bremazocine and morphine

bremazocine has been researched along with morphine in 74 studies

Research

Studies (74)

TimeframeStudies, this research(%)All Research%
pre-199040 (54.05)18.7374
1990's23 (31.08)18.2507
2000's7 (9.46)29.6817
2010's4 (5.41)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujii, H; Hasebe, K; Izumimoto, N; Mochizuki, H; Momen, S; Nagase, H; Nakajima, R; Nemoto, T; Yamamoto, N1
Craft, RM; Dykstra, LA2
al-Shireida, MF; el-Sharkawy, TY; Pilcher, CW1
Muraki, T; Nomoto, T; Oike, N; Shibata, Y1
Buydens, P; Finné, E; Govaerts, J; Matton, A; Vanhaelst, L1
Negus, SS; Picker, MJ; Powell, KR1
Dykstra, LA; Negus, SS; Picker, MJ2
Deviche, P; Lowry, CA; Moore, FL1
Doty, P; Dykstra, LA; Mattox, SR; Negus, SS; Picker, MJ1
Craft, RM; Negus, SS; Picker, MJ1
Coombes, JE; Pumford, KM; Russell, JA; Sumner, BE1
Gyires, K1
Bergman, J; Warren, PH1
Kobylyansky, AG; Nesterenko, PN; Pivovarov, AS; Yarygin, KN1
Brady, LS; Bykov, V; Holaday, JW; Jacobson, AE; Long, JB; Rice, KC; Rothman, RB1
Craft, RM; Dykstra, LA; Picker, MJ1
Makimura, M; Murakoshi, Y1
Huidobro-Toro, JP; Roblero, J; Salas, SP; Ureta, H1
Bhargava, HN; Ramarao, P1
Deviche, P; Moore, FL1
Frey, HH1
Bhargava, HN; Jablonski, HI; Ramarao, P; Rehder, KR1
Di Chiara, G; Imperato, A1
Cooper, SJ; Jackson, A; Kirkham, TC1
Ishihara, K; Iwama, T; Satoh, M; Takagi, H1
Schmauss, C1
Burks, TF; Hirning, LD; Porreca, F1
Grace, M; Kneip, J; Levine, AS; Morley, JE; Shearman, GT; Zeugner, H1
Hayes, AG; Stewart, BR1
Cooper, SJ; Jackson, A1
Conway, S; Koenig, JI; Krulich, L; Mayfield, MA; McCann, SM2
Ignatov, IuD; Zaĭtsev, AA1
Leander, JD1
Bakalkin, GIa; Pivovarov, AS; Romanenko, OK1
Dykstra, LA; Gmerek, DE; Winger, G; Woods, JH1
Dykstra, LA; Heise, JW; Picker, M1
Morozova, AS; Patkina, NA; Zvartau, EE1
Bakalkin, GIa; Bespalova, ZhD; Iakovleva, TV; Korobov, KP; Vinogradov, VA1
Huidobro-Toro, JP; Parada, S1
Goodman, RR; Snyder, SH1
Hayes, AG; Skingle, M; Tyers, MB1
Burkard, WP; Flück, N; Müller, PM1
Akkerman, AM; Bakel, HC; Büscher, H; Hill, RC; Maurer, R; Petcher, TJ; Römer, D; Welle, HB1
Dzoljic, MR; van der Poel-Heisterkamp, AL1
Iwamoto, ET; Martin, WR1
Kattau, RW; Leander, JD; Rathbun, RC1
Ramabadran, K1
Gambino, MC; Petrillo, P; Tavani, A1
Chaillet, P; Costentin, J; Marçais-Collado, H1
Markó, M; Römer, D1
Amico, MC; Morrone, LA; Romanelli, L; Valeri, P1
Alsasua, A; Martín, MI; Parra, L; Pérez-Vizcaíno, F; Tamargo, J1
Alfaro, MJ; Goicoechea, C; Lopez, F; Martin, MI; Ormazabal, MJ1
Agmo, A; Contreras, JL; Paredes, RG1
Nishiyama, N; Schwartz, JP; Taniwaki, T; Wilson, D1
Collins, KA; Tseng, LF1
Chang, KJ; Comer, SD; De Costa, BR; McNutt, RW; Mosberg, HI; Woods, JH1
Morgan, D; Picker, MJ1
Cook, CD; Morgan, D; Negus, SS; Picker, MJ1
Angel, F; Chevalier, E; Dahl, SG; Friese, N; Junien, JL; Pascaud, X; Riviere, PJ1
Picker, MJ1
Ananthanarayanan, VS; Zhorov, BS1
Akil, H; Bonner, G; Meng, F1
Bandari, P; Chaturvedi, K; Chinen, N; Christoffers, KH; Dondio, G; Howells, RD; Jiang, X; Raveglia, LF; Ronzoni, S1
Kuzmin, A; Ogren, SO; Sandin, J; Terenius, L1
Cancela, LM; del Rosario Capriles, N1
da Fonseca Pacheco, CM; da Fonseca Pacheco, D; de Castro Perez, A; de Francischi, JN; Duarte, ID; Klein, A1
Husbands, SM; Ko, MC1
Chen, G; Goddard, WA; Kim, SK; Li, Q; Tan, H1
Fujii, H; Hirono, S; Nagase, H; Yamaotsu, N1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1

