beta-carboline-3-carboxylic acid ethyl ester has been researched along with gamma-aminobutyric acid in 38 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 34 (89.47) | 18.7374 |
1990's | 3 (7.89) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (2.63) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
Blakeman, DP; Im, WB | 1 |
Alho, H; Costa, E; Ferrero, P; Guidotti, A; Santi, MR; Vicini, S | 1 |
Akaike, N; Fukuda, T; Oyama, Y; Yakushiji, T | 1 |
Arbilla, S; Langer, SZ; Lista, A | 1 |
Gobbi, M; Mennini, T; Perin, L; Salmona, M | 1 |
Clow, A; Glover, V; Sandler, M | 1 |
Moura, D; Soares-da-Silva, P | 1 |
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ | 1 |
Cohen, RM; Havoundjian, H; Paul, SM; Skolnick, P | 1 |
Hammond, JR; Martin, IL | 1 |
Chang, LR; Lee, HK; Tao, PL | 1 |
Ciuffi, M; Franchi-Micheli, S; Luzzi, S; Rosi, E; Spagnesi, S; Zilletti, L | 1 |
Morrow, AL; Paul, SM | 1 |
Macdonald, RL; Skerritt, JH | 1 |
Little, HJ | 1 |
Moncada, VY; Paul, SM; Schweri, MM; Skolnick, P; Williams, EF | 1 |
Paul, SM; Skolnick, P | 1 |
Cardinali, DP; Lowenstein, PR | 1 |
Haefely, W | 2 |
Polc, P; Ropert, N; Wright, DM | 1 |
Goodwin, FK; Marangos, PJ; Patel, J | 1 |
Marangos, PJ; Patel, J | 1 |
Cowen, PJ; Little, HJ; Nutt, DJ | 1 |
Hirsch, JD; Kochman, RL | 1 |
Horton, RW; Prestwich, SA; Stapleton, SR | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN | 1 |
Corda, MG; Costa, E; Guidotti, A | 1 |
Brown, CL; Martin, IL | 1 |
Biggio, G; Concas, A; Crisponi, G; Nurchi, V; Salis, M; Serra, M | 1 |
Saneyoshi, M; Sung, SC | 1 |
Biggio, G; Concas, A; Corda, MG; Crisponi, C; Gessa, GL; Nurchi, V; Salis, M; Serra, M | 1 |
Barrett, JE; Martin, JV; Mendelson, WB; Paul, SM; Schweri, MM; Skolnick, P | 1 |
Biggio, G; Concas, A; Corda, MG; Salis, M; Serra, M | 1 |
Braestrup, C; Johnston, GA; Skerritt, JH | 1 |
DaSilva, AM; Gatti, PJ; Gillis, RA; Homby, PJ; Mandal, AK; Norman, WP | 1 |
Hu, HZ; Li, ZW; Shao, M | 1 |
5 review(s) available for beta-carboline-3-carboxylic acid ethyl ester and gamma-aminobutyric acid
Article | Year |
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[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid | 1985 |
The mechanism(s) of action of the benzodiazepines.
Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Caffeine; Carbolines; Cats; Cattle; Diazepam; gamma-Aminobutyric Acid; Humans; Molecular Weight; Muscle Relaxation; Neurotransmitter Agents; Niacinamide; Purines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Sleep Wake Disorders | 1981 |
Antagonists of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding, Competitive; Carbolines; Flumazenil; gamma-Aminobutyric Acid; Humans; Models, Chemical; Molecular Conformation; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptic Transmission | 1983 |
Benzodiazepine receptor ligands with positive and negative efficacy.
Topics: Acoustic Stimulation; Animals; Carbolines; Chlorides; gamma-Aminobutyric Acid; Humans; Ligands; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1983 |
On a brain polypeptide functioning as a putative effector for the recognition sites of benzodiazepine and beta-carboline derivatives.
Topics: Animals; Benzodiazepinones; Brain Chemistry; Carbolines; Carrier Proteins; Chlorides; Flumazenil; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; Ionophores; Ligands; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Organic Anion Transporters; Peptides; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
33 other study(ies) available for beta-carboline-3-carboxylic acid ethyl ester and gamma-aminobutyric acid
Article | Year |
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Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes | 1991 |
Gamma-aminobutyric acid and chloride channels: regulation by neuropeptides.
Topics: Animals; Carbolines; Cells, Cultured; Cerebellum; Chlorides; gamma-Aminobutyric Acid; Hippocampus; Humans; Ion Channels; Muscimol; Nerve Tissue Proteins; Receptors, GABA-A | 1985 |
Effects of benzodiazepines and non-benzodiazepine compounds on the GABA-induced response in frog isolated sensory neurones.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Carbolines; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Neurons, Afferent; Rana catesbeiana | 1989 |
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1988 |
Rapid internalization of benzodiazepine receptors in the rat cortex induced by handling.
