Page last updated: 2024-08-21

bicuculline and naltrexone

bicuculline has been researched along with naltrexone in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19902 (7.69)18.7374
1990's10 (38.46)18.2507
2000's10 (38.46)29.6817
2010's3 (11.54)24.3611
2020's1 (3.85)2.80

Authors

AuthorsStudies
Cheney, DL; Costa, E; Revuelta, AV; Wood, PL1
Pinnock, RD2
Jackson, HC; Nutt, DJ1
Castellano, C; Introini-Collison, IB; McGaugh, JL; Pavone, F1
Lemaire, S; Shukla, VK1
Randić, M; Wang, RA1
Lewis, DV; Xie, CW1
Castellano, C; Introini-Collison, IB; McGaugh, JL1
Brusa, L; D'Amore, A; Lorenzini, P; Massotti, M1
Mulder, AH; Ronken, E; Schoffelmeer, AN1
Fields, HL; Roychowdhury, SM1
Misawa, M; Mizoguchi, H; Nagase, H; Narita, M; Suzuki, T; Takahashi-Nakano, Y; Tseng, LF; Yajima, Y1
Bodnar, RJ; Christian, G; Echo, JA; Lamonte, N; Ragnauth, A; Znamensky, V1
Bhandari, RN; Clarke, RW; Leggett, J1
Chung, J; Kim, C; Kim, E; Kim, Y; Koo, G; Lee, C; Shin, M1
Castellan-Baldan, L; Coimbra, NC; Corrêa, SA; Da Silva, LA; Eichenberger, GC; Maruoka, RY; Osaki, MY; Resende, GC; Ribeiro, SJ1
Chen, SR; Li, DP; Pan, HL; Pan, YZ1
Brailoiu, GC; Dun, NJ; Ohtubo, Y; Wu, SY1
Billi, S; De Laurentiis, A; Fernández-Solari, J; Franchi, A; McCann, SM; Mohn, C; Rettori, V; Scorticati, C1
Carai, MA; Colombo, G; Gessa, GL1
Chen, Q; Dong, L; Fu, CY; Ni, JM; Wang, R; Zhao, YL1
Aicher, SA; Arttamangkul, S; Bobeck, EN; Hegarty, DM; Ingram, SL; Macey, TA; Morgan, MM1
Prado, WA; Silva, JR; Silva, ML1
Almada, RC; Calvo, F; Coimbra, NC; da Silva Soares, R; da Silva, JA; de Paiva, YB; Medeiros, P; Roncon, CM1
Chen, Q; He, W; Ivanova, D; Kuang, Y; Lass, G; Li, X; Liu, Y; Long, H; Lyu, Q; O'Byrne, KT; Wang, L; Wang, Y; Yu, S1

Other Studies

26 other study(ies) available for bicuculline and naltrexone

ArticleYear
GABAergic mediation in the inhibition of hippocampal acetylcholine turnover rate elicited by delta 9-tetrahydrocannabinol.
    Neuropharmacology, 1979, Volume: 18, Issue:6

    Topics: Acetylcholine; Animals; Bicuculline; Dopamine; Dronabinol; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Muscimol; Naltrexone; Norepinephrine; Rats; Substantia Nigra

1979
A highly selective kappa-opioid receptor agonist, CI-977, reduces excitatory synaptic potentials in the rat locus coeruleus in vitro.
    Neuroscience, 1992, Volume: 47, Issue:1

    Topics: Amino Acids; Analgesics; Animals; Benzofurans; Benzomorphans; Bicuculline; Depression, Chemical; Electric Stimulation; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; In Vitro Techniques; Ligands; Locus Coeruleus; Membrane Potentials; Naloxone; Naltrexone; Picrotoxin; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1992
Activation of kappa-opioid receptors depresses electrically evoked excitatory postsynaptic potentials on 5-HT-sensitive neurones in the rat dorsal raphé nucleus in vitro.
    Brain research, 1992, Jun-26, Volume: 583, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Animals; Benzofurans; Bicuculline; Bombesin; Cholecystokinin; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; Glutamates; Glutamic Acid; In Vitro Techniques; Kynurenic Acid; N-Methylaspartate; Naloxone; Naltrexone; Neurons; Picrotoxin; Prazosin; Pyrrolidines; Quinoxalines; Raphe Nuclei; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Synapses; Tetrodotoxin

1992
Differential effects of selective mu-, kappa- and delta-opioid antagonists on electroshock seizure threshold in mice.
    Psychopharmacology, 1991, Volume: 103, Issue:3

    Topics: Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Electroshock; gamma-Aminobutyric Acid; Indoles; Male; Mice; Mice, Inbred Strains; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Phenytoin; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1991
Effects of naloxone and naltrexone on memory consolidation in CD1 mice: involvement of GABAergic mechanisms.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:2

    Topics: Animals; Avoidance Learning; Bicuculline; gamma-Aminobutyric Acid; Male; Memory; Mice; Mice, Inbred Strains; Muscimol; Naloxone; Naltrexone; Picrotoxin

