bremazocine and enkephalin, ala(2)-mephe(4)-gly(5)-

bremazocine has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 59 studies

Research

Studies (59)

Timeframe	Studies, this research(%)	All Research%
pre-1990	22 (37.29)	18.7374
1990's	33 (55.93)	18.2507
2000's	4 (6.78)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Gioannini, TL; Hiller, JM; Liu, YF; Ofri, D; Ritter, AM; Simon, EJ	1
Kowalski, J; Petrillo, P; Sbacchi, M; Tavani, A	1
Barnard, EA; Richardson, A; Simon, J	1
Pinnock, RD	1
Colombo, M; La Regina, A; Petrillo, P; Tavani, A	1
Barnard, EA; Demoliou-Mason, C; Richardson, A	1
Millan, MJ; Morris, BJ	1
Bunn, SJ	1
Bunn, SJ; Dunkley, PR	1
Klein, P; Nelson, WL; Olsen, LD; Simon, EJ; Yao, YH	1
Hammer, RP	1
Baumann, NA; Cabon, F; Cupo, A; Ruiz-Gayo, M; Zalc, B	1
Fields, KL; Kessler, JA; Vaysse, PJ; Zukin, RS	1
Magnan, J; Tiberi, M	1
Heijna, MH; Hogenboom, F; Mulder, AH; Padt, M; Portoghese, PS; Schoffelmeer, AN	1
Dissanayake, VU; Hill, RG; Hughes, J; Hunter, JC	1
Brady, LS; Bykov, V; Holaday, JW; Jacobson, AE; Long, JB; Rice, KC; Rothman, RB	1
Kosterlitz, HW; La Regina, A; Petrillo, P; Robson, LE; Sbacchi, M; Tavani, A	1
Hoffman, PL; Khatami, S; Salafsky, B; Shibuya, T	1
Gauthier, S; Magnan, J; Pilapil, C; Quirion, R; Welner, S	1
La Regina, A; Petrillo, P; Sbacchi, M; Tavani, A	1
Crema, G; Gioannini, TL; Hiller, JM; Simon, EJ	1
Costa, T; Herz, A; Lang, J; Przewłocki, R	1
Bolger, GT; Marcus, KA; Skolnick, P; Thibou, R; Weissman, BA	1
Herz, A; Millan, MJ; Morris, BJ	1
Bunn, SJ; Livett, BG; Marley, PD	1
Frances, B; Meunier, JC; Moisand, C	1
De Montis, GM; Devoto, P; Preti, A; Tagliamonte, A	1
Bidlack, JM; O'Malley, WE	1
Herz, A; Morris, BJ	1
Akil, H; Khachaturian, H; Lewis, ME; Mansour, A; Watson, SJ	2
Ignatov, IuD; Zaĭtsev, AA	1
Itzhak, Y; Simon, EJ	1
Rance, MJ; Traynor, JR	1
Burkard, WP; Flück, N; Müller, PM	1
Burke, TR; Danks, JA; Jacobson, AE; Pert, CB; Rice, KC; Rothman, RB	1
Foote, RW; Maurer, R	1
Alsasua, A; Martín, MI; Parra, L; Pérez-Vizcaíno, F; Tamargo, J	1
Alfaro, MJ; Goicoechea, C; Lopez, F; Martin, MI; Ormazabal, MJ	1
Carr, KD; Hiller, JM; Simon, EJ; Wolinsky, TD	1
Howells, RD; Jin, J; Shahrestanifar, M; Wang, WW	1
Burke, T; Lewis, JW; Woods, JH; Zernig, G	1
Kaputlu, I; Oğütman, C; Sadan, G	1
Fan, LQ; Hiller, JM	1
Abrahamsen, GC; Carr, KD; Wolinsky, TD	1
Nelson, WL; Palmer, RB; Upthagrove, AL	1
Caudle, RM; Dubner, R; Ho, J; Mannes, AJ	1
Mamede Rosa, ML; Prado, WA	1
Adams, DJ; Trequattrini, C	1
Gioannini, TL; Hiller, JM; Onoprishvili, I; Simon, EJ	1
Coirini, H; Ortí, E; Pico, JC	1
Bakalkin, G; Derjabin, V; Hauser, KF; Nazarevskaja, G; Reznikov, K; Trunova, Y	1
Margotta, V; Merante, A; Palladini, G; Passarelli, F; Pontieri, FE; Venturini, G	1
Lia, EN; Prado, WA	1
Cheong, YP; Cho, KP; Kim, CJ; Kim, JK; Kim, KW; Kwun, J; Woo, RS	1
Akil, H; Bonner, G; Meng, F	1
Filliol, D; Goody, RJ; Kieffer, BL; Kitchen, I; Oakley, SM	1
Ballard, ME; Harmon, AC; Holtzman, SG; White, DA	1

Other Studies

59 other study(ies) available for bremazocine and enkephalin, ala(2)-mephe(4)-gly(5)-

Article	Year
Characterization of solubilized opioid receptors: reconstitution and uncoupling of guanine nucleotide-sensitive agonist binding. Journal of neurochemistry, 1992, Volume: 58, Issue:2 Topics: Animals; Benzomorphans; Binding Sites; Binding, Competitive; Cattle; Cholic Acids; Corpus Striatum; Detergents; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Receptors, Opioid; Solubility	1992
Characterization of opioid binding sites in rat spinal cord. Journal of receptor research, 1992, Volume: 12, Issue:1 Topics: Animals; Benzomorphans; Binding Sites; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; In Vitro Techniques; Male; Rats; Receptors, Opioid; Spinal Cord	1992
Protection by opioid ligands against modification of the opioid receptor by a carbodiimide. Biochemical pharmacology, 1992, Apr-01, Volume: 43, Issue:7 Topics: Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Brain Chemistry; Carbodiimides; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Guanylyl Imidodiphosphate; Guinea Pigs; Pyrrolidines; Receptors, Opioid	1992
A highly selective kappa-opioid receptor agonist, CI-977, reduces excitatory synaptic potentials in the rat locus coeruleus in vitro. Neuroscience, 1992, Volume: 47, Issue:1 Topics: Amino Acids; Analgesics; Animals; Benzofurans; Benzomorphans; Bicuculline; Depression, Chemical; Electric Stimulation; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; In Vitro Techniques; Ligands; Locus Coeruleus; Membrane Potentials; Naloxone; Naltrexone; Picrotoxin; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1992
