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bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- and bradykinin

bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- has been researched along with bradykinin in 8 studies

Compound Research Comparison

Studies
(bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-)
Trials
(bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-)
Recent Studies (post-2010)
(bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
80114,1953551,520

Protein Interaction Comparison

ProteinTaxonomybradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (62.50)18.2507
2000's2 (25.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gobeil, F; Regoli, D; Rhaleb, NE1
Schölkens, BA; Wiemer, G; Wirth, KJ1
Lecci, A; Maggi, CA; Meini, S1
Domingues-Costa, A; Magina, S; Moura, D; Vaz-da-Silva, M1
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Tramontana, M1
Greco, S; Marsigliante, S; Storelli, C1
Bujalska, M; Makulska-Nowak, H1
Bogo, MR; Campos, MM; Couture, R; Dias, JP; Gaudreau, P; Lahjouji, K; Talbot, S1

Other Studies

8 other study(ies) available for bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- and bradykinin

ArticleYear
Non-selectivity of new bradykinin antagonists for B1 receptors.
    Life sciences, 1992, Volume: 51, Issue:11

    Topics: Amino Acid Sequence; Animals; Aorta; Binding, Competitive; Bradykinin; Guinea Pigs; Ileum; In Vitro Techniques; Jugular Veins; Kinetics; Molecular Sequence Data; Muscle, Smooth; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Tetrahydroisoquinolines

1992
DesArg10[Hoe 140] is a potent B1 bradykinin antagonist.
    Agents and actions. Supplements, 1992, Volume: 38 ( Pt 2)

    Topics: Animals; Aorta; Bradykinin; Duodenum; Endothelium, Vascular; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Pulmonary Artery; Rabbits; Rats; Receptors, Bradykinin; Receptors, Neurotransmitter; Tetrahydroisoquinolines

1992
The longitudinal muscle of rat ileum as a sensitive monoreceptor assay for bradykinin B1 receptors.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Animals; Bradykinin; Guinea Pigs; Ileum; Male; Muscle, Smooth; Rats; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Tetrahydroisoquinolines; Urinary Bladder

1996
The role of the endocardium in the facilitatory effect of bradykinin on electrically-induced release of noradrenaline in rat cardiac ventricle.
    British journal of pharmacology, 1996, Volume: 118, Issue:2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Captopril; Electric Stimulation; Endocardium; Heart Ventricles; In Vitro Techniques; Male; Norepinephrine; Rats; Rats, Wistar; Tetrahydroisoquinolines; Ventricular Function

1996
Kinin B1 receptor-mediated motor responses in normal or inflamed rat urinary bladder in vivo.
    Regulatory peptides, 1999, Mar-17, Volume: 80, Issue:1-2

    Topics: Administration, Topical; Anesthetics, Intravenous; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Bradykinin Receptor Antagonists; Cyclophosphamide; Cystitis; Dose-Response Relationship, Drug; Ganglia, Parasympathetic; Ganglionectomy; Male; Muscle Contraction; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Reference Values; Tetrahydroisoquinolines; Urethane; Urinary Bladder

1999
Protein kinase C (PKC)-delta/-epsilon mediate the PKC/Akt-dependent phosphorylation of extracellular signal-regulated kinases 1 and 2 in MCF-7 cells stimulated by bradykinin.
    The Journal of endocrinology, 2006, Volume: 188, Issue:1

    Topics: Analysis of Variance; Biological Transport; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Breast Neoplasms; Cell Line, Tumor; Cell Membrane; Cell Proliferation; Chromones; Cytosol; Dose-Response Relationship, Drug; Estrenes; Female; Flavonoids; Humans; Immunoblotting; Indoles; Kallidin; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Morpholines; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-delta; Protein Kinase C-epsilon; Pyrrolidinones; Stimulation, Chemical; Tetrahydroisoquinolines

2006
Bradykinin receptors antagonists and nitric oxide synthase inhibitors in vincristine and streptozotocin induced hyperalgesia in chemotherapy and diabetic neuropathy rat model.
    Neuro endocrinology letters, 2009, Volume: 30, Issue:1

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Drug Evaluation, Preclinical; Enzyme Inhibitors; Hyperalgesia; Hypoglycemic Agents; Indazoles; Lysine; Male; Nitric Oxide Synthase; Nitroarginine; Pain Measurement; Rats; Rats, Wistar; Receptors, Bradykinin; Streptozocin; Tetrahydroisoquinolines; Vincristine

2009
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
    Journal of neuroinflammation, 2012, Jan-20, Volume: 9

    Topics: Acetylcysteine; Analysis of Variance; Anilides; Animals; Antioxidants; Autoradiography; Bradykinin; Bradykinin B1 Receptor Antagonists; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Gene Expression Regulation; Iodine Isotopes; Male; Microglia; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; RNA, Messenger; Sensory System Agents; Spinal Cord; Superoxides; Tetrahydroisoquinolines; Time Factors; TRPV Cation Channels

2012