betaxolol and practolol

betaxolol has been researched along with practolol in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19908 (50.00)18.7374
1990's3 (18.75)18.2507
2000's2 (12.50)29.6817
2010's3 (18.75)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ball, JB; Iakovidis, D; Jackman, G; Louis, WJ; Nero, TL; Tung, L1
Binet, JL; Cavero, IG; Lefèvre-Borg, F; Manoury, PM; Rousseau, J1
Carrupt, PA; el Tayar, N; Testa, B; Van de Waterbeemd, H1
Aué, GH; Bultsma, T; IJzerman, AP; Linschoten, MR; Timmerman, H1
Baldwin, JJ; Denny, GH; Freedman, MB; Gross, DM; Hirschmann, R; Ponticello, GS; Sweet, CS1
Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL1
Abraham, MH; Acree, WE; Ibrahim, A1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brunton, LL; Buxton, IL1
Gomeni, R; Kilborn, JR; Morselli, PL; Saunders, J; Sönksen, PH1
Curtis-Prior, PB; Tan, S1
Engel, G1
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M1

Reviews

1 review(s) available for betaxolol and practolol

ArticleYear
Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:11

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Models, Molecular; Receptors, Adrenergic, beta; Structure-Activity Relationship

1988

Other Studies

15 other study(ies) available for betaxolol and practolol

ArticleYear
Computer-aided mapping of the beta-adrenoceptor. 1. Explanation for effect of para substitution on blocking activity at the beta-1-adrenoceptor.
    Journal of medicinal chemistry, 1992, Dec-11, Volume: 35, Issue:25

    Topics: Adrenergic beta-Antagonists; Computer Simulation; Propanolamines; Stereoisomerism; Structure-Activity Relationship

1992
Synthesis of a series of compounds related to betaxolol, a new beta 1-adrenoceptor antagonist with a pharmacological and pharmacokinetic profile optimized for the treatment of chronic cardiovascular diseases.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:6

    Topics: Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Antihypertensive Agents; Betaxolol; Biotransformation; Cardiovascular Diseases; Chronic Disease; Female; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Propanolamines; Rana esculenta; Rats; Structure-Activity Relationship

1987
Quantitative evaluation of the beta 2-adrenoceptor affinity of phenoxypropanolamines and phenylethanolamines.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Animals; Cattle; Chemical Phenomena; Chemistry; Dihydroalprenolol; Ethanolamines; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Muscles; Propanolamines; Receptors, Adrenergic, beta; Structure-Activity Relationship

1985
Beta 1-selective adrenoceptor antagonists: examples of the 2-[4-[3-(substituted-amino)-2-hydroxypropoxy]phenyl]imidazole class.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Female; Guinea Pigs; Heart; Imidazoles; Indicators and Reagents; Isoproterenol; Magnetic Resonance Spectroscopy; Receptors, Adrenergic; Receptors, Adrenergic, beta; Structure-Activity Relationship

1983
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea

1999
Air to lung partition coefficients for volatile organic compounds and blood to lung partition coefficients for volatile organic compounds and drugs.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Air; Animals; Humans; Lung; Organic Chemicals; Probability; Rats; Tissue Distribution; Volatilization

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Direct analysis of beta-adrenergic receptor subtypes on intact adult ventricular myocytes of the rat.
    Circulation research, 1985, Volume: 56, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Betaxolol; Binding Sites; Cells, Cultured; Ethanolamines; Heart; Iodine Radioisotopes; Iodocyanopindolol; Male; Myocardium; Pindolol; Practolol; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1985
A comparison between propranolol, practolol and betaxolol (SL75212) on the circulatory and metabolic responses to insulin-induced hypoglycaemia.
    European journal of clinical pharmacology, 1981, Volume: 21, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Betaxolol; Blood Glucose; Blood Pressure; Fatty Acids, Nonesterified; Glycerol; Growth Hormone; Heart Rate; Humans; Hypoglycemia; Insulin; Male; Practolol; Propanolamines; Propranolol

1981
Characterization of the beta-adrenoceptor of the adipose cell of the rat.
    International journal of obesity, 1983, Volume: 7, Issue:5

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Albuterol; Animals; Betaxolol; Dose-Response Relationship, Drug; Isoproterenol; Lipolysis; Norepinephrine; Practolol; Prenalterol; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta

1983
Subclasses of beta-adrenoceptors--a quantitative estimation of beta 1- and beta 2- adrenoceptors in guinea pig and human lung.
    Postgraduate medical journal, 1981, Volume: 57 Suppl 1

    Topics: Aged; Animals; Atenolol; Betaxolol; Cell Membrane; Guinea Pigs; Humans; Iodocyanopindolol; Lung; Metoprolol; Middle Aged; Models, Biological; Pindolol; Practolol; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta

1981
Constitutively active mutants of the beta1-adrenergic receptor.
    FEBS letters, 1999, Sep-03, Volume: 457, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol

1999