Page last updated: 2024-08-21

bicuculline and 8-hydroxy-2-(di-n-propylamino)tetralin

bicuculline has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.85)18.7374
1990's9 (34.62)18.2507
2000's11 (42.31)29.6817
2010's5 (19.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bobker, DH; Williams, JT1
Kelder, D; Ross, SB1
Alkadhi, KA; Salgado, D1
Gale, K; Pasini, A; Tortorella, A1
Alkadhi, KA; Salgado-Commissariat, D1
Colwell, DD; Kavaliers, M; Perrot-Sinal, TS1
Draguhn, A; Empson, RM; Gloveli, T; Heinemann, U; Schmitz, D1
Bischoff, AM; Pierrefiche, O; Richter, DW; Schwarzacher, SW1
Fernández-Guasti, A; López-Rubalcava, C1
Rainnie, DG1
Abe, K; Edagawa, Y; Saito, H1
Akaike, N; Kishimoto, K; Koyama, S1
Crochet, S; Sakai, K1
Akasu, T; Hasuo, H1
Mogil, JS; Nemmani, KV1
Guptarak, J; Selvamani, A; Uphouse, L1
Bannatyne, BA; Dougherty, KJ; Jankowska, E; Krutki, P; Maxwell, DJ1
Forsberg, T; Gabrielsson, J; Martinsson, S; Pozarek, S; Ross, SB; Visser, SA1
Dampney, RA; Horiuchi, J; Wakabayashi, S1
Cheng, HY; Hsieh, CC; Hsieh, MT; Lin, YT; Lu, MC; Peng, WH; Wu, CR1
Belzung, C; Chapouthier, G; Clément, Y; Le Guisquet, AM; Venault, P1
Congleton, MR; Duncan, MJ1
Ferreira, MD; Menescal-de-Oliveira, L1
Kallingal, GJ; Mintz, EM1
Biagioni, AF; Coimbra, NC; Corrado, AP; da Silva, JA; de Oliveira, R; de Oliveira, RC; dos Anjos-Garcia, T; Roncon, CM; Zangrossi, H1
Geijo-Barrientos, E; Rovira, V1

Other Studies

26 other study(ies) available for bicuculline and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
Serotonin agonists inhibit synaptic potentials in the rat locus ceruleus in vitro via 5-hydroxytryptamine1A and 5-hydroxytryptamine1B receptors.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Cocaine; Electric Stimulation; In Vitro Techniques; Kinetics; Locus Coeruleus; Male; Neurons; Picrotoxin; Piperazines; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Synapses; Tetrahydronaphthalenes

1989
Counteraction of the rapid tolerance to 8-OH-DPAT-induced corticosterone secretion in rats by activation of the GABAA receptor-chloride channel complex.
    British journal of pharmacology, 1993, Volume: 109, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzodiazepines; Bicuculline; Chloride Channels; Chlormethiazole; Corticosterone; Drug Tolerance; Ion Channels; Male; Membrane Proteins; Muscimol; Pentobarbital; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Inhibition of epileptiform activity by serotonin in rat CA1 neurons.
    Brain research, 1995, Jan-16, Volume: 669, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Electric Stimulation; Epilepsy; Evoked Potentials; Hippocampus; Male; Membrane Potentials; Neurons; Rats; Rats, Sprague-Dawley; Serotonin

1995
The anticonvulsant action of fluoxetine in substantia nigra is dependent upon endogenous serotonin.
    Brain research, 1996, Jun-10, Volume: 724, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anticonvulsants; Bicuculline; Convulsants; Fenclonine; Fluoxetine; gamma-Aminobutyric Acid; Male; Microinjections; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Seizures; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Substantia Nigra

1996
Effects of serotonin on induced epileptiform activity in CA1 pyramidal neurons of genetically epilepsy prone rats.
    Brain research, 1996, Dec-16, Volume: 743, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Convulsants; Drug Evaluation, Preclinical; Electric Stimulation; Epilepsy; Evoked Potentials; Genetic Predisposition to Disease; In Vitro Techniques; Male; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists

1996
Opioid and non-opioid NMDA-mediated predator-induced analgesia in mice and the effects of parasitic infection.
    Brain research, 1997, Aug-22, Volume: 766, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amino Acids; Analgesia; Animals; Behavior, Animal; Bicuculline; Butyrates; Butyric Acid; Excitatory Amino Acid Antagonists; GABA Antagonists; Histamine Antagonists; Host-Parasite Interactions; Male; Mice; Mice, Inbred Strains; Naloxone; Narcotic Antagonists; Nematospiroides dubius; Nociceptors; Odorants; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Serotonin Receptor Agonists; Stress, Physiological; Strongylida Infections; Time Factors

