bremazocine and dynorphins

bremazocine has been researched along with dynorphins in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199012 (52.17)18.7374
1990's10 (43.48)18.2507
2000's1 (4.35)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bunn, SJ; Dunkley, PR1
Fiorica-Howells, E; Spector, S1
Devlin, T; Shoemaker, WJ1
Cross, AJ; Hewitt, L; Savage, WJ; Slater, P1
Rodriguez, FD; Traynor, JR; Wood, MS1
Gillan, MG; Kosterlitz, HW; McKnight, AT; Robson, LE1
Cooper, SJ; Jackson, A; Kirkham, TC1
Ishihara, K; Iwama, T; Satoh, M; Takagi, H1
Schmauss, C1
De Montis, GM; Devoto, P; Preti, A; Tagliamonte, A1
Brady, LS; Herkenham, M; Rothman, RB1
Hayes, AG; Skingle, M; Tyers, MB1
Faden, AI; Feuerstein, G; Hassen, AH1
Burkard, WP; Flück, N; Müller, PM1
Akil, H; Khachaturian, H; Lewis, ME; Watson, SJ1
Berzetei-Gurske, IP; Brandt, SR; Polgar, WE; Toll, L; Webster, JL1
Collins, KA; Tseng, LF1
Akil, H; Ardati, A; Civelli, O; Hoversten, MT; Meng, F; Monsma, FJ; Reinscheid, RK; Taylor, LP; Ueda, Y; Watson, SJ1
Adams, DJ; Trequattrini, C1
Childers, SR; Sim, LJ; Vogt, L; Xiao, R1
Butelman, ER; Ko, MC; Woods, JH1
Lishmanov, YB; Maslov, LN; Ugdyzhekova, DS1
Horie, S; Ishihara, S; Minowa, S; Murayama, T; Tsuchiya, S; Watanabe, K1

Reviews

1 review(s) available for bremazocine and dynorphins

ArticleYear
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response

1985

Other Studies

22 other study(ies) available for bremazocine and dynorphins

ArticleYear
Opioid inhibition of nicotine-induced 45Ca2(+)-uptake into cultured bovine adrenal medullary cells.
    Biochemical pharmacology, 1991, Mar-01, Volume: 41, Issue:5

    Topics: Adrenal Medulla; Animals; Benzomorphans; Calcium; Cattle; Cells, Cultured; Chromaffin System; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Methionine; Enkephalins; Nicotine; Oligopeptides

1991
Selectivity of some "specific" opioid ligands?
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Dynorphins; Female; Haloperidol; In Vitro Techniques; Mice; Morphinans; Peptide Fragments; Phencyclidine; Piperidines; Receptors, Opioid

1990
Characterization of kappa opioid binding using dynorphin A1-13 and U69,593 in the rat brain.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Culture Techniques; Dynorphins; Ligands; Male; Morphinans; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Tritium

1990
Autoradiographic visualization of kappa opioid receptors with labelled dynorphins in guinea pig brain.
    Journal of receptor research, 1989, Volume: 9, Issue:2

    Topics: Animals; Autoradiography; Benzomorphans; Brain Chemistry; Dynorphins; Guinea Pigs; In Vitro Techniques; Male; Receptors, Opioid; Receptors, Opioid, kappa

1989
Characterisation of kappa-opioid binding sites in rat and guinea-pig spinal cord.
    Neuropharmacology, 1989, Volume: 28, Issue:10

    Topics: Animals; Benzeneacetamides; Benzomorphans; Captopril; Diprenorphine; Dynorphins; Guinea Pigs; In Vitro Techniques; Leucine; Ligands; Male; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord

1989
Kappa-binding and degradation of [3H]dynorphin A (1-8) and [3H]dynorphin A (1-9) in suspensions of guinea pig brain membranes.
    Journal of neurochemistry, 1985, Volume: 45, Issue:4

    Topics: Animals; Benzomorphans; Binding Sites; Brain; Dynorphins; Guinea Pigs; Kinetics; Membranes; Peptide Fragments; Protease Inhibitors; Receptors, Opioid; Receptors, Opioid, kappa; Substrate Specificity; Temperature

1985
Different effects of dynorphin A on in vitro guinea pig hippocampal CA3 pyramidal cells with various degrees of paired-pulse facilitation.
    Neuroscience letters, 1986, Jan-16, Volume: 63, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Drug Interactions; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Morphine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptic Transmission

1986
Spinal kappa-opioid receptor-mediated antinociception is stimulus-specific.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Dynorphins; Ethylketocyclazocine; Injections, Spinal; Male; Morphine; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord

1987
Differential effect of mu, delta, and kappa opioid agonists on adenylate cyclase activity.
    Journal of neuroscience research, 1987, Volume: 17, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Analgesics; Animals; Benzeneacetamides; Benzomorphans; Corpus Striatum; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Male; Morphinans; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid

1987
Physiological regulation of neurohypophyseal kappa-opiate receptors.
    Brain research, 1988, Mar-08, Volume: 443, Issue:1-2

    Topics: Analgesics; Animals; Benzomorphans; Dynorphins; Etorphine; Homeostasis; Kinetics; Male; Pituitary Gland, Posterior; Rats; Rats, Brattleboro; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1988
Antinociceptive profile of dynorphin in the rat.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Analgesics; Animals; Benzomorphans; Dynorphins; Endorphins; Male; Morphine; Nociceptors; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1983
Kappa opioid receptors modulate cardiorespiratory function in hindbrain nuclei of rat.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1984, Volume: 4, Issue:9

    Topics: Animals; Benzomorphans; Blood Pressure; Dynorphins; Heart; Heart Rate; Male; Medulla Oblongata; Microinjections; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Respiration; Respiration, Artificial; Respiratory Physiological Phenomena; Tidal Volume

1984
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid

1984
Anatomical relationship between opioid peptides and receptors in rhesus monkey brain.
    Brain research bulletin, 1984, Volume: 13, Issue:6

    Topics: Animals; Benzomorphans; Brain; Brain Mapping; Dynorphins; Endorphins; Enkephalins; Macaca mulatta; Naloxone; Pro-Opiomelanocortin; Radioligand Assay; Receptors, Opioid; Synaptic Transmission

1984
Comparison of kappa 2-opioid receptors in guinea pig brain and guinea pig ileum membranes.
    European journal of pharmacology, 1993, Feb-09, Volume: 231, Issue:2

    Topics: Analgesics; Animals; Benzomorphans; Brain Chemistry; Dynorphins; Ethylketocyclazocine; Guanylyl Imidodiphosphate; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Ligands; Male; Membranes; Myenteric Plexus; Receptors, Opioid, kappa

1993
Spinal involvement of both dynorphin A and Met-enkephalin in the antinociception induced by intracerebroventricularly administered bremazocine but not morphine in the mouse.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Benzomorphans; beta-Endorphin; Drug Interactions; Dynorphins; Enkephalin, Leucine; Enkephalin, Methionine; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphine; Nociceptors; Pain Measurement; Pyrrolidines; Spinal Cord; Time Factors

1993
Moving from the orphanin FQ receptor to an opioid receptor using four point mutations.
    The Journal of biological chemistry, 1996, Dec-13, Volume: 271, Issue:50

    Topics: Analgesics; Animals; Benzomorphans; Dynorphins; Models, Molecular; Naltrexone; Narcotic Antagonists; Nociceptin Receptor; Point Mutation; Rats; Receptors, Opioid

1996
Opioid receptor-mediated inhibition of omega-conotoxin GVIA-sensitive calcium channel currents in rat intracardiac neurons.
    Journal of neurophysiology, 1998, Volume: 79, Issue:2

    Topics: Acetylcholine; Animals; Animals, Newborn; Anti-Arrhythmia Agents; Benzomorphans; Calcium; Calcium Channels; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Heart Conduction System; Ion Channel Gating; Ion Transport; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; omega-Conotoxin GVIA; Parasympathetic Nervous System; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Virulence Factors, Bordetella

1998
Lack of evidence of kappa2-selective activation of G-proteins: kappa opioid receptor stimulation of [35S] GTPgammaS binding in guinea pig brain.
    Biochemical pharmacology, 1998, Jul-01, Volume: 56, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Autoradiography; Benzomorphans; Brain; Dynorphins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; In Vitro Techniques; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Sulfur Radioisotopes

1998
Activation of peripheral kappa opioid receptors inhibits capsaicin-induced thermal nociception in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Azocines; Benzomorphans; Capsaicin; Dynorphins; Female; Hot Temperature; Ligands; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Pain Measurement; Peptide Fragments; Receptors, Opioid, kappa

1999
Participation of central and peripheral kappa 1 and kappa 2 opioid receptors in arrhythmogenesis.
    Clinical and experimental pharmacology & physiology, 1999, Volume: 26, Issue:9

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Arrhythmias, Cardiac; Benzomorphans; Dynorphins; Male; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa

1999
Involvement of glutamate and gamma-amino-butyric acid receptor systems on gastric acid secretion induced by activation of kappa-opioid receptors in the central nervous system in rats.
    British journal of pharmacology, 2003, Volume: 138, Issue:6

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Bicuculline; Brain; Dynorphins; gamma-Aminobutyric Acid; Gastric Acid; Injections, Intraventricular; Ketanserin; Male; Perfusion; Piperazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, Serotonin; Stomach

2003