Binding capacities and affinities at mu-, delta- and kappa-opioid sites in membrane suspensions from guinea-pig brain regions. Journal of receptor research, 1992, Volume: 12, Issue:2 Topics: Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; In Vitro Techniques; Male; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1992
Guanine nucleotide-binding protein-coupled and -uncoupled states of opioid receptors and their relevance to the determination of subtypes. Proceedings of the National Academy of Sciences of the United States of America, 1992, Nov-01, Volume: 89, Issue:21 Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Cell Membrane; Cerebellum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Etorphine; Female; GTP-Binding Proteins; Guinea Pigs; Humans; Kinetics; Ligands; Placenta; Pregnancy; Prosencephalon; Protein Binding; Pyrrolidines; Rats; Receptors, Opioid	1992
Inability of an opioid antagonist lacking negative intrinsic activity to induce opioid receptor up-regulation in vivo. British journal of pharmacology, 1991, Volume: 102, Issue:4 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Binding, Competitive; Drinking; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Narcotic Antagonists; Pain; Pain Measurement; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Sensory Thresholds; Up-Regulation	1991
Localisation and pharmacological characterisation of [3H]bremazocine binding in the bovine adrenal medulla. Neuroscience letters, 1991, Apr-29, Volume: 125, Issue:2 Topics: Adrenal Medulla; Animals; Autoradiography; Benzomorphans; Binding, Competitive; Cattle; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Kinetics; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1991
Opioid inhibition of nicotine-induced 45Ca2(+)-uptake into cultured bovine adrenal medullary cells. Biochemical pharmacology, 1991, Mar-01, Volume: 41, Issue:5 Topics: Adrenal Medulla; Animals; Benzomorphans; Calcium; Cattle; Cells, Cultured; Chromaffin System; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Methionine; Enkephalins; Nicotine; Oligopeptides	1991
Conjugate addition ligands of opioid antagonists. Methacrylate esters and ethers of 6 alpha- and 6 beta-naltrexol. Journal of medicinal chemistry, 1990, Volume: 33, Issue:2 Topics: Animals; Benzomorphans; Binding, Competitive; Cattle; Caudate Nucleus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Esters; Ethers; In Vitro Techniques; Ligands; Methacrylates; Naltrexone; Receptors, Opioid; Structure-Activity Relationship	1990
Mu-opiate receptor binding in the medial preoptic area is cyclical and sexually dimorphic. Brain research, 1990, May-07, Volume: 515, Issue:1-2 Topics: Animals; Benzomorphans; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estrus; Female; Male; Naloxone; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Sex Characteristics	1990
Pharmacological and molecular properties of opioid binding sites synthesized in a cell-free translation system. Journal of neuroscience research, 1990, Volume: 26, Issue:2 Topics: Animals; Benzomorphans; Binding, Competitive; Cell Line; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hybridomas; Mice; Molecular Weight; Morphinans; Oligopeptides; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger	1990
Characterization of opioid receptors in cultured neurons. Journal of neurochemistry, 1990, Volume: 55, Issue:2 Topics: Animals; Benzomorphans; Brain; Cell Membrane; Cells, Cultured; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Fluorescent Antibody Technique; Hippocampus; Hypothalamus; Neurons; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1990
Demonstration of the heterogeneity of the kappa-opioid receptors in guinea-pig cerebellum using selective and nonselective drugs. European journal of pharmacology, 1990, Jun-12, Volume: 188, Issue:6 Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Cerebellum; Computers; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1990
