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beta-carboline-3-carboxylic acid ethyl ester and ro 15-4513

beta-carboline-3-carboxylic acid ethyl ester has been researched along with ro 15-4513 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19903 (30.00)18.7374
1990's2 (20.00)18.2507
2000's3 (30.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W1
Crawley, JN; Paul, SM; Suzdak, PD1
Miller, DW; Tessel, RE; Yourick, DL1
Eichinger, A; Möhler, H; Richards, JG; Sieghart, W1
Estupinan, LE; France, CP; Gerak, LR1
France, CP; Gerak, LR1
France, CP; Gerak, LR; Lelas, S1
Abe, K; Hosoi, R; Inoue, O; Momosaki, S1
Meera, P; Olsen, RW; Otis, TS; Wallner, M1

Other Studies

10 other study(ies) available for beta-carboline-3-carboxylic acid ethyl ester and ro 15-4513

ArticleYear
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Effects of Ro15-4513 and other benzodiazepine receptor inverse agonists on alcohol-induced intoxication in the rat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: Alcoholic Intoxication; Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Ion Channels; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Antagonism of methoxyflurane-induced anesthesia in rats by benzodiazepine inverse agonists.
    European journal of pharmacology, 1989, Nov-28, Volume: 173, Issue:1

    Topics: Anesthesia; Animals; Azides; Benzodiazepines; Carbolines; Electric Stimulation; Ketamine; Male; Methoxyflurane; Pain; Pain Measurement; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reflex; Respiration

1989
Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.
    Journal of neurochemistry, 1987, Volume: 48, Issue:1

    Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Molecular Weight; Photochemistry; Pyridazines; Rats; Receptors, GABA-A

1987
Ventilatory effects of negative GABA(A) modulators in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 61, Issue:4

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Female; GABA Modulators; Macaca mulatta; Male; Receptors, GABA-A; Respiration, Artificial

1998
Discriminative stimulus effects of flumazenil in untreated and in diazepam-treated rhesus monkeys.
    Psychopharmacology, 1999, Volume: 146, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Receptors, GABA-A

1999
Antagonism of the discriminative stimulus effects of positive gamma-aminobutyric acid(A) modulators in rhesus monkeys discriminating midazolam.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Drug Antagonism; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Midazolam; Receptors, GABA-A

2000
Remarkable selectivity of the in vivo binding of [3H]Ro15-4513 to α5 subtype of benzodiazepine receptor in the living mouse brain.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:12

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Male; Mice; Protein Subunits; Receptors, GABA-A; Tritium

2010
Alcohol- and alcohol antagonist-sensitive human GABAA receptors: tracking δ subunit incorporation into functional receptors.
    Molecular pharmacology, 2010, Volume: 78, Issue:5

    Topics: Allosteric Regulation; Animals; Azides; Benzodiazepines; Carbolines; Cations, Divalent; Cell Line; Diazepam; Ethanol; Humans; Mutation; Patch-Clamp Techniques; Protein Subunits; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Zinc

2010