kappa opioid agonists.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Male; Methadone; Morphine; Naloxone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Opioid receptor-mediated inhibition of dopamine and acetylcholine release from slices of rat nucleus accumbens, olfactory tubercle and frontal cortex.
    European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Animals; Benzomorphans; Cerebral Cortex; Corpus Striatum; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ergolines; In Vitro Techniques; Male; Naloxone; Naltrexone; Nucleus Accumbens; Olfactory Bulb; Oxymetazoline; Pyrrolidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Opioid; Septal Nuclei

1990
Characterization of kappa-opioid receptors in the guinea-pig ileum.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Naloxone; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Thiophenes

1990
Evidence that bremazocine prevents urine retention induced by intraspinal cord injection of colchicine in rats.
    Journal of the autonomic nervous system, 1990, Volume: 30 Suppl

    Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Colchicine; Eledoisin; Hypertrophy; Injections, Spinal; Naloxone; Pyrrolidines; Rats; Receptors, Opioid; Spinal Cord; Urinary Bladder; Urination

1990
The effect of different opiates on acidified ethanol-induced gastric lesions in rats.
    Acta physiologica Hungarica, 1990, Volume: 75 Suppl

    Topics: Animals; Benzomorphans; Enkephalin, Methionine; Ethanol; Morphine; Naloxone; Narcotics; Rats; Stomach Ulcer

1990
Opioid binding properties of the purified kappa receptor from human placenta.
    Life sciences, 1989, Volume: 44, Issue:13

    Topics: Benzomorphans; Binding, Competitive; Chromatography; Cyclazocine; Electrophoresis, Polyacrylamide Gel; Ethylketocyclazocine; Etorphine; Humans; Molecular Weight; Naloxone; Narcotics; Placenta; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, kappa

1989
Lateralization of opioid receptors in turtle visual cortex.
    Brain research, 1989, Feb-20, Volume: 480, Issue:1-2

    Topics: Animals; Benzomorphans; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Evoked Potentials, Visual; Functional Laterality; Morphine; Naloxone; Receptors, Opioid; Turtles; Visual Cortex

1989
Opioids induce postural asymmetry in spinal rat: the side of the flexed limb depends upon the type of opioid agonist.
    Brain research, 1989, Feb-20, Volume: 480, Issue:1-2

    Topics: Animals; Benzomorphans; Decerebrate State; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Functional Laterality; Male; Muscles; Naloxone; Narcotics; Phenazocine; Posture; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord; Time Factors

1989
Kappa-opioid agonists do not inhibit adenylate cyclase.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclase Inhibitors; Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Cell Membrane; Enkephalin, Methionine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Levorphanol; Morphine; Naloxone; Pentazocine; Pyrrolidines; Rana catesbeiana; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride

1989
Diuretic effect of bremazocine, a kappa-opioid with central and peripheral sites of action.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Animals; Benzomorphans; Blood Pressure; Brain; Diuresis; Female; Glomerular Filtration Rate; Kidney; Kidney Concentrating Ability; Male; Morphinans; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Water-Electrolyte Balance

1989
Biphasic effect of a kappa-opioid receptor agonist on plasma oxytocin levels in rats.
    European journal of pharmacology, 1989, Jul-04, Volume: 166, Issue:1

    Topics: Analgesics; Animals; Benzomorphans; Body Water; Brain Chemistry; Female; In Vitro Techniques; Male; Morphinans; Naloxone; Oxytocin; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Time Factors

1989
Opiate control of spontaneous locomotor activity in a urodele amphibian.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 34, Issue:4

    Topics: Animals; Benzomorphans; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Morphinans; Motor Activity; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Salamandridae

1989
Discriminative stimulus effects of mu and kappa opioids in the pigeon: analysis of the effects of full and partial mu and kappa agonists.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Columbidae; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Morphinans; Naloxone; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1989
5-HT3 receptor binding sites are on capsaicin-sensitive fibres in the rat spinal cord.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Animals; Animals, Newborn; Antiemetics; Autoradiography; Benzamides; Benzomorphans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Male; Naloxone; Nerve Tissue Proteins; Neurons; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord

