Page last updated: 2024-08-21

bicuculline and phenobarbital

bicuculline has been researched along with phenobarbital in 49 studies

Research

Studies (49)

TimeframeStudies, this research(%)All Research%
pre-199028 (57.14)18.7374
1990's12 (24.49)18.2507
2000's7 (14.29)29.6817
2010's1 (2.04)24.3611
2020's1 (2.04)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Haefely, W; Polc, P1
Kozhechkin, SN; Markovich, VV; Molodavkin, GM; Ostrovskaya, RU; Voronina, TA; Zakusov, VV1
Javid, MJ; Stone, WE1
Enna, SJ; Maggi, A1
Frey, HH; Löscher, W1
Gardner, CR; Webster, RA1
Amabeoku, GJ; Chikuni, O2
Cairns, A; Schneiderman, JH; Sterling, CA1
Faktorová, M; Kubová, H; Mares, P1
Alpern, HP; McIntyre, TD1
Hascoet, JM; Monin, P; Vert, P1
Mehta, AK; Ticku, MK2
Gross, RA; Macdonald, RL; Weddle, MG1
Fujiwara, M; Kurahashi, K; Okamoto, T; Tsubomura, T1
Sedlácek, J1
Lloyd, KG1
Benowitz, NL; Bronstein, J; Copeland, JR; Jacob, P; Simon, RP1
Chatt, AB; Ebersole, JS1
Armstrong, DR; Ault, B; Gruenthal, M; Nadler, JV; Okazaki, MM1
Chweh, AY; Coleman, JC; Shenoy, AK; Swinyard, EA1
Clozel, M; Daval, JL; Dubruc, C; Monin, P; Morselli, PL; Vert, P1
Nicoll, RA; Wojtowicz, JM1
Macdonald, RL; Schulz, DW1
Vellucci, SV; Webster, RA1
Bourgeois, BF; Dodson, WE; Ferrendelli, JA1
Clineschmidt, BV1
Macdonald, RL; McLean, MJ1
Gormley, JM; Holtman, JR; Richter, JA; Simon, JR1
Astrup, J; Rehncrona, S; Siesjö, BK1
Obara, N1
Alleva, FR; Alleva, JJ1
Amabeoku, G; Chikuni, O1
Golovko, AI; Sofronov, GA1
Stringer, JL1
Liljequist, S; Tabakoff, B1
Fueta, Y; Janjua, NA; Mita, T; Murai, Y; Ohmori, O; Ohno, K; Ono, T1
Greenfield, LJ; Macdonald, RL; Neelands, TR; Turner, RS; Zhang, J1
Francischi, JN; Pesquero, SM; Tatsuo, MA; Turchetti-Maia, RM; Yokoro, CM1
Hamann, M; Richter, A1
Matsuoka, N; Mochizuki, Y; Mutoh, S; Sugimoto, M; Terai, T; Uchida, I; Yamazaki, S1
Klitgaard, H; Margineanu, DG1
Asimiadou, S; Bittigau, P; Dzietko, M; Felderhoff-Mueser, U; Ikonomidou, C; Kaindl, AM; Manthey, D; Mozrzymas, JW; Pesditschek, S; Pytel, M; Sifringer, M; Studniarczyk, D1
Rahman, M; Wang, MD; Zhu, D1
Mathers, DA; Puil, E; Wan, X1
Behrens, CJ; Caliskan, G; Heinemann, U; Hollnagel, JO; Liotta, A; Rösler, A; ul Haq, R1
Gharpure, A; Hibbs, RE; Howard, RJ; Kim, JJ; Lindahl, E; Noviello, CM; Teng, J; Walsh, RM; Zhu, S; Zhuang, Y1

Reviews

1 review(s) available for bicuculline and phenobarbital

ArticleYear
[GABAergic theory of epilepsy].
    La Revue du praticien, 1986, Jan-21, Volume: 36, Issue:5

