Page last updated: 2024-09-03

bradykinin, leu(8)-des-arg(9)- and bradykinin

bradykinin, leu(8)-des-arg(9)- has been researched along with bradykinin in 97 studies

Compound Research Comparison

Studies
(bradykinin, leu(8)-des-arg(9)-)
Trials
(bradykinin, leu(8)-des-arg(9)-)
Recent Studies (post-2010)
(bradykinin, leu(8)-des-arg(9)-)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
1020714,1953551,520

Protein Interaction Comparison

ProteinTaxonomybradykinin, leu(8)-des-arg(9)- (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (97)

TimeframeStudies, this research(%)All Research%
pre-19906 (6.19)18.7374
1990's58 (59.79)18.2507
2000's22 (22.68)29.6817
2010's11 (11.34)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Escher, E; Guillemette, G; Laczkó, E; Regoli, D1
Borkowski, JA; Derrick, AW; Hess, JF; MacNeil, T1
Austin, CE; Bathon, JM; Chakravarty, S; Faussner, A; Kyle, DJ; Proud, D; Robinson, HE1
Aramori, I; Asano, M; Iwami, M; Kojo, H; Morikawa, N; Nakamura, K; Notsu, Y; O'Donnell, N; Zenkoh, J1
Arbuckle, J; Bevan, SJ; Burgess, GM; Davis, C; Docherty, RJ; Jones, C; McIntyre, P; Phillips, E; Webb, M; Yaqoob, M1
Amblard, M; Bedos, P; Daffix, I; Dodey, P; Luccarini, JM; Martinez, J; Olivier, C; Paquet, JL; Pruneau, D1
Alvarez, AL; Delorenzi, A; Finkielman, S; Nahmod, VE; Pirola, CJ; Santajuliana, D1
Campbell, JN; Khan, AA; Manning, DC; Meyer, RA; Raja, SN1
Gobeil, F; Regoli, D; Rhaleb, NE1
Illiano, S; Mombouli, JV; Vanhoutte, PM1
Blöchl, A; Brenner, P; Dominiak, P; Simon, M1
Harik, SI; Homayoun, P1
Staszewska-Woolley, J; Woodman, OL1
Mantione, CR; Rodriguez, R1
Okabe, E; Sugihara, M; Todoki, K1
Northover, AM1
Barnes, PJ; Ichinose, M1
Kumazawa, T; Minagawa, M; Mizumura, K; Tsujii, Y1
McFadden, RG; Vickers, KE1
Churchill, L; Ward, PE1
Bettaney, J; Dray, A; Forster, P; Perkins, MN1
Marceau, F; Tremblay, B1
Couture, R; Laneuville, O1
Advenier, C; Hirsch, A; Martin, CA; Molimard, M; Naline, E1
Chulak, C; Couture, R; Foucart, S1
Andreeva, L; Rang, HP1
Fan, TP; Hu, DE1
Fu, T; Gu, ZL; Xu, YH1
Butt, SK; Dawson, LG; Hall, JM1
Oh-ishi, S; Tokumasu, T; Ueno, A1
Davis, AJ; Perkins, MN1
Butt, SK; Field, JL; Hall, JM; Morton, IK1
Griesbacher, T; Legat, FJ; Lembeck, F1
Hsia, HC; Hsieh, JT; Luo, SF; Ong, R; Yang, CM1
Berezin, M; Prior, T; Rangachari, PK1
Campbell, E; Dray, A; Perkins, MN1
Brown, M; McIntyre, P; Phillips, E; Skidmore, E; Webb, M1
Cocks, TM; Drummond, GR1
Ahluwalia, A; Perretti, M1
Kato, M; Kobayashi, I; Saito, Y; Tatemoto, K1
Lecci, A; Maggi, CA; Meini, S1
Burkard, MR; Cuadrado, DK; Greer, RA; Selig, WM; Whalley, ET; Zuzack, JS1
Catanzaro, O; Cueva, F; Frontera, M; Navarro, M; Zuccollo, A1
Roach, TJ; Sufka, KJ1
Catanzaro, O; Navarro, M; Zuccollo, A1
Dedio, J; Schölkens, BA; Wiemer, G; Wirth, K; Wohlfart, P1
Antúnez, P; Pérez, H; Rothlin, RP; Sardi, SP1
Ferreira, SH; Tonussi, CR2
Borkowski, JA; Boyce, S; Carlson, EJ; Hess, JF; Hill, RG; Rupniak, NM; Webb, JK; Williams, AR1
Cuthbert, AW; Teather, S2
Buchinger, P; Chondromatidou, A; Hermann, A; Miska, K; Rehbock, J1
Arakawa, M; Fujimura, A; Ohmori, M; Sakamoto, K; Sugimoto, K1
Knox, AJ; Pang, L1
Gao, XP; Oda, D; Pakhlevaniants, S; Rubinstein, I1
Andersson, RG; Persson, K1
Abbas, F; Clayton, JK; Marshall, KM; Senior, J1
Da Silva, A; Gies, JP; Lach, E; Landry, Y; Scherrer, D; Schmidlin, F1
Habib, S; Jaggar, SI; Rice, AS1
Cheronis, JC; Fritz, H; Lehner, M; Schorr, M; Siebeck, M; Spannagl, E; Whalley, ET1
Calixto, JB; de Campos, RO; Henriques, MG1
Charland, S; Filteau, C; Gobeil, F; Neugebauer, W; Perron, SI; Regoli, D1
Cunha, FQ; Cunha, JM; Ferreira, SH; Lorenzetti, BB; Poole, S1
Bateson, EA; Olley, PM; Schulz, R1
Al-Rashed, S; Brain, SD; Cao, T; Gerard, N; Hoult, JR; Pintér, E1
Levy, D; Zochodne, DW1
Bentley, KR; Jarrott, B1
Bader, M; Bonaria Salis, M; Cayla, C; Emanueli, C; Gaspa, L; Isner, JM; Kirchmair, R; Madeddu, P; Pesquero, JB; Pinna, A; Pintus, G; Regoli, D; Stacca, T1
Calixto, JB; Cordeiro, RS; e Silva, PM; Lavich, TR; Martins, MA1
Daaka, Y; Guo, R; Leeb-Lundberg, LM; Madden, JF; Taub, JS1
Kohno, S; Mizutani, N; Nabe, T; Sugahara, S; Takenaka, H1
Caruso-Neves, C; Corrêa da Costa, VM; Gomes, VO; Lopes, AG; Lóss, FF; Malaquias, AT1
Asada, A; Maeda, K; Nakamura, M; Watanabe, T; Yasunari, K; Yoshikawa, J1
Chichorro, JG; Lorenzetti, BB; Zampronio, AR1
Arunkumar, R; Brennan, TJ; Leonard, PA1
Araújo, RC; Bader, M; Beirith, A; Calixto, JB; Ferreira, J; Mori, MA; Pesquero, JB1
Cidlowski, JA; Rhen, T1
Farias, NC; Feres, T; Paiva, AC; Paiva, TB1
Ghilardi, JR; Halvorson, KG; Kubota, K; Lindsay, TH; Mantyh, PW; Sevcik, MA1
Bergren, DR1
Calixto, JB; Ferreira, J; Kassuya, CA; Rae, GA; Werner, MF; Zampronio, AR1
Cunha, FQ; Cunha, TM; Ferreira, SH; Fukada, SY; Guerrero, AT; Parada, CA; Poole, S; Santodomingo-Garzón, T; Verri, WA1
Bader, M; Cheung, G; Färber, K; Ifuku, M; Ishikawa, E; Iwamoto, T; Kettenmann, H; Kita, S; Komuro, I; Merrino, VF; Miyamoto, T; Noda, M; Nolte, C; Okuno, Y; Ooboshi, H; Wada, K; Wang, B; Yamakawa, Y1
Aoki, M; Inoue, N; Kobayashi, K; Kondo, T; Li, P; Murohara, T; Numaguchi, Y; Okumura, K1
Calixto, JB; Campos, MM; Duarte, FS; Medeiros, R; Pandolfo, P; Passos, GF; Pesquero, JB; Prediger, RD; Takahashi, RN1
Calixto, JB; Chichorro, JG; Luiz, AP; Rae, GA; Schroeder, SD; Zampronio, AR1
Akira, A; Andoh, T; Kuraishi, Y; Saiki, I1
Calixto, JB; Costa, R; Juliano, L; Manjavachi, MN; Marotta, DM; Motta, EM; Pesquero, JB; Torres, HA1
Chen, Q; Lai, J; Ossipov, MH; Porreca, F; Vardanyan, M; Vera-Portocarrero, LP1
Araújo, RC; Braga, TT; Buscariollo, BN; Câmara, NO; Corrêa-Costa, M; Filho, AP; Keller, AC; Malheiros, DM; Maquigussa, E; Moura, IC; Oliveira, CD; Pereira, RL; Reis, VO; Semedo, P; Soares, MF1
Bento, AF; Calixto, JB; Costa, R; Dutra, RC; Malinsky, FR; Manjavachi, MN; Motta, EM; Pesquero, JB1
Bento, AF; Bouzon, ZL; Calixto, JB; Claudino, RF; Dutra, RC; Marcon, R; Morais, RL; Pesquero, JB; Schmidt, EC; Sordi, R1
Bobinski, F; Brum, JS; de Barros, CS; de Campos Velho Gewehr, C; de Oliveira, CV; Della-Pace, ID; dos Santos, AR; Ferreira, AP; Ferreira, J; Fighera, MR; Furian, AF; Mota, BC; Oliveira, MS; Oliveira, SM; Rodrigues, FS; Royes, LF1
Calixto, JB; Chichorro, JG; Luiz, AP; Rae, GA; Schroeder, SD1
Bicca, MA; Bitencourt, RM; Calixto, JB; de Mello, N; Guerra de Souza, AC; Medeiros, R; Pamplona, FA; Passos, GF; Prediger, RD; Takahashi, RN1
Dąbrowska-Bouta, B; Podsiadło, K; Strużyńska, L; Sulkowski, G1

