bisindolylmaleimide v and bisindolylmaleimide i

bisindolylmaleimide v has been researched along with bisindolylmaleimide i in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's8 (88.89)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ajakane, M; Baudet, V; Bellevergue, P; Boissin, P; Boursier, E; Coste, H; Grand-Perret, T; Loriolle, F; Pianetti, P; Toullec, D1
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
Goekjian, P; Jochum, A; Jung, M; Kunick, C; Marshall, B; Meier, R; Saunders, L; Sippl, W; Trapp, J; Verdin, E1
Bekker, OB; Danilenko, VN; Elizarov, SM; Kubbutat, MH; Lakatosh, SA; Luzikov, YN; Preobrazhenskaya, MN; Printsevskaya, SS; Reznikova, MI; Schächtele, C; Shtil, AA; Simonov, AY; Totzke, F1
Hunter, ES; Rogers, EH; Ward, KW1
Booth, G; Lefer, AM; Scalia, R; Stalker, TJ1
Aoyama, Y; Asakai, R; Fujimoto, T1
Carrico-Moniz, D; Imperiali, B; Shults, MD1
Gozal, D; Reeves, SR1

Other Studies

9 other study(ies) available for bisindolylmaleimide v and bisindolylmaleimide i

ArticleYear
The bisindolylmaleimide GF 109203X is a potent and selective inhibitor of protein kinase C.
    The Journal of biological chemistry, 1991, Aug-25, Volume: 266, Issue:24

    Topics: Adenosine Triphosphate; Alkaloids; Animals; Blood Platelets; Bombesin; Collagen; DNA; Electrophoresis, Polyacrylamide Gel; Epidermal Growth Factor; Fibroblasts; Humans; Indoles; Maleimides; Mice; Phorbol 12,13-Dibutyrate; Phosphorylation; Platelet Aggregation; Protein Kinase C; Staurosporine; Structure-Activity Relationship; Thymidine; Vimentin

1991
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition.
    Journal of medicinal chemistry, 2006, Dec-14, Volume: 49, Issue:25

    Topics: Acetylation; Adenosine; Binding Sites; Cell Line, Tumor; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Models, Molecular; Molecular Mimicry; Protein Kinase Inhibitors; Sirtuins; Structure-Activity Relationship; Tubulin

2006
Search for inhibitors of bacterial and human protein kinases among derivatives of diazepines[1,4] annelated with maleimide and indole cycles.
    Journal of medicinal chemistry, 2008, Dec-25, Volume: 51, Issue:24

    Topics: Chemistry, Pharmaceutical; Humans; Indoles; Inhibitory Concentration 50; Maleimides; Models, Chemical; Molecular Conformation; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Recombinant Proteins; Serine; Streptomyces lividans; Thiourea; Threonine

2008
Comparative pathogenesis of haloacetic acid and protein kinase inhibitor embryotoxicity in mouse whole embryo culture.
    Toxicological sciences : an official journal of the Society of Toxicology, 2000, Volume: 53, Issue:1

    Topics: Animals; Apoptosis; Cell Cycle; Culture Techniques; Embryonic and Fetal Development; Enzyme Inhibitors; Female; Flow Cytometry; Indoles; Male; Maleimides; Mice; Pregnancy; Protein Kinase C; Staurosporine

2000
Mechanisms of amelioration of glucose-induced endothelial dysfunction following inhibition of protein kinase C in vivo.
    Diabetes, 2002, Volume: 51, Issue:5

    Topics: Animals; Aorta; Cell Adhesion; Diabetic Angiopathies; Endothelium, Vascular; Enzyme Inhibitors; Glucose; Immunohistochemistry; Indoles; Intercellular Adhesion Molecule-1; Male; Maleimides; Neutrophils; Nitric Oxide; Oxidative Stress; P-Selectin; Protein Kinase C; Rats; Rats, Sprague-Dawley

2002
Bisindolylmaleimide I and V inhibit necrosis induced by oxidative stress in a variety of cells including neurons.
    Neuroscience research, 2002, Volume: 44, Issue:3

    Topics: Adenosine Triphosphate; Animals; Cell Death; Cell Survival; Cells, Cultured; Free Radicals; Indicators and Reagents; Indoles; Maleimides; Microscopy, Electron; Necrosis; Neurons; Oxidation-Reduction; Oxidative Stress; Swine

2002
Optimal Sox-based fluorescent chemosensor design for serine/threonine protein kinases.
    Analytical biochemistry, 2006, May-15, Volume: 352, Issue:2

    Topics: Enzyme Activation; Enzyme Inhibitors; Fluorescence; Fluorescent Dyes; Indoles; Kinetics; Maleimides; Phosphorylation; Protein Serine-Threonine Kinases; Sensitivity and Specificity; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Transcription Factors

2006
Protein kinase C activity in the nucleus tractus solitarii is critically involved in the acute hypoxic ventilatory response, but is not required for intermittent hypoxia-induced phrenic long-term facilitation in adult rats.
    Experimental physiology, 2007, Volume: 92, Issue:6

    Topics: Animals; Behavior, Animal; Diaphragm; Enzyme Inhibitors; Hypoxia, Brain; Indoles; Male; Maleimides; Phrenic Nerve; Protein Kinase C; Pulmonary Ventilation; Rats; Rats, Sprague-Dawley; Respiratory Physiological Phenomena; Solitary Nucleus

2007