1989
Opioid kappa-receptor agonists suppress sexual behaviors in male rough-skinned newts (Taricha granulosa).
    Hormones and behavior, 1987, Volume: 21, Issue:3

    Topics: Analgesics; Animals; Benzomorphans; Cyclazocine; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Receptors, Opioid; Salamandridae; Sexual Behavior, Animal

1987
Interaction of U-69,593 with mu-, alpha- and kappa-opioid binding sites and its analgesic and intestinal effects in rats.
    Life sciences, 1988, Volume: 42, Issue:3

    Topics: Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Gastrointestinal Motility; In Vitro Techniques; Male; Naloxone; Nociceptors; Pyrrolidines; Rats; Receptors, Opioid

1988
Enhancement of [3H]DAGO1 binding to rat brain by low concentrations of monovalent cations.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:11

    Topics: Animals; Batrachotoxins; Benzomorphans; Brain Chemistry; Cations, Monovalent; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Naloxone; Rats; Receptors, Opioid; Temperature

1987
Effect of mu- and kappa-opioid agonists on the electroconvulsive seizure threshold in mice and antagonism by naloxone and MR 2266.
    Pharmacology & toxicology, 1988, Volume: 62, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzodiazepines; Benzomorphans; Electroshock; Fentanyl; Male; Mice; Morphinans; Morphine; Nalbuphine; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures

1988
Long-term blockade of mu-opioid receptors suggests a role in control of ingestive behaviour, body weight and core temperature in the rat.
    Brain research, 1988, May-31, Volume: 450, Issue:1-2

    Topics: Animals; Benzomorphans; Body Temperature Regulation; Body Weight; Circadian Rhythm; Drinking Behavior; Feeding Behavior; Fentanyl; Male; Naloxone; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Sufentanil

1988
Antagonist-induced opioid receptor up-regulation. II. Regionally specific modulation of mu, delta and kappa binding sites in rat brain revealed by quantitative autoradiography.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2

    Topics: Animals; Autoradiography; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Kinetics; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord; Substantia Nigra

1988
A novel series of potent and selective agonists at the opioid kappa-receptor.
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Mice; Morphinans; Muscle Contraction; Muscle, Smooth; Naloxone; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1988
Opposite effects of mu and kappa opiate agonists on dopamine release in the nucleus accumbens and in the dorsal caudate of freely moving rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Benzomorphans; Caudate Nucleus; Dopamine; Male; Methadone; Morphine; Motor Activity; Naloxone; Naltrexone; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reward; Septal Nuclei

1988
Na+ ions and Gpp(NH)p selectively inhibit agonist interactions at mu- and kappa-opioid receptor sites in rabbit and guinea-pig cerebellum membranes.
    European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzomorphans; Binding, Competitive; Cerebellum; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium

1985
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
Profile of activity of kappa receptor agonists in the rabbit vas deferens.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
The kappa opioid receptor and food intake.
    European journal of pharmacology, 1985, May-28, Volume: 112, Issue:1

    Topics: Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Diprenorphine; Eating; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Time Factors

1985
Effect of mu and kappa opioid receptor agonists on rat plasma corticosterone levels.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Corticosterone; Dose-Response Relationship, Drug; Fentanyl; Male; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Effects of tifluadom on food consumption compared with chlordiazepoxide and kappa agonists in the rat.
    Neuropharmacology, 1985, Volume: 24, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzodiazepinones; Benzomorphans; Chlordiazepoxide; Convulsants; Cyclazocine; Drug Interactions; Eating; Ethylketocyclazocine; Flumazenil; Male; Naloxone; Pyrazoles; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
Multiple opiate receptors may be involved in suppressing gamma-aminobutyrate release in substantia nigra.
    Life sciences, 1985, Dec-16, Volume: 37, Issue:24

    Topics: Aminooxyacetic Acid; Animals; Benzomorphans; Dopamine; Enkephalin, Methionine; Female; gamma-Aminobutyric Acid; Male; Naloxone; Nialamide; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Secretory Rate; Substantia Nigra