Reviews

2 review(s) available for bremazocine and morphine

ArticleYear
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response

1985
Multiple opioid receptors.
    Medicinal research reviews, 1981,Winter, Volume: 1, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Benzomorphans; Cyclazocine; Discrimination Learning; Dogs; Dopamine; Drug Tolerance; Electroencephalography; Humans; Macaca mulatta; Mice; Morphine; Morphine Dependence; Motor Activity; Nalorphine; Pain; Rabbits; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, kappa; Seizures; Temperature

1981

Other Studies

72 other study(ies) available for bremazocine and morphine

ArticleYear
Synthesis of new opioid derivatives with a propellane skeleton and their pharmacology: part 1.
    Bioorganic & medicinal chemistry letters, 2011, Jul-01, Volume: 21, Issue:13

    Topics: Analgesics, Opioid; Animals; Bridged-Ring Compounds; Cells, Cultured; Mice; Molecular Structure; Protein Binding; Receptors, Opioid, kappa; Structure-Activity Relationship; Substrate Specificity

2011
Agonist and antagonist activity of kappa opioids in the squirrel monkey: I. Antinociception and urine output.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Benzodiazepines; Benzomorphans; Drug Interactions; Ethylketocyclazocine; Male; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptors; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Urination

1992
Agonist and antagonist activity of kappa opioids in the squirrel monkey: II. Effect of chronic morphine treatment.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Drug Interactions; Drug Tolerance; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptors; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Saimiri; Shock; Time Factors

1992
Vascular effects of some opioid receptor agonists.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Calcium Channel Blockers; Dinoprost; Endothelium, Vascular; Ethylketocyclazocine; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Narcotic Antagonists; Norepinephrine; Potassium; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Vasodilation

1991
Analgesic effect of mu- and kappa-opioid agonists in beige and CXBK mice.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetates; Acetic Acid; Analgesics; Animals; Benzodiazepines; Benzomorphans; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Female; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Morphine; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1991
Analysis of the receptor specificity of tolerance induction in stress versus opioid-related prolactin secretion in rats.
    The Journal of endocrinology, 1991, Volume: 128, Issue:2

    Topics: Animals; Benzomorphans; Dose-Response Relationship, Drug; Drug Tolerance; Haloperidol; Male; Morphine; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid; Stress, Psychological

1991
Differential cross-tolerance to mu and kappa opioid agonists in morphine-tolerant rats responding under a schedule of food presentation.
    Psychopharmacology, 1991, Volume: 103, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Chlorpromazine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Fentanyl; Food; Male; Methadone; Morphine; Naloxone; Narcotics; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule

1991
Interactions between mu and kappa opioid agonists in the rat drug discrimination procedure.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Buprenorphine; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Fentanyl; Male; Morphine; Pentobarbital; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Effects of corticotropin-releasing factor (CRF) and opiates on amphibian locomotion.
    Brain research, 1990, Apr-09, Volume: 513, Issue:1

    Topics: Animals; Benzomorphans; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Locomotion; Male; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Salamandridae

