bmy 7378 has been researched along with nan 190 in 15 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 11 (73.33) | 18.2507 |
2000's | 4 (26.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Barrett, JE; Gleeson, S | 1 |
Ahlers, ST; Barrett, JE; Weissman, BA | 1 |
Glaser, T; Greuel, JM | 1 |
Moser, PC | 1 |
Fornal, CA; Jacobs, BL; Marrosu, F; Metzler, CW; Tada, K | 1 |
Newman, ME | 1 |
Fozard, JR; Hoyer, D; McQuade, R; Sharp, T | 1 |
Bervoets, K; Brocco, M; Canton, H; Gobert, A; Lejeune, F; Millan, MJ; Peglion, JL; Rivet, JM; Widdowson, P | 1 |
Harrington, ME; Lall, GS | 1 |
Audinot, V; Bervoets, K; Brocco, M; Canton, H; Gobert, A; Le Marouille-Girardon, S; Millan, MJ; Peglion, JL | 1 |
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B | 1 |
Bojarski, AJ; Chojnacka-Wójcik, E; Dereń-Wesołek, A; Duszyńska, B; Mokrosz, JL; Mokrosz, MJ; Tatarczyńska, E | 1 |
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R | 1 |
Li, MY; Tsai, KC; Xia, L | 1 |
Pedretti, A; Testa, B; Villa, L; Vistoli, G | 1 |
15 other study(ies) available for bmy 7378 and nan 190
Article | Year |
---|---|
Discriminative stimulus effects of 8-OH-DPAT in pigeons: antagonism studies with the putative 5-HT1A receptor antagonists BMY 7378 and NAN-190.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Pindolol; Piperazines; Prazosin; Serotonin Antagonists | 1992 |
Antagonism studies with BMY-7378 and NAN-190: effects on 8-hydroxy-2-(di-n-propylamino)tetralin-induced increases in punished responding of pigeons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Brain; Columbidae; Dose-Response Relationship, Drug; Drug Antagonism; Midazolam; Piperazines; Radioligand Assay; Serotonin Antagonists; Tetrahydronaphthalenes | 1992 |
The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Electrophysiology; In Vitro Techniques; Male; Piperazines; Propranolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tetrahydronaphthalenes | 1992 |
The effect of putative 5-HT1A receptor antagonists on 8-OH-DPAT-induced hypothermia in rats and mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dioxanes; Dose-Response Relationship, Drug; Hypothermia, Induced; Male; Mice; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1991 |
Effects of the putative 5-hydroxytryptamine1A antagonists BMY 7378, NAN 190 and (-)-propranolol on serotonergic dorsal raphe unit activity in behaving cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Cats; Female; Male; Neurons; Piperazines; Propranolol; Raphe Nuclei; Serotonin; Serotonin Antagonists | 1994 |
Serotonin inhibition of adenylate cyclase in human platelet membranes; relation to 5-HT-1A receptor-mediated activity.
Topics: Adenylyl Cyclase Inhibitors; Blood Platelets; Cell Membrane; Dose-Response Relationship, Drug; Epinephrine; Humans; Piperazines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Sodium Chloride | 1994 |
The novel 5-HT1A receptor antagonist, SDZ 216-525, decreases 5-HT release in rat hippocampus in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dialysis; Electrophysiology; GTP-Binding Proteins; Hippocampus; Indoles; Male; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Thiazoles | 1993 |
S 15535: a highly selective benzodioxopiperazine 5-HT1A receptor ligand which acts as an agonist and an antagonist at presynaptic and postsynaptic sites respectively.
Topics: Animals; Behavior, Animal; Blepharoptosis; Body Temperature; Brain Chemistry; Ligands; Male; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses | 1993 |
Potentiation of the resetting effects of light on circadian rhythms of hamsters using serotonin and neuropeptide Y receptor antagonists.
Topics: Animals; Circadian Rhythm; Cricetinae; Drug Interactions; Humans; Light; Mesocricetus; Piperazines; Receptor, Serotonin, 5-HT1A; Receptors, Neuropeptide Y; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Time Factors | 2006 |
Characterization of potent and selective antagonists at postsynaptic 5-HT1A receptors in a series of N4-substituted arylpiperazines.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Male; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Structure-Activity Relationship | 1995 |
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes | 1996 |
8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Buspirone; Hippocampus; Ligands; Male; Molecular Structure; Peptide Fragments; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Serotonin Receptor Agonists; Tetrahydroisoquinolines | 1996 |
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
Pharmacophore identification of alpha(1A)-adrenoceptor antagonists.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Drug Evaluation, Preclinical; Expert Systems; Humans; Models, Molecular; Receptors, Adrenergic, alpha-1; Software; Structure-Activity Relationship | 2005 |
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents | 2005 |