1997
Serotonin reduces synaptic excitation in the superficial medial entorhinal cortex of the rat via a presynaptic mechanism.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Entorhinal Cortex; Excitatory Postsynaptic Potentials; Female; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Male; Patch-Clamp Techniques; Piperazines; Potassium Channels; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Synapses; Synaptic Transmission; Tetrodotoxin

1998
Blockade of synaptic inhibition within the pre-Bötzinger complex in the cat suppresses respiratory rhythm generation in vivo.
    The Journal of physiology, 1998, May-15, Volume: 509 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Cats; Female; GABA Antagonists; GABA-A Receptor Antagonists; Glycine Agents; Male; Medulla Oblongata; Microinjections; Phrenic Nerve; Receptors, Glycine; Respiratory Mechanics; Serotonin Receptor Agonists; Strychnine; Synapses; Tetrodotoxin

1998
Modification of the anxiolytic action of 5-HT1A compounds by GABA-benzodiazepine agents in rats.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:1

    Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anxiety; Bicuculline; Buspirone; Diazepam; Drug Interactions; Flumazenil; GABA Agonists; Male; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1

1998
Serotonergic modulation of neurotransmission in the rat basolateral amygdala.
    Journal of neurophysiology, 1999, Volume: 82, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amygdala; Animals; Bicuculline; Evoked Potentials; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; In Vitro Techniques; Interneurons; Male; Neurons; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Synaptic Transmission; Tetrodotoxin

1999
The serotonin 5-HT2 receptor-phospholipase C system inhibits the induction of long-term potentiation in the rat visual cortex.
    The European journal of neuroscience, 2000, Volume: 12, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Bicuculline; Electrophysiology; Estrenes; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Long-Term Potentiation; Male; Phosphodiesterase Inhibitors; Piperazines; Pyrrolidinones; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Type C Phospholipases; Visual Cortex

2000
Presynaptic modulation of synaptic gamma-aminobutyric acid transmission by tandospirone in rat basolateral amygdala.
    European journal of pharmacology, 2000, Nov-03, Volume: 407, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Amygdala; Animals; Bicuculline; GABA Antagonists; gamma-Aminobutyric Acid; Isoindoles; Neurons; Piperazines; Presynaptic Terminals; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission

2000
Role of dorsal raphe neurons in paradoxical sleep generation in the cat: no evidence for a serotonergic mechanism.
    The European journal of neuroscience, 2001, Volume: 13, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Cats; Excitatory Amino Acid Agonists; Female; GABA Agonists; GABA Antagonists; Kainic Acid; Male; Microdialysis; Muscimol; Neurons; Piperazines; Pyridines; Raphe Nuclei; Serotonin; Serotonin Antagonists; Sleep Stages; Sleep, REM; Wakefulness

2001
5-Hydroxytryptamine facilitates spatiotemporal propagation of optical signals in the hippocampal-septal pathway.
    Neuroscience research, 2001, Volume: 40, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Bicuculline; Electric Stimulation; Electronic Data Processing; Excitatory Amino Acid Antagonists; Fornix, Brain; GABA Antagonists; Hippocampus; Male; Neural Conduction; Neurons; Phosphinic Acids; Piperazines; Propanolamines; Rats; Rats, Wistar; Receptors, Serotonin; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Tetrodotoxin

2001
Serotonin-GABA interactions in the modulation of mu- and kappa-opioid analgesia.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesia; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Fenclonine; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Morphine; Pain Threshold; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Serotonin Agents; Serotonin Antagonists

2003
GABAA-5-HT1A receptor interaction in the mediobasal hypothalamus.
    Brain research, 2004, Nov-19, Volume: 1027, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Bicuculline; Drug Interactions; Estradiol; Female; GABA Agonists; GABA Antagonists; Hypothalamus, Middle; Muscimol; Ovariectomy; Posture; Progesterone; Rats; Rats, Inbred F344; Receptor, Serotonin, 5-HT1A; Receptors, GABA-A; Serotonin Agents; Sexual Behavior, Animal; Time Factors

2004
Membrane receptors involved in modulation of responses of spinal dorsal horn interneurons evoked by feline group II muscle afferents.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jan-19, Volume: 25, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Cats; Electric Stimulation; Evoked Potentials; Immunohistochemistry; Interneurons; Iontophoresis; Muscles; Oxazines; Piperazines; Posterior Horn Cells; Pyridines; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin

