Page last updated: 2024-08-26

bicuculline methochloride and bicuculline

bicuculline methochloride has been researched along with bicuculline in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-199023 (45.10)18.7374
1990's14 (27.45)18.2507
2000's8 (15.69)29.6817
2010's5 (9.80)24.3611
2020's1 (1.96)2.80

Authors

AuthorsStudies
Redman, SJ; Stuart, GJ1
Field, JL; Newberry, NR1
Han, JS; Yu, LC1
Murphy, PC; Sillito, AM1
Arakawa, T; Okada, Y1
Kemp, JA; Salt, TE; Sillito, AM1
Olsen, RW; Snowman, AM2
Lee, RJ; Lomax, P; McCabe, RT; Olsen, RW; Wamsley, JK1
Curtis, DR; Falch, E; Krogsgaard-Larsen, P; Nielsen, L1
McCabe, RT; Wamsley, JK1
Curtis, DR; Gynther, BD1
Bonds, AB; DeBruyn, EJ1
Sato, H; Tsumoto, T1
Herrling, PL1
Collingridge, GL; Davies, J1
Champagnat, J; Denavit-Saubié, M; Moyanova, S; Rondouin, G1
St Péteri, AK; Todd, JA; Tökés, ZA1
Mayer, ML1
Simmonds, MA1
Bornstein, JC; Curtis, DR; Leah, JD; Lodge, D; Peet, MJ1
Olsen, RW; Snowhill, EW; Wamsley, JK1
Lam, DM; Lasater, EM1
Kerr, DI; Ong, J1
Gmelin, G; Zimmermann, M1
Blakemore, C; Kemp, JA; Sillito, AM1
Dirksen, R; Maksay, G; van Rijn, CM; Willems-van Bree, E1
Bonds, AB; Pfleger, B1
Fonia, O; Gavish, M; Katz, Y; Liu, L; Pasternak, GW; Pick, CG; Weizman, A1
Gähwiler, BH; Müller, M; Rietschin, L; Thompson, SM1
Maksay, G; van Rijn, CM1
Dowling, JE; Qian, H1
Heggelund, P; Paulsen, O1
Gisselmann, G; Gottmann, K; Hatt, H; Mehrle, A1
Li, Z; Massengill, JL; O'Dowd, DK; Smith, MA1
Grant, AL; Mellor, JR; Randall, AD; Williamson, AV1
Boonen, G; Häberlein, H1
Hopp, FA; Kampine, JP; Krolo, M; Stucke, AG; Stuth, EA; Tonkovic-Capin, M; Tonkovic-Capin, V; Zuperku, EJ1
Akerman, S; Goadsby, PJ; Storer, RJ1
Kawai, N; Konno, K; Masuzawa, T; Miyawaki, T; Nakayama, H; Tsubokawa, H; Yokota, H1
Barnes, LU; Egland, MC; Martin, DS; Vogel, EM1
Debanne, D; Gähwiler, BH; Thompson, SM1
Inquimbert, P; Rodeau, JL; Schlichter, R1
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD1
Billings, HJ; Bogusz, AL; Connors, JM; Coolen, LM; Goodman, RL; Hardy, SL; Hileman, SM; Lehman, MN; McManus, CJ; Nestor, CC; Singh, SR; Sliwowska, JH; Valent, M1
Einstein, EB; Hon, BJ; Johnson, BN; Mateer, MJ; Melnikoff, DE; Patterson, CA; Reddi, J; Regan, KA; Schulz, S; Tallent, MK1
Green, CR; Nicholson, LF; O'Carroll, SJ; Yoon, JJ1
Blain, EJ; Dachtler, J; Fox, K; Glazewski, S; Hardingham, NR; Wright, NF1
Agudelo-Toro, A; Moses, E; Neef, A; Rotem, A; Stern, S1
Ginty, DD; Kovatsis, EM; Pozsgai, RY; Tasnim, A; Zhang, Q; Zimmerman, AL1
Dawson, A; Hales, TG; Hunter, WN; Jones, MJ1

Other Studies

51 other study(ies) available for bicuculline methochloride and bicuculline

ArticleYear
The role of GABAA and GABAB receptors in presynaptic inhibition of Ia EPSPs in cat spinal motoneurones.
    The Journal of physiology, 1992, Volume: 447

    Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; Membrane Potentials; Motor Neurons; Receptors, GABA-A; Receptors, Neurotransmitter; Spinal Cord

1992
On the histamine-induced depolarization of the isolated superior cervical ganglion of the rat.
    British journal of pharmacology, 1991, Volume: 103, Issue:3

    Topics: Animals; Atropine Derivatives; Bicuculline; Calcium Chloride; Ganglia, Sympathetic; Histamine; In Vitro Techniques; Male; Methylhistamines; Neuromuscular Depolarizing Agents; Nicotine; Parasympatholytics; Propranolol; Rats; Rats, Inbred Strains; Tetrodotoxin; Tubocurarine

1991
Habenula as a relay in the descending pathway from nucleus accumbens to periaqueductal grey subserving antinociception.
    The International journal of neuroscience, 1990, Volume: 54, Issue:3-4

    Topics: Animals; Bicuculline; Efferent Pathways; Enkephalin, Methionine; Immune Sera; Injections; Morphine; Muscimol; Naloxone; Nociceptors; Nucleus Accumbens; Periaqueductal Gray; Rabbits; Thalamic Nuclei

1990
The binocular input to cells in the feline dorsal lateral geniculate nucleus (dLGN).
    The Journal of physiology, 1989, Volume: 415

    Topics: Action Potentials; Animals; Bicuculline; Cats; Feedback; Female; GABA Antagonists; Geniculate Bodies; Membrane Potentials; Neurons; Ocular Physiological Phenomena; Photic Stimulation; Retina; Visual Cortex

1989
Excitatory and inhibitory action of GABA on synaptic transmission in slices of guinea pig superior colliculus.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Muscimol; Nipecotic Acids; Perfusion; Proline; Receptors, GABA-A; Superior Colliculi; Synaptic Membranes; Synaptic Transmission

1988
Modulatory and inhibitory processes in the visual cortex.
    Vision research, 1985, Volume: 25, Issue:3

    Topics: Acetylcholine; Action Potentials; Animals; Bicuculline; Cats; gamma-Aminobutyric Acid; Interneurons; Neural Conduction; Neural Inhibition; Somatostatin; Visual Cortex

1985
Avermectin B1a modulation of gamma-aminobutyric acid/benzodiazepine receptor binding in mammalian brain.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Animals; Bicuculline; Brain; Cattle; Cell Membrane; Cerebral Cortex; Etazolate; gamma-Aminobutyric Acid; Isonicotinic Acids; Ivermectin; Lactones; Muscimol; Pentobarbital; Rats; Receptors, GABA-A

1985
Benzodiazepine/gamma-aminobutyric acid receptor deficit in the midbrain of the seizure-susceptible gerbil.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:19

    Topics: Animals; Bicuculline; Diazepam; Disease Models, Animal; Flunitrazepam; Gerbillinae; Mesencephalon; Muscimol; Pentobarbital; Receptors, GABA-A; Seizures

1985
GABA agonists. Resolution, absolute stereochemistry, and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:11

    Topics: Animals; Bicuculline; Brain; Cats; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Molecular Conformation; Muscimol; Neurons; Oxazolidinones; Piperidines; Rats; Receptors, GABA-A; Spinal Cord; Stereoisomerism; Structure-Activity Relationship; Synaptic Membranes

1985
Autoradiographic localization of subcomponents of the macromolecular GABA receptor complex.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Animals; Autoradiography; Baclofen; Bicuculline; Binding, Competitive; Brain Chemistry; Flunitrazepam; Macromolecular Substances; Muscimol; Rats; Receptors, GABA-A; Tissue Distribution; Tritium

1986
Divalent cations reduce depolarization of primary afferent terminations by GABA.
    Brain research, 1987, Sep-29, Volume: 422, Issue:1

    Topics: Action Potentials; Animals; Bicuculline; Cations, Divalent; Cats; Electric Stimulation; gamma-Aminobutyric Acid; Interneurons; Membrane Potentials; Muscles; Neurons, Afferent; Piperidines; Spinal Cord

1987
Contrast adaptation in cat visual cortex is not mediated by GABA.
    Brain research, 1986, Sep-24, Volume: 383, Issue:1-2

    Topics: Adaptation, Physiological; Animals; Bicuculline; Cats; gamma-Aminobutyric Acid; Neural Inhibition; Visual Cortex; Visual Perception