1985
Opioid kappa receptors and the secretion of prolactin (PRL) and growth hormone (GH) in the rat. I. Effects of opioid kappa receptor agonists bremazocine and U-50,488 on secretion of PRL and GH: comparison with morphine.
    Neuroendocrinology, 1986, Volume: 42, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Dose-Response Relationship, Drug; Growth Hormone; Injections, Intravenous; Male; Morphinans; Morphine; Naloxone; Prolactin; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Time Factors

1986
Bremazocine-induced backwards walking behavior in rats is mediated via opioid kappa receptors.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:4

    Topics: Animals; Benzomorphans; Brain; Hallucinogens; Locomotion; Male; Morphinans; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1986
Delineation of mu-antagonist, partial kappa agonist and non-opioid agonist activity of cyclazocine using urinary output of rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 26, Issue:4

    Topics: Animals; Benzomorphans; Cyclazocine; Diuresis; Dose-Response Relationship, Drug; Male; Morphine; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Water Deprivation

1987
[Effect of the opiate antagonist naloxone on the electrical activity of identified neurons in the edible snail].
    Nauchnye doklady vysshei shkoly. Biologicheskie nauki, 1987, Issue:6

    Topics: Animals; Benzomorphans; beta-Endorphin; Drug Interactions; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Helix, Snails; Membrane Potentials; Morphine; Naloxone; Neurons; Receptors, Opioid

1987
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule

1987
A novel phencyclidine analog interacts selectively with mu opioid receptors.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:2

    Topics: Analgesia; Animals; Benzomorphans; Binding, Competitive; Cerebellum; Dihydromorphine; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; Male; Mice; Muscle Contraction; Naloxone; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, mu; Vas Deferens

1984
[Binding sites of opiates and endogenous opioids in the oocytes of the toad Bufo viridis].
    Biokhimiia (Moscow, Russia), 1984, Volume: 49, Issue:6

    Topics: Animals; Benzomorphans; Binding Sites; Bufonidae; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Female; In Vitro Techniques; Kinetics; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Oocytes; Rabbits; Receptors, Opioid; Vas Deferens

1984
Kappa opioid agonists and antagonists: effects on drinking and urinary output.
    Appetite, 1984, Volume: 5, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Clonidine; Cyclazocine; Drinking; Ethylketocyclazocine; Naloxone; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Urination; Vasopressins

1984
Kappa-opiates and urination: pharmacological evidence for an endogenous role of the kappa-opiate receptor in fluid and electrolyte balance.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Female; Injections, Intraperitoneal; Morphinans; Morphine; Naloxone; Potassium; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium; Water-Electrolyte Balance

1984
Radioligands for probing opioid receptors.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Pro-Opiomelanocortin; Protein Precursors; Pyrrolidines; Radioligand Assay; Rats; Receptors, Opioid; Vas Deferens

1984
Further study of kappa opioids on increased urination.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Male; Morphinans; Naloxone; Narcotic Antagonists; Narcotics; Piperidines; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Urination

1983
Elevation of serum corticosterone in rats by bremazocine, a kappa-opioid agonist.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:5

    Topics: Animals; Benzomorphans; Corticosterone; Dose-Response Relationship, Drug; Male; Morphinans; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1984
Anatomical relationship between opioid peptides and receptors in rhesus monkey brain.
    Brain research bulletin, 1984, Volume: 13, Issue:6

    Topics: Animals; Benzomorphans; Brain; Brain Mapping; Dynorphins; Endorphins; Enkephalins; Macaca mulatta; Naloxone; Pro-Opiomelanocortin; Radioligand Assay; Receptors, Opioid; Synaptic Transmission

1984
Bremazocine: a potent, long-acting opiate kappa-agonist.
    Life sciences, 1980, Sep-15, Volume: 27, Issue:11

    Topics: Analgesia; Animals; Benzomorphans; Brain; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; Macaca mulatta; Male; Mice; Morphinans; Morphine; Naloxone; Pentazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1980
Effects of mu- and kappa-opioid receptor agonists on urinary output in mice.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:5

    Topics: Animals; Benzomorphans; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Male; Mice; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Species Specificity; Stimulation, Chemical; Urination

1983
Discriminative stimulus properties of nalorphine in the rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:3

    Topics: Animals; Benzodiazepines; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Macaca mulatta; Male; Nalorphine; Naloxone; Phenazocine; Receptors, Opioid; Receptors, Opioid, kappa

