Page last updated: 2024-09-03

bradykinin, leu(8)-des-arg(9)- and fr 173657

bradykinin, leu(8)-des-arg(9)- has been researched along with fr 173657 in 3 studies

Compound Research Comparison

Studies
(bradykinin, leu(8)-des-arg(9)-)
Trials
(bradykinin, leu(8)-des-arg(9)-)
Recent Studies (post-2010)
(bradykinin, leu(8)-des-arg(9)-)
Studies
(fr 173657)
Trials
(fr 173657)
Recent Studies (post-2010) (fr 173657)
102077005

Protein Interaction Comparison

ProteinTaxonomybradykinin, leu(8)-des-arg(9)- (IC50)fr 173657 (IC50)
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0014
B2 bradykinin receptorHomo sapiens (human)0.0014

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aramori, I; Asano, M; Iwami, M; Kojo, H; Morikawa, N; Nakamura, K; Notsu, Y; O'Donnell, N; Zenkoh, J1
Bentley, KR; Jarrott, B1
Calixto, JB; Costa, R; Juliano, L; Manjavachi, MN; Marotta, DM; Motta, EM; Pesquero, JB; Torres, HA1

Other Studies

3 other study(ies) available for bradykinin, leu(8)-des-arg(9)- and fr 173657

ArticleYear
Novel subtype-selective nonpeptide bradykinin receptor antagonists FR167344 and FR173657.
    Molecular pharmacology, 1997, Volume: 51, Issue:2

    Topics: Animals; Aorta; Bradykinin Receptor Antagonists; Cricetinae; Dose-Response Relationship, Drug; Humans; Kidney; Pyridines; Quinolines

1997
Lipopolysaccharide decreases bradykinin receptor-induced acidification responses in cultured bovine aortic endothelial cells.
    European journal of pharmacology, 2000, Aug-18, Volume: 402, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Endothelium, Vascular; Endotoxins; Lipopolysaccharides; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

2000
The role of kinin B1 and B2 receptors in the scratching behaviour induced by proteinase-activated receptor-2 agonists in mice.
    British journal of pharmacology, 2010, Volume: 159, Issue:4

    Topics: Animals; Antipruritics; Behavior, Animal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dioxoles; Disease Models, Animal; Dose-Response Relationship, Drug; Injections, Intradermal; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Spinal; Mice; Mice, Inbred C57BL; Mice, Knockout; Oligopeptides; Pain Threshold; Pruritus; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptor, PAR-2; Sulfonamides; Trypsin

2010