1986
GABAergic inhibition and orientation selectivity of neurons in the kitten visual cortex at the time of eye opening.
    Vision research, 1985, Volume: 25, Issue:3

    Topics: Animals; Animals, Newborn; Bicuculline; Brain Mapping; Cats; Evoked Potentials, Visual; Eyelids; gamma-Aminobutyric Acid; Neurons; Rotation; Visual Cortex

1985
Evidence for GABA as the transmitter for early cortically evoked inhibition of cat caudate neurons.
    Experimental brain research, 1984, Volume: 55, Issue:3

    Topics: Animals; Bicuculline; Cats; Caudate Nucleus; Cerebral Cortex; Evoked Potentials; Female; gamma-Aminobutyric Acid; Hippocampus; Male; Neural Inhibition; Neural Pathways; Synaptic Transmission

1984
The influence of striatal stimulation and putative neurotransmitters on identified neurones in the rat substantia nigra.
    Brain research, 1981, May-18, Volume: 212, Issue:2

    Topics: Animals; Bicuculline; Corpus Striatum; Dominance, Cerebral; Electric Stimulation; Evoked Potentials; Female; gamma-Aminobutyric Acid; Glycine; Male; Neural Inhibition; Neural Pathways; Neurons; Neurotransmitter Agents; Rats; Reticular Formation; Substantia Nigra; Superior Colliculi; Synaptic Transmission; Thalamic Nuclei

1981
Involvement of amino acids in periodic inhibitions of bulbar respiratory neurones.
    Brain research, 1982, Apr-15, Volume: 237, Issue:2

    Topics: Alanine; Amino Acids; Animals; Bicuculline; Cats; Glutamates; Glutamic Acid; Glycine; Kinetics; Medulla Oblongata; Methylene Blue; Muscimol; Neurons; Nipecotic Acids; Oxygen Consumption; Picrotoxin; Strychnine

1982
Availability of liposome content to the nervous system. Liposomes and the blood-brain barrier.
    Brain research, 1980, Apr-21, Volume: 188, Issue:1

    Topics: Animals; Bicuculline; Blood-Brain Barrier; Bordetella pertussis; Brain; Cholesterol; gamma-Aminobutyric Acid; Liposomes; Mice; Phosphatidylcholines; Serotonin; Trypan Blue

1980
Inhibitory actions of amino acids in the preoptic-anterior hypothalamus of the rat.
    Experimental brain research, 1981, Volume: 43, Issue:2

    Topics: Amino Acids; Animals; beta-Alanine; Bicuculline; Female; gamma-Aminobutyric Acid; Glycine; Hypothalamus; Hypothalamus, Anterior; Neural Inhibition; Neurons; Preoptic Area; Rats; Strychnine; Synaptic Transmission; Taurine

1981
Classification of some GABA antagonists with regard to site of action and potency in slices of rat cuneate nucleus.
    European journal of pharmacology, 1982, Jun-04, Volume: 80, Issue:4

    Topics: Animals; Bicuculline; Cyclic P-Oxides; Furosemide; GABA Antagonists; In Vitro Techniques; Medulla Oblongata; Organophosphorus Compounds; Pentylenetetrazole; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, GABA-A; Strychnine; Tubocurarine

1982
The dual effects of GABA and related amino acids on the electrical threshold of ventral horn group Ia afferent terminations in the cat.
    Experimental brain research, 1982, Volume: 48, Issue:3

    Topics: Afferent Pathways; Amino Acids; Animals; Bicuculline; Cats; Electric Stimulation; gamma-Aminobutyric Acid; Interneurons; Ion Channels; Membrane Potentials; Motor Neurons; Nerve Fibers; Ouabain; Sensory Thresholds; Sodium; Spinal Cord; Synaptic Transmission

1982
[3H]bicuculline methochloride binding to low-affinity gamma-aminobutyric acid receptor sites.
    Journal of neurochemistry, 1983, Volume: 41, Issue:6

    Topics: Animals; Bicuculline; Binding, Competitive; Brain; Cattle; gamma-Aminobutyric Acid; Membranes; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Autoradiographic localization of low affinity GABA receptors with [3H]bicuculline methochloride.
    European journal of pharmacology, 1984, Mar-23, Volume: 99, Issue:2-3

