Page last updated: 2024-09-04

birb 796 and ceritinib

birb 796 has been researched along with ceritinib in 1 studies

Compound Research Comparison

Studies
(birb 796)
Trials
(birb 796)
Recent Studies (post-2010)
(birb 796)
Studies
(ceritinib)
Trials
(ceritinib)
Recent Studies (post-2010) (ceritinib)
13758032935322

Protein Interaction Comparison

ProteinTaxonomybirb 796 (IC50)ceritinib (IC50)
Tyrosine-protein kinase JAK2Homo sapiens (human)1.385
Rho-associated protein kinase 2Homo sapiens (human)1.27
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)3.7
Tyrosine-protein kinase ABL1Homo sapiens (human)1.25
Epidermal growth factor receptorHomo sapiens (human)0.7757
High affinity nerve growth factor receptorHomo sapiens (human)2.727
Insulin receptorHomo sapiens (human)0.1525
Tyrosine-protein kinase LckHomo sapiens (human)0.616
NucleophosminHomo sapiens (human)0.026
Tyrosine-protein kinase LynHomo sapiens (human)1.573
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)1.352
Insulin-like growth factor 1 receptorHomo sapiens (human)0.209
Hepatocyte growth factor receptorHomo sapiens (human)1.5933
Cytochrome P450 3A4Homo sapiens (human)3.36
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)0.2697
Tyrosine-protein kinase FgrHomo sapiens (human)1.947
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 22.86
Mast/stem cell growth factor receptor KitHomo sapiens (human)2.0675
Cyclin-dependent kinase 4Homo sapiens (human)4.72
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)1.694
Platelet-derived growth factor receptor alphaHomo sapiens (human)1.14
Fibroblast growth factor receptor 2Homo sapiens (human)0.26
Fibroblast growth factor receptor 4Homo sapiens (human)0.95
Fibroblast growth factor receptor 3Homo sapiens (human)0.43
Tyrosine-protein kinase JAK1Homo sapiens (human)3.73
Cyclin-dependent kinase 2Homo sapiens (human)3.97
Vascular endothelial growth factor receptor 2Homo sapiens (human)4.21
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)1.0965
Transcription factor ETV6Homo sapiens (human)3.25
Tyrosine-protein kinase ZAP-70Homo sapiens (human)9.7
Tyrosine-protein kinase SYKHomo sapiens (human)3.05
Tyrosine-protein kinase JAK3Homo sapiens (human)7.92
Tyrosine-protein kinase BTKHomo sapiens (human)3.36
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.25
BDNF/NT-3 growth factors receptorHomo sapiens (human)1.829
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)0.023
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)2.24
Echinoderm microtubule-associated protein-like 4Homo sapiens (human)0.5935
ALK tyrosine kinase receptorHomo sapiens (human)0.1102

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Juvale, K; Kharkar, PS; Sahu, NU; Shah, CP; Silbermann, K; Stefan, SM; Wiese, M1

Other Studies

1 other study(ies) available for birb 796 and ceritinib

ArticleYear
Novel chalcone and flavone derivatives as selective and dual inhibitors of the transport proteins ABCB1 and ABCG2.
    European journal of medicinal chemistry, 2019, Feb-15, Volume: 164

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Chalcones; Drug Resistance, Multiple; Flavones; Humans; Structure-Activity Relationship

2019