1990
Discriminative stimulus properties of U50,488 and morphine: effects of training dose on stimulus substitution patterns produced by mu and kappa opioid agonists.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Male; Methadone; Morphine; Naloxone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Butorphanol's efficacy at mu and kappa opioid receptors: inferences based on the schedule-controlled behavior of nontolerant and morphine-tolerant rats and on the responding of rats under a drug discrimination procedure.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:3

    Topics: Analgesics; Animals; Behavior, Animal; Benzomorphans; Butorphanol; Discrimination, Psychological; Drug Tolerance; Male; Morphinans; Morphine; Narcotic Antagonists; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reinforcement Schedule

1990
Opioid receptor subtypes in the supraoptic nucleus and posterior pituitary gland of morphine-tolerant rats.
    Neuroscience, 1990, Volume: 37, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Autoradiography; Benzomorphans; Binding, Competitive; Drug Tolerance; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; Female; Injections, Intraventricular; Morphine; Pituitary Gland, Posterior; Plasma; Preoptic Area; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Supraoptic Nucleus

1990
The effect of different opiates on acidified ethanol-induced gastric lesions in rats.
    Acta physiologica Hungarica, 1990, Volume: 75 Suppl

    Topics: Animals; Benzomorphans; Enkephalin, Methionine; Ethanol; Morphine; Naloxone; Narcotics; Rats; Stomach Ulcer

1990
Effects of kappa opioids on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Conditioning, Psychological; Dose-Response Relationship, Drug; Electroshock; Male; Morphinans; Morphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Saimiri

1989
Lateralization of opioid receptors in turtle visual cortex.
    Brain research, 1989, Feb-20, Volume: 480, Issue:1-2

    Topics: Animals; Benzomorphans; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Evoked Potentials, Visual; Functional Laterality; Morphine; Naloxone; Receptors, Opioid; Turtles; Visual Cortex

1989
Chronic administration of morphine and naltrexone up-regulate mu-opioid binding sites labeled by [3H][D-Ala2,MePhe4,Gly-ol5]enkephalin: further evidence for two mu-binding sites.
    European journal of pharmacology, 1989, Jan-24, Volume: 160, Issue:1

    Topics: Animals; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; In Vitro Techniques; Male; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1989
Differential cross-tolerance to opioid agonists in morphine-tolerant pigeons responding under a schedule of food presentation.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Chlorpromazine; Columbidae; Conditioning, Operant; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Female; Morphine; Pyrrolidines; Receptors, Opioid

1989
Kappa antagonist properties of buprenorphine in non-tolerant and morphine-tolerant rats.
    Psychopharmacology, 1989, Volume: 98, Issue:1

    Topics: Animals; Behavior, Animal; Benzomorphans; Buprenorphine; Dose-Response Relationship, Drug; Drug Tolerance; Male; Morphine; Narcotic Antagonists; Rats; Receptors, Opioid, kappa; Reinforcement Schedule

1989
Kappa-opioid agonists do not inhibit adenylate cyclase.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclase Inhibitors; Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Cell Membrane; Enkephalin, Methionine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Levorphanol; Morphine; Naloxone; Pentazocine; Pyrrolidines; Rana catesbeiana; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride

1989
Diuretic effect of bremazocine, a kappa-opioid with central and peripheral sites of action.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Animals; Benzomorphans; Blood Pressure; Brain; Diuresis; Female; Glomerular Filtration Rate; Kidney; Kidney Concentrating Ability; Male; Morphinans; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Water-Electrolyte Balance

1989
Effects of kappa-opioid receptor agonists and morphine on food intake and urinary output in food-deprived and nondeprived rats.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Dose-Response Relationship, Drug; Feeding Behavior; Food Deprivation; Male; Morphine; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Time Factors; Urination

1989
Opioid kappa-receptor agonists suppress sexual behaviors in male rough-skinned newts (Taricha granulosa).
    Hormones and behavior, 1987, Volume: 21, Issue:3

    Topics: Analgesics; Animals; Benzomorphans; Cyclazocine; Ethylketocyclazocine; Male; Morphinans; Morphine; Naloxone; Receptors, Opioid; Salamandridae; Sexual Behavior, Animal

1987
Effect of mu- and kappa-opioid agonists on the electroconvulsive seizure threshold in mice and antagonism by naloxone and MR 2266.
    Pharmacology & toxicology, 1988, Volume: 62, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzodiazepines; Benzomorphans; Electroshock; Fentanyl; Male; Mice; Morphinans; Morphine; Nalbuphine; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures

1988
Effect of kappa-opioid receptor agonists on morphine analgesia in morphine-naive and morphine-tolerant rats.
    European journal of pharmacology, 1988, Nov-01, Volume: 156, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Male; Morphine; Narcotic Antagonists; Pain Measurement; Pyrrolidines; Rats; Rats, Inbred Strains; Tail

1988
Opposite effects of mu and kappa opiate agonists on dopamine release in the nucleus accumbens and in the dorsal caudate of freely moving rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Benzomorphans; Caudate Nucleus; Dopamine; Male; Methadone; Morphine; Motor Activity; Naloxone; Naltrexone; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reward; Septal Nuclei

1988
Different effects of dynorphin A on in vitro guinea pig hippocampal CA3 pyramidal cells with various degrees of paired-pulse facilitation.
    Neuroscience letters, 1986, Jan-16, Volume: 63, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Drug Interactions; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Morphine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptic Transmission

1986
Spinal kappa-opioid receptor-mediated antinociception is stimulus-specific.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Dynorphins; Ethylketocyclazocine; Injections, Spinal; Male; Morphine; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord

1987
Mu, but not kappa, opioid agonists induce contractions of the canine small intestine ex vivo.
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Dimethylphenylpiperazinium Iodide; Dogs; Ethylketocyclazocine; Gastrointestinal Motility; In Vitro Techniques; Intestine, Small; Morphine; Nalorphine; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
The kappa opioid receptor and food intake.
    European journal of pharmacology, 1985, May-28, Volume: 112, Issue:1

    Topics: Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Diprenorphine; Eating; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Time Factors

1985
Effect of mu and kappa opioid receptor agonists on rat plasma corticosterone levels.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Corticosterone; Dose-Response Relationship, Drug; Fentanyl; Male; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Effects of kappa opiate agonists on palatable food consumption in non-deprived rats, with and without food preloads.
    Brain research bulletin, 1985, Volume: 15, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Eating; Ethylketocyclazocine; Male; Morphine; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Satiety Response

1985
Opioid kappa receptors and the secretion of prolactin (PRL) and growth hormone (GH) in the rat. I. Effects of opioid kappa receptor agonists bremazocine and U-50,488 on secretion of PRL and GH: comparison with morphine.
    Neuroendocrinology, 1986, Volume: 42, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Dose-Response Relationship, Drug; Growth Hormone; Injections, Intravenous; Male; Morphinans; Morphine; Naloxone; Prolactin; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Time Factors

1986
Opioid kappa receptors and the secretion of prolactin (PRL) and growth hormone (GH) in the rat. II. GH and PRL release-inhibiting effects of the opioid kappa receptor agonists bremazocine and U-50,488.
    Neuroendocrinology, 1986, Volume: 42, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Clonidine; Growth Hormone; Injections, Intravenous; Male; Morphinans; Morphine; Prolactin; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Serotonin; Time Factors

1986
[The role of various opiate receptors in the regulation of the nociceptive reaction of the arterial pressure].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 103, Issue:4

    Topics: Animals; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Hemodynamics; Morphine; Nociceptors; Rats; Receptors, Opioid

1987
Delineation of mu-antagonist, partial kappa agonist and non-opioid agonist activity of cyclazocine using urinary output of rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 26, Issue:4

    Topics: Animals; Benzomorphans; Cyclazocine; Diuresis; Dose-Response Relationship, Drug; Male; Morphine; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Water Deprivation

1987
[Effect of the opiate antagonist naloxone on the electrical activity of identified neurons in the edible snail].
    Nauchnye doklady vysshei shkoly. Biologicheskie nauki, 1987, Issue:6

    Topics: Animals; Benzomorphans; beta-Endorphin; Drug Interactions; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Helix, Snails; Membrane Potentials; Morphine; Naloxone; Neurons; Receptors, Opioid

1987
Kappa opioids in rhesus monkeys. II. Analysis of the antagonistic actions of quadazocine and beta-funaltrexamine.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Azocines; Benzomorphans; Cyclazocine; Diuresis; Endorphins; Ethylketocyclazocine; Female; Hot Temperature; Macaca mulatta; Male; Morphine; Naltrexone; Narcotic Antagonists; Pyrrolidines; Reaction Time; Tail

