Page last updated: 2024-09-04

birb 796 and sotrastaurin

birb 796 has been researched along with sotrastaurin in 2 studies

Compound Research Comparison

Studies
(birb 796)
Trials
(birb 796)
Recent Studies (post-2010)
(birb 796)
Studies
(sotrastaurin)
Trials
(sotrastaurin)
Recent Studies (post-2010) (sotrastaurin)
137580881269

Protein Interaction Comparison

ProteinTaxonomybirb 796 (IC50)sotrastaurin (IC50)
Serine/threonine-protein kinase D3Homo sapiens (human)0.0021
Tyrosine-protein kinase ABL1Homo sapiens (human)3.3
Protein kinase C beta typeHomo sapiens (human)0.0025
Tyrosine-protein kinase FynHomo sapiens (human)5.5
Cytochrome P450 3A4Homo sapiens (human)0.001
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.0501
Protein kinase C alpha typeHomo sapiens (human)0.0026
Cyclin-A2Homo sapiens (human)2.3
Tyrosine-protein kinase JAK1Homo sapiens (human)7.3
Protein kinase C eta typeHomo sapiens (human)0.0041
Cyclin-dependent kinase 2Homo sapiens (human)2.3
Tyrosine-protein kinase receptor UFOHomo sapiens (human)9.1
Vascular endothelial growth factor receptor 3Homo sapiens (human)4.6
Vascular endothelial growth factor receptor 2Homo sapiens (human)3.9
Glycogen synthase kinase-3 betaHomo sapiens (human)0.87
Tyrosine-protein kinase JAK3Homo sapiens (human)1.5
Protein kinase C beta type Mus musculus (house mouse)0.234
Cyclin-A1Homo sapiens (human)2.3
Protein kinase C epsilon typeHomo sapiens (human)0.0041
Protein kinase C theta typeHomo sapiens (human)0.0094
Focal adhesion kinase 1Homo sapiens (human)8.3
Protein kinase C zeta typeHomo sapiens (human)5.4
Protein kinase C delta typeHomo sapiens (human)0.0025
Peroxisome proliferator-activated receptor alphaHomo sapiens (human)0.0031
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialHomo sapiens (human)6.7

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1
Cahya, S; Cummins, DJ; Gao, C; Iversen, PW; Nicolaou, CA; Vieth, M; Wang, J; Watson, IA1

Other Studies

2 other study(ies) available for birb 796 and sotrastaurin

ArticleYear
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011
Selectivity data: assessment, predictions, concordance, and implications.
    Journal of medicinal chemistry, 2013, Sep-12, Volume: 56, Issue:17

    Topics: Computer Simulation; Drug Discovery

2013