Page last updated: 2024-09-03

blonanserin and mdl 100907

blonanserin has been researched along with mdl 100907 in 5 studies

Compound Research Comparison

Studies
(blonanserin)
Trials
(blonanserin)
Recent Studies (post-2010)
(blonanserin)
Studies
(mdl 100907)
Trials
(mdl 100907)
Recent Studies (post-2010) (mdl 100907)
12121931,24165539

Protein Interaction Comparison

ProteinTaxonomyblonanserin (IC50)mdl 100907 (IC50)
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0048

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ishibashi, T; Nakamura, H; Nishikawa, H; Une, T1
Imaki, J; Ohno, Y; Okano, M; Okumura, T; Shimizu, S; Tatara, A1
Horiguchi, M; Meltzer, HY1
Huang, M; Kwon, S; Meltzer, HY; Oyamada, Y; Panos, JJ; Rajagopal, L1
Baba, S; Enomoto, T; Hashimoto, T; Horisawa, T; Ono, M1

Reviews

1 review(s) available for blonanserin and mdl 100907

ArticleYear
[Pharmacological profiles and clinical effects of blonanserin (Lonasen) on schizophrenia].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2008, Volume: 132, Issue:6

    Topics: Animals; Antidepressive Agents, Second-Generation; Cognition Disorders; Dopamine D2 Receptor Antagonists; Double-Blind Method; Drug Discovery; Drug-Related Side Effects and Adverse Reactions; Humans; Piperazines; Piperidines; Randomized Controlled Trials as Topic; Schizophrenia; Serotonin 5-HT2 Receptor Antagonists; Treatment Outcome

2008

Other Studies

4 other study(ies) available for blonanserin and mdl 100907

ArticleYear
Atypical antipsychotic properties of blonanserin, a novel dopamine D2 and 5-HT2A antagonist.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 96, Issue:2

    Topics: Animals; Antipsychotic Agents; Catalepsy; Corpus Striatum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; Haloperidol; Male; Mice; Mice, Inbred Strains; Nucleus Accumbens; Piperazines; Piperidines; Proto-Oncogene Proteins c-fos; Pyridines; Serotonin 5-HT2 Receptor Antagonists

2010
Blonanserin reverses the phencyclidine (PCP)-induced impairment in novel object recognition (NOR) in rats: role of indirect 5-HT(1A) partial agonism.
    Behavioural brain research, 2013, Jun-15, Volume: 247

    Topics: Animals; Female; Isoindoles; Phencyclidine; Piperazines; Piperidines; Pyridines; Pyrimidines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1A; Recognition, Psychology; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2013
Comparative effect of lurasidone and blonanserin on cortical glutamate, dopamine, and acetylcholine efflux: role of relative serotonin (5-HT)2A and DA D2 antagonism and 5-HT1A partial agonism.
    Journal of neurochemistry, 2014, Volume: 128, Issue:6

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Brain; Cerebral Cortex; Dopamine; Glutamic Acid; Hippocampus; Isoindoles; Lurasidone Hydrochloride; Male; Microdialysis; Neurotransmitter Agents; Nucleus Accumbens; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Synaptic Transmission; Thiazoles

2014
Blonanserin extensively occupies rat dopamine D3 receptors at antipsychotic dose range.
    Journal of pharmacological sciences, 2015, Volume: 127, Issue:3

    Topics: Animals; Antipsychotic Agents; Cells, Cultured; Cricetinae; Cricetulus; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Hyperkinesis; Male; Piperazines; Piperidines; Protein Binding; Rats, Sprague-Dawley; Receptors, Dopamine D3; Serotonin 5-HT2 Receptor Antagonists

2015