    Topics: Animals; Autoradiography; Bicuculline; Brain; Rats; Receptors, Cell Surface; Receptors, GABA-A

1984
The identification and some functions of GABAergic neurons in the proximal retina of the catfish.
    Vision research, 1984, Volume: 24, Issue:8

    Topics: Action Potentials; Animals; Autoradiography; Bicuculline; Fishes; gamma-Aminobutyric Acid; Neurons; Pattern Recognition, Visual; Retina; Retinal Ganglion Cells

1984
Evidence for a physiological role of GABA in the control of guinea-pig intestinal motility.
    Neuroscience letters, 1984, Sep-07, Volume: 50, Issue:1-3

    Topics: Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Gastrointestinal Motility; Guinea Pigs; Ileum; Male; Muscle, Smooth; Myenteric Plexus; Picrotoxin; Sesterterpenes; Tachyphylaxis

1984
Effects of gamma-aminobutyrate and bicuculline on primary afferent depolarization of cutaneous fibres in the cat spinal cord.
    Neuroscience, 1983, Volume: 10, Issue:3

    Topics: Afferent Pathways; Animals; Bicuculline; Cats; Electric Stimulation; Female; gamma-Aminobutyric Acid; Male; Nerve Fibers; Neural Inhibition; Spinal Cord; Spinal Nerves; Sural Nerve; Time Factors

1983
The role of GABAergic inhibition in the cortical effects of monocular deprivation.
    Nature, 1981, May-28, Volume: 291, Issue:5813

    Topics: Animals; Bicuculline; Cats; Functional Laterality; gamma-Aminobutyric Acid; Sensory Deprivation; Vision, Ocular; Visual Cortex

1981
Diazepam biphasically modulates [3H]TBOB binding to the convulsant site of the GABAA receptor complex.
    Journal of receptor and signal transduction research, 1995, Volume: 15, Issue:6

    Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA-A

1995
Dynamic differentiation of GABAA-sensitive influences on orientation selectivity of complex cells in the cat striate cortex.
    Experimental brain research, 1995, Volume: 104, Issue:1

    Topics: Animals; Bicuculline; Cats; GABA Antagonists; GABA-A Receptor Antagonists; Iontophoresis; Orientation; Photic Stimulation; Receptors, GABA-A; Visual Cortex

1995
Interactions between laudanosine, GABA, and opioid subtype receptors: implication for laudanosine seizure activity.
    Brain research, 1994, May-23, Volume: 646, Issue:2

    Topics: Animals; Bicuculline; Binding, Competitive; Brain; Cell Membrane; Cerebral Ventricles; GABA Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Injections, Spinal; Isoquinolines; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Narcotic Antagonists; Pain; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures; Spinal Cord; Substance Withdrawal Syndrome

1994
Reversible loss of dendritic spines and altered excitability after chronic epilepsy in hippocampal slice cultures.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jan-01, Volume: 90, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Bicuculline; Dendrites; Electric Stimulation; Epilepsy; Evoked Potentials; Hippocampus; Membrane Potentials; Organ Culture Techniques; Organophosphorus Compounds; Pyramidal Tracts; Quinoxalines; Rats; Synapses

1993
Interconvertible kinetic states of t-butylbicycloorthobenzoate binding sites of the gamma-aminobutyric acidA ionophores.
    Journal of neurochemistry, 1993, Volume: 61, Issue:6

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Fractionation; Cell Membrane; Cerebral Cortex; Convulsants; gamma-Aminobutyric Acid; Intracellular Membranes; Kinetics; Ligands; Male; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Synaptosomes; Tritium

1993
Novel GABA responses from rod-driven retinal horizontal cells.
    Nature, 1993, Jan-14, Volume: 361, Issue:6408

    Topics: Animals; Bicuculline; Chlorides; Crotonates; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Muscimol; Pentobarbital; Perches; Photoreceptor Cells; Receptors, GABA; Retina

1993
Quantal properties of spontaneous EPSCs in neurones of the guinea-pig dorsal lateral geniculate nucleus.
    The Journal of physiology, 1996, Nov-01, Volume: 496 ( Pt 3)

