bmy 7378 and nan 190

bmy 7378 has been researched along with nan 190 in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (73.33)18.2507
2000's4 (26.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barrett, JE; Gleeson, S1
Ahlers, ST; Barrett, JE; Weissman, BA1
Glaser, T; Greuel, JM1
Moser, PC1
Fornal, CA; Jacobs, BL; Marrosu, F; Metzler, CW; Tada, K1
Newman, ME1
Fozard, JR; Hoyer, D; McQuade, R; Sharp, T1
Bervoets, K; Brocco, M; Canton, H; Gobert, A; Lejeune, F; Millan, MJ; Peglion, JL; Rivet, JM; Widdowson, P1
Harrington, ME; Lall, GS1
Audinot, V; Bervoets, K; Brocco, M; Canton, H; Gobert, A; Le Marouille-Girardon, S; Millan, MJ; Peglion, JL1
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B1
Bojarski, AJ; Chojnacka-Wójcik, E; Dereń-Wesołek, A; Duszyńska, B; Mokrosz, JL; Mokrosz, MJ; Tatarczyńska, E1
Itoh, H; Muramatsu, I; Taniguchi, T; Yoshio, R1
Li, MY; Tsai, KC; Xia, L1
Pedretti, A; Testa, B; Villa, L; Vistoli, G1

Other Studies

15 other study(ies) available for bmy 7378 and nan 190

ArticleYear
Discriminative stimulus effects of 8-OH-DPAT in pigeons: antagonism studies with the putative 5-HT1A receptor antagonists BMY 7378 and NAN-190.
    European journal of pharmacology, 1992, Jul-07, Volume: 217, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Pindolol; Piperazines; Prazosin; Serotonin Antagonists

1992
Antagonism studies with BMY-7378 and NAN-190: effects on 8-hydroxy-2-(di-n-propylamino)tetralin-induced increases in punished responding of pigeons.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Brain; Columbidae; Dose-Response Relationship, Drug; Drug Antagonism; Midazolam; Piperazines; Radioligand Assay; Serotonin Antagonists; Tetrahydronaphthalenes

1992
The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Electrophysiology; In Vitro Techniques; Male; Piperazines; Propranolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tetrahydronaphthalenes

1992
The effect of putative 5-HT1A receptor antagonists on 8-OH-DPAT-induced hypothermia in rats and mice.
    European journal of pharmacology, 1991, Feb-07, Volume: 193, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dioxanes; Dose-Response Relationship, Drug; Hypothermia, Induced; Male; Mice; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Effects of the putative 5-hydroxytryptamine1A antagonists BMY 7378, NAN 190 and (-)-propranolol on serotonergic dorsal raphe unit activity in behaving cats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Cats; Female; Male; Neurons; Piperazines; Propranolol; Raphe Nuclei; Serotonin; Serotonin Antagonists

1994
Serotonin inhibition of adenylate cyclase in human platelet membranes; relation to 5-HT-1A receptor-mediated activity.
    Biochemical pharmacology, 1994, Nov-01, Volume: 48, Issue:9

    Topics: Adenylyl Cyclase Inhibitors; Blood Platelets; Cell Membrane; Dose-Response Relationship, Drug; Epinephrine; Humans; Piperazines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Sodium Chloride

1994
The novel 5-HT1A receptor antagonist, SDZ 216-525, decreases 5-HT release in rat hippocampus in vivo.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Dialysis; Electrophysiology; GTP-Binding Proteins; Hippocampus; Indoles; Male; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Thiazoles

1993
S 15535: a highly selective benzodioxopiperazine 5-HT1A receptor ligand which acts as an agonist and an antagonist at presynaptic and postsynaptic sites respectively.
    European journal of pharmacology, 1993, Jan-05, Volume: 230, Issue:1

    Topics: Animals; Behavior, Animal; Blepharoptosis; Body Temperature; Brain Chemistry; Ligands; Male; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses

1993
Potentiation of the resetting effects of light on circadian rhythms of hamsters using serotonin and neuropeptide Y receptor antagonists.
    Neuroscience, 2006, Sep-01, Volume: 141, Issue:3

    Topics: Animals; Circadian Rhythm; Cricetinae; Drug Interactions; Humans; Light; Mesocricetus; Piperazines; Receptor, Serotonin, 5-HT1A; Receptors, Neuropeptide Y; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Time Factors

2006
Characterization of potent and selective antagonists at postsynaptic 5-HT1A receptors in a series of N4-substituted arylpiperazines.
    Journal of medicinal chemistry, 1995, Sep-29, Volume: 38, Issue:20

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Male; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Structure-Activity Relationship

1995
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
8-[4-[2-(1,2,3,4-Tetrahydroisoquinolinyl]butyl-8-azaspiro[4.5]decane-7,9-dione: a new 5-HT1A receptor ligand with the same activity profile as buspirone.
    Journal of medicinal chemistry, 1996, Mar-01, Volume: 39, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Buspirone; Hippocampus; Ligands; Male; Molecular Structure; Peptide Fragments; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Serotonin Receptor Agonists; Tetrahydroisoquinolines

1996
Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:2

    Topics: Animals; Aorta, Thoracic; Carotid Arteries; Dogs; Humans; Male; Organ Culture Techniques; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists

2001
Pharmacophore identification of alpha(1A)-adrenoceptor antagonists.
    Bioorganic & medicinal chemistry letters, 2005, Feb-01, Volume: 15, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Drug Evaluation, Preclinical; Expert Systems; Humans; Models, Molecular; Receptors, Adrenergic, alpha-1; Software; Structure-Activity Relationship

2005
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005