Page last updated: 2024-08-21

bicuculline and flurazepam

bicuculline has been researched along with flurazepam in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-199024 (75.00)18.7374
1990's5 (15.63)18.2507
2000's3 (9.38)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dray, A; Straughan, DW1
Bowery, NG; Dray, A1
Franco, S; Schlosser, W1
Ferrendelli, JA; Miller, JW1
Chiu, TH; Ngur, DO; Rosenberg, HC1
Chiu, TH; Rosenberg, HC; Tietz, EI1
Haji, A; Takeda, R1
Gale, RG; Little, HJ; Nutt, DJ; Standing, BL; Taylor, SC1
Greentree, SG; Pertwee, RG; Swift, PA1
Vellucci, SV; Webster, RA1
Agardh, E; Herrmann, R; Puro, DG; Yeh, HH1
Hicks, TP; Jang, EK1
Little, H; Nutt, DJ1
Simmonds, MA2
Gray, JA; Green, AR1
Caspary, DM; Faingold, CL; Gehlbach, G1
Little, HJ1
Lorens, SA; Sainati, SM1
Cowen, PJ; Green, AR; Nutt, DJ1
Bichard, AR; Little, HJ2
Starr, MS; Summerhayes, M1
Coward, DM1
Lee, EK; Ross, RJ; Walters, JR; Waszczak, BL1
Kilpatrick, IC; Starr, MS; Summerhayes, M1
Bourn, WM; Reigel, CE1
Smart, TG; Xie, X1
Delaney, AJ; Sah, P1
Hamann, M; Richter, A1
Popova, E1
Cherubini, E; Conti, F; Fattorini, G; Safiulina, VF1

Reviews

1 review(s) available for bicuculline and flurazepam

ArticleYear
Classification of inhibitory amino acid receptors in the mammalian nervous system.
    Medical biology, 1986, Volume: 64, Issue:6

    Topics: Animals; Barbiturates; Bicuculline; Flurazepam; Humans; Muscimol; Nervous System; Picrotoxin; Receptors, GABA-A; Receptors, Glycine; Receptors, Neurotransmitter; Taurine

1986

Other Studies

31 other study(ies) available for bicuculline and flurazepam

ArticleYear
Benzodiazepines: GABA and glycine receptors on single neurons in the rat medulla.
    The Journal of pharmacy and pharmacology, 1976, Volume: 28, Issue:4

    Topics: Aminobutyrates; Animals; Benzodiazepines; Bicuculline; Chlordiazepoxide; Evoked Potentials; Flurazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Medulla Oblongata; Neurons; Neurotransmitter Agents; Nitrazepam; Rats; Receptors, Drug; Strychnine

1976
Reversal of the action of amino acid antagonists by barbiturates and other hypnotic drugs.
    British journal of pharmacology, 1978, Volume: 63, Issue:1

    Topics: Aminobutyrates; Animals; Benzodiazepines; Bicuculline; Central Nervous System; Chlordiazepoxide; Dose-Response Relationship, Drug; Drug Interactions; Flurazepam; GABA Antagonists; Hypnotics and Sedatives; Male; Pentobarbital; Rats; Secobarbital; Strychnine; Synaptic Transmission

1978
Modification of GABA-mediated depolarization of the cat ganglion by pentobarbital and two benzodiazepines.
    Neuropharmacology, 1979, Volume: 18, Issue:4

    Topics: Animals; Benzodiazepines; Bicuculline; Cats; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Spinal; Pentobarbital; Picrotoxin

1979
Characterization of GABAergic seizure regulation in the midline thalamus.
    Neuropharmacology, 1990, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Bicuculline; Electroencephalography; Epilepsy; Female; Flurazepam; gamma-Aminobutyric Acid; Pentobarbital; Pentylenetetrazole; Piperidines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thalamic Nuclei

1990
Modulation of GABA-stimulated Cl- flux by a benzodiazepine agonist and an 'inverse agonist' after chronic flurazepam treatment.
    European journal of pharmacology, 1990, Feb-13, Volume: 176, Issue:3

    Topics: Animals; Benzodiazepines; Bicuculline; Brain Chemistry; Carbolines; Chlorides; Dose-Response Relationship, Drug; Flurazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains

1990
Regional GABA/benzodiazepine receptor/chloride channel coupling after acute and chronic benzodiazepine treatment.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Bicuculline; Brain; Chlorides; Diazepam; Flunitrazepam; Flurazepam; gamma-Aminobutyric Acid; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical

1989
Microiontophoresis of flurazepam on inspiratory and postinspiratory neurons in the ventrolateral medulla of cats: an intracellular study in vivo.
    Neuroscience letters, 1989, Jul-31, Volume: 102, Issue:2-3