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Dogs; Epilepsy; gamma-Aminobutyric Acid; Humans; Mice; Nerve Endings; Pentylenetetrazole; Phenobarbital; Phenytoin; Rats; Receptors, GABA-A; Synapses; Valproic Acid

1986

Other Studies

48 other study(ies) available for bicuculline and phenobarbital

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Effects of two benzodiazepines, phenobarbitone, and baclofen on synaptic transmission in the cat cuneate nucleus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 294, Issue:2

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Cats; Diazepam; Drug Interactions; Evoked Potentials; Flunitrazepam; Glutamate Decarboxylase; Medulla Oblongata; Neural Inhibition; Phenobarbital; Picrotoxin; Propionates; Semicarbazides; Synapses; Synaptic Transmission

1976
Further evidence for GABA-ergic mechanisms in the action of benzodiazepines.
    Archives internationales de pharmacodynamie et de therapie, 1977, Volume: 229, Issue:2

    Topics: Aminobutyrates; Animals; Anti-Anxiety Agents; Benzodiazepines; Bicuculline; Cats; Cerebral Cortex; Electric Stimulation; gamma-Aminobutyric Acid; Male; Mice; Phenobarbital; Phenytoin; Rabbits; Rats; Reflex; Sciatic Nerve; Thiosemicarbazones

1977
Benzodiazepines and phenobarbital as antagonists of dissimilar chemical convulsants.
    Epilepsia, 1978, Volume: 19, Issue:4

    Topics: 3-Mercaptopropionic Acid; Animals; Anti-Anxiety Agents; Anticonvulsants; Bicuculline; Chlordiazepoxide; Convulsants; Diazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Mice; Nitrazepam; Pentylenetetrazole; Phenobarbital; Picrotoxin; Therapeutic Equivalency

1978
Characteristics of muscimol accumulation in mouse brain after systemic administration.
    Neuropharmacology, 1979, Volume: 18, Issue:4

    Topics: Animals; Bicuculline; Brain; gamma-Aminobutyric Acid; History, 18th Century; Injections, Intravenous; Mice; Muscimol; Oxazoles; Phenobarbital; Time Factors

1979
Di-n-propylacetic acid--profile of anticonvulsant activity in mice.
    Arzneimittel-Forschung, 1976, Volume: 26, Issue:2

    Topics: Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Electroshock; Ethosuximide; Female; Male; Mice; Pentylenetetrazole; Phenobarbital; Picrotoxin; Seizures; Strychnine; Trimethadione; Valerates; Valproic Acid

1976
Convulsant-anticonvulsant interactions on seizure activity and cortical acetylcholine release.
    European journal of pharmacology, 1977, Apr-07, Volume: 42, Issue:3

    Topics: Acetylcholine; Animals; Anticonvulsants; Bicuculline; Blood Pressure; Cerebral Cortex; Convulsants; Drug Interactions; Electroencephalography; Male; Pentylenetetrazole; Phenobarbital; Phenytoin; Rats; Seizures; Time Factors; Trimethadione

1977
Effects of some GABAergic agents on quinine-induced seizures in mice.
    Experientia, 1992, Jul-15, Volume: 48, Issue:7

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Diazepam; Male; Mice; Mice, Inbred Strains; Muscimol; Phenobarbital; Phenytoin; Quinine; Receptors, GABA-A; Seizures

1992
Evoked CA3 field potentials corresponding to both EPSPs and IPSPs in hippocampal slice.
    Brain research, 1992, Jan-13, Volume: 569, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Dendrites; Electric Stimulation; Evoked Potentials; Guinea Pigs; Hippocampus; In Vitro Techniques; Penicillins; Pentobarbital; Phenobarbital; Pyramidal Tracts; Quinoxalines; Receptors, GABA-A; Synapses

1992
Effect of phenobarbital on motor seizures elicited by picrotoxin and bicuculline in rats.
    Homeostasis in health and disease : international journal devoted to integrative brain functions and homeostatic systems, 1991, Volume: 33, Issue:3