1983
A comparative study of the respiratory depressant and analgesic effects of bremazocine, a kappa-agonist.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Analgesia; Analgesics; Animals; Benzomorphans; Drug Antagonism; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Respiration

1983
Bremazocine induces antinociception, but prevents opioid-induced constipation and catatonia in rats and precipitates withdrawal in morphine-dependent rats.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Analgesics; Animals; Benzomorphans; Catatonia; Constipation; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Gastrointestinal Motility; Humans; Male; Morphinans; Morphine; Naloxone; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
Catatonic or hypotonic immobility induced in mice by intracerebroventricular injection of mu or kappa opioid receptor agonists as well as enkephalins or inhibitors of their degradation.
    Life sciences, 1983, Nov-21, Volume: 33, Issue:21

    Topics: Animals; Benzomorphans; Catatonia; Cyclazocine; Enkephalins; Ethylketocyclazocine; Fentanyl; Humans; Immobilization; Injections, Intraventricular; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics

1983
Inhibitory effect of a new opioid agonist on reproductive endocrine activity in rats of both sexes.
    Life sciences, 1983, Jul-18, Volume: 33, Issue:3

    Topics: Animals; Benzomorphans; Castration; Cells, Cultured; Female; In Vitro Techniques; Luteinizing Hormone; Male; Morphinans; Morphine; Naloxone; Ovulation; Pituitary Gland; Rats; Rats, Inbred Strains; Reproduction; Testis; Time Factors

1983
Acute withdrawal after bremazocine and the interaction between mu- and kappa-opioid receptors in isolated gut tissues.
    British journal of pharmacology, 1995, Volume: 114, Issue:6

    Topics: Animals; Benzomorphans; Guinea Pigs; In Vitro Techniques; Intestine, Small; Male; Morphine; Muscle Contraction; Naloxone; Rabbits; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance Withdrawal Syndrome

1995
Opioids and sexual behavior in the male rabbit: the role of central and peripheral opioid receptors.
    Journal of neural transmission. General section, 1994, Volume: 97, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Central Nervous System; Dose-Response Relationship, Drug; Ejaculation; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Loperamide; Male; Morphine; Naloxone; Narcotics; Oxymorphone; Peripheral Nervous System; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Sexual Behavior, Animal

1994
Characterization of opioid binding sites in the neural and intermediate lobe of the rat pituitary gland by quantitative receptor autoradiography.
    Journal of neuroendocrinology, 1994, Volume: 6, Issue:1

    Topics: Amino Acid Sequence; Analgesics; Animals; Autoradiography; Benzomorphans; Binding, Competitive; Densitometry; Enkephalins; Ligands; Male; Molecular Sequence Data; Naloxone; Naltrexone; Pituitary Gland; Pituitary Gland, Posterior; Protein Precursors; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, kappa

1994
Studies on mu and delta opioid receptor selectivity utilizing chimeric and site-mutagenized receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Dec-19, Volume: 92, Issue:26

    Topics: Amino Acid Sequence; Analgesics; Base Sequence; Benzomorphans; Binding, Competitive; Cell Line; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Etorphine; GTP-Binding Proteins; Humans; Kidney; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Naloxone; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Protein Structure, Secondary; Receptors, Opioid, delta; Receptors, Opioid, mu; Recombinant Fusion Proteins; Substrate Specificity; Transfection

1995
Effects of the delta opioid against BW373U86 in pigeons trained to discriminate fentanyl, bremazocine and water in a three-choice drug discrimination procedure.
    Psychopharmacology, 1996, Volume: 126, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Columbidae; Discrimination, Psychological; Female; Fentanyl; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Piperazines; Receptors, Opioid, delta

1996
Cardiovascular effects of intrathecally injected mu, delta and kappa opioid receptor agonists in rabbits.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:6

    Topics: Animals; Baroreflex; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Spinal; Naloxone; Narcotic Antagonists; Rabbits; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord

1995
Reversal by kappa-agonists of peritoneal irritation-induced ileus and visceral pain in rats.
    Life sciences, 1997, Volume: 60, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetic Acid; Analgesics; Animals; Benzofurans; Benzomorphans; Cyclazocine; Fentanyl; Gastric Emptying; Intestinal Pseudo-Obstruction; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Peritoneum; Pyrroles; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thiophenes