1987
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule

1987
[Reinforcing, but no analgesic, effect of opioid stimulation of the ventral tegmental area].
    Biulleten' eksperimental'noi biologii i meditsiny, 1986, Volume: 102, Issue:8

    Topics: Analgesics; Animals; Benzomorphans; Male; Morphine; Phencyclidine; Rats; Reinforcement, Psychology; Tegmentum Mesencephali

1986
[Binding sites of opiates and endogenous opioids in the oocytes of the toad Bufo viridis].
    Biokhimiia (Moscow, Russia), 1984, Volume: 49, Issue:6

    Topics: Animals; Benzomorphans; Binding Sites; Bufonidae; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Female; In Vitro Techniques; Kinetics; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Oocytes; Rabbits; Receptors, Opioid; Vas Deferens

1984
Kappa-opiates and urination: pharmacological evidence for an endogenous role of the kappa-opiate receptor in fluid and electrolyte balance.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Female; Injections, Intraperitoneal; Morphinans; Morphine; Naloxone; Potassium; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium; Water-Electrolyte Balance

1984
Kappa opiate receptors localized by autoradiography to deep layers of cerebral cortex: relation to sedative effects.
    Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:18

    Topics: Analgesics; Analgesics, Opioid; Animals; Autoradiography; Benzomorphans; Brain Stem; Cerebral Cortex; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Morphine; Organ Specificity; Receptors, Opioid; Receptors, Opioid, kappa; Tritium

1982
Antinociceptive profile of dynorphin in the rat.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Analgesics; Animals; Benzomorphans; Dynorphins; Endorphins; Male; Morphine; Nociceptors; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1983
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid

1984
Bremazocine: a potent, long-acting opiate kappa-agonist.
    Life sciences, 1980, Sep-15, Volume: 27, Issue:11

    Topics: Analgesia; Animals; Benzomorphans; Brain; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; Macaca mulatta; Male; Mice; Morphinans; Morphine; Naloxone; Pentazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1980
Delta opiate receptors are involved in the endopioid-induced myoclonic contractions.
    Brain research bulletin, 1982, Volume: 8, Issue:1

    Topics: Analgesics; Animals; Benzomorphans; Endorphins; Enkephalins; Female; Male; Morphine; Muscle Contraction; Myoclonus; Rats; Rats, Inbred Strains; Receptors, Opioid

1982
Effects of mu- and kappa-opioid receptor agonists on urinary output in mice.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:5

    Topics: Animals; Benzomorphans; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Male; Mice; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Species Specificity; Stimulation, Chemical; Urination

1983
Hyperalgesic effect of the selective kappa opioid agonist, U-50488H in mice.
    Japanese journal of pharmacology, 1983, Volume: 33, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Male; Mice; Morphine; Nociceptors; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1983
Bremazocine induces antinociception, but prevents opioid-induced constipation and catatonia in rats and precipitates withdrawal in morphine-dependent rats.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Analgesics; Animals; Benzomorphans; Catatonia; Constipation; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Gastrointestinal Motility; Humans; Male; Morphinans; Morphine; Naloxone; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
Catatonic or hypotonic immobility induced in mice by intracerebroventricular injection of mu or kappa opioid receptor agonists as well as enkephalins or inhibitors of their degradation.
    Life sciences, 1983, Nov-21, Volume: 33, Issue:21

    Topics: Animals; Benzomorphans; Catatonia; Cyclazocine; Enkephalins; Ethylketocyclazocine; Fentanyl; Humans; Immobilization; Injections, Intraventricular; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics

1983
Inhibitory effect of a new opioid agonist on reproductive endocrine activity in rats of both sexes.
    Life sciences, 1983, Jul-18, Volume: 33, Issue:3

    Topics: Animals; Benzomorphans; Castration; Cells, Cultured; Female; In Vitro Techniques; Luteinizing Hormone; Male; Morphinans; Morphine; Naloxone; Ovulation; Pituitary Gland; Rats; Rats, Inbred Strains; Reproduction; Testis; Time Factors

