bq 610 has been researched along with bq 123 in 17 studies
| Studies (bq 610) | Trials (bq 610) | Recent Studies (post-2010) (bq 610) | Studies (bq 123) | Trials (bq 123) | Recent Studies (post-2010) (bq 123) |
|---|---|---|---|---|---|
| 124 | 1 | 3 | 1,391 | 63 | 152 |
| Protein | Taxonomy | bq 610 (IC50) | bq 123 (IC50) |
|---|---|---|---|
| Endothelin-1 receptor | Homo sapiens (human) | 0.017 | |
| Endothelin-1 receptor | Rattus norvegicus (Norway rat) | 0.014 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 9 (52.94) | 18.2507 |
| 2000's | 7 (41.18) | 29.6817 |
| 2010's | 1 (5.88) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Doualla-Bell Kotto Maka, F; Ferré, F; Mondon, F; Sabry, S | 1 |
| Featherstone, RL; Uhlig, S; von Bethmann, AN; Wendel, A | 1 |
| Fukami, T; Ihara, M; Ishikawa, K; Ohwaki, K; Ozaki, S; Towers, P; Yamanaka, R; Yano, M | 1 |
| Braeker, B; Ertl, G; Han, H; Neubauer, S | 1 |
| Deng, LY; Li, JS; Schiffrin, EL | 1 |
| Brichard, MH; Demaude, T; Paye, I; Scarso, A; Van Assche, I; Van Binst, G; Verheyden, P | 1 |
| Brelinska, R; De Caro, R; Malendowicz, LK; Nussdorfer, GG; Trejer, M | 1 |
| Appalsamy, M; Fernandez-Violante, R; Hamakubo, T; Mosqueda-Garcia, R | 1 |
| Freeman, ME; Kanyicska, B; Lerant, A | 1 |
| Foster, HE; Ikeda, K; Latifpour, J; Nishi, K; Saito, M; Smith, SD; Wada, Y; Wang, Z; Weiss, RM | 1 |
| Damon, DH | 1 |
| Gavin, JB; Harrison, WR; Maxwell, L | 1 |
| Garrido, Mdel R; Israel, A | 1 |
| Chen, ZC; Cheng, BC; Lin, MT; Liu, CC | 1 |
| Doerr, MD; Flores, JA; Goravanahally, MP; Inskeep, EK; Rhinehart, JD | 1 |
| Bai, J; Lin, L; Lu, H; Ren, A; Shi, J; Yan, X; Yin, Y; Yuan, W | 1 |
| Rapoport, RM; Yoon, S; Zuccarello, M | 1 |
17 other study(ies) available for bq 610 and bq 123
| Article | Year |
|---|---|
Endothelin-induced phosphoinositide hydrolysis in the muscular layer of stem villi vessels of human term placenta.
Topics: Amino Acid Sequence; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Female; Humans; Hydrolysis; Molecular Sequence Data; Muscle, Smooth, Vascular; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Phosphatidylinositols; Placenta; Pregnancy; Receptors, Endothelin; Type C Phospholipases; Vasoconstrictor Agents; Viper Venoms | 1995 |
Pharmacologic characterization of endothelin receptor responses in the isolated perfused rat lung.
Topics: Analysis of Variance; Animals; Bosentan; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Epoprostenol; Female; In Vitro Techniques; Lung; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Rats; Rats, Wistar; Receptors, Endothelin; Respiratory Mechanics; Sulfonamides; Thromboxanes; Time Factors; Vascular Resistance | 1995 |
[3H]BQ-123, a highly specific and reversible radioligand for the endothelin ETA receptor subtype.
Topics: Amino Acid Sequence; Azepines; Binding, Competitive; Endothelin Receptor Antagonists; Endothelins; Humans; Indoles; Isotope Labeling; Molecular Sequence Data; Neuroblastoma; Oligopeptides; Peptides, Cyclic; Radioligand Assay; Receptor, Endothelin A; Receptors, Endothelin; Structure-Activity Relationship; Tritium; Tumor Cells, Cultured | 1995 |
Endothelin-1 contributes to ischemia/reperfusion injury in isolated rat heart-attenuation of ischemic injury by the endothelin-1 antagonists BQ123 and BQ610.
Topics: Animals; Endothelin Receptor Antagonists; Endothelins; Heart; Heart Rate; In Vitro Techniques; Myocardium; Oligopeptides; Peptides, Cyclic; Rats; Rats, Wistar; Reperfusion Injury; Ventricular Function, Left | 1995 |
Endothelin receptor subtypes in resistance arteries from humans and rats.