1989
Norbinaltorphimine protection against N-methyl-D-aspartic acid-induced convulsions and mortality.
    European journal of pharmacology, 1993, Feb-09, Volume: 231, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Bicuculline; Binding, Competitive; Brain; Ibotenic Acid; Injections, Intraventricular; Kainic Acid; Male; Mice; N-Methylaspartate; Naltrexone; Receptors, N-Methyl-D-Aspartate; Seizures

1993
Activation of mu-opioid receptor modulates GABAA receptor-mediated currents in isolated spinal dorsal horn neurons.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Action Potentials; Amino Acid Sequence; Animals; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Molecular Sequence Data; Muscimol; Naloxone; Naltrexone; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Opioid, mu; Spinal Cord

1994
Endogenous opioids regulate long-term potentiation of synaptic inhibition in the dentate gyrus of rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:5 Pt 2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Bicuculline; Electric Stimulation; GABA-A Receptor Antagonists; Hippocampus; Homeostasis; In Vitro Techniques; Long-Term Potentiation; Male; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; Opioid Peptides; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Time Factors

1995
Interaction of beta-endorphin and GABAergic drugs in the regulation of memory storage.
    Behavioral and neural biology, 1993, Volume: 60, Issue:2

    Topics: Animals; Avoidance Learning; beta-Endorphin; Bicuculline; Conditioning, Classical; Dose-Response Relationship, Drug; Electroshock; Fear; Injections, Intraperitoneal; Male; Mice; Muscimol; Naloxone; Naltrexone; Picrotoxin; Reaction Time; Receptors, GABA; Receptors, Opioid; Retention, Psychology

1993
Area tempestas modulates the behavioural responses to nociceptive stimuli in rats.
    Annali dell'Istituto superiore di sanita, 1993, Volume: 29, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anticonvulsants; Azocines; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Escape Reaction; Foot; Hot Temperature; Male; Morphine; Naltrexone; Narcotic Antagonists; Olfactory Pathways; Pain; Phenazocine; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Seizures; Tail

1993
Interacting presynaptic kappa-opioid and GABAA receptors modulate dopamine release from rat striatal synaptosomes.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: Analysis of Variance; Animals; Benzeneacetamides; Bicuculline; Corpus Striatum; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; gamma-Aminobutyric Acid; Kinetics; Male; Naltrexone; Narcotics; Oligopeptides; Picrotoxin; Potassium; Pyrrolidines; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Opioid, kappa; Synaptosomes

1993
Endogenous opioids acting at a medullary mu-opioid receptor contribute to the behavioral antinociception produced by GABA antagonism in the midbrain periaqueductal gray.
    Neuroscience, 1996, Volume: 74, Issue:3

    Topics: Animals; Bicuculline; Brain Mapping; GABA Antagonists; Male; Medulla Oblongata; Mesencephalon; Microinjections; Models, Neurological; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Somatostatin; Spinal Cord; Time Factors

1996
Effects of differential modulation of mu-, delta- and kappa-opioid systems on bicuculline-induced convulsions in the mouse.
    Brain research, 2000, Apr-17, Volume: 862, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Bicuculline; Brain Chemistry; Convulsants; Enkephalin, D-Penicillamine (2,5)-; Epilepsy, Tonic-Clonic; Injections, Intraventricular; Injections, Subcutaneous; Male; Mice; Morphine; Naltrexone; Narcotic Antagonists; Quinolines; Receptors, GABA-A; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures; Synaptic Transmission

2000
gamma-Aminobutyric acid receptor subtype antagonists differentially alter opioid-induced feeding in the shell region of the nucleus accumbens in rats.
    Brain research, 2001, Jul-06, Volume: 906, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Naltrexone; Narcotic Antagonists; Narcotics; Neurons; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Opioid

2001
Opioid and GABA receptors involved in mediation and modulation of tonic and stimulus-evoked inhibition of a spinal reflex in the decerebrated and spinalized rabbit.
    Neuropharmacology, 2001, Volume: 41, Issue:3

    Topics: Animals; Bicuculline; Conditioning, Classical; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Methionine; Female; GABA Antagonists; Male; Muscle Tonus; Naloxone; Naltrexone; Narcotic Antagonists; Organophosphorus Compounds; Rabbits; Receptors, GABA; Receptors, Opioid; Receptors, Opioid, mu; Receptors, sigma; Reflex

2001
Modulation of Chelidonii herba on GABA activated chloride current in rat PAG neurons.
    The American journal of Chinese medicine, 2001, Volume: 29, Issue:2

    Topics: Animals; Bicuculline; Chelidonium; Chloride Channels; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Naltrexone; Narcotic Antagonists; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Plant Preparations; Rats; Rats, Sprague-Dawley

2001
Neuroanatomical and psychopharmacological evidence for interaction between opioid and GABAergic neural pathways in the modulation of fear and defense elicited by electrical and chemical stimulation of the deep layers of the superior colliculus and dorsal
    Neuropharmacology, 2002, Volume: 42, Issue:1