Opioid receptor-mediated inhibition of dopamine and acetylcholine release from slices of rat nucleus accumbens, olfactory tubercle and frontal cortex. European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Animals; Benzomorphans; Cerebral Cortex; Corpus Striatum; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ergolines; In Vitro Techniques; Male; Naloxone; Naltrexone; Nucleus Accumbens; Olfactory Bulb; Oxymetazoline; Pyrrolidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Opioid; Septal Nuclei	1990
Characterization of kappa-opioid receptors in the guinea-pig ileum. European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1 Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Naloxone; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Thiophenes	1990
Chronic administration of morphine and naltrexone up-regulate mu-opioid binding sites labeled by [3H][D-Ala2,MePhe4,Gly-ol5]enkephalin: further evidence for two mu-binding sites. European journal of pharmacology, 1989, Jan-24, Volume: 160, Issue:1 Topics: Animals; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; In Vitro Techniques; Male; Morphine; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu	1989
Regional variations in binding capacities at mu-, delta- and kappa-opioid sites in membrane suspensions from rabbit brain. European journal of pharmacology, 1989, Jul-18, Volume: 166, Issue:2 Topics: Analgesics; Animals; Benzomorphans; Binding, Competitive; Body Weight; Brain Chemistry; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; In Vitro Techniques; Male; Membranes; Nerve Tissue Proteins; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1989
Selective effects of ethanol on opiate receptor subtypes in brain. Neuropharmacology, 1987, Volume: 26, Issue:10 Topics: Animals; Benzomorphans; Binding, Competitive; Brain Chemistry; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethanol; In Vitro Techniques; Limbic System; Male; Mice; Mice, Inbred C57BL; Narcotics; Oligopeptides; Receptors, Opioid	1987
Autoradiographic distribution of multiple classes of opioid receptor binding sites in human forebrain. Brain research bulletin, 1987, Volume: 19, Issue:5 Topics: Aged; Autoradiography; Benzomorphans; Binding Sites; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Female; Humans; Male; Middle Aged; Oligopeptides; Receptors, Opioid; Tissue Distribution	1987
Interaction of U-69,593 with mu-, alpha- and kappa-opioid binding sites and its analgesic and intestinal effects in rats. Life sciences, 1988, Volume: 42, Issue:3 Topics: Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Gastrointestinal Motility; In Vitro Techniques; Male; Naloxone; Nociceptors; Pyrrolidines; Rats; Receptors, Opioid	1988
The direct demonstration of binding of mu, delta and kappa agonists to digitonin-solubilized opioid receptors from bovine striatum. NIDA research monograph, 1986, Volume: 75 Topics: Analgesics; Animals; Benzomorphans; Cattle; Cell Membrane; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Kinetics; Morphinans; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1986
Pertussis toxin abolishes the antinociception mediated by opioid receptors in rat spinal cord. European journal of pharmacology, 1987, Nov-24, Volume: 144, Issue:1 Topics: Adenosine Diphosphate; Analgesics; Animals; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Membranes; Nociceptors; Pertussis Toxin; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Ribose; Spinal Cord; Virulence Factors, Bordetella	1987
Enhancement of [3H]DAGO1 binding to rat brain by low concentrations of monovalent cations. Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:11 Topics: Animals; Batrachotoxins; Benzomorphans; Brain Chemistry; Cations, Monovalent; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Naloxone; Rats; Receptors, Opioid; Temperature	1987
Antagonist-induced opioid receptor up-regulation. II. Regionally specific modulation of mu, delta and kappa binding sites in rat brain revealed by quantitative autoradiography. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2 Topics: Animals; Autoradiography; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Kinetics; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord; Substantia Nigra	1988
The distribution of opioid binding subtypes in the bovine adrenal medulla. Neuroscience, 1988, Volume: 27, Issue:3 Topics: Adrenal Medulla; Animals; Benzomorphans; Cattle; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1988
