bisindolylmaleimide iii and ro 31-7549

bisindolylmaleimide iii has been researched along with ro 31-7549 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
Alessi, DR; Bain, J; Deak, M; Elliott, M; Garrido-Franco, M; Komander, D; Kozikowski, AP; Kular, GS; Prakash, KR; Schüttelkopf, AW; van Aalten, DM1
Chen, Z; Dong, H; Dugar, S; Higaki, J; Laney, M; Levy, DE; Liclican, A; Lu, Q; Mavunkel, B; Perumattam, J; Wang, DX; Xu, YJ2

Other Studies

4 other study(ies) available for bisindolylmaleimide iii and ro 31-7549

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Interactions of LY333531 and other bisindolyl maleimide inhibitors with PDK1.
    Structure (London, England : 1993), 2004, Volume: 12, Issue:2

    Topics: 3-Phosphoinositide-Dependent Protein Kinases; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Indoles; Maleimides; Models, Molecular; Protein Kinase C; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Signal Transduction

2004
Aryl-indolyl maleimides as inhibitors of CaMKIIdelta. Part 1: SAR of the aryl region.
    Bioorganic & medicinal chemistry letters, 2008, Apr-01, Volume: 18, Issue:7

    Topics: Adenosine Triphosphate; Benzene Derivatives; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Drug Design; Enzyme Inhibitors; Indoles; Maleimides; Models, Chemical; Structure-Activity Relationship; Substrate Specificity

2008
Aryl-indolyl maleimides as inhibitors of CaMKIIdelta. Part 2: SAR of the amine tether.
    Bioorganic & medicinal chemistry letters, 2008, Apr-01, Volume: 18, Issue:7

    Topics: Adenosine Triphosphate; Amines; Benzene Derivatives; Binding Sites; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Drug Design; Enzyme Inhibitors; Indoles; Maleimides; Models, Chemical; Structure-Activity Relationship; Substrate Specificity

2008