Page last updated: 2024-08-21

bicuculline and picrotoxinin

bicuculline has been researched along with picrotoxinin in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199011 (40.74)18.7374
1990's11 (40.74)18.2507
2000's4 (14.81)29.6817
2010's1 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Pencheva, N; Radomirov, R; Venkova, K1
Bowman, JW; Lee, BL; Thompson, DP; Whaley, HA1
Isenberg, KE; Yang, J; Zorumski, CF1
Fincher, AS; Frye, GD; Griffith, WH; Lorenzetti, M; Trzeciakowski, J1
Fukuda, H; Matsumoto, K; Ono, H; Yamazaki, J1
Crema, A; De Petris, G; Manzo, L; Onori, L; Rizzi, CA; Tonini, M1
Bhadra, S; Idemudia, SO; Lal, H1
Johnston, GA; Kerr, DI; Ong, J1
Ong, J1
Leeb-Lundberg, LM; Olsen, RW; Snowman, AM; Wong, EH1
Kerr, DI; Ong, J2
Kerr, DI; Krantis, A1
Sarhan, S; Seiler, N1
Pokras, R; Tabakoff, B1
Bormann, J; Feigenspan, A1
Bormann, J; Enz, R1
Bormann, J; Feigenspan, A; Wässle, H1
Morishita, W; Sastry, BR1
Pencheva, N; Radomirov, R1
Fiszer de Plazas, S; Mitridate de Novara, A; Viapiano, MS1
Buckingham, SD; Rauh, J; Sattelle, DB; Schnee, M1
Feigenspan, A; Gustincich, S; Raviola, E1
Baufreton, J; Bioulac, B; Dovero, S; Dufy, B; Garret, M; Taupignon, A1
Chebib, M; Duke, RK; Huang, SH; Johnston, GA; Sasaki, K; Wada, K1
Amin, J; Hadley, SH1

Other Studies

27 other study(ies) available for bicuculline and picrotoxinin

ArticleYear
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
GABAA and GABAB receptor-mediated effects on the spontaneous activity of the longitudinal layer in cat terminal ileum.
    General pharmacology, 1991, Volume: 22, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Cats; GABA Antagonists; gamma-Aminobutyric Acid; Gastrointestinal Motility; Ileum; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Tetrodotoxin

1991
Effects of dihydroavermectin B1a and analogs on stretcher muscle of the lined shore crab, Pachygrapsus crassipes.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1991, Volume: 99, Issue:3

    Topics: Animals; Anthelmintics; Bicuculline; Brachyura; Caenorhabditis; Chlorides; Cobalt; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; In Vitro Techniques; Ivermectin; Membrane Potentials; Membranes; Motor Endplate; Muscimol; Muscles; Picrotoxin; Sesterterpenes; Structure-Activity Relationship; Synapses; Time Factors

1991
Volatile anesthetics gate a chloride current in postnatal rat hippocampal neurons.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1992, Feb-01, Volume: 6, Issue:3

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Anesthetics; Animals; Animals, Newborn; Bicuculline; Chlorine; Chromatography, Gas; Culture Techniques; Dose-Response Relationship, Drug; Electrophysiology; Enflurane; gamma-Aminobutyric Acid; Halothane; Hippocampus; Ion Channel Gating; Isoflurane; Neurons; Picrotoxin; Rats; Sesterterpenes; Strychnine

1992
Comparison of contractile responses of the guinea pig ileum longitudinal muscle to ethanol and GABAA agonists.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:2

    Topics: Animals; Atropine; Bicuculline; Chlorides; Ethanol; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Pentobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Taurine; Tetrodotoxin

1990
Macrolide compounds, ivermectin and milbemycin D, stimulate chloride channels sensitive to GABAergic drugs in cultured chick spinal neurons.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1989, Volume: 93, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Bicuculline; Cells, Cultured; Chick Embryo; Chlorides; Diazepam; gamma-Aminobutyric Acid; Ion Channels; Ivermectin; Lactones; Macrolides; Membrane Potentials; Muscimol; Neurons; Picrotoxin; Sesterterpenes; Spinal Cord