    Topics: Animals; Bicuculline; Male; Pentylenetetrazole; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Seizures

1991
Patterns of convulsive susceptibility in the long-sleep and short-sleep selected mouse lines.
    Brain research bulletin, 1989, Volume: 22, Issue:5

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Female; Flumazenil; Male; Mice; Pentylenetetrazole; Phenobarbital; Reaction Time; Seizures; Sleep

1989
Autoregulation of cerebral blood flow. Effect of phenobarbital and pancuronium in the newborn piglet.
    Developmental pharmacology and therapeutics, 1989, Volume: 13, Issue:2-4

    Topics: Animals; Animals, Newborn; Bicuculline; Blood Gas Analysis; Cardiac Output; Cerebrovascular Circulation; Pancuronium; Phenobarbital; Seizures; Swine

1989
Interactions of pentobarbital and phenobarbital with GABAergic drugs against chemoconvulsants in rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Diazepam; Drug Interactions; Isoxazoles; Male; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Strychnine

1988
Benzodiazepine, beta-carboline, and barbiturate actions on GABA responses.
    Advances in biochemical psychopharmacology, 1986, Volume: 41

    Topics: Animals; Anti-Anxiety Agents; Barbiturates; Bicuculline; Carbolines; Cells, Cultured; Clonazepam; Diazepam; gamma-Aminobutyric Acid; Membrane Potentials; Mice; Neurons; Nitrazepam; Pentobarbital; Phenobarbital; Picrotoxin; Receptors, GABA-A; Spinal Cord

1986
Effects of barbiturates on the inhibitory action of GABA on excitatory response of the stomach to stimulation of vagal afferent fibers in cat.
    Life sciences, 1987, Jul-27, Volume: 41, Issue:4

    Topics: Afferent Pathways; Animals; Bicuculline; Cats; Chloralose; Electric Stimulation; Female; gamma-Aminobutyric Acid; Hexamethonium; Hexamethonium Compounds; Kinetics; Male; Phenobarbital; Picrotoxin; Stomach; Vagus Nerve

1987
Consequences of chronic phenobarbital blockade of spontaneous motility in chick embryos for the development of central motor output activity.
    Physiologia Bohemoslovaca, 1988, Volume: 37, Issue:2

    Topics: Animals; Bicuculline; Central Nervous System; Chick Embryo; gamma-Aminobutyric Acid; Motor Activity; Oxazepam; Pentylenetetrazole; Phenobarbital; Strychnine

1988
Comparison of anticonvulsant effect of pentobarbital and phenobarbital against seizures induced by maximal electroshock and picrotoxin in rats.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:5

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Anticonvulsants; Bicuculline; Electroshock; Male; Muscimol; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1986
Brain phenobarbital uptake during prolonged status epilepticus.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1987, Volume: 7, Issue:6

    Topics: Animals; Bicuculline; Blood; Blood Pressure; Blood-Brain Barrier; Brain; Cerebrovascular Circulation; Electroencephalography; Female; Hydrogen-Ion Concentration; Kinetics; Lactates; Lactic Acid; Phenobarbital; Sheep; Status Epilepticus

1987
Spread and arrest of seizures: the importance of layer 4 in laminar interactions during neocortical epileptogenesis.
    Advances in neurology, 1986, Volume: 44

    Topics: Action Potentials; Animals; Anticonvulsants; Bicuculline; Biomechanical Phenomena; Cats; Cerebral Cortex; Disease Susceptibility; Epilepsy; Models, Neurological; Neural Pathways; Neurons; Penicillins; Phenobarbital; Phenytoin; Reaction Time

1986
Kainic acid seizures and neuronal cell death: insights from studies of selective lesions and drugs.
    Advances in experimental medicine and biology, 1986, Volume: 203

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Convulsants; Hippocampus; Kainic Acid; Limbic System; Male; Nerve Degeneration; Neural Inhibition; Neural Pathways; Phenobarbital; Rats; Seizures; Time Factors