1983
Acute withdrawal after bremazocine and the interaction between mu- and kappa-opioid receptors in isolated gut tissues.
    British journal of pharmacology, 1995, Volume: 114, Issue:6

    Topics: Animals; Benzomorphans; Guinea Pigs; In Vitro Techniques; Intestine, Small; Male; Morphine; Muscle Contraction; Naloxone; Rabbits; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance Withdrawal Syndrome

1995
mu- and delta-opioid receptor-mediated contractile effects on rat aortic vascular smooth muscle.
    European journal of pharmacology, 1995, Apr-13, Volume: 277, Issue:1

    Topics: Amino Acid Sequence; Analgesics; Analysis of Variance; Animals; Aorta; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Molecular Sequence Data; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Naltrexone; Norepinephrine; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu

1995
Analgesic effect of two calcitonins and in vitro interaction with opioids.
    General pharmacology, 1995, Volume: 26, Issue:3

    Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Dose-Response Relationship, Drug; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guinea Pigs; In Vitro Techniques; Male; Mice; Morphine; Muscle Contraction; Muscle, Smooth; Narcotics; Pain Measurement; Pain Threshold; Rabbits; Rats; Rats, Wistar

1995
Opioids and sexual behavior in the male rabbit: the role of central and peripheral opioid receptors.
    Journal of neural transmission. General section, 1994, Volume: 97, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Central Nervous System; Dose-Response Relationship, Drug; Ejaculation; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Loperamide; Male; Morphine; Naloxone; Narcotics; Oxymorphone; Peripheral Nervous System; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Sexual Behavior, Animal

1994
Receptor-mediated regulation of neuropeptide gene expression in astrocytes.
    Glia, 1994, Volume: 11, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Benzomorphans; Brain; Enkephalin, Methionine; Etorphine; Gene Expression Regulation; Morphine; Naltrexone; Nerve Tissue Proteins; Neuropeptides; Organ Specificity; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Opioid

1994
Spinal involvement of both dynorphin A and Met-enkephalin in the antinociception induced by intracerebroventricularly administered bremazocine but not morphine in the mouse.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Benzomorphans; beta-Endorphin; Drug Interactions; Dynorphins; Enkephalin, Leucine; Enkephalin, Methionine; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphine; Nociceptors; Pain Measurement; Pyrrolidines; Spinal Cord; Time Factors

1993
Discriminative stimulus effects of BW373U86: a nonpeptide ligand with selectivity for delta opioid receptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Amino Acid Sequence; Analgesics; Animals; Benzamides; Benzomorphans; Columbidae; Discrimination Learning; Enkephalin, Leucine; Molecular Sequence Data; Morphine; Naltrexone; Narcotic Antagonists; Piperazines; Receptors, Opioid, delta; Receptors, Opioid, mu

1993
Discriminative stimulus effects of the 5HT1A agonist 8-OH-DPAT: attenuation by mu but not by kappa opioids.
    Psychopharmacology, 1995, Volume: 122, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Benzomorphans; Discrimination Learning; Drug Therapy, Combination; Fentanyl; Male; Morphine; Narcotics; Pyrimidines; Pyrrolidines; Rats; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin Receptor Agonists

1995
Effects of the delta opioid against BW373U86 in pigeons trained to discriminate fentanyl, bremazocine and water in a three-choice drug discrimination procedure.
    Psychopharmacology, 1996, Volume: 126, Issue:3

    Topics: Analgesics; Animals; Benzamides; Benzomorphans; Columbidae; Discrimination, Psychological; Female; Fentanyl; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Piperazines; Receptors, Opioid, delta

1996
Reversal by kappa-agonists of peritoneal irritation-induced ileus and visceral pain in rats.
    Life sciences, 1997, Volume: 60, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetic Acid; Analgesics; Animals; Benzofurans; Benzomorphans; Cyclazocine; Fentanyl; Gastric Emptying; Intestinal Pseudo-Obstruction; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Peritoneum; Pyrroles; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thiophenes

1997
Drug discrimination history: pigeons trained to discriminate opioids with activity at different receptor types.
    Experimental and clinical psychopharmacology, 1998, Volume: 6, Issue:2

    Topics: Animals; Benzomorphans; Butorphanol; Discrimination Learning; Dose-Response Relationship, Drug; Female; Fentanyl; Guinea Pigs; Morphine; Narcotics; Receptors, Opioid