1997
Comparison of the effects of a series of kappa-opioid receptor agonists upon sodium channel function in rat brain miniprisms.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1997, Volume: 117, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzeneacetamides; Benzomorphans; Brain; Disease Models, Animal; Inositol Phosphates; Naloxone; Pyrrolidines; Rats; Receptors, Opioid, kappa; Sodium Channels

1997
Opioid receptor-mediated inhibition of omega-conotoxin GVIA-sensitive calcium channel currents in rat intracardiac neurons.
    Journal of neurophysiology, 1998, Volume: 79, Issue:2

    Topics: Acetylcholine; Animals; Animals, Newborn; Anti-Arrhythmia Agents; Benzomorphans; Calcium; Calcium Channels; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Heart Conduction System; Ion Channel Gating; Ion Transport; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; omega-Conotoxin GVIA; Parasympathetic Nervous System; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Virulence Factors, Bordetella

1998
Inactivation of the purified bovine mu opioid receptor by sulfhydryl reagents.
    Neurochemical research, 1999, Volume: 24, Issue:1

    Topics: Animals; Benzomorphans; Cattle; Cell Membrane; Corpus Striatum; Cysteine; Dithionitrobenzoic Acid; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylmaleimide; Kinetics; Ligands; Naloxone; Radioligand Assay; Receptors, Opioid, mu; Sulfhydryl Reagents; Tritium

1999
Opioids modulate cell division in the germinal zone of the late embryonic neocortex.
    The European journal of neuroscience, 1999, Volume: 11, Issue:8

    Topics: Animals; Benzomorphans; Cell Division; Cerebral Ventricles; Embryo, Mammalian; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Female; Mice; Mice, Inbred CBA; Mitotic Index; Naloxone; Narcotic Antagonists; Narcotics; Neocortex; Pregnancy; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1999
Homology models of mu-opioid receptor with organic and inorganic cations at conserved aspartates in the second and third transmembrane domains.
    Archives of biochemistry and biophysics, 2000, Mar-01, Volume: 375, Issue:1

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Aspartic Acid; Benzomorphans; Binding Sites; Cations; Cattle; Computer Simulation; Conserved Sequence; Fentanyl; Humans; Ligands; Metals; Models, Molecular; Molecular Sequence Data; Morphine; Naloxone; Narcotic Antagonists; Protein Binding; Protein Structure, Tertiary; Rats; Receptors, Opioid, mu; Sequence Alignment; Sequence Homology, Amino Acid; Structure-Activity Relationship

2000
Receptor selectivity of Met-enkephalin-Arg6-Phe7, an endogenous opioid peptide, in cerebral cortex of human and rat.
    Life sciences, 2000, May-26, Volume: 67, Issue:1

    Topics: Adult; Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Ethylketocyclazocine; Female; Humans; Male; Naloxone; Naltrexone; Norepinephrine; Oligopeptides; Peptide Fragments; Peptides; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Somatostatin

2000
Selectivity of mu-opioid receptor determined by interfacial residues near third extracellular loop.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Amino Acid Substitution; Animals; Benzamides; Benzomorphans; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Morphine; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Peptides; Piperazines; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid, mu; Signal Transduction; Sulfur Radioisotopes

2000
Pharmacological profiles of selective non-peptidic delta opioid receptor ligands.
    Brain research. Molecular brain research, 2000, Sep-15, Volume: 80, Issue:2

    Topics: Amino Acid Sequence; Analgesics; Analgesics, Opioid; Benzomorphans; Binding, Competitive; Cells, Cultured; Cloning, Molecular; Down-Regulation; Enkephalin, Leucine-2-Alanine; GTP-Binding Proteins; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Isoquinolines; Kidney; Ligands; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Morphine; Mutagenesis, Site-Directed; Naloxone; Narcotic Antagonists; Quinolines; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, mu; Tritium

2000
The conserved cysteine 7.38 residue is differentially accessible in the binding-site crevices of the mu, delta, and kappa opioid receptors.
    Biochemistry, 2000, Nov-14, Volume: 39, Issue:45

