birb 796 has been researched along with axitinib in 2 studies
Studies (birb 796) | Trials (birb 796) | Recent Studies (post-2010) (birb 796) | Studies (axitinib) | Trials (axitinib) | Recent Studies (post-2010) (axitinib) |
---|---|---|---|---|---|
137 | 5 | 80 | 765 | 145 | 683 |
Protein | Taxonomy | birb 796 (IC50) | axitinib (IC50) |
---|---|---|---|
Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | 0.045 | |
Tyrosine-protein kinase ABL1 | Homo sapiens (human) | 0.0658 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 0.046 | |
Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | 0.0001 | |
Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | 0.0001 | |
Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | 0.0079 | |
Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | 0.47 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP | 1 |
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ | 1 |
2 other study(ies) available for birb 796 and axitinib
Article | Year |
---|---|
Comprehensive analysis of kinase inhibitor selectivity.
Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity | 2011 |
Identification of potent Yes1 kinase inhibitors using a library screening approach.
Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship | 2013 |