1989
The role of GABAA receptor function in peristaltic activity of the guinea-pig ileum: a comparative study with bicuculline, SR 95531 and picrotoxinin.
    British journal of pharmacology, 1989, Volume: 97, Issue:2

    Topics: Animals; Bicuculline; Electric Stimulation; GABA Antagonists; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Peristalsis; Picrotoxin; Pyridazines; Receptors, GABA-A; Sesterterpenes

1989
The pentylenetetrazol-like interoceptive stimulus produced by ethanol withdrawal is potentiated by bicuculline and picrotoxinin.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1989, Volume: 2, Issue:2

    Topics: Animals; Anxiety; Bicuculline; Discrimination Learning; Dose-Response Relationship, Drug; Ethanol; GABA Antagonists; Male; Pentylenetetrazole; Picrotoxin; Rats; Seizures; Sesterterpenes; Substance Withdrawal Syndrome

1989
Alfaxalone potentiates and mimics GABA-induced contractile responses in the guinea-pig isolated ileum.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Anesthetics; Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Picrotoxin; Pregnanediones; Sesterterpenes

1988
Uptake inhibitors potentiate gamma-aminobutyric acid-induced contractile responses in the isolated ileum of the guinea-pig.
    British journal of pharmacology, 1987, Volume: 91, Issue:1

    Topics: Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Muscle, Smooth; Picrotoxin; Sesterterpenes; Taurine

1987
Barbiturates allosterically inhibit GABA antagonist and benzodiazepine inverse agonist binding.
    European journal of pharmacology, 1984, Jul-13, Volume: 102, Issue:2

    Topics: Allosteric Regulation; Animals; Barbiturates; Benzodiazepines; Bicuculline; Binding, Competitive; Carbolines; Etazolate; GABA Antagonists; In Vitro Techniques; Kinetics; Picrotoxin; Rats; Receptors, GABA-A; Sesterterpenes; Stereoisomerism

1984
Potentiation of GABAA-receptor-mediated responses by barbiturates in the guinea-pig ileum.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Barbiturates; Bicuculline; Drug Interactions; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pentobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes

1984
Gaba induced excitatory responses in the guinea-pig small intestine are antagonized by bicuculline, picrotoxinin and chloride ion blockers.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:3

    Topics: Animals; Bicuculline; Chlorides; Diuretics; Female; Furosemide; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Ion Channels; Male; Muscle Contraction; Myenteric Plexus; Picrotoxin; Sesterterpenes; Sulfonamides

1981
Synergistic anticonvulsant effects of GABA-T inhibitors and glycine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 326, Issue:1

    Topics: 3-Mercaptopropionic Acid; 4-Aminobutyrate Transaminase; Amino Acids; Aminocaproates; Aminooxyacetic Acid; Animals; Anticonvulsants; Bicuculline; Brain Chemistry; Drug Synergism; Ethanolamines; Glycine; Male; Mice; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Sesterterpenes; Strychnine; Vigabatrin

1984
Evidence for a physiological role of GABA in the control of guinea-pig intestinal motility.
    Neuroscience letters, 1984, Sep-07, Volume: 50, Issue:1-3

    Topics: Animals; Bicuculline; Female; gamma-Aminobutyric Acid; Gastrointestinal Motility; Guinea Pigs; Ileum; Male; Muscle, Smooth; Myenteric Plexus; Picrotoxin; Sesterterpenes; Tachyphylaxis

1984
On the mechanism by which dopamine inhibits prolactin release in the anterior pituitary.
    Life sciences, 1982, Dec-06, Volume: 31, Issue:23

    Topics: Animals; Bicuculline; Chlorpromazine; Depression, Chemical; Dopamine; gamma-Aminobutyric Acid; Haloperidol; Male; Mice; Mice, Inbred C57BL; Muscimol; Picrotoxin; Pituitary Gland, Anterior; Prolactin; Sesterterpenes

1982
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction

1994
A single point mutation decreases picrotoxinin sensitivity of the human GABA receptor rho 1 subunit.
    Neuroreport, 1995, Jul-31, Volume: 6, Issue:11