Topics: Adipose Tissue; Adult; Animals; Arginine; Arteries; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Male; Mesenteric Arteries; Middle Aged; NG-Nitroarginine Methyl Ester; Oligopeptides; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Receptors, Endothelin; Stimulation, Chemical; Vascular Resistance; Viper Venoms | 1995 |
Conformational study of three endothelin antagonists with 1H NMR at low temperature and molecular dynamics.
Topics: Amino Acid Sequence; Cold Temperature; Endothelins; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Oligopeptides; Peptides, Cyclic; Protein Conformation | 1994 |
Endothelin-1, acting via the A receptor subtype, stimulates thymocyte proliferation in the rat.
Topics: Animals; Cell Division; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Female; Kinetics; Mitotic Index; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Piperidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptors, Endothelin; Thymus Gland | 1998 |
Modulatory effects of endothelin on baroreflex activation in the nucleus of the solitary tract.
Topics: Animals; Baroreflex; Endothelin Receptor Antagonists; Endothelins; Male; Microinjections; Oligopeptides; Peptides, Cyclic; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Endothelin; Solitary Nucleus | 1998 |
Endothelin is an autocrine regulator of prolactin secretion.
Topics: Animals; Autocrine Communication; Endothelin Receptor Antagonists; Endothelins; Female; Immunohistochemistry; Male; Oligopeptides; Peptides, Cyclic; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Sex Characteristics | 1998 |
Gene expression, localization, and pharmacological characterization of endothelin receptors in diabetic rat bladder dome.
Topics: Animals; Autoradiography; Diabetes Mellitus, Experimental; Endothelin-1; Male; Oligopeptides; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Receptors, Endothelin; RNA, Messenger; Streptozocin; Urinary Bladder | 2000 |
VSM growth is stimulated in sympathetic neuron/VSM cocultures: role of TGF-beta2 and endothelin.
Topics: Animals; Coculture Techniques; Endothelin Receptor Antagonists; Endothelins; Male; Muscle Development; Muscle, Smooth, Vascular; Neurons; Oligopeptides; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Superior Cervical Ganglion; Sympathetic Nervous System; Transforming Growth Factor beta | 2000 |
Endothelin antagonists diminish postischemic microvascular incompetence and necrosis in the heart.
Topics: Animals; Calcium; Capillaries; Coronary Vessels; Drug Evaluation, Preclinical; Endothelin Receptor Antagonists; Endothelins; Heart; Heart Ventricles; Ion Transport; Myocardial Stunning; Myocardium; Necrosis; Oligopeptides; Peptides, Cyclic; Rats; Rats, Inbred WKY; Receptor, Endothelin A; Receptors, Endothelin | 2000 |
Endothelin ETB receptor signaling in the median eminence and subfornical organ of the rat brain.
Topics: Animals; Antihypertensive Agents; Binding Sites; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Endothelin-3; Male; Median Eminence; Oligopeptides; Peptides, Cyclic; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Signal Transduction; Subfornical Organ | 2004 |
Prior antagonism of endothelin-1A receptors alleviates circulatory shock and cerebral ischemia during rat heatstroke.
Topics: Animals; Brain Ischemia; Endothelin-1; Heat Stroke; Male; Oligopeptides; Peptides, Cyclic; Rats; Rats, Sprague-Dawley; Shock; Time Factors | 2004 |
Effects of endothelin receptor type-A and type-B antagonists on prostaglandin F2alpha-induced luteolysis of the sheep corpus luteum.
Topics: Animals; Corpus Luteum; Dinoprost; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Female; Gene Expression; Luteolysis; Oligopeptides; Peptides, Cyclic; Piperidines; Progesterone; Receptor, Endothelin A; Receptor, Endothelin B; RNA; Sheep | 2008 |
Antagonism of endothelin-1 inhibits hypoxia-induced apoptosis in cardiomyocytes.
Topics: Animals; Animals, Newborn; Apoptosis; Cell Hypoxia; Dose-Response Relationship, Drug; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Flow Cytometry; In Situ Nick-End Labeling; L-Lactate Dehydrogenase; Myocytes, Cardiac; Oligopeptides; Peptides, Cyclic; Piperidines; Rats; Rats, Sprague-Dawley; Superoxide Dismutase | 2008 |
EndothelinA-endothelinB receptor cross-talk in rat basilar artery in situ.
Topics: Animals; Antihypertensive Agents; Basilar Artery; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Male; Oligopeptides; Peptides, Cyclic; Piperidines; Rats; Rats, Sprague-Dawley; Receptor Cross-Talk; Receptor, Endothelin A; Receptor, Endothelin B; Vasoconstrictor Agents; Vasodilator Agents; Viper Venoms | 2012 |