Other Studies

97 other study(ies) available for bradykinin, leu(8)-des-arg(9)- and bradykinin

ArticleYear
Biological activities of photoaffinity labeling analogues of kinins and their irreversible effects on kinin receptors.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:12

    Topics: Affinity Labels; Animals; Binding, Competitive; In Vitro Techniques; Kinins; Muscle Contraction; Muscle, Smooth; Rabbits; Receptors, Bradykinin; Receptors, Cell Surface; Structure-Activity Relationship

1981
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cattle; Cloning, Molecular; COS Cells; DNA Primers; DNA, Complementary; Humans; Kallidin; Mice; Molecular Sequence Data; Rabbits; Receptor, Bradykinin B1; Receptors, Bradykinin; Sequence Homology, Amino Acid; Species Specificity; Transfection

1996
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
    The Journal of biological chemistry, 1997, Apr-25, Volume: 272, Issue:17

    Topics: Animals; Binding, Competitive; Biological Transport; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Inositol Phosphates; Kallidin; Ligands; Oligopeptides; Precipitin Tests; Protein Binding; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Recombinant Proteins; Signal Transduction; Type C Phospholipases

1997
Novel subtype-selective nonpeptide bradykinin receptor antagonists FR167344 and FR173657.
    Molecular pharmacology, 1997, Volume: 51, Issue:2

    Topics: Animals; Aorta; Bradykinin Receptor Antagonists; Cricetinae; Dose-Response Relationship, Drug; Humans; Kidney; Pyridines; Quinolines

1997
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
    European journal of pharmacology, 1999, Jun-25, Volume: 374, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Cloning, Molecular; COS Cells; DNA, Complementary; Female; Gene Expression; Genes; Humans; Kallidin; Molecular Sequence Data; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Tissue Distribution; Tritium

1999
Synthesis and biological evaluation of bradykinin B(1)/B(2) and selective B(1) receptor antagonists.
    Journal of medicinal chemistry, 2000, Jun-15, Volume: 43, Issue:12

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; CHO Cells; Cricetinae; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Structure-Activity Relationship; Transfection; Umbilical Veins

2000
Central bradykininergic system in normotensive and hypertensive rats.
    Clinical science (London, England : 1979), 1992, Volume: 82, Issue:5

    Topics: Animals; Blood Pressure; Bradykinin; Brain; Dose-Response Relationship, Drug; Heart Rate; Male; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Bradykinin; Receptors, Neurotransmitter

1992
The effects of bradykinin and sequence-related analogs on the response properties of cutaneous nociceptors in monkeys.
    Somatosensory & motor research, 1992, Volume: 9, Issue:2

    Topics: Afferent Pathways; Analgesics; Animals; Bradykinin; Evoked Potentials, Somatosensory; Macaca fascicularis; Nerve Fibers; Nerve Fibers, Myelinated; Nociceptors; Sensory Thresholds; Skin; Synaptic Transmission