    Topics: Animals; Bicuculline; Cats; Electrophysiology; Flurazepam; gamma-Aminobutyric Acid; Iontophoresis; Medulla Oblongata; Membrane Potentials; Microelectrodes; Neurons; Respiration; Synaptic Transmission

1989
Changes in benzodiazepine/GABA receptor complex function in benzodiazepine-tolerant mice.
    Psychopharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Anticonvulsants; Bicuculline; Body Temperature; Drug Tolerance; Flurazepam; gamma-Aminobutyric Acid; Infusions, Intravenous; Male; Mice; Motor Activity; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors

1988
Drugs which stimulate or facilitate central GABAergic transmission interact synergistically with delta-9-tetrahydrocannabinol to produce marked catalepsy in mice.
    Neuropharmacology, 1988, Volume: 27, Issue:12

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Catalepsy; Dronabinol; Drug Synergism; Flumazenil; Flupenthixol; Flurazepam; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Nipecotic Acids; Receptors, GABA-A; Strychnine; Taurine; Tiagabine

1988
GABA and benzodiazepine-induced modification of [14C]L-glutamic acid release from rat spinal cord slices.
    Brain research, 1985, Mar-25, Volume: 330, Issue:2

    Topics: Aminooxyacetic Acid; Animals; Bicuculline; Drug Interactions; Flurazepam; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Potassium; Rats; Spinal Cord

1985
gamma-Aminobutyric acid-mediated inhibition at cholinergic synapses formed by cultured retinal neurons.
    Brain research, 1985, Mar-25, Volume: 330, Issue:2

    Topics: Animals; Bicuculline; Cells, Cultured; Chick Embryo; Cholinergic Fibers; Flurazepam; gamma-Aminobutyric Acid; Neural Inhibition; Neurons; Retina; Synaptic Transmission

1985
The gamma-aminobutyric acid-mimetic action of omega-aminocaprylic acid in rat cortex.
    Neuroscience letters, 1985, Jun-24, Volume: 57, Issue:3

    Topics: Animals; Bicuculline; Caprylates; Cerebral Cortex; Drug Interactions; Flurazepam; gamma-Aminobutyric Acid; Models, Chemical; Rats; Receptors, GABA-A

1985
Benzodiazepine-receptor mediated convulsions in infant rats: effects of beta-carbolines.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:4

    Topics: Animals; Bicuculline; Carbolines; Convulsants; Flurazepam; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1986
GABAB-receptor mediated inhibition of potassium-evoked release of endogenous 5-hydroxytryptamine from mouse frontal cortex.
    British journal of pharmacology, 1987, Volume: 91, Issue:3

    Topics: Animals; Anticonvulsants; Baclofen; Bicuculline; Calcium; Cerebral Cortex; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Potassium; Receptors, GABA-A; Serotonin; Stereoisomerism

1987
Decreased effectiveness of GABA-mediated inhibition in the inferior colliculus of the genetically epilepsy-prone rat.
    Experimental neurology, 1986, Volume: 93, Issue:1

    Topics: Animals; Bicuculline; Epilepsy; Flurazepam; GABA Antagonists; gamma-Aminobutyric Acid; Inferior Colliculi; Rats; Rats, Inbred Strains

1986
The effects of benzodiazepine agonists, inverse agonists and Ro 15-1788 on the responses of the superior cervical ganglion to GABA in vitro.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepinones; Bicuculline; Carbolines; Chlordiazepoxide; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Sympathetic; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Intra-raphe benzodiazepines enhance rat locomotor activity: interactions with GABA.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Bicuculline; Brain Stem; Chlordiazepoxide; Dose-Response Relationship, Drug; Flurazepam; gamma-Aminobutyric Acid; Male; Midazolam; Motor Activity; Muscimol; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1983
A site for the potentiation of GABA-mediated responses by benzodiazepines.
    Nature, 1980, Apr-10, Volume: 284, Issue:5756

    Topics: Afferent Pathways; Animals; Bicuculline; Drug Synergism; Flurazepam; gamma-Aminobutyric Acid; Ion Channels; Medulla Oblongata; Membrane Potentials; Muscimol; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter

1980
Ethyl beta-carboline carboxylate lowers seizure threshold and antagonizes flurazepam-induced sedation in rats.
    Nature, 1981, Mar-05, Volume: 290, Issue:5801

    Topics: Animals; Bicuculline; Carbolines; Dose-Response Relationship, Drug; Flurazepam; Indoles; Rats; Receptors, Drug; Receptors, GABA-A; Seizures

1981
Drugs that increase gamma-aminobutyric acid transmission protect against the high pressure neurological syndrome.
    British journal of pharmacology, 1982, Volume: 76, Issue:3

    Topics: Anesthetics; Animals; Bicuculline; Body Temperature; Flurazepam; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Muscimol; Pressure; Seizures; Synaptic Transmission; Tremor; Valproic Acid