1998
Homology models of mu-opioid receptor with organic and inorganic cations at conserved aspartates in the second and third transmembrane domains.
    Archives of biochemistry and biophysics, 2000, Mar-01, Volume: 375, Issue:1

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Aspartic Acid; Benzomorphans; Binding Sites; Cations; Cattle; Computer Simulation; Conserved Sequence; Fentanyl; Humans; Ligands; Metals; Models, Molecular; Molecular Sequence Data; Morphine; Naloxone; Narcotic Antagonists; Protein Binding; Protein Structure, Tertiary; Rats; Receptors, Opioid, mu; Sequence Alignment; Sequence Homology, Amino Acid; Structure-Activity Relationship

2000
Selectivity of mu-opioid receptor determined by interfacial residues near third extracellular loop.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Amino Acid Substitution; Animals; Benzamides; Benzomorphans; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Morphine; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Peptides; Piperazines; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid, mu; Signal Transduction; Sulfur Radioisotopes

2000
Pharmacological profiles of selective non-peptidic delta opioid receptor ligands.
    Brain research. Molecular brain research, 2000, Sep-15, Volume: 80, Issue:2

    Topics: Amino Acid Sequence; Analgesics; Analgesics, Opioid; Benzomorphans; Binding, Competitive; Cells, Cultured; Cloning, Molecular; Down-Regulation; Enkephalin, Leucine-2-Alanine; GTP-Binding Proteins; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Isoquinolines; Kidney; Ligands; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Morphine; Mutagenesis, Site-Directed; Naloxone; Narcotic Antagonists; Quinolines; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, mu; Tritium

2000
Dose- and time-dependent bimodal effects of kappa-opioid agonists on locomotor activity in mice.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetamides; Animals; Benzomorphans; Dose-Response Relationship, Drug; Isothiocyanates; Male; Mice; Morphine; Motor Activity; Naloxone; Naltrexone; Receptors, Opioid, kappa; Time Factors

2000
Motivational effects mu- and kappa-opioid agonists following acute and chronic restraint stress: involvement of dopamine D(1) and D(2) receptors.
    Behavioural brain research, 2002, May-14, Volume: 132, Issue:2

    Topics: Acute Disease; Animals; Behavior, Animal; Benzomorphans; Chronic Disease; Conditioning, Operant; Injections, Intraventricular; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stress, Psychological

2002
The mu-opioid receptor agonist morphine, but not agonists at delta- or kappa-opioid receptors, induces peripheral antinociception mediated by cannabinoid receptors.
    British journal of pharmacology, 2008, Volume: 154, Issue:5

    Topics: Amidohydrolases; Analgesics, Opioid; Animals; Arachidonic Acids; Benzamides; Benzomorphans; Cannabinoid Receptor Modulators; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hyperalgesia; Indoles; Male; Morphine; Organophosphonates; Pain; Pain Measurement; Piperazines; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2008
Effects of atypical kappa-opioid receptor agonists on intrathecal morphine-induced itch and analgesia in primates.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 328, Issue:1

    Topics: Analgesia; Animals; Benzomorphans; Female; Hot Temperature; Injections, Spinal; Macaca mulatta; Male; Morphinans; Morphine; Neurons; Piperazines; Pyrrolidines; Reaction Time; Receptors, Opioid, kappa; Restraint, Physical; Spiro Compounds

2009
Predicted structures for kappa opioid G-protein coupled receptor bound to selective agonists.
    Journal of chemical information and modeling, 2015, Mar-23, Volume: 55, Issue:3

    Topics: Benzomorphans; Binding Sites; Drug Design; Ethylketocyclazocine; Humans; Ligands; Models, Molecular; Molecular Docking Simulation; Morphine; Nalorphine; Pentazocine; Protein Conformation; Receptors, G-Protein-Coupled; Receptors, Opioid, kappa; Structure-Activity Relationship

2015
Identification of the three-dimensional pharmacophore of kappa-opioid receptor agonists.
    Bioorganic & medicinal chemistry, 2010, Jun-15, Volume: 18, Issue:12

    Topics: Models, Chemical; Models, Molecular; Receptors, Opioid, kappa

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011