1992
Non-selectivity of new bradykinin antagonists for B1 receptors.
    Life sciences, 1992, Volume: 51, Issue:11

    Topics: Amino Acid Sequence; Animals; Aorta; Binding, Competitive; Bradykinin; Guinea Pigs; Ileum; In Vitro Techniques; Jugular Veins; Kinetics; Molecular Sequence Data; Muscle, Smooth; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Tetrahydroisoquinolines

1992
Local production of kinins contributes to the endothelium dependent relaxations evoked by converting enzyme inhibitors in isolated arteries.
    Agents and actions. Supplements, 1992, Volume: 38 ( Pt 3)

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Arginine; Bradykinin; Carotid Arteries; Dogs; Endothelium, Vascular; In Vitro Techniques; Indoles; Indomethacin; Kininogens; Kinins; Muscle, Smooth, Vascular; Nitroarginine; Nitroprusside; Vasodilation

1992
Modulation of presynaptic sympathetic activity by kinins and related compounds: influence of converting enzyme inhibition.
    Agents and actions. Supplements, 1992, Volume: 38 ( Pt 3)

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Electric Stimulation; Epinephrine; Male; Norepinephrine; Ramipril; Rats; Rats, Inbred BN; Rats, Inbred SHR; Sympathetic Nervous System; Synapses

1992
Bradykinin receptors of cerebral microvessels stimulate phosphoinositide turnover.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1991, Volume: 11, Issue:4

    Topics: Animals; Binding, Competitive; Bradykinin; Brain; Hydrolysis; Inositol Phosphates; Male; Microcirculation; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Swine

1991
Kinin receptors mediating the effects of bradykinin on the coronary circulation in anaesthetized greyhounds.
    European journal of pharmacology, 1991, Apr-10, Volume: 196, Issue:1

    Topics: Animals; Blood Pressure; Bradykinin; Coronary Circulation; Coronary Vessels; Dogs; Fluoroacetates; Heart Rate; Receptors, Bradykinin; Receptors, Neurotransmitter; Reflex; Vagus Nerve; Vascular Resistance

1991
A bradykinin (BK)1 receptor antagonist blocks capsaicin-induced ear inflammation in mice.
    British journal of pharmacology, 1990, Volume: 99, Issue:3

    Topics: Animals; Bradykinin; Capsaicin; Ear, External; Edema; Inflammation; Male; Mice; Receptors, Bradykinin; Receptors, Neurotransmitter; Substance P

1990
[The contractile response of isolated lingual arteries from rabbits treated with bacterial lipopolysaccharide via the stimulation of B1-receptors for kinins].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 98, Issue:2

    Topics: Animals; Arteries; Bradykinin; Cycloheximide; Dactinomycin; Endotoxins; Escherichia coli; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Rabbits; Tongue

1991
Modification by some antagonists of the shape changes of venous endothelial cells in response to inflammatory agents in vitro.
    Agents and actions, 1990, Volume: 29, Issue:3-4

    Topics: Aminoquinolines; Animals; Bradykinin; Calcimycin; Calcium; Cimetidine; Endothelium, Vascular; Guinea Pigs; Histamine; Histamine Antagonists; Isoproterenol; Platelet Activating Factor; Pyrilamine; Vena Cava, Inferior

1990
Bradykinin-induced airway microvascular leakage and bronchoconstriction are mediated via a bradykinin B2 receptor.
    The American review of respiratory disease, 1990, Volume: 142, Issue:5

    Topics: Animals; Bradykinin; Bronchoconstriction; Capillary Permeability; Guinea Pigs; Male; Receptors, Bradykinin; Receptors, Neurotransmitter; Respiratory System

1990
The effects of bradykinin agonists and antagonists on visceral polymodal receptor activities.
    Pain, 1990, Volume: 40, Issue:2

    Topics: Animals; Bradykinin; Dogs; Epididymis; In Vitro Techniques; Male; Neurons, Afferent; Testis

1990
Bradykinin augments the in vitro migration of nonsensitized lymphocytes.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1989, Volume: 12, Issue:4

    Topics: Angiotensin II; Animals; Bradykinin; Chemotaxis, Leukocyte; Concanavalin A; Humans; Kallidin; Lymphocytes; Rats; Rats, Inbred Strains; Receptors, Bradykinin; Receptors, Neurotransmitter; Spleen

1989
Conversion of B1 kinin receptor-mediated vascular relaxation to contraction.
    Hypertension (Dallas, Tex. : 1979), 1987, Volume: 9, Issue:6 Pt 2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Bradykinin; Dose-Response Relationship, Drug; Indomethacin; Kallidin; Male; Pyrazoles; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Vasoconstriction; Vasodilation

1987
Activation of a bradykinin receptor in peripheral nerve and spinal cord in the neonatal rat in vitro.
    British journal of pharmacology, 1988, Volume: 95, Issue:4

    Topics: Animals; Animals, Newborn; Bradykinin; In Vitro Techniques; Membrane Potentials; Peripheral Nerves; Rats; Receptors, Bradykinin; Receptors, Neurotransmitter; Spinal Cord

1988
Mitogenic effect of bradykinin and of des-Arg9-bradykinin on cultured fibroblasts.
    Life sciences, 1986, Dec-15, Volume: 39, Issue:24

    Topics: Animals; Bradykinin; Dinoprostone; Fibroblasts; Humans; Mitosis; Prostaglandins E; Rabbits; Thymidine

1986
Bradykinin analogue blocks bradykinin-induced inhibition of a spinal nociceptive reflex in the rat.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: Animals; Bradykinin; Male; Nociceptors; Rats; Rats, Inbred Strains; Reaction Time; Reflex; Spinal Cord

1987
Contractile effects of bradykinin on the isolated human small bronchus.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Acetylcholine; Aged; Atropine; Benzamides; Biphenyl Compounds; Bradykinin; Bronchi; Bronchoconstriction; Capsaicin; Humans; In Vitro Techniques; Indomethacin; Middle Aged; Muscle, Smooth; Nerve Fibers; Neurokinin A; Neurons, Afferent; Piperidines; Receptors, Bradykinin; Ruthenium Red; Tetrodotoxin

1994
Modulatory effect of bradykinin on the release of noradrenaline from rat isolated atria.
    British journal of pharmacology, 1995, Volume: 115, Issue:2

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Angiotensin II; Animals; Bradykinin; Diclofenac; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Fenoterol; Heart Atria; Indoles; Male; Maleimides; Norepinephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar

1995
Effect of bradykinin and prostaglandins on the release of calcitonin gene-related peptide-like immunoreactivity from the rat spinal cord in vitro.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Amino Acid Sequence; Animals; Bradykinin; Calcitonin Gene-Related Peptide; Colforsin; Electric Stimulation; Female; In Vitro Techniques; Indomethacin; Male; Molecular Sequence Data; Prostaglandins; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Spinal Cord

1993
[Leu8]des-Arg9-bradykinin inhibits the angiogenic effect of bradykinin and interleukin-1 in rats.
    British journal of pharmacology, 1993, Volume: 109, Issue:1

    Topics: Animals; Bradykinin; Hemoglobins; Humans; Inflammation; Interleukin-1; Male; Neovascularization, Pathologic; Rats; Rats, Wistar; Receptors, Bradykinin; Receptors, Neurotransmitter; Recombinant Proteins

1993
Modulation of bradykinin-induced intracellular Ca2+ oscillations in v-Ki-ras-transformed fibroblasts.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:6

    Topics: 3T3 Cells; Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium Channels; Calcium-Transporting ATPases; Genes, ras; Mice; Terpenes; Thapsigargin

1994
Bradykinin B1 receptors in the rabbit urinary bladder: induction of responses, smooth muscle contraction, and phosphatidylinositol hydrolysis.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Amino Acid Sequence; Animals; Bradykinin; Hydrolysis; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Rabbits; Receptors, Bradykinin; Urinary Bladder

1995
A hypotensive response induced by des-Arg9-bradykinin in young brown/Norway rats pretreated with endotoxin.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Amino Acid Sequence; Analysis of Variance; Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Drug Interactions; Escherichia coli; Hypotension; Lipopolysaccharides; Male; Molecular Sequence Data; Rats; Rats, Inbred BN; Specific Pathogen-Free Organisms

1995
The involvement of bradykinin B1 and B2 receptor mechanisms in cytokine-induced mechanical hyperalgesia in the rat.
    British journal of pharmacology, 1994, Volume: 113, Issue:1

    Topics: Animals; Bradykinin; Cytokines; Female; Hyperalgesia; Indomethacin; Injections, Intra-Articular; Interleukins; Knee Joint; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin

1994
Bradykinin B2 receptors and coupling mechanisms in the smooth muscle of the guinea-pig taenia caeci.
    British journal of pharmacology, 1994, Volume: 113, Issue:2

    Topics: Amino Acid Sequence; Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Cecum; Culture Media; Guinea Pigs; Hydrolysis; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phosphatidylinositols; Potassium; Receptors, Bradykinin; Sodium

1994
Mediation by bradykinin of rat paw oedema induced by collagenase from Clostridium histolyticum.
    British journal of pharmacology, 1994, Volume: 112, Issue:2

    Topics: Animals; Biphenyl Compounds; Bradykinin; Capillary Permeability; Capsaicin; Edema; Female; Foot; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypnotics and Sedatives; Microbial Collagenase; Motor Activity; Neurokinin-1 Receptor Antagonists; Rats; Rats, Sprague-Dawley

1994
Bradykinin-stimulated calcium mobilization in cultured canine tracheal smooth muscle cells.
    Cell calcium, 1994, Volume: 16, Issue:2

    Topics: Animals; Bradykinin; Calcium; Carbachol; Cells, Cultured; Diltiazem; Dogs; Dose-Response Relationship, Drug; Egtazic Acid; Female; Fura-2; Kallidin; Male; Muscle, Smooth; Trachea; Verapamil

1994
Effects of bradykinin on the canine proximal colon.
    Regulatory peptides, 1993, Jul-23, Volume: 46, Issue:3

    Topics: Amino Acid Sequence; Animals; Bradykinin; Colon; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Epithelium; Female; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Male; Molecular Sequence Data; Tetrodotoxin

1993
Antinociceptive activity of the bradykinin B1 and B2 receptor antagonists, des-Arg9, [Leu8]-BK and HOE 140, in two models of persistent hyperalgesia in the rat.
    Pain, 1993, Volume: 53, Issue:2

    Topics: Analgesics; Animals; Bradykinin; Disease Models, Animal; Female; Freund's Adjuvant; Hindlimb; Hot Temperature; Hyperalgesia; Inflammation; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Bradykinin; Receptors, Neurotransmitter; Ultraviolet Rays

1993
Cloned murine bradykinin receptor exhibits a mixed B1 and B2 pharmacological selectivity.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bradykinin; Cell Line; Cloning, Molecular; DNA; Humans; Mice; Molecular Sequence Data; Oocytes; Polymerase Chain Reaction; Rats; Receptors, Bradykinin; Receptors, Neurotransmitter; Transfection; Tumor Cells, Cultured; Xenopus laevis

1993
Endothelium-dependent relaxations mediated by inducible B1 and constitutive B2 kinin receptors in the bovine isolated coronary artery.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arginine; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Coronary Vessels; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitroarginine; Protein Synthesis Inhibitors

1995
Involvement of bradykinin B1 receptors in the polymorphonuclear leukocyte accumulation induced by IL-1 beta in vivo in the mouse.
    Journal of immunology (Baltimore, Md. : 1950), 1996, Jan-01, Volume: 156, Issue:1

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Chemotaxis, Leukocyte; Interleukin-1; Male; Mice; Neutrophil Activation; Neutrophils; Receptors, Bradykinin

1996
Effects of bradykinin on the intracellular calcium concentration of pancreatic acinar AR42J cells.
    Life sciences, 1996, Volume: 58, Issue:18

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Cell Line; Dexamethasone; Dose-Response Relationship, Drug; Intracellular Fluid; Neomycin; Pancreas; Rats

1996
The longitudinal muscle of rat ileum as a sensitive monoreceptor assay for bradykinin B1 receptors.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Animals; Bradykinin; Guinea Pigs; Ileum; Male; Muscle, Smooth; Rats; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Tetrahydroisoquinolines; Urinary Bladder

1996
Inducible bradykinin B1 receptor in isolated human ileum.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Bradykinin; Humans; Ileum; In Vitro Techniques; Kallidin; Muscle Contraction; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

1996
The role of the kallikrein-kinin system in type I diabetes (insulitis).
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Kallikrein-Kinin System; Male; Mice; Mice, Inbred C57BL; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

