Page last updated: 2024-08-21

bicuculline and colforsin

bicuculline has been researched along with colforsin in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19904 (25.00)18.7374
1990's1 (6.25)18.2507
2000's8 (50.00)29.6817
2010's3 (18.75)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Hampson, EC; Vaney, DI; Weiler, R1
Wojcik, WJ; Xu, J1
Baes, M; Vale, WW1
Georgieva, J1
Beltrán-Parrazal, L; Clapp, C; Martínez de la Escalera, G; Noris, G1
Bali, B; Kovács, KJ1
Billi, S; De Laurentiis, A; Fernández-Solari, J; Franchi, A; McCann, SM; Mohn, C; Rettori, V; Scorticati, C1
Gainer, H; Rusnak, M1
Chen, JF; Cunha, RA; Domenici, MR; Grò, MC; Martire, A; Pepponi, R; Popoli, P; Rebola, N; Schwarzschild, MA; Tebano, MT1
Beltran-Parrazal, L; Brennan, KC; Charles, AC; de Vellis, J; Díaz-Muñoz, M; López-Valdés, HE1
Krueger, DD; Nairn, AC1
Einstein, EB; Hon, BJ; Johnson, BN; Mateer, MJ; Melnikoff, DE; Patterson, CA; Reddi, J; Regan, KA; Schulz, S; Tallent, MK1
Bobeck, EN; Chen, Q; Ingram, SL; Morgan, MM1

Other Studies

16 other study(ies) available for bicuculline and colforsin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Dopaminergic modulation of gap junction permeability between amacrine cells in mammalian retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Bicuculline; Cadmium; Cadmium Chloride; Cell Membrane Permeability; Chlorides; Colforsin; Dopamine; Ergolines; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Intercellular Junctions; Male; Quinpirole; Rabbits; Retina; Synapses; Veratridine

1992
Gamma aminobutyric acid B receptor-mediated inhibition of adenylate cyclase in cultured cerebellar granule cells: blockade by islet-activating protein.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Autoradiography; Baclofen; Bicuculline; Cerebellum; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Pertussis Toxin; Rats; Receptors, GABA-A; Time Factors; Virulence Factors, Bordetella

1986
Growth hormone-releasing factor secretion from fetal hypothalamic cell cultures is modulated by forskolin, phorbol esters, and muscimol.
    Endocrinology, 1989, Volume: 124, Issue:1

    Topics: Animals; Bicuculline; Cells, Cultured; Chromatography, High Pressure Liquid; Colforsin; Growth Hormone-Releasing Hormone; Hypothalamus; Muscimol; Picrotoxin; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tetradecanoylphorbol Acetate; Verapamil

1989
Effects of the diterpene sclareol glycol on convulsive seizures.
    Methods and findings in experimental and clinical pharmacology, 1989, Volume: 11, Issue:5

    Topics: Animals; Bicuculline; Colforsin; Convulsants; Diterpenes; Drug Synergism; Male; Mice; Pentylenetetrazole; Picrotoxin; Seizures

1989
GABA inhibition of immortalized gonadotropin-releasing hormone neuronal excitability involves GABA(A) receptors negatively coupled to cyclic adenosine monophosphate formation.
    Endocrine, 2001, Volume: 14, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Baclofen; Bicuculline; Calcium; Calcium Channels; Cell Line, Transformed; Cell Membrane; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Kinetics; Muscimol; Neurons; Potassium; Receptors, GABA-A

2001
GABAergic control of neuropeptide gene expression in parvocellular neurons of the hypothalamic paraventricular nucleus.
    The European journal of neuroscience, 2003, Volume: 18, Issue:6

    Topics: Animals; Animals, Newborn; Arginine Vasopressin; Autoradiography; Bicuculline; Cell Count; Colforsin; Corticotropin-Releasing Hormone; Female; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Glutamate Decarboxylase; Immunohistochemistry; In Situ Hybridization; Isoenzymes; Male; Microinjections; Microscopy, Immunoelectron; Neurons; Neuropeptides; Organ Culture Techniques; Paraventricular Hypothalamic Nucleus; Potassium; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; RNA, Messenger