Na+ ions and Gpp(NH)p selectively inhibit agonist interactions at mu- and kappa-opioid receptor sites in rabbit and guinea-pig cerebellum membranes. European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzomorphans; Binding, Competitive; Cerebellum; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium	1985
Differential effect of mu, delta, and kappa opioid agonists on adenylate cyclase activity. Journal of neuroscience research, 1987, Volume: 17, Issue:4 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Analgesics; Animals; Benzeneacetamides; Benzomorphans; Corpus Striatum; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Male; Morphinans; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid	1987
Inhibition of mu and delta but not kappa opioid binding to membranes by Fab fragments from a monoclonal antibody directed against the opioid receptor. The Journal of biological chemistry, 1986, Dec-05, Volume: 261, Issue:34 Topics: Animals; Antibodies, Monoclonal; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guinea Pigs; Immunoglobulin Fab Fragments; In Vitro Techniques; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1986
Autoradiographic localization in rat brain of kappa opiate binding sites labelled by [3H]bremazocine. Neuroscience, 1986, Volume: 19, Issue:3 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Autoradiography; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Morphinans; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa	1986
Pharmacological and anatomical evidence of selective mu, delta, and kappa opioid receptor binding in rat brain. Brain research, 1986, Dec-03, Volume: 399, Issue:1 Topics: Animals; Autoradiography; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalins; Male; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1986
[The role of various opiate receptors in the regulation of the nociceptive reaction of the arterial pressure]. Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 103, Issue:4 Topics: Animals; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Hemodynamics; Morphine; Nociceptors; Rats; Receptors, Opioid	1987
Autoradiographic differentiation of mu, delta, and kappa opioid receptors in the rat forebrain and midbrain. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:8 Topics: Animals; Autoradiography; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1987
A novel phencyclidine analog interacts selectively with mu opioid receptors. The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:2 Topics: Analgesia; Animals; Benzomorphans; Binding, Competitive; Cerebellum; Dihydromorphine; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; Male; Mice; Muscle Contraction; Naloxone; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, mu; Vas Deferens	1984
Opiate binding in the rat spinal cord: evidence for mu and delta sites. Neuropeptides, 1984, Volume: 5, Issue:1-3 Topics: Animals; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; In Vitro Techniques; Male; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Spinal Cord	1984
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes. Journal of receptor research, 1984, Volume: 4, Issue:1-6 Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid	1984
Tritiated-6-beta-fluoro-6-desoxy-oxymorphone: a highly selective ligand for the opiate mu receptor whose binding is characterized by low nonspecific binding. Neuropeptides, 1984, Volume: 4, Issue:4 Topics: Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Fentanyl; Hydromorphone; Isothiocyanates; Kinetics; Oxymorphone; Rats; Receptors, Opioid; Receptors, Opioid, mu; Thiocyanates; Tomography, Emission-Computed	1984
Autoradiographic localization of opiate kappa-receptors in the guinea-pig brain. European journal of pharmacology, 1982, Nov-05, Volume: 85, Issue:1 Topics: Animals; Autoradiography; Benzomorphans; Binding, Competitive; Brain; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Hypothalamus, Middle; Male; Receptors, Opioid; Receptors, Opioid, kappa	1982
mu- and delta-opioid receptor-mediated contractile effects on rat aortic vascular smooth muscle. European journal of pharmacology, 1995, Apr-13, Volume: 277, Issue:1 Topics: Amino Acid Sequence; Analgesics; Analysis of Variance; Animals; Aorta; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Molecular Sequence Data; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Naltrexone; Norepinephrine; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu	1995
