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beta-carboline-3-carboxylic acid ethyl ester and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

beta-carboline-3-carboxylic acid ethyl ester has been researched along with methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19909 (75.00)18.7374
1990's2 (16.67)18.2507
2000's1 (8.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Adler-Graschinsky, E; Elgoyhen, B; Lorenzo, PS; Tellez-Iñón, MT1
Arbilla, S; Langer, SZ; Lista, A1
Sieghart, W1
Morrow, AL; Paul, SM1
Braestrup, C; Honoré, T; Jensen, LH; Petersen, EN1
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN3
Biggio, G; Concas, A; Corda, MG; Crisponi, C; Gessa, GL; Nurchi, V; Salis, M; Serra, M1
Barrett, JE; Martin, JV; Mendelson, WB; Paul, SM; Schweri, MM; Skolnick, P1

Reviews

3 review(s) available for beta-carboline-3-carboxylic acid ethyl ester and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Differential pharmacological effects of benzodiazepine receptor inverse agonists.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Carbolines; Convulsants; Electroshock; Humans; Mice; Pentylenetetrazole; Rats; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
Benzodiazepine receptor ligands with positive and negative efficacy.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Acoustic Stimulation; Animals; Carbolines; Chlorides; gamma-Aminobutyric Acid; Humans; Ligands; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
Benzodiazepine receptor ligands with negative efficacy: chloride channel coupling.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Barbiturates; Brain; Carbolines; Chlorides; Flunitrazepam; Humans; Ion Channels; Ligands; Membranes; Receptors, Cell Surface; Receptors, GABA-A

1983

Other Studies

9 other study(ies) available for beta-carboline-3-carboxylic acid ethyl ester and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
    Journal of medicinal chemistry, 1998, Jul-02, Volume: 41, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship

1998
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Relaxant effects of beta-carbolines on rat aortic rings.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:2

    Topics: Animals; Aorta; Benzodiazepines; Carbolines; Convulsants; Female; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Vasoconstrictor Agents

1992
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1988
Benzodiazepine receptors: multiple receptors or multiple conformations?
    Journal of neural transmission, 1985, Volume: 63, Issue:3-4

    Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A

1985
Benzodiazepine enhancement of gamma-aminobutyric acid-mediated chloride ion flux in rat brain synaptoneurosomes.
    Journal of neurochemistry, 1988, Volume: 50, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chlorides; Clonazepam; Diazepam; Drug Synergism; Flurazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Inbred Strains; Synaptosomes

1988
Ligands for benzodiazepine receptors with positive and negative efficacy.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A

1984
Stress and beta-carbolines decrease the density of low affinity GABA binding sites; an effect reversed by diazepam.
    Brain research, 1984, Jul-02, Volume: 305, Issue:1

    Topics: Animals; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Handling, Psychological; Indoles; Male; Rats; Rats, Inbred Strains; Stress, Physiological

1984
Pharmacokinetic and pharmacodynamic factors contributing to the convulsant action of beta-carboline-3-carboxylic acid esters.
    Life sciences, 1983, Oct-10, Volume: 33, Issue:15

    Topics: Animals; Brain; Carbolines; Convulsants; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Indoles; Kinetics; Male; Rats; Rats, Inbred Strains; Saimiri

1983