2003
Alcohol inhibits luteinizing hormone-releasing hormone release by activating the endocannabinoid system.
    Proceedings of the National Academy of Sciences of the United States of America, 2004, Mar-02, Volume: 101, Issue:9

    Topics: Animals; Arachidonic Acids; Bicuculline; Cannabinoid Receptor Modulators; Colforsin; Cyclic AMP; Endocannabinoids; Ethanol; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; Kinetics; Male; N-Methylaspartate; Naltrexone; Polyunsaturated Alkamides; Radioimmunoassay; Rats; Rats, Wistar

2004
Differential effects of forskolin on tyrosine hydroxylase gene transcription in identified brainstem catecholaminergic neuronal subtypes in organotypic culture.
    The European journal of neuroscience, 2005, Volume: 21, Issue:4

    Topics: Animals; Animals, Newborn; Bicuculline; Brain Stem; Catecholamines; Cell Count; Colforsin; Drug Interactions; GABA Antagonists; Gene Expression Regulation, Developmental; Immunohistochemistry; In Situ Hybridization; In Vitro Techniques; Isoquinolines; Membrane Glycoproteins; Membrane Transport Proteins; Neurons; Norepinephrine Plasma Membrane Transport Proteins; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Sulfonamides; Symporters; Tetrodotoxin; Tyrosine 3-Monooxygenase; Vesicular Biogenic Amine Transport Proteins; Vesicular Monoamine Transport Proteins

2005
Adenosine A2A receptors and metabotropic glutamate 5 receptors are co-localized and functionally interact in the hippocampus: a possible key mechanism in the modulation of N-methyl-D-aspartate effects.
    Journal of neurochemistry, 2005, Volume: 95, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Animals; Bicuculline; Blotting, Western; Colforsin; Disks Large Homolog 4 Protein; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Female; Fluorescent Antibody Technique; GABA Antagonists; Glycine; Hippocampus; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Phenethylamines; Phenylacetates; Pregnancy; Presynaptic Terminals; Pyridines; Qa-SNARE Proteins; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Adenosine A2; Receptors, Metabotropic Glutamate; Synaptophysin; Vesicular Glutamate Transport Protein 1

2005
Mitochondrial transport in processes of cortical neurons is independent of intracellular calcium.
    American journal of physiology. Cell physiology, 2006, Volume: 291, Issue:6

    Topics: Aldehydes; Animals; Bicuculline; Biological Transport; Calcium; Calcium Signaling; Cells, Cultured; Cerebral Cortex; Colforsin; Female; GABA Antagonists; Glutamic Acid; Image Processing, Computer-Assisted; Mitochondria; Neurons; Pregnancy; Rats; Rats, Sprague-Dawley

2006
Expression of PKC substrate proteins, GAP-43 and neurogranin, is downregulated by cAMP signaling and alterations in synaptic activity.
    The European journal of neuroscience, 2007, Volume: 26, Issue:11

    Topics: Animals; Bicuculline; Cerebral Cortex; Colforsin; Cyclic AMP; Down-Regulation; Drug Interactions; Embryo, Mammalian; Enzyme Activators; Enzyme Inhibitors; GABA Antagonists; GAP-43 Protein; Neurogranin; Neurons; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2007
Somatostatin signaling in neuronal cilia is critical for object recognition memory.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-24, Volume: 30, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Adenylyl Cyclases; Amides; Animals; Behavior, Animal; Bicuculline; Biophysics; CA1 Region, Hippocampal; Cilia; Colforsin; Cyclic AMP; Discrimination, Psychological; Electric Stimulation; Female; GABA Antagonists; In Vitro Techniques; Isoquinolines; Locomotion; Long-Term Potentiation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Neuropsychological Tests; Nitrobenzenes; Phosphodiesterase Inhibitors; Receptors, Somatostatin; Recognition, Psychology; Signal Transduction; Somatostatin

2010
Contribution of adenylyl cyclase modulation of pre- and postsynaptic GABA neurotransmission to morphine antinociception and tolerance.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:9

    Topics: Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Analgesics, Opioid; Animals; Bicuculline; Colforsin; Drug Tolerance; Enzyme Activators; Enzyme Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Morphine; Nociception; Presynaptic Terminals; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptic Transmission

2014