    Topics: Aggression; Animals; Bicuculline; Electric Stimulation; Fear; GABA Antagonists; Immunohistochemistry; Male; Mesencephalon; Microinjections; Naloxone; Naltrexone; Narcotic Antagonists; Neural Pathways; Neurons; Periaqueductal Gray; Rats; Rats, Wistar; Receptors, GABA; Receptors, Opioid; Stimulation, Chemical; Superior Colliculi

2002
Activation of delta-opioid receptors excites spinally projecting locus coeruleus neurons through inhibition of GABAergic inputs.
    Journal of neurophysiology, 2002, Volume: 88, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics, Opioid; Animals; Bicuculline; Dopamine beta-Hydroxylase; Electrophysiology; Enkephalin, D-Penicillamine (2,5)-; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Immunohistochemistry; Locus Coeruleus; Naltrexone; Narcotic Antagonists; Neural Pathways; Neurons; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Spinal Cord

2002
Effects of endomorphin on substantia gelatinosa neurons in rat spinal cord slices.
    British journal of pharmacology, 2003, Volume: 140, Issue:6

    Topics: Animals; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Excitatory Postsynaptic Potentials; Female; Male; Membrane Potentials; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; Oligopeptides; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Spinal Cord; Substantia Gelatinosa; Tetrodotoxin; Time Factors

2003
Alcohol inhibits luteinizing hormone-releasing hormone release by activating the endocannabinoid system.
    Proceedings of the National Academy of Sciences of the United States of America, 2004, Mar-02, Volume: 101, Issue:9

    Topics: Animals; Arachidonic Acids; Bicuculline; Cannabinoid Receptor Modulators; Colforsin; Cyclic AMP; Endocannabinoids; Ethanol; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; Kinetics; Male; N-Methylaspartate; Naltrexone; Polyunsaturated Alkamides; Radioimmunoassay; Rats; Rats, Wistar

2004
Resuscitative effect of a gamma-aminobutyric acid B receptor antagonist on gamma-hydroxybutyric acid mortality in mice.
    Annals of emergency medicine, 2005, Volume: 45, Issue:6

    Topics: Animals; Benzocycloheptenes; Bicuculline; Drug Overdose; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Morpholines; Naltrexone; Neuroprotective Agents; Neurotransmitter Agents; Survival Rate; Taurine

2005
In vivo characterization of the effects of human hemokinin-1 and human hemokinin-1(4-11), mammalian tachykinin peptides, on the modulation of pain in mice.
    Brain, behavior, and immunity, 2008, Volume: 22, Issue:6

    Topics: Analgesics; Animals; Benzamides; Bicuculline; Dose-Response Relationship, Drug; GABA Antagonists; Humans; Injections, Intraventricular; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Neurokinin-1 Receptor Antagonists; Pain; Pain Measurement; Peptide Fragments; Piperidines; Receptors, Neurokinin-2; Tachykinins; Tropanes

2008
Opioid receptor internalization contributes to dermorphin-mediated antinociception.
    Neuroscience, 2010, Jun-30, Volume: 168, Issue:2

    Topics: Analgesics, Opioid; Animals; Bicuculline; Concanavalin A; Dynamins; Fluorescent Dyes; GABA-A Receptor Antagonists; Male; Microinjections; Naltrexone; Neurons; Opioid Peptides; Pain; Pain Measurement; Peptides; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2010
Analgesia induced by 2- or 100-Hz electroacupuncture in the rat tail-flick test depends on the anterior pretectal nucleus.
    Life sciences, 2013, Nov-06, Volume: 93, Issue:20

    Topics: Analgesia; Animals; Atropine; Bicuculline; Electroacupuncture; GABA-A Receptor Antagonists; Male; Mesencephalon; Methiothepin; Methysergide; Muscarinic Antagonists; Naloxone; Naltrexone; Narcotic Antagonists; Pain Management; Rats; Rats, Wistar; Serotonin Antagonists; Somatostatin

2013
The Blockade of µ1- and κ-Opioid Receptors in the Inferior Colliculus Decreases the Expression of Panic Attack-Like Behaviours Induced by Chemical Stimulation of the Dorsal Midbrain.
    Neuropsychobiology, 2019, Volume: 78, Issue:4

    Topics: Animals; Behavior, Animal; Bicuculline; Exploratory Behavior; GABA-A Receptor Antagonists; Inferior Colliculi; Male; Mesencephalon; Naloxone; Naltrexone; Narcotic Antagonists; Neurons; Panic; Rats; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu

2019
Dynorphin and GABAA Receptor Signaling Contribute to Progesterone's Inhibition of the LH Surge in Female Mice.
    Endocrinology, 2020, 05-01, Volume: 161, Issue:5

    Topics: Animals; Bicuculline; Dynorphins; Estradiol; Female; GABA Antagonists; Hypothalamus; Hypothalamus, Anterior; Kisspeptins; Luteinizing Hormone; Mice, Inbred C57BL; Naltrexone; Neurons; Organophosphorus Compounds; Ovariectomy; Progesterone; Receptors, GABA-A; Signal Transduction

2020