1996
Stimulus properties and antinociceptive effects of selective bradykinin B1 and B2 receptor antagonists in rats.
    Pain, 1996, Volume: 66, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Bradykinin Receptor Antagonists; Choice Behavior; Dose-Response Relationship, Drug; Formaldehyde; Male; Nociceptors; Rats; Rats, Sprague-Dawley; Stimulation, Chemical

1996
Effects of B1 and B2 kinin receptor antagonists in diabetic mice.
    Canadian journal of physiology and pharmacology, 1996, Volume: 74, Issue:5

    Topics: Analysis of Variance; Animals; Blood Glucose; Body Weight; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Male; Mice; Mice, Inbred C57BL; Streptozocin

1996
Different B1 kinin receptor expression and pharmacology in endothelial cells of different origins and species.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Aorta; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Coronary Vessels; Cyclic GMP; DNA Primers; Endothelium, Vascular; Humans; Microcirculation; Naphthalenes; Organophosphorus Compounds; Polymerase Chain Reaction; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Species Specificity; Transcription, Genetic; Umbilical Veins

1997
Bradykinin B1 receptors in human umbilical vein.
    European journal of pharmacology, 1997, Feb-19, Volume: 321, Issue:1

    Topics: Anti-Inflammatory Agents; Bradykinin; Bradykinin Receptor Antagonists; Cyclooxygenase Inhibitors; Dexamethasone; Female; Humans; In Vitro Techniques; Muscle Contraction; Pregnancy; Receptor, Bradykinin B1; Receptors, Bradykinin; Umbilical Veins; Up-Regulation

1997
Bradykinin-induced knee joint incapacitation involves bradykinin B2 receptor mediated hyperalgesia and bradykinin B1 receptor-mediated nociception.
    European journal of pharmacology, 1997, May-12, Volume: 326, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis; Behavior, Animal; Bradykinin; Bradykinin Receptor Antagonists; Dinoprostone; Hindlimb; Hyperalgesia; Indomethacin; Joints; Male; Nociceptors; Pain Measurement; Rats; Rats, Wistar; Receptors, Bradykinin

1997
Effects of the bradykinin B1 receptor antagonist des-Arg9[Leu8]bradykinin and genetic disruption of the B2 receptor on nociception in rats and mice.
    Pain, 1997, Volume: 71, Issue:1

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Carrageenan; Edema; Female; Formaldehyde; Freund's Adjuvant; Hindlimb; Male; Mice; Mice, Transgenic; Nociceptors; Pain; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Reflex

1997
Induction of bradykinin B1 receptors in rat colonic epithelium.
    British journal of pharmacology, 1997, Volume: 121, Issue:5

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Chloride Channels; Colon; Cycloheximide; Cystic Fibrosis Transmembrane Conductance Regulator; Dactinomycin; Epithelial Cells; Epithelium; In Vitro Techniques; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Transcription, Genetic

1997
Evidence for bradykinin B2-receptors on cultured human decidua cells.
    Immunopharmacology, 1997, Volume: 36, Issue:2-3

    Topics: Adrenergic beta-Antagonists; Base Sequence; Binding, Competitive; Bradykinin; Bradykinin Receptor Antagonists; Cells, Cultured; Decidua; Electrophoresis, Polyacrylamide Gel; Female; Humans; Immunohistochemistry; Inflammation; Isotope Labeling; Labor, Induced; Molecular Sequence Data; Polymerase Chain Reaction; Pregnancy; Radioligand Assay; Receptor, Bradykinin B2; Receptors, Bradykinin; RNA, Messenger; Tritium

1997
Expression of bradykinin B1 receptors in colonic epithelia.
    Immunopharmacology, 1997, Volume: 36, Issue:2-3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Chlorides; Colon; Cycloheximide; Dactinomycin; Diuretics; Epithelium; Furosemide; In Vitro Techniques; Ion Channels; Ion Transport; Lethal Dose 50; Protein Biosynthesis; Protein Synthesis Inhibitors; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Transcription, Genetic

1997
Daily variation in an intensity of kaolin-induced writhing reaction in mice.
    Life sciences, 1997, Volume: 61, Issue:13

    Topics: Analgesia; Animals; Bradykinin; Bradykinin Receptor Antagonists; Circadian Rhythm; Kaolin; Kinetics; Male; Mice; Mice, Inbred ICR; Pain; Photoperiod

1997
PGE2 release by bradykinin in human airway smooth muscle cells: involvement of cyclooxygenase-2 induction.
    The American journal of physiology, 1997, Volume: 273, Issue:6

    Topics: Adult; Arachidonic Acid; Bradykinin; Bradykinin Receptor Antagonists; Cell Survival; Cells, Cultured; Cyclooxygenase 2; Dinoprostone; Enzyme Induction; Female; Humans; Isoenzymes; Kinetics; Male; Membrane Proteins; Middle Aged; Muscle, Smooth; Prostaglandin-Endoperoxide Synthases; Receptors, Bradykinin; Trachea

1997
Smokeless tobacco-exposed oral keratinocytes increase macromolecular efflux from the in situ oral mucosa.
    The American journal of physiology, 1998, Volume: 274, Issue:1

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Cells, Cultured; Cheek; Cricetinae; Dextrans; Fluorescein-5-isothiocyanate; Humans; Keratinocytes; Kinetics; Leupeptins; Male; Mesocricetus; Microcirculation; Mouth Mucosa; Plants, Toxic; Tobacco, Smokeless

1998
Biphasic response to bradykinin in isolated porcine iliac arteries is mediated by bradykinin B1 and B2 receptors.
    Journal of cardiovascular pharmacology, 1998, Volume: 31, Issue:2

    Topics: 3-Mercaptopropionic Acid; Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cilazapril; Cycloheximide; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Enalaprilat; Endothelium, Vascular; Enzyme Inhibitors; Iliac Artery; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Protease Inhibitors; Protein Synthesis Inhibitors; Receptors, Bradykinin; Swine; Vasoconstriction; Vasodilation

1998
Characterisation of kinin receptors on the human isolated umbilical artery.
    The Journal of endocrinology, 1998, Volume: 156, Issue:2

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Bradykinin; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Adrenergic, beta-1; Umbilical Arteries

1998
Effect of WIN 64338, a B2 bradykinin receptor antagonist on guinea-pig tracheal smooth muscle cells in culture.
    Fundamental & clinical pharmacology, 1998, Volume: 12, Issue:2