1986
An analysis of the in vivo interactions between chemical convulsants and anticonvulsants.
    Life sciences, 1985, Aug-26, Volume: 37, Issue:8

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Mice; Pentylenetetrazole; Phenobarbital; Picrotoxin; Valproic Acid

1985
Regional cerebral blood flow during bicuculline-induced seizures in the newborn piglet: effect of phenobarbital.
    Developmental pharmacology and therapeutics, 1985, Volume: 8, Issue:3

    Topics: Acid-Base Equilibrium; Animals; Animals, Newborn; Bicuculline; Blood Gas Analysis; Blood Pressure; Cerebrovascular Circulation; Microspheres; Phenobarbital; Potassium Chloride; Seizures; Swine; Time Factors

1985
The effects of pentobarbital and related compounds on frog motoneurons.
    Brain research, 1980, Jun-02, Volume: 191, Issue:1

    Topics: Amino Acids; Animals; Anura; Bicuculline; Chloralose; Chlordiazepoxide; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glutamates; Motor Neurons; Muscimol; Pentobarbital; Phenobarbital; Phenytoin; Picrotoxin; Spinal Cord; Strychnine; Synaptic Transmission

1980
Barbiturate enhancement of GABA-mediated inhibition and activation of chloride ion conductance: correlation with anticonvulsant and anesthetic actions.
    Brain research, 1981, Mar-23, Volume: 209, Issue:1

    Topics: Animals; Bicuculline; Chlorides; Dose-Response Relationship, Drug; Evoked Potentials; gamma-Aminobutyric Acid; Ion Channels; Mice; Neural Inhibition; Neurons; Pentobarbital; Phenobarbital; Spinal Cord

1981
Is Ro15-1788 a partial agonist at benzodiazepine receptors?
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Animals; Benzodiazepinones; Bicuculline; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C3H; Phenobarbital; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
Primidone, phenobarbital, and PEMA: I. Seizure protection, neurotoxicity, and therapeutic index of individual compounds in mice.
    Neurology, 1983, Volume: 33, Issue:3

    Topics: Animals; Bicuculline; Brain; Brain Chemistry; Electroshock; Female; Malonates; Mice; Mice, Inbred Strains; Pentylenetetrazole; Phenobarbital; Phenylethylmalonamide; Primidone; Seizures

1983
Effect of the benzodiazepine receptor antagonist Ro 15-1788 on the anticonvulsant and anticonflict actions of MK-801.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepinones; Bicuculline; Chlordiazepoxide; Clonazepam; Conflict, Psychological; Dibenzocycloheptenes; Dizocilpine Maleate; Drug Interactions; Female; Flumazenil; Mice; Phenobarbital; Rats; Rats, Inbred Strains

1982
Cellular bases of barbiturate and phenytoin anticonvulsant drug action.
    Epilepsia, 1982, Volume: 23 Suppl 1

    Topics: Animals; Barbiturates; Bicuculline; Drug Interactions; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Neurons; Pentobarbital; Phenobarbital; Phenytoin; Synapses

1982
High-affinity choline uptake in the hippocampus: its relationship to the physiological state produced by administration of barbiturates and other treatments.
    Journal of neurochemistry, 1982, Volume: 39, Issue:5

    Topics: Animals; Barbiturates; Bicuculline; Choline; Convulsants; Hippocampus; Kinetics; Male; Mice; Pentobarbital; Phenobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Septum Pellucidum; Synaptosomes

1982
The increase in extracellular potassium concentration in the ischemic brain in relation to the preischemic functional activity and cerebral metabolic rate.
    Brain research, 1980, Oct-13, Volume: 199, Issue:1

    Topics: Adenosine Triphosphate; Amphetamine; Animals; Bicuculline; Blood Pressure; Body Temperature; Brain Ischemia; Cerebral Cortex; Energy Metabolism; Extracellular Space; Male; Phenobarbital; Potassium; Rats