Analgesic effect of two calcitonins and in vitro interaction with opioids. General pharmacology, 1995, Volume: 26, Issue:3 Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Dose-Response Relationship, Drug; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guinea Pigs; In Vitro Techniques; Male; Mice; Morphine; Muscle Contraction; Muscle, Smooth; Narcotics; Pain Measurement; Pain Threshold; Rabbits; Rats; Rats, Wistar	1995
Effects of chronic food restriction on mu and kappa opioid binding in rat forebrain: a quantitative autoradiographic study. Brain research, 1994, Sep-12, Volume: 656, Issue:2 Topics: Analgesics; Animals; Autoradiography; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Food Deprivation; Hypothalamus; Image Processing, Computer-Assisted; Male; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Self Stimulation	1994
Studies on mu and delta opioid receptor selectivity utilizing chimeric and site-mutagenized receptors. Proceedings of the National Academy of Sciences of the United States of America, 1995, Dec-19, Volume: 92, Issue:26 Topics: Amino Acid Sequence; Analgesics; Base Sequence; Benzomorphans; Binding, Competitive; Cell Line; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Etorphine; GTP-Binding Proteins; Humans; Kidney; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Naloxone; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Protein Structure, Secondary; Receptors, Opioid, delta; Receptors, Opioid, mu; Recombinant Fusion Proteins; Substrate Specificity; Transfection	1995
Mechanism of clocinnamox blockade of opioid receptors: evidence from in vitro and ex vivo binding and behavioral assays. The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:1 Topics: Animals; Behavior, Animal; Benzomorphans; Cinnamates; Cycloheximide; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Mice; Morphine Derivatives; Narcotic Antagonists; Receptors, Opioid, mu	1996
Cardiovascular effects of intrathecally injected mu, delta and kappa opioid receptor agonists in rabbits. Journal of autonomic pharmacology, 1995, Volume: 15, Issue:6 Topics: Animals; Baroreflex; Benzomorphans; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Spinal; Naloxone; Narcotic Antagonists; Rabbits; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1995
Laminar distribution of the multiple opioid receptors in the human cerebral cortex. Neurochemical research, 1996, Volume: 21, Issue:11 Topics: Aged; Aged, 80 and over; Analgesics; Autoradiography; Benzomorphans; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Female; Humans; Male; Organ Specificity; Postmortem Changes; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tritium	1996
Diabetes alters mu and kappa opioid binding in rat brain regions: comparison with effects of food restriction. Brain research, 1996, Oct-28, Volume: 738, Issue:1 Topics: Animals; Autoradiography; Benzomorphans; Brain; Diabetes Mellitus, Experimental; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tissue Distribution	1996
(E)- and (Z)-7-arylidenenaltrexones: synthesis and opioid receptor radioligand displacement assays. Journal of medicinal chemistry, 1997, Feb-28, Volume: 40, Issue:5 Topics: Animals; Benzeneacetamides; Benzomorphans; Benzylidene Compounds; Binding, Competitive; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guinea Pigs; Magnetic Resonance Spectroscopy; Mass Spectrometry; Models, Molecular; Molecular Conformation; Molecular Structure; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid, delta; Spectroscopy, Fourier Transform Infrared	1997
Putative kappa-2 opioid agonists are antihyperalgesic in a rat model of inflammation. The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1 Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Hyperalgesia; Male; Piperazines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa	1997
Antinociception induced by opioid or 5-HT agonists microinjected into the anterior pretectal nucleus of the rat. Brain research, 1997, May-16, Volume: 757, Issue:1 Topics: Analgesics; Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Microinjections; Pain; Phenazocine; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Serotonin Receptor Agonists	1997