1982
Role of the ventromedial nucleus of the thalamus in motor behaviour--I. Effects of focal injections of drugs.
    Neuroscience, 1983, Volume: 10, Issue:4

    Topics: Amino Acids; Amino Acids, Cyclic; Aminocaproates; Animals; Bicuculline; Corpus Striatum; Cyclohexanecarboxylic Acids; Flurazepam; gamma-Aminobutyric Acid; Humans; Male; Motor Activity; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stereotyped Behavior; Substantia Nigra; Synaptic Transmission; Thalamic Nuclei; Vigabatrin

1983
Nigral actions of GABA agonists are enhanced by chronic fluphenazine and differentiated by concomitant flurazepam.
    Psychopharmacology, 1982, Volume: 76, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Female; Fluphenazine; Flurazepam; gamma-Aminobutyric Acid; Humans; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substantia Nigra

1982
Effects of benzodiazepines on single unit activity in the substantia nigra pars reticulata.
    Life sciences, 1982, Sep-06, Volume: 31, Issue:10

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Dose-Response Relationship, Drug; Electric Conductivity; Flumazenil; Flurazepam; Male; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Substantia Nigra; Theophylline

1982
The benzodiazepine antagonist, Ro 15-1788, prevents the effects of flurazepam on the high pressure neurological syndrome.
    Neuropharmacology, 1982, Volume: 21, Issue:9

    Topics: Animals; Benzodiazepinones; Bicuculline; Flumazenil; Flurazepam; Male; Mice; Nervous System Diseases; Pressure; Seizures; Tremor

1982
Interactions between dopamine and gamma-aminobutyrate in the substantia nigra: implications for the striatonigral output hypothesis.
    Neuroscience, 1983, Volume: 8, Issue:3

    Topics: Amino Acids; Amino Acids, Cyclic; Aminocaproates; Animals; Apomorphine; Bicuculline; Corpus Striatum; Cyclohexanecarboxylic Acids; Dopamine; Ethanolamines; Female; Flurazepam; gamma-Aminobutyric Acid; Locomotion; Male; Neural Pathways; Procaine; Rats; Rats, Inbred Strains; Substantia Nigra; Thalamus; Vigabatrin

1983
Effects of barbital or diazepam withdrawal on seizure thresholds to bicuculline, picrotoxin and flurazepam.
    Proceedings of the Western Pharmacology Society, 1995, Volume: 38

    Topics: Animals; Barbital; Bicuculline; Convulsants; Diazepam; Flurazepam; Male; Picrotoxin; Rats; Rats, Sprague-Dawley; Seizures; Substance Withdrawal Syndrome

1995
Properties of GABA-mediated synaptic potentials induced by zinc in adult rat hippocampal pyramidal neurones.
    The Journal of physiology, 1993, Volume: 460

    Topics: Action Potentials; Animals; Bicuculline; Culture Techniques; Flurazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Membrane Potentials; Pentobarbital; Picrotoxin; Rats; Synapses; Synaptic Transmission; Zinc

1993
GABA receptors inhibited by benzodiazepines mediate fast inhibitory transmission in the central amygdala.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Nov-15, Volume: 19, Issue:22

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Bicuculline; Evoked Potentials; Flurazepam; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Neurons; Nipecotic Acids; Nitrazepam; Oximes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Strychnine; Synaptic Transmission

1999
Effects of striatal injections of GABA(A) receptor agonists and antagonists in a genetic animal model of paroxysmal dystonia.
    European journal of pharmacology, 2002, May-17, Volume: 443, Issue:1-3

    Topics: Animals; Bicuculline; Binding Sites; Corpus Striatum; Cricetinae; Dystonia; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Mesocricetus; Microinjections; Muscimol; Pentylenetetrazole; Phenobarbital

2002
Effects of benzodiazepines on frog ERG.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2003, Volume: 134, Issue:4

    Topics: Animals; Benzodiazepines; Bicuculline; Electroretinography; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Rana ridibunda; Retina

2003
GABAergic signaling at mossy fiber synapses in neonatal rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-11, Volume: 26, Issue:2

    Topics: Action Potentials; Aminobutyrates; Animals; Animals, Newborn; Bicuculline; Cation Transport Proteins; Dentate Gyrus; Electric Stimulation; Excitatory Amino Acid Agonists; Flurazepam; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Glutamic Acid; Interneurons; Mossy Fibers, Hippocampal; Nipecotic Acids; Oximes; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Propanolamines; Pyramidal Cells; Quinoxalines; Rats; Rats, Wistar; Reaction Time; Receptors, AMPA; Receptors, GABA-A; Synaptic Transmission; Vesicular Glutamate Transport Protein 1

2006