1980
[Involvement of GABAergic and NMDA systems in drug-induced convulsions in mice].
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1995, Volume: 15, Issue:1

    Topics: Animals; Anticonvulsants; Bicuculline; Calcium Channels; Chloride Channels; Male; Mice; Mice, Inbred Strains; Muscimol; Phenobarbital; Picrotoxin; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Seizures

1995
Synergistic inhibition by benzodiazepine and barbiturate drugs of the clock control of ovulation in hamsters.
    Chronobiology international, 1995, Volume: 12, Issue:1

    Topics: Animals; Bicuculline; Circadian Rhythm; Cricetinae; Drug Synergism; Estrus; Female; GABA-A Receptor Antagonists; Luteinizing Hormone; Mesocricetus; Ovulation; Phenobarbital; Time Factors; Triazolam

1995
GABAergic and dopaminergic systems may be involved in seizures induced by pyrimethamine in mice.
    General pharmacology, 1994, Volume: 25, Issue:6

    Topics: Animals; Bicuculline; Diazepam; Dopamine; Drug Interactions; gamma-Aminobutyric Acid; Levodopa; Mice; Mice, Inbred Strains; Muscimol; Phenobarbital; Pyrimethamine; Seizures

1994
[Effect of preliminary administration of phenobarbital on the toxicity of GABA-lytics in mice].
    Biulleten' eksperimental'noi biologii i meditsiny, 1993, Volume: 115, Issue:5

    Topics: 3-Mercaptopropionic Acid; Animals; Antidotes; Barbiturates; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Male; Mice; Phenobarbital; Picrotoxin; Time Factors

1993
Alterations in both excitation and inhibition occur before the onset of seizure activity in the hippocampus.
    Epilepsy research, 1993, Volume: 16, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Diazepam; Electric Stimulation; Evoked Potentials; Hippocampus; Ketamine; Kindling, Neurologic; Limbic System; Male; Neurons; Phenobarbital; Pyramidal Tracts; Rats; Rats, Sprague-Dawley; Seizures; Stereotaxic Techniques; Synapses

1993
Cimetidine-induced seizures in mice. Antagonism by some GABAergic agents.
    Biochemical pharmacology, 1993, Dec-14, Volume: 46, Issue:12

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Cimetidine; Diazepam; Female; Mice; Muscimol; Phenobarbital; Phenytoin; Picrotoxin; Receptors, GABA; Seizures; Strychnine

1993
Bicuculline-produced regional differences in the modulation of 35S-TBPS binding by GABA, pentobarbital and diazepam in mouse cerebellum and cortex.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Receptors, GABA-A

1993
Granule cell disinhibition in dentate gyrus of genetically seizure susceptible El mice.
    Brain research, 1997, Jan-16, Volume: 745, Issue:1-2

    Topics: Aging; Animals; Anticonvulsants; Bicuculline; Chromatography, High Pressure Liquid; Dentate Gyrus; Electrophysiology; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Phenobarbital; Seizures

1997
GABAA receptor pharmacology and subtype mRNA expression in human neuronal NT2-N cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jul-01, Volume: 18, Issue:13

    Topics: Anticonvulsants; Bicuculline; Carbolines; Convulsants; Diazepam; Diuretics; DNA Primers; Furosemide; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Hypnotics and Sedatives; Lanthanum; Neurons; Patch-Clamp Techniques; Pentobarbital; Phenobarbital; Picrotoxin; Polymerase Chain Reaction; Pregnanediones; Pregnenolone; Pyridines; Receptors, GABA-A; RNA, Messenger; Teratocarcinoma; Triazoles; Tumor Cells, Cultured; Zinc; Zolpidem

1998
Acute phenobarbital administration induces hyperalgesia: pharmacological evidence for the involvement of supraspinal GABA-A receptors.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2001, Volume: 34, Issue:3

    Topics: Analysis of Variance; Animals; Bicuculline; Dose-Response Relationship, Drug; GABA Antagonists; Hyperalgesia; Hypnotics and Sedatives; Male; Pain Measurement; Pain Threshold; Phenobarbital; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord

2001
Effects of striatal injections of GABA(A) receptor agonists and antagonists in a genetic animal model of paroxysmal dystonia.
    European journal of pharmacology, 2002, May-17, Volume: 443, Issue:1-3

    Topics: Animals; Bicuculline; Binding Sites; Corpus Striatum; Cricetinae; Dystonia; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Mesocricetus; Microinjections; Muscimol; Pentylenetetrazole; Phenobarbital

2002
Intracerebroventricular injection of the antibiotic cefoselis produces convulsion in mice via inhibition of GABA receptors.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 74, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Anticonvulsants; Bicuculline; Carbamazepine; Ceftizoxime; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; N-Methylaspartate; Phenobarbital; Phenytoin; Receptors, GABA; Seizures; Sodium Channel Blockers

2002
Levetiracetam has no significant gamma-aminobutyric acid-related effect on paired-pulse interaction in the dentate gyrus of rats.
    European journal of pharmacology, 2003, Apr-18, Volume: 466, Issue:3

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Clonazepam; Convulsants; Dentate Gyrus; Diazepam; Electric Stimulation; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Levetiracetam; Male; Phenobarbital; Piracetam; Rats; Rats, Sprague-Dawley; Receptors, GABA; Synaptic Transmission; Time Factors

2003
Protection with estradiol in developmental models of apoptotic neurodegeneration.
    Annals of neurology, 2005, Volume: 58, Issue:2

    Topics: Animals; Animals, Newborn; Apoptosis; Bicuculline; Blotting, Western; Brain; Caenorhabditis elegans Proteins; Cell Count; Cells, Cultured; Cerebral Cortex; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Estradiol; Estrogen Antagonists; Extracellular Signal-Regulated MAP Kinases; GABA Antagonists; Hypoxia; Immunohistochemistry; In Situ Nick-End Labeling; Membrane Potentials; Neurodegenerative Diseases; Neurons; Neuroprotective Agents; Patch-Clamp Techniques; Phenobarbital; Phenytoin; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Rats, Wistar; Receptors, GABA-A; Silver Staining; Tamoxifen

2005
Protons inhibit Cl- conductance by direct or allosteric interaction with the GABA-binding site in the rat recombinant alpha1beta2gamma2L and alpha1beta2 GABAA receptor.
    European journal of pharmacology, 2005, Dec-28, Volume: 528, Issue:1-3

    Topics: Allosteric Regulation; Animals; Bicuculline; Chlorides; Dose-Response Relationship, Drug; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Ion Channel Gating; Membrane Potentials; Oocytes; Phenobarbital; Protons; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Xenopus laevis

2005
Barbiturate activation and modulation of GABA(A) receptors in neocortex.
    Neuropharmacology, 2007, Volume: 52, Issue:4

    Topics: Animals; Animals, Newborn; Barbiturates; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Neocortex; Neurons; Patch-Clamp Techniques; Pentobarbital; Phenobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Thalamus

2007
Partial disinhibition is required for transition of stimulus-induced sharp wave-ripple complexes into recurrent epileptiform discharges in rat hippocampal slices.
    Journal of neurophysiology, 2011, Volume: 105, Issue:1

    Topics: Action Potentials; Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Electric Stimulation; Epilepsy; Female; Hippocampus; Long-Term Potentiation; Male; Models, Animal; Nicotine; Phenobarbital; Potassium; Pyramidal Cells; Rats; Rats, Wistar

2011
Shared structural mechanisms of general anaesthetics and benzodiazepines.
    Nature, 2020, Volume: 585, Issue:7824

    Topics: Allosteric Regulation; Anesthetics, General; Barbiturates; Benzodiazepines; Bicuculline; Binding Sites; Binding, Competitive; Cryoelectron Microscopy; Diazepam; Electrophysiology; Etomidate; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Phenobarbital; Picrotoxin; Propofol; Receptors, GABA-A

2020