Opioid receptor-mediated inhibition of omega-conotoxin GVIA-sensitive calcium channel currents in rat intracardiac neurons. Journal of neurophysiology, 1998, Volume: 79, Issue:2 Topics: Acetylcholine; Animals; Animals, Newborn; Anti-Arrhythmia Agents; Benzomorphans; Calcium; Calcium Channels; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Heart Conduction System; Ion Channel Gating; Ion Transport; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; omega-Conotoxin GVIA; Parasympathetic Nervous System; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Virulence Factors, Bordetella	1998
Inactivation of the purified bovine mu opioid receptor by sulfhydryl reagents. Neurochemical research, 1999, Volume: 24, Issue:1 Topics: Animals; Benzomorphans; Cattle; Cell Membrane; Corpus Striatum; Cysteine; Dithionitrobenzoic Acid; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylmaleimide; Kinetics; Ligands; Naloxone; Radioligand Assay; Receptors, Opioid, mu; Sulfhydryl Reagents; Tritium	1999
Site-specific effects of the nonsteroidal anti-inflammatory drug lysine clonixinate on rat brain opioid receptors. Pharmacology, 1999, Volume: 58, Issue:4 Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Clonixin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Lysine; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sensitivity and Specificity; Tritium	1999
Opioids modulate cell division in the germinal zone of the late embryonic neocortex. The European journal of neuroscience, 1999, Volume: 11, Issue:8 Topics: Animals; Benzomorphans; Cell Division; Cerebral Ventricles; Embryo, Mammalian; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Female; Mice; Mice, Inbred CBA; Mitotic Index; Naloxone; Narcotic Antagonists; Narcotics; Neocortex; Pregnancy; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1999
Opioid-dopamine interaction in planaria: a behavioral study. Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1999, Volume: 124, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Dopamine; Dopamine Antagonists; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Motor Activity; Narcotic Antagonists; Planarians; Receptors, Opioid; Receptors, Opioid, kappa; Sulpiride	1999
Effects of intrathecal L- and N-type calcium channel blockers on the antinociception evoked by opioid agonists in the rat tail flick test. Acta physiologica, pharmacologica et therapeutica latinoamericana : organo de la Asociacion Latinoamericana de Ciencias Fisiologicas y [de] la Asociacion Latinoamericana de Farmacologia, 1999, Volume: 49, Issue:4 Topics: Analgesics; Analgesics, Opioid; Animals; Benzomorphans; Calcium Channel Blockers; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Injections, Spinal; Male; Nimodipine; omega-Conotoxins; Pain Measurement; Rats; Rats, Wistar; Tail	1999
Receptor selectivity of Met-enkephalin-Arg6-Phe7, an endogenous opioid peptide, in cerebral cortex of human and rat. Life sciences, 2000, May-26, Volume: 67, Issue:1 Topics: Adult; Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Ethylketocyclazocine; Female; Humans; Male; Naloxone; Naltrexone; Norepinephrine; Oligopeptides; Peptide Fragments; Peptides; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Somatostatin	2000
Selectivity of mu-opioid receptor determined by interfacial residues near third extracellular loop. European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2 Topics: Amino Acid Substitution; Animals; Benzamides; Benzomorphans; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Ligands; Morphine; Mutation; Naloxone; Naltrexone; Narcotic Antagonists; Peptides; Piperazines; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid, mu; Signal Transduction; Sulfur Radioisotopes	2000
Quantitative autoradiographic mapping of opioid receptors in the brain of delta-opioid receptor gene knockout mice. Brain research, 2002, Jul-26, Volume: 945, Issue:1 Topics: Animals; Autoradiography; Benzofurans; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Female; Heterozygote; Homozygote; Male; Mice; Mice, Knockout; Oligopeptides; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	2002
Acute delta- and kappa-opioid agonist pretreatment potentiates opioid antagonist-induced suppression of water consumption. Brain research bulletin, 2008, Aug-15, Volume: 76, Issue:6 Topics: Analgesics, Opioid; Animals; Benzamides; Benzomorphans; Discrimination, Psychological; Dose-Response Relationship, Drug; Drinking; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Injections, Subcutaneous; Male; Naltrexone; Narcotic Antagonists; Pain Measurement; Piperazines; Pyrrolidines; Rats; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Water Deprivation	2008