Page last updated: 2024-08-26

bicuculline methiodide and sr 95531

bicuculline methiodide has been researched along with sr 95531 in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.69)18.7374
1990's2 (15.38)18.2507
2000's8 (61.54)29.6817
2010's2 (15.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Mienville, JM; Vicini, S1
Maksay, G1
Hess, A; Richter, K; Scheich, H1
Margineanu, DG; Wülfert, E1
Karnup, S; Stelzer, A1
Howard, J; Lambert, TD; Plant, A; Roberts, A; Soffe, S1
Goshgarian, HG; Zimmer, MB1
Osaka, T1
Kamphausen, S; Pedroarena, CM1
Birabil, CG; Marks, GA; Sachs, OW1
Dvorzhak, A; Grantyn, R; Kirischuk, S; Kirmse, K1
Gire, DH; Pandipati, S; Schoppa, NE1
Fehérvári, TD; Okazaki, Y; Sawai, H; Yagi, T1

Other Studies

13 other study(ies) available for bicuculline methiodide and sr 95531

ArticleYear
A pyridazinyl derivative of gamma-aminobutyric acid (GABA), SR 95531, is a potent antagonist of Cl- channel opening regulated by GABAA receptors.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Bicuculline; Chlorides; Electrophysiology; Ion Channels; Pyridazines; Rats; Receptors, GABA-A; Synapses

1987
Differential effects of thiocyanate on the binding thermodynamics of bicuculline methiodide versus SR95531 (gabazine) to the gamma-aminobutyric acid receptor-ionophore complex.
    Biochemical pharmacology, 1998, Sep-15, Volume: 56, Issue:6

    Topics: Animals; Bicuculline; Coloring Agents; GABA Antagonists; Ionophores; Kinetics; Male; Protein Binding; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Temperature; Thermodynamics; Thiocyanates

1998
Functional mapping of transsynaptic effects of local manipulation of inhibition in gerbil auditory cortex.
    Brain research, 1999, Jun-12, Volume: 831, Issue:1-2

    Topics: Animals; Auditory Cortex; Auditory Pathways; Bicuculline; Binding, Competitive; Brain Mapping; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Gerbillinae; Male; Pyridazines; Synapses

1999
Differential paired-pulse effects of gabazine and bicuculline in rat hippocampal CA3 area.
    Brain research bulletin, 2000, Jan-01, Volume: 51, Issue:1

    Topics: Animals; Bicuculline; Electric Stimulation; Epilepsy; Evoked Potentials; Functional Laterality; GABA Antagonists; Hippocampus; Male; Pyridazines; Rats; Rats, Sprague-Dawley

2000
Seizure-like activity in the disinhibited CA1 minislice of adult guinea-pigs.
    The Journal of physiology, 2001, May-01, Volume: 532, Issue:Pt 3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Age Factors; Animals; Bicuculline; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glycine; Guinea Pigs; Hippocampus; Neural Inhibition; Neurons, Afferent; Organ Culture Techniques; Picrotoxin; Pyridazines; Receptors, AMPA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols

2001
Mechanisms and significance of reduced activity and responsiveness in resting frog tadpoles.
    The Journal of experimental biology, 2004, Volume: 207, Issue:Pt 7

    Topics: Animals; Bicuculline; Electrophysiology; Exocrine Glands; GABA Antagonists; Insecta; Larva; Neural Inhibition; NG-Nitroarginine Methyl Ester; Organophosphorus Compounds; Physical Stimulation; Predatory Behavior; Pyridazines; Rest; Swimming; Trigeminal Nerve; Xenopus laevis

2004
GABA, not glycine, mediates inhibition of latent respiratory motor pathways after spinal cord injury.
    Experimental neurology, 2007, Volume: 203, Issue:2

    Topics: Animals; Bicuculline; Body Weight; Efferent Pathways; Female; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Phrenic Nerve; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Respiratory Mechanics; Respiratory Muscles; Spinal Cord Injuries; Stereotaxic Techniques; Strychnine; Vagotomy

2007
Prostaglandin E(2) fever mediated by inhibition of the GABAergic transmission in the region immediately adjacent to the organum vasculosum of the lamina terminalis.
    Pflugers Archiv : European journal of physiology, 2008, Volume: 456, Issue:5

    Topics: Animals; Bicuculline; Body Temperature; Dinoprostone; Dose-Response Relationship, Drug; Fever; GABA Antagonists; gamma-Aminobutyric Acid; Heart Rate; Hypothalamus; Male; Muscimol; Preoptic Area; Pyridazines; Rats; Rats, Wistar; Synaptic Transmission; Vasoconstriction

2008
Glycinergic synaptic currents in the deep cerebellar nuclei.
    Neuropharmacology, 2008, Volume: 54, Issue:5

    Topics: Age Factors; Animals; Animals, Newborn; Bicuculline; Cerebellar Nuclei; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Glycine; Glycine Agents; Glycine Plasma Membrane Transport Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Strychnine; Synapses

2008
Blockade of GABA, type A, receptors in the rat pontine reticular formation induces rapid eye movement sleep that is dependent upon the cholinergic system.
    Neuroscience, 2008, Sep-22, Volume: 156, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Bicuculline; Carbachol; Cholinergic Agonists; Cholinergic Fibers; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscarinic Antagonists; Neural Inhibition; Neural Pathways; Pons; Pyridazines; Rats; Rats, Long-Evans; Receptors, GABA-A; Reticular Formation; Sleep, REM; Synaptic Transmission

2008
GABA transporter 1 tunes GABAergic synaptic transmission at output neurons of the mouse neostriatum.
    The Journal of physiology, 2008, Dec-01, Volume: 586, Issue:23

    Topics: Action Potentials; Animals; Animals, Newborn; Baclofen; Bicuculline; Electric Impedance; Electric Stimulation; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Neostriatum; Neurons; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Presynaptic Terminals; Propanolamines; Pyridazines; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Tetrodotoxin

2008
Adrenergic receptor-mediated disinhibition of mitral cells triggers long-term enhancement of synchronized oscillations in the olfactory bulb.
    Journal of neurophysiology, 2010, Volume: 104, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Agonists; Animals; Animals, Newborn; Bicuculline; Biological Clocks; Biophysical Phenomena; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Inhibitory Postsynaptic Potentials; N-Methylaspartate; Neurons; Norepinephrine; Olfactory Bulb; Pyridazines; Quinoxalines; Rats; Receptors, Adrenergic; Valine

2010
In Vivo Voltage-Sensitive Dye Study of Lateral Spreading of Cortical Activity in Mouse Primary Visual Cortex Induced by a Current Impulse.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Animals; Bicuculline; Electric Stimulation; Evoked Potentials, Visual; GABA Antagonists; Mice; Mice, Inbred C57BL; Photic Stimulation; Pyridazines; Retina; Visual Cortex; Visual Pathways

2015