Page last updated: 2024-09-05

bradykinin, sar-(d-phe(8))des-arg(9) and bradykinin

bradykinin, sar-(d-phe(8))des-arg(9) has been researched along with bradykinin in 18 studies

Compound Research Comparison

Studies
(bradykinin, sar-(d-phe(8))des-arg(9))
Trials
(bradykinin, sar-(d-phe(8))des-arg(9))
Recent Studies (post-2010)
(bradykinin, sar-(d-phe(8))des-arg(9))
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
180114,1953551,520

Protein Interaction Comparison

ProteinTaxonomybradykinin, sar-(d-phe(8))des-arg(9) (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (50.00)18.2507
2000's8 (44.44)29.6817
2010's1 (5.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M1
deBlois, D; Drapeau, G; Marceau, F1
Advenier, C; Hirsch, A; Martin, CA; Molimard, M; Naline, E1
Davis, AJ; Perkins, MN1
Audet, R; Drapeau, G; Godin, D; Levesque, L; Marceau, F1
Bachvarov, DR; Drapeau, G; Larrivée, JF; Levesque, L; Marceau, F; Rioux, F1
Feltrin, MR; Nicolau, M; Regoli, D1
Audet, R; Drapeau, G; Marceau, F; Rioux, F1
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Tramontana, M1
Antel, JP; Biernacki, K; Couture, R; Nalbantoglu, J; Pouly, S; Prat, A1
Adam, A; Bachvarov, DR; Bouthillier, J; Guay, K; Houle, S; Marceau, F; Sabourin, T1
Gabilan, NH; Nicolau, M; Vitor, R; Wille, PR1
Bader, M; Bonaria Salis, M; Cayla, C; Emanueli, C; Gaspa, L; Isner, JM; Kirchmair, R; Madeddu, P; Pesquero, JB; Pinna, A; Pintus, G; Regoli, D; Stacca, T1
Duret, JF; El Habach, T; Haury, L; Tiritilli, A1
Alvarez-Silva, M; Bianchin, MM; Cardoso, RC; Carlotti, CG; Lobão-Soares, B; Nicolau, M; Trentin, AG; Walz, R1
Adam, A; Marceau, F; Morissette, G; Sabourin, T1
Daray, FM; Errasti, AE; Falcioni, AG; Gago, JE; Goldschmidt, ED; Nowak, W; Pelorosso, FG; Pugliese, MI; Rothlin, RP1
Bhat, M; Couture, R; Hachana, S; Huppé-Gourgues, F; Sénécal, J; Vaucher, E1

Other Studies

18 other study(ies) available for bradykinin, sar-(d-phe(8))des-arg(9) and bradykinin

ArticleYear
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
    European journal of pharmacology, 1999, Jun-25, Volume: 374, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

1999
Hypotensive effects of Lys-des-Arg9-bradykinin and metabolically protected agonists of B1 receptors for kinins.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:3

    Topics: Animals; Blood Pressure; Bradykinin; Cardiovascular System; Female; Hypotension; Kallidin; Kinins; Lipopolysaccharides; Male; Prostaglandins; Protease Inhibitors; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter

1991
Contractile effects of bradykinin on the isolated human small bronchus.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Acetylcholine; Aged; Atropine; Benzamides; Biphenyl Compounds; Bradykinin; Bronchi; Bronchoconstriction; Capsaicin; Humans; In Vitro Techniques; Indomethacin; Middle Aged; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Bradykinin; Ruthenium Red; Tetrodotoxin

1994
Induction of B1 receptors in vivo in a model of persistent inflammatory mechanical hyperalgesia in the rat.
    Neuropharmacology, 1994, Volume: 33, Issue:1

    Topics: Animals; Arthritis, Experimental; Bradykinin; Bradykinin Receptor Antagonists; Female; Freund's Adjuvant; Hindlimb; Hyperalgesia; Injections, Intra-Articular; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin

1994
Development and in vivo evaluation of metabolically resistant antagonists of B1 receptors for kinins.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Amino Acid Sequence; Animals; Bradykinin; Drug Evaluation, Preclinical; Drug Stability; Female; Kallidin; Kidney; Male; Molecular Sequence Data; Peptide Hydrolases; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Structure-Activity Relationship

1993
Regulation of kinin-induced contraction and DNA synthesis by inflammatory cytokines in the smooth muscle of the rabbit aorta.
    British journal of pharmacology, 1995, Volume: 116, Issue:1

    Topics: Angiotensin II; Animals; Aorta, Thoracic; Bradykinin; Cells, Cultured; Cytokines; DNA; Endothelins; Female; Humans; Interleukin-1; Macrophage Migration-Inhibitory Factors; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oncostatin M; Peptides; Phenylephrine; Rabbits; Receptors, Bradykinin; Vasoconstrictor Agents

1995
Induction of bradykinin B1 hypotensive receptors in rats by lipopolysaccharide.
    Canadian journal of physiology and pharmacology, 1996, Volume: 74, Issue:3

    Topics: Animals; Bradykinin; Dose-Response Relationship, Drug; Hypotension; Lipopolysaccharides; Male; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin

1996
Cardiovascular effects of Sar-[D-Phe8]des-Arg9-bradykinin, a metabolically protected agonist of B1 receptor for kinins, in the anesthetized rabbit pretreated with a sublethal dose of bacterial lipopolysaccharide.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:1

    Topics: Anesthesia; Animals; Bradykinin; Female; Halothane; Hemodynamics; Lipopolysaccharides; Male; Nitric Oxide; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin

1997
Capsaicin pretreatment does not alter rat urinary bladder motor responses induced by a kinin B1 receptor agonist after endotoxin treatment.
    Neuroscience letters, 1999, Mar-05, Volume: 262, Issue:2

    Topics: Administration, Intravesical; Animals; Bradykinin; Capsaicin; Gene Expression; Lipopolysaccharides; Male; Muscle Contraction; Muscle, Smooth; Protamines; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Reflex, Abnormal; Sodium Chloride; Urinary Bladder

1999
Kinin B1 receptor expression and function on human brain endothelial cells.
    Journal of neuropathology and experimental neurology, 2000, Volume: 59, Issue:10

    Topics: Adult; Blood-Brain Barrier; Bradykinin; Brain Chemistry; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Gene Expression; Humans; Inositol Phosphates; Interferon-gamma; Interleukin-8; NG-Nitroarginine Methyl Ester; Nitric Oxide; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Serum Albumin, Bovine; Temporal Lobe

2000
Absence of ligand-induced regulation of kinin receptor expression in the rabbit.
    British journal of pharmacology, 2001, Volume: 133, Issue:7

    Topics: Anesthesia; Animals; Aorta; Bradykinin; Bradykinin Receptor Antagonists; Captopril; Cells, Cultured; Dextran Sulfate; Dose-Response Relationship, Drug; Gene Expression Regulation; Hypotension; Interleukin-1; Kininogens; Ligands; Lipopolysaccharides; Male; Muscle, Smooth, Vascular; Rabbits; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Vasoconstriction

2001
Plasma extravasation mediated by lipopolysaccharide-induction of kinin B1 receptors in rat tissues.
    Mediators of inflammation, 2001, Volume: 10, Issue:3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Duodenum; Ileum; Kallidin; Lipopolysaccharides; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Trachea; Urinary Bladder

2001
Targeting kinin B(1) receptor for therapeutic neovascularization.
    Circulation, 2002, Jan-22, Volume: 105, Issue:3

    Topics: Animals; Apoptosis; Bradykinin; Bradykinin Receptor Antagonists; Cell Division; Cells, Cultured; Endothelium, Vascular; Extremities; Humans; Ischemia; Laser-Doppler Flowmetry; Mice; Mice, Knockout; Muscle, Skeletal; Neovascularization, Physiologic; Perfusion; Receptor, Bradykinin B1; Receptors, Bradykinin; Signal Transduction

2002
BK2 but not BK1 receptors mediating contractile response in human umbilical arteries: role of thromboxane A2.
    Methods and findings in experimental and clinical pharmacology, 2004, Volume: 26, Issue:4

    Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dose-Response Relationship, Drug; Endothelium; Humans; Imidazoles; Indomethacin; Masoprocol; Muscle Contraction; Muscle, Smooth, Vascular; Quinacrine; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Thromboxane A2; Umbilical Arteries

2004
Enhancement of blood-tumor barrier permeability by Sar-[D-Phe8]des-Arg9BK, a metabolically resistant bradykinin B1 agonist, in a rat C6 glioma model.
    BMC neuroscience, 2004, Sep-30, Volume: 5

    Topics: Animals; Blood Proteins; Blood-Brain Barrier; Bradykinin; Brain Neoplasms; Cell Line, Tumor; Cell Membrane Permeability; Disease Models, Animal; Glioma; Male; Rats; Rats, Wistar; Receptor, Bradykinin B1

2004
Inhibition of human and rabbit arterial smooth muscle cell migration mediated by the kinin B1 receptor: role of receptor density and released mediators.
    Canadian journal of physiology and pharmacology, 2006, Volume: 84, Issue:11

    Topics: Animals; Aorta; Bradykinin; Cell Movement; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nitric Oxide; Phosphatidylinositol 3-Kinases; Prostaglandins; Rabbits; Receptor, Bradykinin B1; Signal Transduction; Time Factors; Umbilical Veins; Wound Healing

2006
Functional evidence of des-Arg10-kallidin enzymatic inactivating pathway in isolated human umbilical vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Bradykinin; Captopril; CD13 Antigens; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Female; Glycopeptides; Humans; In Vitro Techniques; Kallidin; Metalloproteases; Neprilysin; Peptides; Protease Inhibitors; Receptor, Bradykinin B1; Umbilical Veins; Vasoconstriction

2007
Expression, distribution and function of kinin B
    British journal of pharmacology, 2018, Volume: 175, Issue:6

    Topics: Administration, Ophthalmic; Animals; Bradykinin; Capillary Permeability; Diabetes Mellitus, Experimental; Diabetic Retinopathy; Gene Expression Regulation; Leukostasis; Male; Rats; Rats, Wistar; Receptor, Bradykinin B1; Retina; RNA, Messenger; RNA, Small Interfering; Streptozocin

2018