    Topics: 2-Amino-5-phosphonovalerate; Animals; Bicuculline; Electric Stimulation; Evoked Potentials; Geniculate Bodies; Guinea Pigs; In Vitro Techniques; Kinetics; Neurons; Patch-Clamp Techniques; Picrotoxin; Quantum Theory; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin

1996
Presynaptic control of subunit composition of NMDA receptors mediating synaptic plasticity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Apr-15, Volume: 17, Issue:8

    Topics: Animals; Bicuculline; Cells, Cultured; Coculture Techniques; Embryo, Mammalian; Evoked Potentials; Excitatory Amino Acid Antagonists; Hippocampus; Kinetics; Macromolecular Substances; Magnesium; N-Methylaspartate; Neuronal Plasticity; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Piperidines; Polymerase Chain Reaction; Presynaptic Terminals; Quinoxalines; Rats; Receptors, N-Methyl-D-Aspartate; Synapses

1997
Agrin gene expression in mouse somatosensory cortical neurons during development in vivo and in cell culture.
    Neuroscience, 1997, Volume: 79, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; Agrin; Alternative Splicing; Animals; Bicuculline; Cells, Cultured; Cellular Senescence; DNA Primers; Gene Expression Regulation, Developmental; Genetic Variation; Mice; Mice, Inbred ICR; Neurons; Patch-Clamp Techniques; Polymerase Chain Reaction; Receptors, Cholinergic; RNA, Messenger; Somatosensory Cortex; Synapses; Transcription, Genetic

1997
Properties of GABA(A) receptors in cultured rat oligodendrocyte progenitor cells.
    Neuropharmacology, 1998, Volume: 37, Issue:7

    Topics: Acrylates; Animals; Animals, Newborn; Bicuculline; Brain; Cells, Cultured; GABA Agonists; gamma-Aminobutyric Acid; Membrane Potentials; Oligodendroglia; Patch-Clamp Techniques; Potassium; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; Stem Cells

1998
Influence of genuine kavapyrone enantiomers on the GABA-A binding site.
    Planta medica, 1998, Volume: 64, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Plants, Medicinal; Pyrans; Pyrones; Rats; Receptors, GABA-A; Stereoisomerism; Tritium

1998
Effects of halothane on excitatory neurotransmission to medullary expiratory neurons in a decerebrate dog model.
    Anesthesiology, 2000, Volume: 93, Issue:6

    Topics: Anesthetics, Inhalation; Animals; Bicuculline; Decerebrate State; Dogs; Excitatory Amino Acid Agonists; GABA Antagonists; Halothane; Models, Animal; N-Methylaspartate; Phrenic Nerve; Pulmonary Alveoli; Respiration; Respiratory Center; Synaptic Transmission

2000
GABA receptors modulate trigeminovascular nociceptive neurotransmission in the trigeminocervical complex.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Muscimol; Neurons; Nociceptors; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors; Trigeminal Nuclei

2001
Modulation of synaptic transmission in hippocampal CA1 neurons by a novel neurotoxin (beta-pompilidotoxin) derived from wasp venom.
    Neuroscience research, 2001, Volume: 41, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Bicuculline; Dendrites; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Gerbillinae; Hippocampus; Insect Proteins; Interneurons; Neurons; Neurotoxins; Phosphinic Acids; Propanolamines; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Sodium Channels; Synaptic Transmission; Wasp Venoms

2001
Adrenergic nerves mediate the venoconstrictor response to PVN stimulation.
    Brain research, 2006, Mar-03, Volume: 1076, Issue:1

    Topics: Adrenal Medulla; Adrenergic Agents; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Bicuculline; Blood Circulation; Blood Pressure; Epinephrine; GABA Antagonists; Ganglionic Blockers; Guanethidine; Heart Rate; Male; Paraventricular Hypothalamic Nucleus; Propanolamines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Vasoconstriction; Veins; Venous Pressure

2006
A brief period of epileptiform activity strengthens excitatory synapses in the rat hippocampus in vitro.
    Epilepsia, 2006, Volume: 47, Issue:2

    Topics: Animals; Bicuculline; Cells, Cultured; Disease Models, Animal; Electric Stimulation; Epilepsy; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; Humans; In Vitro Techniques; Interneurons; Long-Term Potentiation; Memory Disorders; Pyramidal Cells; Rats; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

