bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- has been researched along with bradykinin in 8 studies
Studies (bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-) | Trials (bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-) | Recent Studies (post-2010) (bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)-) | Studies (bradykinin) | Trials (bradykinin) | Recent Studies (post-2010) (bradykinin) |
---|---|---|---|---|---|
8 | 0 | 1 | 14,195 | 355 | 1,520 |
Protein | Taxonomy | bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- (IC50) | bradykinin (IC50) |
---|---|---|---|
B2 bradykinin receptor | Homo sapiens (human) | 0.0018 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (62.50) | 18.2507 |
2000's | 2 (25.00) | 29.6817 |
2010's | 1 (12.50) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Gobeil, F; Regoli, D; Rhaleb, NE | 1 |
Schölkens, BA; Wiemer, G; Wirth, KJ | 1 |
Lecci, A; Maggi, CA; Meini, S | 1 |
Domingues-Costa, A; Magina, S; Moura, D; Vaz-da-Silva, M | 1 |
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Tramontana, M | 1 |
Greco, S; Marsigliante, S; Storelli, C | 1 |
Bujalska, M; Makulska-Nowak, H | 1 |
Bogo, MR; Campos, MM; Couture, R; Dias, JP; Gaudreau, P; Lahjouji, K; Talbot, S | 1 |
8 other study(ies) available for bradykinin, hyp(3)-thi(5)-tic(7)-oic(8)-desarg(9)- and bradykinin
Article | Year |
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Non-selectivity of new bradykinin antagonists for B1 receptors.
Topics: Amino Acid Sequence; Animals; Aorta; Binding, Competitive; Bradykinin; Guinea Pigs; Ileum; In Vitro Techniques; Jugular Veins; Kinetics; Molecular Sequence Data; Muscle, Smooth; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Receptors, Bradykinin; Receptors, Neurotransmitter; Tetrahydroisoquinolines | 1992 |
DesArg10[Hoe 140] is a potent B1 bradykinin antagonist.
Topics: Animals; Aorta; Bradykinin; Duodenum; Endothelium, Vascular; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Pulmonary Artery; Rabbits; Rats; Receptors, Bradykinin; Receptors, Neurotransmitter; Tetrahydroisoquinolines | 1992 |
The longitudinal muscle of rat ileum as a sensitive monoreceptor assay for bradykinin B1 receptors.
Topics: Adrenergic beta-Antagonists; Analysis of Variance; Animals; Bradykinin; Guinea Pigs; Ileum; Male; Muscle, Smooth; Rats; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Tetrahydroisoquinolines; Urinary Bladder | 1996 |
The role of the endocardium in the facilitatory effect of bradykinin on electrically-induced release of noradrenaline in rat cardiac ventricle.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Captopril; Electric Stimulation; Endocardium; Heart Ventricles; In Vitro Techniques; Male; Norepinephrine; Rats; Rats, Wistar; Tetrahydroisoquinolines; Ventricular Function | 1996 |
Kinin B1 receptor-mediated motor responses in normal or inflamed rat urinary bladder in vivo.
Topics: Administration, Topical; Anesthetics, Intravenous; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bradykinin; Bradykinin Receptor Antagonists; Cyclophosphamide; Cystitis; Dose-Response Relationship, Drug; Ganglia, Parasympathetic; Ganglionectomy; Male; Muscle Contraction; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptors, Bradykinin; Reference Values; Tetrahydroisoquinolines; Urethane; Urinary Bladder | 1999 |
Protein kinase C (PKC)-delta/-epsilon mediate the PKC/Akt-dependent phosphorylation of extracellular signal-regulated kinases 1 and 2 in MCF-7 cells stimulated by bradykinin.
Topics: Analysis of Variance; Biological Transport; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Breast Neoplasms; Cell Line, Tumor; Cell Membrane; Cell Proliferation; Chromones; Cytosol; Dose-Response Relationship, Drug; Estrenes; Female; Flavonoids; Humans; Immunoblotting; Indoles; Kallidin; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Morpholines; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-delta; Protein Kinase C-epsilon; Pyrrolidinones; Stimulation, Chemical; Tetrahydroisoquinolines | 2006 |
Bradykinin receptors antagonists and nitric oxide synthase inhibitors in vincristine and streptozotocin induced hyperalgesia in chemotherapy and diabetic neuropathy rat model.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Drug Evaluation, Preclinical; Enzyme Inhibitors; Hyperalgesia; Hypoglycemic Agents; Indazoles; Lysine; Male; Nitric Oxide Synthase; Nitroarginine; Pain Measurement; Rats; Rats, Wistar; Receptors, Bradykinin; Streptozocin; Tetrahydroisoquinolines; Vincristine | 2009 |
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
Topics: Acetylcysteine; Analysis of Variance; Anilides; Animals; Antioxidants; Autoradiography; Bradykinin; Bradykinin B1 Receptor Antagonists; Capsaicin; Cinnamates; Dose-Response Relationship, Drug; Gene Expression Regulation; Iodine Isotopes; Male; Microglia; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B1; RNA, Messenger; Sensory System Agents; Spinal Cord; Superoxides; Tetrahydroisoquinolines; Time Factors; TRPV Cation Channels | 2012 |