bradykinin, leu(8)-des-arg(9)- has been researched along with fr 173657 in 3 studies
Studies (bradykinin, leu(8)-des-arg(9)-) | Trials (bradykinin, leu(8)-des-arg(9)-) | Recent Studies (post-2010) (bradykinin, leu(8)-des-arg(9)-) | Studies (fr 173657) | Trials (fr 173657) | Recent Studies (post-2010) (fr 173657) |
---|---|---|---|---|---|
102 | 0 | 7 | 70 | 0 | 5 |
Protein | Taxonomy | bradykinin, leu(8)-des-arg(9)- (IC50) | fr 173657 (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 0.0014 | |
B2 bradykinin receptor | Homo sapiens (human) | 0.0014 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 1 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Aramori, I; Asano, M; Iwami, M; Kojo, H; Morikawa, N; Nakamura, K; Notsu, Y; O'Donnell, N; Zenkoh, J | 1 |
Bentley, KR; Jarrott, B | 1 |
Calixto, JB; Costa, R; Juliano, L; Manjavachi, MN; Marotta, DM; Motta, EM; Pesquero, JB; Torres, HA | 1 |
3 other study(ies) available for bradykinin, leu(8)-des-arg(9)- and fr 173657
Article | Year |
---|---|
Novel subtype-selective nonpeptide bradykinin receptor antagonists FR167344 and FR173657.
Topics: Animals; Aorta; Bradykinin Receptor Antagonists; Cricetinae; Dose-Response Relationship, Drug; Humans; Kidney; Pyridines; Quinolines | 1997 |
Lipopolysaccharide decreases bradykinin receptor-induced acidification responses in cultured bovine aortic endothelial cells.
Topics: Animals; Aorta, Thoracic; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Endothelium, Vascular; Endotoxins; Lipopolysaccharides; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin | 2000 |
The role of kinin B1 and B2 receptors in the scratching behaviour induced by proteinase-activated receptor-2 agonists in mice.
Topics: Animals; Antipruritics; Behavior, Animal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dioxoles; Disease Models, Animal; Dose-Response Relationship, Drug; Injections, Intradermal; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Spinal; Mice; Mice, Inbred C57BL; Mice, Knockout; Oligopeptides; Pain Threshold; Pruritus; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptor, PAR-2; Sulfonamides; Trypsin | 2010 |