2006
Differential contribution of GABAergic and glycinergic components to inhibitory synaptic transmission in lamina II and laminae III-IV of the young rat spinal cord.
    The European journal of neuroscience, 2007, Volume: 26, Issue:10

    Topics: Analysis of Variance; Animals; Bicuculline; Carrageenan; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Patch-Clamp Techniques; Posterior Horn Cells; Progesterone; Progestins; Rats; Rats, Wistar; Spinal Cord; Strychnine; Synapses; Synaptic Transmission

2007
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
    Psychopharmacology, 2008, Volume: 197, Issue:4

    Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem

2008
Evidence that gamma-aminobutyric acid is part of the neural circuit mediating estradiol negative feedback in anestrous ewes.
    Endocrinology, 2008, Volume: 149, Issue:6

    Topics: Anestrus; Animals; Baclofen; Bicuculline; Dopamine; Estradiol; Feedback; Female; gamma-Aminobutyric Acid; Muscimol; Neurons; Ovariectomy; Sheep

2008
Somatostatin signaling in neuronal cilia is critical for object recognition memory.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-24, Volume: 30, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Adenylyl Cyclases; Amides; Animals; Behavior, Animal; Bicuculline; Biophysics; CA1 Region, Hippocampal; Cilia; Colforsin; Cyclic AMP; Discrimination, Psychological; Electric Stimulation; Female; GABA Antagonists; In Vitro Techniques; Isoquinolines; Locomotion; Long-Term Potentiation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Neuropsychological Tests; Nitrobenzenes; Phosphodiesterase Inhibitors; Receptors, Somatostatin; Recognition, Psychology; Signal Transduction; Somatostatin

2010
Dose-dependent protective effect of connexin43 mimetic peptide against neurodegeneration in an ex vivo model of epileptiform lesion.
    Epilepsy research, 2010, Volume: 92, Issue:2-3

    Topics: Animals; Animals, Newborn; Bicuculline; CA1 Region, Hippocampal; Cell Death; Connexin 43; Culture Media, Serum-Free; Dose-Response Relationship, Drug; GABA Antagonists; In Vitro Techniques; Microtubule-Associated Proteins; Nerve Degeneration; Peptides; Rats; Rats, Wistar; Time Factors

2010
Experience-dependent plasticity acts via GluR1 and a novel neuronal nitric oxide synthase-dependent synaptic mechanism in adult cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Aug-03, Volume: 31, Issue:31

    Topics: Analysis of Variance; Animals; Bicuculline; Cerebral Cortex; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Long-Term Potentiation; Magnesium; Mice; Mice, Inbred C57BL; Mice, Knockout; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; Patch-Clamp Techniques; Receptors, AMPA; Synapses; Synaptic Transmission; Valine; Vibrissae

2011
Chronaxie Measurements in Patterned Neuronal Cultures from Rat Hippocampus.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: 2-Amino-5-phosphonovalerate; 4-Aminopyridine; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Axons; Bicuculline; Calcium; Chronaxy; Dendrites; Embryo, Mammalian; Excitatory Amino Acid Antagonists; GABA Antagonists; Hippocampus; Potassium Channel Blockers; Primary Cell Culture; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA; Receptors, N-Methyl-D-Aspartate

2015
Distinct Modes of Presynaptic Inhibition of Cutaneous Afferents and Their Functions in Behavior.
    Neuron, 2019, 04-17, Volume: 102, Issue:2

    Topics: Animals; Behavior, Animal; Bicuculline; Discrimination, Psychological; GABA-A Receptor Antagonists; Hyperesthesia; Mice; Nerve Tissue Proteins; Neural Inhibition; Neurons, Afferent; Presynaptic Terminals; Pyridazines; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Sensory Receptor Cells; Skin; Spinal Cord Dorsal Horn; Touch

2019
A Structural Rationale for N-Methylbicuculline Acting as a Promiscuous Competitive Antagonist of Inhibitory Pentameric Ligand-Gated Ion Channels.
    Chembiochem : a European journal of chemical biology, 2020, 05-15, Volume: 21, Issue:10

    Topics: Amino Acid Sequence; Bicuculline; Binding Sites; GABA Antagonists; Humans; Ion Channel Gating; Models, Molecular; Protein Conformation; Receptors, GABA-A; Receptors, Glycine; Sequence Homology

2020