Page last updated: 2024-09-03

bradykinin, leu(8)-des-arg(9)- and kallidin, des-arg(10)-

bradykinin, leu(8)-des-arg(9)- has been researched along with kallidin, des-arg(10)- in 7 studies

Compound Research Comparison

Studies
(bradykinin, leu(8)-des-arg(9)-)
Trials
(bradykinin, leu(8)-des-arg(9)-)
Recent Studies (post-2010)
(bradykinin, leu(8)-des-arg(9)-)
Studies
(kallidin, des-arg(10)-)
Trials
(kallidin, des-arg(10)-)
Recent Studies (post-2010) (kallidin, des-arg(10)-)
1020780417

Protein Interaction Comparison

ProteinTaxonomybradykinin, leu(8)-des-arg(9)- (IC50)kallidin, des-arg(10)- (IC50)
B1 bradykinin receptorHomo sapiens (human)0.0009

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19901 (14.29)18.7374
1990's5 (71.43)18.2507
2000's1 (14.29)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Borkowski, JA; Derrick, AW; Hess, JF; MacNeil, T1
Austin, CE; Bathon, JM; Chakravarty, S; Faussner, A; Kyle, DJ; Proud, D; Robinson, HE1
Bastian, S; Loillier, B; Paquet, JL; Pruneau, D1
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M1
Churchill, L; Ward, PE1
Calixto, JB; de Campos, RO; Henriques, MG1
Kohno, S; Mizutani, N; Nabe, T; Sugahara, S; Takenaka, H1

Other Studies

7 other study(ies) available for bradykinin, leu(8)-des-arg(9)- and kallidin, des-arg(10)-

ArticleYear
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cattle; Cloning, Molecular; COS Cells; DNA Primers; DNA, Complementary; Humans; Kallidin; Mice; Molecular Sequence Data; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Sequence Homology, Amino Acid; Species Specificity; Transfection

1996
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
    The Journal of biological chemistry, 1997, Apr-25, Volume: 272, Issue:17

    Topics: Animals; Binding, Competitive; Biological Transport; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Inositol Phosphates; Kallidin; Ligands; Oligopeptides; Precipitin Tests; Protein Binding; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Signal Transduction; Type C Phospholipases

1997
Stable expression of human kinin B1 receptor in 293 cells: pharmacological and functional characterization.
    British journal of pharmacology, 1997, Volume: 122, Issue:2

    Topics: Calcium; Cell Line; Enzyme Activation; Humans; Kallidin; Receptor, Bradykinin B1; Receptors, Bradykinin; Transfection; Type C Phospholipases

1997
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
    European journal of pharmacology, 1999, Jun-25, Volume: 374, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

1999
Conversion of B1 kinin receptor-mediated vascular relaxation to contraction.
    Hypertension (Dallas, Tex. : 1979), 1987, Volume: 9, Issue:6 Pt 2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bradykinin; Dose-Response Relationship, Drug; Indomethacin; Kallidin; Male; Pyrazoles; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Vasoconstriction; Vasodilation

1987
Systemic treatment with Mycobacterium bovis bacillus Calmette-Guérin (BCG) potentiates kinin B1 receptor agonist-induced nociception and oedema formation in the formalin test in mice.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Animals; Bradykinin; Dexamethasone; Dose-Response Relationship, Drug; Drug Synergism; Edema; Formaldehyde; Hindlimb; Indomethacin; Kallidin; Male; Mice; Mycobacterium bovis; Pain; Pain Measurement; Pyrazoles; Receptor, Bradykinin B1; Receptors, Bradykinin

1998
Kinins are involved in the development of allergic nasal hyperresponsiveness in guinea pigs.
    European journal of pharmacology, 2003, Aug-29, Volume: 476, Issue:3

    Topics: Airway Resistance; Allergens; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Guinea Pigs; Kallidin; Kinins; Leukotriene D4; Male; Nasal Lavage Fluid; Pollen; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Rhinitis, Allergic, Seasonal; Time Factors

2003