    Topics: Adrenergic beta-Antagonists; Analgesics; Animals; Binding, Competitive; Bradykinin; Bradykinin Receptor Antagonists; Cells, Cultured; Fluorescent Antibody Technique; Guinea Pigs; Inositol Phosphates; Male; Muscle, Smooth; Naphthalenes; Oligopeptides; Organophosphorus Compounds; Receptor, Bradykinin B2; Receptors, Bradykinin; Trachea

1998
The modulatory effects of bradykinin B1 and B2 receptor antagonists upon viscero-visceral hyper-reflexia in a rat model of visceral hyperalgesia.
    Pain, 1998, Volume: 75, Issue:2-3

    Topics: Adrenergic beta-Antagonists; Animals; Bradykinin; Bradykinin Receptor Antagonists; Coloring Agents; Cystitis; Evans Blue; Female; Hyperalgesia; Rats; Rats, Wistar; Reflex, Abnormal; Urinary Bladder; Viscera

1998
B1 kinin receptor activity in pigs is associated with pre-existing infection.
    Immunopharmacology, 1998, Volume: 40, Issue:1

    Topics: Acetylcholine; Animals; Bacterial Infections; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Gram-Negative Bacteria; Heart Rate; Lipopolysaccharides; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Swine

1998
Systemic treatment with Mycobacterium bovis bacillus Calmette-Guérin (BCG) potentiates kinin B1 receptor agonist-induced nociception and oedema formation in the formalin test in mice.
    Neuropeptides, 1998, Volume: 32, Issue:5

    Topics: Animals; Bradykinin; Dexamethasone; Dose-Response Relationship, Drug; Drug Synergism; Edema; Formaldehyde; Hindlimb; Indomethacin; Kallidin; Male; Mice; Mycobacterium bovis; Pain; Pain Measurement; Pyrazoles; Receptor, Bradykinin B1; Receptors, Bradykinin

1998
Kinin B1 receptor antagonists containing alpha-methyl-L-phenylalanine: in vitro and in vivo antagonistic activities.
    Hypertension (Dallas, Tex. : 1979), 1999, Volume: 33, Issue:3

    Topics: Animals; Blood Pressure; Bradykinin; Humans; Kallidin; Peptides; Peptidyl-Dipeptidase A; Phenylalanine; Plasma; Rabbits; Receptors, Neurokinin-3; Time Factors

1999
Bradykinin B1 and B2 receptors, tumour necrosis factor alpha and inflammatory hyperalgesia.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Bradykinin; Bradykinin Receptor Antagonists; Carrageenan; Dinoprostone; Dose-Response Relationship, Drug; Drug Synergism; Hyperalgesia; Indomethacin; Inflammation; Interleukin-8; Kallidin; Lipopolysaccharides; Male; Mice; Pain Measurement; Pain Threshold; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Sheep; Time Factors; Tumor Necrosis Factor-alpha

1999
Response of fetal rabbit ductus arteriosus to bradykinin: role of nitric oxide, prostaglandins, and bradykinin receptors.
    Pediatric research, 1999, Volume: 45, Issue:4 Pt 1

    Topics: Animals; Animals, Newborn; Bradykinin; Dinoprostone; Ductus Arteriosus; Endothelium, Vascular; Female; In Vitro Techniques; Isometric Contraction; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; omega-N-Methylarginine; Pregnancy; Prostaglandins; Rabbits; Receptors, Bradykinin

1999
Tumour necrosis factor-alpha mediates carrageenin-induced knee-joint incapacitation and also triggers overt nociception in previously inflamed rat knee-joints.
    Pain, 1999, Volume: 82, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis; Bradykinin; Bradykinin Receptor Antagonists; Carrageenan; Dinoprostone; Inflammation Mediators; Injections, Intra-Articular; Knee Joint; Male; Pain; Rats; Rats, Wistar; Stimulation, Chemical; Substance P; Tumor Necrosis Factor-alpha

1999
Neurokinin-1 receptor agonists are involved in mediating neutrophil accumulation in the inflamed, but not normal, cutaneous microvasculature: an in vivo study using neurokinin-1 receptor knockout mice.
    Journal of immunology (Baltimore, Md. : 1950), 2000, May-15, Volume: 164, Issue:10

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Carrageenan; Cell Movement; Drug Combinations; Female; Injections, Intradermal; Injections, Intravenous; Interleukin-1; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Microcirculation; Neutrophils; Receptors, Neurokinin-1; Skin; Substance P; Zymosan

2000
Increased mRNA expression of the B1 and B2 bradykinin receptors and antinociceptive effects of their antagonists in an animal model of neuropathic pain.
    Pain, 2000, Volume: 86, Issue:3

    Topics: Animals; Bradykinin; Constriction, Pathologic; Ganglia, Spinal; Hot Temperature; Lumbosacral Region; Male; Nervous System Diseases; Nociceptors; Pain; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; RNA, Messenger; Sciatic Nerve; Wounds and Injuries

2000
Lipopolysaccharide decreases bradykinin receptor-induced acidification responses in cultured bovine aortic endothelial cells.
    European journal of pharmacology, 2000, Aug-18, Volume: 402, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Endothelium, Vascular; Endotoxins; Lipopolysaccharides; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin

2000
Targeting kinin B(1) receptor for therapeutic neovascularization.
    Circulation, 2002, Jan-22, Volume: 105, Issue:3

    Topics: Animals; Apoptosis; Bradykinin; Bradykinin Receptor Antagonists; Cell Division; Cells, Cultured; Endothelium, Vascular; Extremities; Humans; Ischemia; Laser-Doppler Flowmetry; Mice; Mice, Knockout; Muscle, Skeletal; Neovascularization, Physiologic; Perfusion; Receptor, Bradykinin B1; Receptors, Bradykinin; Signal Transduction

2002
Combined action of vasoactive amines and bradykinin mediates allergen-evoked thermal hyperalgesia in rats.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: Allergens; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cyproheptadine; Dinitrophenols; Dose-Response Relationship, Drug; Drug Synergism; Edema; Histamine; Histamine H1 Antagonists; Hyperalgesia; Immunoglobulin E; Male; Meclizine; Methysergide; Pain; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Serum Albumin, Bovine; Time Factors

2003
Bradykinin receptor subtype 1 expression and function in prostate cancer.
    Cancer research, 2003, May-01, Volume: 63, Issue:9

    Topics: Biopsy; Bradykinin; Bradykinin Receptor Antagonists; Cell Division; Cell Movement; Enzyme Activation; Humans; Male; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neoplasm Invasiveness; Prostatic Neoplasms; Receptors, Bradykinin; Signal Transduction