    Topics: Amino Acid Sequence; Animals; Benzomorphans; Binding Sites; Cell Line; Conserved Sequence; Cysteine; Diprenorphine; Dose-Response Relationship, Drug; Ethyl Methanesulfonate; Glutamic Acid; Humans; Indicators and Reagents; Mesylates; Methionine; Molecular Sequence Data; Mutagenesis, Site-Directed; Naloxone; Narcotic Antagonists; Protein Structure, Secondary; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serine; Time Factors; Tritium

2000
Dose- and time-dependent bimodal effects of kappa-opioid agonists on locomotor activity in mice.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetamides; Animals; Benzomorphans; Dose-Response Relationship, Drug; Isothiocyanates; Male; Mice; Morphine; Motor Activity; Naloxone; Naltrexone; Receptors, Opioid, kappa; Time Factors

2000
Motivational effects mu- and kappa-opioid agonists following acute and chronic restraint stress: involvement of dopamine D(1) and D(2) receptors.
    Behavioural brain research, 2002, May-14, Volume: 132, Issue:2

    Topics: Acute Disease; Animals; Behavior, Animal; Benzomorphans; Chronic Disease; Conditioning, Operant; Injections, Intraventricular; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stress, Psychological

2002
Autoradiography of opioid and ORL1 ligands in opioid receptor triple knockout mice.
    The European journal of neuroscience, 2002, Volume: 16, Issue:9

    Topics: Animals; Autoradiography; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Mice; Mice, Knockout; Naloxone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid; Spinal Cord; Vasodilator Agents

2002
Reciprocal regulation of agonist and inverse agonist signaling efficacy upon short-term treatment of the human delta-opioid receptor with an inverse agonist.
    Molecular pharmacology, 2005, Volume: 67, Issue:1

    Topics: Benzomorphans; Binding Sites; Cell Line; Cell Membrane; Cyclic AMP; Cycloheximide; DNA, Complementary; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kinetics; Naloxone; Phosphorylation; Receptors, Opioid, delta; Recombinant Proteins; Transfection

2005
Electrophilic opioid ligands. Oxygen tethered alpha-methylene-gamma-lactone, acrylate, isothiocyanate, and epoxide derivatives of 6 beta-naltrexol.
    Journal of medicinal chemistry, 1992, Jun-26, Volume: 35, Issue:13

    Topics: Acrylates; Animals; Binding Sites; Brain; Endorphins; Epoxy Compounds; Guinea Pigs; Lactones; Ligands; Naltrexone; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stereoisomerism; Thiocyanates

1992
O3-(2-carbomethoxyallyl) ethers of opioid ligands derived from oxymorphone, naltrexone, etorphine, diprenorphine, norbinaltorphimine, and naltrindole. Unexpected O3-dealkylation in the opioid radioligand displacement assay.
    Journal of medicinal chemistry, 1992, Nov-27, Volume: 35, Issue:24

    Topics: Alkylation; Animals; Brain; Diprenorphine; Drug Stability; Ethers; Etorphine; Guinea Pigs; Indoles; Methacrylates; Molecular Structure; Morphinans; Naltrexone; Narcotic Antagonists; Narcotics; Oxymorphone; Phenols; Radioligand Assay; Receptors, Opioid; Tritium

1992
Conjugate addition ligands of opioid antagonists. Methacrylate esters and ethers of 6 alpha- and 6 beta-naltrexol.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:2

    Topics: Animals; Benzomorphans; Binding, Competitive; Cattle; Caudate Nucleus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Esters; Ethers; In Vitro Techniques; Ligands; Methacrylates; Naltrexone; Receptors, Opioid; Structure-Activity Relationship

1990
Electrophilic alpha-methylene-gamma-lactone and isothiocyanate opioid ligands related to etorphine.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:8

    Topics: Chemical Phenomena; Chemistry; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Isothiocyanates; Lactones; Ligands; Magnetic Resonance Spectroscopy; Molecular Structure; Morphinans; Naloxone; Receptors, Opioid; Receptors, Opioid, mu; Spectrophotometry, Infrared; Stereoisomerism; Thebaine; Thiocyanates

1990
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011