2005
Rapid and long-lasting tolerance to clomethiazole-induced hypothermia in the rat.
    European journal of pharmacology, 2005, Apr-11, Volume: 512, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Body Temperature; Chlormethiazole; Dizocilpine Maleate; Drug Tolerance; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; GABA Modulators; Hypothermia; Injections, Subcutaneous; Male; Muscimol; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Time Factors

2005
Activation of 5-hydroxytryptamine 1A receptors suppresses the cardiovascular response evoked from the dorsomedial hypothalamic nucleus.
    Hypertension (Dallas, Tex. : 1979), 2005, Volume: 46, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Baroreflex; Bicuculline; Blood Pressure; Cardiovascular System; Chemoreceptor Cells; Dorsomedial Hypothalamic Nucleus; GABA Antagonists; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Kidney; Male; Microinjections; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Psychological; Sympathetic Nervous System

2005
Ameliorating effect of emodin, a constitute of Polygonatum multiflorum, on cycloheximide-induced impairment of memory consolidation in rats.
    Journal of ethnopharmacology, 2007, Jul-25, Volume: 112, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Animals; Baclofen; Bicuculline; Cycloheximide; Dose-Response Relationship, Drug; Emodin; GABA Agonists; GABA Antagonists; Injections, Subcutaneous; Learning; Male; Memory; Memory Disorders; Plant Roots; Polygonatum; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Ritanserin; Scopolamine; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2007
Pharmacological alterations of anxious behaviour in mice depending on both strain and the behavioural situation.
    PloS one, 2009, Nov-11, Volume: 4, Issue:11

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Behavior, Animal; Benzodiazepines; Bicuculline; Chlordiazepoxide; Female; Indoles; Light; Male; Maze Learning; Mice; Mice, Inbred C57BL; Phosphorylation

2009
Neural mechanisms mediating circadian phase resetting by activation of 5-HT(7) receptors in the dorsal raphe: roles of GABAergic and glutamatergic neurotransmission.
    Brain research, 2010, Dec-17, Volume: 1366

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Circadian Rhythm; Cricetinae; Dizocilpine Maleate; Drug Administration Schedule; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Mesocricetus; Microinjections; Muscimol; N-Methylaspartate; Raphe Nuclei; Receptors, Serotonin; Serotonin Receptor Agonists; Synaptic Transmission

2010
Opioidergic, GABAergic and serotonergic neurotransmission in the dorsal raphe nucleus modulates tonic immobility in guinea pigs.
    Physiology & behavior, 2012, May-15, Volume: 106, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics, Opioid; Animals; Bicuculline; Drug Interactions; GABAergic Neurons; Guinea Pigs; Immobility Response, Tonic; Male; Microinjections; Morphine; Muscimol; Naloxone; Opioid Peptides; Raphe Nuclei; Serotonergic Neurons; Serotonin; Serotonin 5-HT2 Receptor Agonists; Synaptic Transmission

2012
Site-specific effects of gastrin-releasing peptide in the suprachiasmatic nucleus.
    The European journal of neuroscience, 2014, Volume: 39, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bicuculline; Circadian Rhythm; Cricetinae; Extracellular Signal-Regulated MAP Kinases; GABA-A Receptor Antagonists; Gastrin-Releasing Peptide; Gastrointestinal Agents; Male; Mesocricetus; Organ Specificity; Paraventricular Hypothalamic Nucleus; Proto-Oncogene Proteins c-fos; Serotonin Receptor Agonists; Suprachiasmatic Nucleus; Supraoptic Nucleus

2014
5-Hydroxytryptamine 1A receptors in the dorsomedial hypothalamus connected to dorsal raphe nucleus inputs modulate defensive behaviours and mediate innate fear-induced antinociception.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2016, Volume: 26, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Bicuculline; Biotin; Dextrans; Dorsal Raphe Nucleus; Dorsomedial Hypothalamic Nucleus; Dose-Response Relationship, Drug; Escape Reaction; Fear; GABA-A Receptor Antagonists; Male; Microinjections; Neural Pathways; Pain Measurement; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists

2016
Intra- and Interhemispheric Propagation of Electrophysiological Synchronous Activity and Its Modulation by Serotonin in the Cingulate Cortex of Juvenile Mice.
    PloS one, 2016, Volume: 11, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Bicuculline; Electric Stimulation; Electrophysiological Phenomena; GABA-A Receptor Antagonists; Gyrus Cinguli; Male; Mice, Inbred C57BL; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Receptor Agonists; Time Factors

2016