2003
Kinins are involved in the development of allergic nasal hyperresponsiveness in guinea pigs.
    European journal of pharmacology, 2003, Aug-29, Volume: 476, Issue:3

    Topics: Airway Resistance; Allergens; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Guinea Pigs; Kallidin; Kinins; Leukotriene D4; Male; Nasal Lavage Fluid; Pollen; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Rhinitis, Allergic, Seasonal; Time Factors

2003
Bradykinin B1 receptor stimulates the proximal tubule Na(+)-ATPase activity through protein kinase C pathway.
    Regulatory peptides, 2003, Oct-15, Volume: 115, Issue:3

    Topics: Adenosine Triphosphatases; Animals; Bradykinin; Cation Transport Proteins; Enzyme Inhibitors; Kidney Tubules, Proximal; Naphthalenes; Phosphatidylinositols; Phosphorylation; Phosphoserine; Protein Kinase C; Receptor, Bradykinin B1; Swine

2003
Converting enzyme inhibitor temocaprilat prevents high glucose-mediated suppression of human aortic endothelial cell proliferation.
    Journal of cardiovascular pharmacology, 2003, Volume: 42 Suppl 1

    Topics: Alkaloids; Angiotensin-Converting Enzyme Inhibitors; Aorta; Benzophenanthridines; Bradykinin; Bradykinin B2 Receptor Antagonists; Cell Division; Cell Membrane; Cells, Cultured; Coronary Vessels; Dose-Response Relationship, Drug; Endothelial Cells; Glucose; Humans; Naphthalenes; Oxidative Stress; Phenanthridines; Protein Kinase C; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Thiazepines; Time Factors

2003
Involvement of bradykinin, cytokines, sympathetic amines and prostaglandins in formalin-induced orofacial nociception in rats.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: Animals; Arachidonic Acids; Atenolol; Behavior, Animal; Biogenic Amines; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Captopril; Celecoxib; Cytokines; Dose-Response Relationship, Drug; Drug Synergism; Facial Pain; Formaldehyde; Guanethidine; Hindlimb; Indomethacin; Injections, Subcutaneous; Interleukin-6; Interleukin-8; Lip; Male; Meloxicam; Nociceptors; Prostaglandins; Pyrazoles; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Sulfonamides; Thiazines; Thiazoles; Tumor Necrosis Factor-alpha; Tyramine

2004
Bradykinin antagonists have no analgesic effect on incisional pain.
    Anesthesia and analgesia, 2004, Volume: 99, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Bradykinin; Dose-Response Relationship, Drug; Foot; Hot Temperature; Male; Pain Measurement; Pain, Postoperative; Physical Stimulation; Rats; Rats, Sprague-Dawley

2004
Reduced nerve injury-induced neuropathic pain in kinin B1 receptor knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Mar-02, Volume: 25, Issue:9

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Female; Functional Laterality; Gene Expression; Hyperalgesia; Male; Mice; Mice, Knockout; Neuralgia; Pain Measurement; Receptor, Bradykinin B1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sciatic Neuropathy; Skin; Skin Temperature; Time Factors

2005
Estrogens and glucocorticoids have opposing effects on the amount and latent activity of complement proteins in the rat uterus.
    Biology of reproduction, 2006, Volume: 74, Issue:2

    Topics: Animals; Body Fluids; Bradykinin; Complement C1 Inactivator Proteins; Complement C1 Inhibitor Protein; Complement System Proteins; Dexamethasone; Escherichia coli; Estradiol; Estrogens; Female; Glucocorticoids; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Serpins; Uterus

2006
Ca2+-dependent K+ channels are targets for bradykinin B1 receptor ligands and for lipopolysaccharide in the rat aorta.
    European journal of pharmacology, 2005, Nov-21, Volume: 525, Issue:1-3

    Topics: Animals; Aorta; Bradykinin; Bradykinin B1 Receptor Antagonists; Calcium; Calcium-Transporting ATPases; In Vitro Techniques; Kallidin; Ligands; Lipopolysaccharides; Male; Membrane Potentials; Myocytes, Smooth Muscle; Peptides; Potassium Channels, Calcium-Activated; Rats; Rats, Wistar; Receptor, Bradykinin B1; Thapsigargin

2005
Analgesic efficacy of bradykinin B1 antagonists in a murine bone cancer pain model.
    The journal of pain, 2005, Volume: 6, Issue:11

    Topics: Animals; Bone Neoplasms; Bradykinin; Bradykinin B1 Receptor Antagonists; Injections, Subcutaneous; Male; Mice; Mice, Inbred C3H; Neoplasm Transplantation; Pain; Sarcoma

2005
Prostaglandin involvement in lung C-fiber activation by substance P in guinea pigs.
    Journal of applied physiology (Bethesda, Md. : 1985), 2006, Volume: 100, Issue:6

    Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Asthma; Blood Pressure; Bradykinin; Capsaicin; Cyclooxygenase Inhibitors; Dinoprost; Dinoprostone; Guinea Pigs; Heart Rate; Indomethacin; Lung; Nerve Fibers, Unmyelinated; Prostaglandins; Respiratory Hypersensitivity; Substance P

2006
Peripheral kinin B(1) and B(2) receptor-operated mechanisms are implicated in neuropathic nociception induced by spinal nerve ligation in rats.
    Neuropharmacology, 2007, Volume: 53, Issue:1

    Topics: Animals; Behavior, Animal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Drug Administration Routes; Functional Laterality; Hyperalgesia; Ligation; Male; Neuralgia; Pain Measurement; Pain Threshold; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Spinal Nerves; Time Factors

2007
TNF-alpha and IL-1beta mediate inflammatory hypernociception in mice triggered by B1 but not B2 kinin receptor.
    European journal of pharmacology, 2007, Nov-14, Volume: 573, Issue:1-3

    Topics: Animals; Antibodies; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Bradykinin Receptor Antagonists; Carrageenan; Dose-Response Relationship, Drug; Guanethidine; Hyperalgesia; Indomethacin; Inflammation; Interleukin-1beta; Lipopolysaccharides; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Prostaglandins; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Tumor Necrosis Factor, Type I; Tumor Necrosis Factor-alpha

2007
Bradykinin-induced microglial migration mediated by B1-bradykinin receptors depends on Ca2+ influx via reverse-mode activity of the Na+/Ca2+ exchanger.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Nov-28, Volume: 27, Issue:48