    Topics: Base Sequence; Bicuculline; Cell Line; Humans; Molecular Sequence Data; Patch-Clamp Techniques; Peptide Fragments; Picrotoxin; Point Mutation; Proline; Protein Structure, Tertiary; Receptors, GABA; Serine; Sesterterpenes

1995
Pharmacology of GABA receptor Cl- channels in rat retinal bipolar cells.
    Nature, 1993, Jan-14, Volume: 361, Issue:6408

    Topics: Animals; Animals, Newborn; Bicuculline; Cells, Cultured; Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Membrane Potentials; Membrane Proteins; Neurons; Pentobarbital; Photoreceptor Cells; Picrotoxin; Pregnanediones; Rats; Receptors, GABA-A; Sesterterpenes; Strychnine

1993
Presynaptic actions of GABA and baclofen in CA1 region of the guinea-pig hippocampus in vitro.
    Neuroscience, 1994, Volume: 61, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Calcium; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neuromuscular Depolarizing Agents; Organophosphorus Compounds; Picrotoxin; Receptors, Presynaptic; Sesterterpenes; Tetrodotoxin

1994
Biphasic GABA-A receptor-mediated effect on the spontaneous activity of the circular layer in cat terminal ileum.
    General pharmacology, 1993, Volume: 24, Issue:4

    Topics: Animals; Atropine; Baclofen; Bicuculline; Cats; gamma-Aminobutyric Acid; Ileum; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Tetrodotoxin

1993
Pentobarbital modulatory effect on GABA binding sites in developing chick optic lobe.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1995, Volume: 13, Issue:8

    Topics: Animals; Bicuculline; Brain; Chick Embryo; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Pentobarbital; Picrotoxin; Sesterterpenes; Synaptic Membranes

1995
Pharmacology of skeletal muscle GABA-gated chloride channels in the cockroach Periplaneta americana.
    The Journal of experimental biology, 1997, Volume: 200, Issue:Pt 23

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Isonicotinic Acids; Male; Motor Neurons; Muscle, Skeletal; Periplaneta; Picrotoxin; Receptors, GABA; Sesterterpenes

1997
Pharmacology of GABA(A) receptors of retinal dopaminergic neurons.
    Journal of neurophysiology, 2000, Volume: 84, Issue:4

    Topics: Alkaline Phosphatase; Animals; Benzodiazepines; Bicuculline; Binding Sites; Dopamine; Dose-Response Relationship, Drug; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Mice; Mice, Transgenic; Neurons; Osmolar Concentration; Patch-Clamp Techniques; Picrotoxin; Pregnanediones; Protein Isoforms; Receptors, GABA-A; Retina; Sesterterpenes; Triazoles; Zinc

2000
Activation of GABA(A) receptors in subthalamic neurons in vitro: properties of native receptors and inhibition mechanisms.
    Journal of neurophysiology, 2001, Volume: 86, Issue:1

    Topics: Animals; Bicarbonates; Bicuculline; Chlorides; Diazepam; Electrophysiology; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; Organ Culture Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Subthalamic Nucleus

2001
Bilobalide, a sesquiterpene trilactone from Ginkgo biloba, is an antagonist at recombinant alpha1beta2gamma2L GABA(A) receptors.
    European journal of pharmacology, 2003, Mar-07, Volume: 464, Issue:1

    Topics: Animals; Bicuculline; Cyclopentanes; Diterpenes; Dose-Response Relationship, Drug; Furans; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ginkgo biloba; Ginkgolides; Humans; Membrane Potentials; Oocytes; Picrotoxin; Receptors, GABA-A; Recombinant Proteins; Sesterterpenes; Xenopus laevis

2003
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities.
    The Journal of physiology, 2007, Jun-15, Volume: 581, Issue:Pt 3

    Topics: Action Potentials; Animals; beta-Alanine; Bicuculline; Crotonates; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Furosemide; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Microinjections; Mutation; Neural Inhibition; Neurons; Oocytes; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Sesterterpenes; Taurine; Xenopus laevis; Zinc

2007