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Calcium; Cell Movement; Cells, Cultured; Cerebellar Cortex; Chemotaxis; Dose-Response Relationship, Drug; Mice; Mice, Knockout; Microglia; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Signal Transduction; Sodium-Calcium Exchanger; Time Factors

2007
Role of bradykinin, nitric oxide, and angiotensin II type 2 receptor in imidapril-induced angiogenesis.
    Hypertension (Dallas, Tex. : 1979), 2008, Volume: 51, Issue:2

    Topics: Angiogenesis Inducing Agents; Angiotensin II Type 2 Receptor Blockers; Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Capillaries; Enzyme Inhibitors; Hindlimb; Imidazoles; Imidazolidines; Ischemia; Male; Mice; Mice, Knockout; Neovascularization, Physiologic; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type III; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; RNA, Messenger; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factor Receptor-2

2008
Genetic deletion or antagonism of kinin B(1) and B(2) receptors improves cognitive deficits in a mouse model of Alzheimer's disease.
    Neuroscience, 2008, Feb-06, Volume: 151, Issue:3

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Analysis of Variance; Animals; Behavior, Animal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cerebral Cortex; Cognition Disorders; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Hippocampus; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Peptide Fragments; Reaction Time; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Time Factors

2008
Kinin B(1) and B(2) receptors contribute to orofacial heat hyperalgesia induced by infraorbital nerve constriction injury in mice and rats.
    Neuropeptides, 2010, Volume: 44, Issue:2

    Topics: Analysis of Variance; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cranial Nerve Injuries; Facial Pain; Hot Temperature; Hyperalgesia; Male; Maxillary Nerve; Mice; Pain Measurement; Pain Threshold; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2010
Bradykinin increases the secretion and expression of endothelin-1 through kinin B2 receptors in melanoma cells.
    Peptides, 2010, Volume: 31, Issue:2

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Cell Line, Tumor; Endothelin-1; Gene Expression; Gene Expression Regulation, Neoplastic; Melanoma, Experimental; Mice; Receptor, Bradykinin B1; Receptor, Bradykinin B2

2010
The role of kinin B1 and B2 receptors in the scratching behaviour induced by proteinase-activated receptor-2 agonists in mice.
    British journal of pharmacology, 2010, Volume: 159, Issue:4

    Topics: Animals; Antipruritics; Behavior, Animal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dioxoles; Disease Models, Animal; Dose-Response Relationship, Drug; Injections, Intradermal; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Spinal; Mice; Mice, Inbred C57BL; Mice, Knockout; Oligopeptides; Pain Threshold; Pruritus; Quinolines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptor, PAR-2; Sulfonamides; Trypsin

2010
Attenuation of persistent experimental pancreatitis pain by a bradykinin b2 receptor antagonist.
    Pancreas, 2010, Volume: 39, Issue:8

    Topics: Abdominal Pain; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dynorphins; Ganglia, Spinal; Gene Expression; Immune Sera; Injections, Intraperitoneal; Injections, Intravenous; Injections, Spinal; Male; Organotin Compounds; Pain; Pancreas; Pancreatitis; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Reverse Transcriptase Polymerase Chain Reaction; Spinal Cord

2010
Bradykinin receptor 1 activation exacerbates experimental focal and segmental glomerulosclerosis.
    Kidney international, 2011, Volume: 79, Issue:11

    Topics: Actinin; Albuminuria; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Disease Models, Animal; Doxorubicin; Gene Expression Regulation; Glomerulosclerosis, Focal Segmental; Heme Oxygenase-1; Interleukin-1beta; Intracellular Signaling Peptides and Proteins; Macrophages; Male; Matrix Metalloproteinase 9; Membrane Proteins; Mice; Mice, Inbred BALB C; Podocytes; Receptor, Bradykinin B1; RNA, Messenger; Signal Transduction; Time Factors; Tissue Inhibitor of Metalloproteinase-1

2011
Anti-nociceptive effect of kinin B₁ and B₂ receptor antagonists on peripheral neuropathy induced by paclitaxel in mice.
    British journal of pharmacology, 2011, Volume: 164, Issue:2b

    Topics: Analgesics; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Hyperalgesia; Kinins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Paclitaxel; Peripheral Nervous System Diseases; Receptor, Bradykinin B1; Receptor, Bradykinin B2; RNA, Messenger

2011
Exacerbation of DSS-induced colitis in mice lacking kinin B(1) receptors through compensatory up-regulation of kinin B(2) receptors: the role of tight junctions and intestinal homeostasis.
    British journal of pharmacology, 2013, Volume: 168, Issue:2

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Colitis; Cytokines; Dextran Sulfate; Dioxoles; Homeostasis; Intestinal Mucosa; Intestines; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Peroxidase; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Sulfonamides; Tight Junctions; Up-Regulation

2013
HOE-140, an antagonist of B2 receptor, protects against memory deficits and brain damage induced by moderate lateral fluid percussion injury in mice.
    Psychopharmacology, 2014, Volume: 231, Issue:9

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Brain; Brain Edema; Brain Injuries; Disease Models, Animal; Male; Maze Learning; Memory Disorders; Mice; Motor Activity; NADPH Oxidases; Neuroprotective Agents; Oxidative Stress; Recognition, Psychology; Time Factors

2014
Contribution and interaction of kinin receptors and dynorphin A in a model of trigeminal neuropathic pain in mice.
    Neuroscience, 2015, Aug-06, Volume: 300

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Disease Models, Animal; Dynorphins; Facial Pain; Hot Temperature; Hyperalgesia; Male; Mice, Inbred C57BL; Mice, Knockout; Neuralgia; Neurotransmitter Agents; Pain Measurement; Receptors, Bradykinin; Touch

2015
Blockade of hippocampal bradykinin B1 receptors improves spatial learning and memory deficits in middle-aged rats.
    Behavioural brain research, 2017, 01-01, Volume: 316

    Topics: Aging; Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Disease Models, Animal; Hippocampus; Male; Maze Learning; Memory Disorders; Rats; Rats, Wistar; Receptor, Bradykinin B1; Spatial Learning; Up-Regulation

2017
Blockade of the kinin B1 receptor affects the cytokine/chemokine profile in rat brain subjected to autoimmune encephalomyelitis.
    Inflammopharmacology, 2017, Volume: 25, Issue:4

    Topics: Animals; Bradykinin; Bradykinin B1 Receptor Antagonists; Brain; Chemokines; Cytokines; Encephalomyelitis, Autoimmune, Experimental; Female; Rats; Rats, Inbred Lew; Receptor, Bradykinin B1

2017