Topics: Animals; Bicuculline; Carbolines; Cerebral Cortex; Corticosterone; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Ligands; Male; Rats; Receptors, GABA-A; Stress, Physiological; Synaptic Membranes; Viscosity | 1988 |
Triazolam, an anomalous benzodiazepine receptor ligand: in vitro characterization of alprazolam and triazolam binding.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Triazolam | 1985 |
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A | 1985 |
Differential sensitivity of "central" and "peripheral" type benzodiazepine receptors to phospholipase A2.
Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kidney; Male; Myocardium; Pentobarbital; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1986 |
Solubilization of the benzodiazepine/gamma-aminobutyric acid receptor complex: comparison of the detergents octylglucopyranoside and 3-[(3-cholamidopropyl)-dimethylammonio]1-propanesulfonate (CHAPS).
Topics: Animals; Carbolines; Cerebellum; Chlorides; Cholic Acids; Drug Stability; Flunitrazepam; gamma-Aminobutyric Acid; Glucosides; Glycosides; Male; Phospholipids; Pyrazoles; Rats; Receptors, GABA-A; Solubility; Synaptic Membranes | 1986 |
Heterogeneity of [3H]ethyl beta-carboline-3-carboxylate binding sites and [3H]gamma-aminobutyric acid binding sites.
Topics: Animals; Binding, Competitive; Carbolines; Cattle; Cerebral Cortex; Detergents; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Molecular Weight; Muscimol; Photolysis; Radioligand Assay; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptosomes | 1986 |
Diazepam potentiates GABA-contraction in guinea-pig ileum.
Topics: Animals; Baclofen; Benzodiazepinones; Carbolines; Diazepam; Drug Synergism; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth | 1986 |
Benzodiazepine enhancement of gamma-aminobutyric acid-mediated chloride ion flux in rat brain synaptoneurosomes.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chlorides; Clonazepam; Diazepam; Drug Synergism; Flurazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Inbred Strains; Synaptosomes | 1988 |
Benzodiazepine receptor ligand actions on GABA responses. Beta-carbolines, purines.
Topics: Animals; Carbolines; Cells, Cultured; Diazepam; Drug Interactions; gamma-Aminobutyric Acid; Indoles; Ligands; Mice; Neurons; Purines; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord | 1984 |
The effects of benzodiazepine agonists, inverse agonists and Ro 15-1788 on the responses of the superior cervical ganglion to GABA in vitro.
Topics: Animals; Barbiturates; Benzodiazepinones; Bicuculline; Carbolines; Chlordiazepoxide; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Sympathetic; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
An in vitro binding assay which differentiates benzodiazepine 'agonists' and 'antagonists'.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding, Competitive; Carbolines; Flumazenil; gamma-Aminobutyric Acid; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A | 1982 |
Characterization of flunitrazepam and beta-carboline high affinity binding in bovine pineal gland.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Carbolines; Cattle; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Kinetics; Pentobarbital; Pineal Gland; Rats; Species Specificity | 1983 |
Antagonists of benzodiazepines: functional aspects.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Chlorides; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channels; Narcotic Antagonists; Parasympathomimetics; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Substance-Related Disorders; Xanthines | 1983 |
Ethyl beta-carboline-3-carboxylate antagonizes the action of GABA and benzodiazepines in the hippocampus.
Topics: Animals; Benzodiazepines; Carbolines; Diazepam; Electric Stimulation; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Indoles; Male; Midazolam; Neural Inhibition; Neurons; Rats; Receptors, Drug; Receptors, GABA-A | 1981 |
[3H] Ethyl beta-carboline-3-carboxylate binding to the benzodiazepine receptor is not affected by GABA.
Topics: Animals; Brain; Carbolines; Cell Membrane; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Rats; Receptors, Drug; Receptors, GABA-A | 1981 |
Properties of [3H] beta-carboline-3-carboxylate ethyl ester binding to the benzodiazepine receptor.
Topics: Animals; Benzodiazepines; Brain; Carbolines; Diazepam; gamma-Aminobutyric Acid; Indoles; Kidney; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A | 1981 |
Unusual interactions of benzodiazepine receptor antagonists.
Topics: Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Biological Assay; Carbolines; Flumazenil; gamma-Aminobutyric Acid; Ganglia, Sympathetic; Indoles; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures | 1982 |
Thermodynamic changes associated with benzodiazepine and alkyl beta-carboline-3-carboxylate binding to rat brain homogenates.
Topics: Animals; Benzodiazepines; Brain; Carbolines; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Nickel; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Temperature; Thermodynamics | 1982 |
Regional heterogeneity of benzodiazepine binding sites in rat brain.
Topics: Animals; Binding, Competitive; Brain; Carbolines; Cerebellum; Chlorides; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1982 |
Interactions of different ligand classes with the benzodiazepine receptor.
Topics: Affinity Labels; Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Flumazenil; gamma-Aminobutyric Acid; Humans; Ligands; Membranes; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sodium Chloride | 1983 |
Evidence for an involvement of GABA receptors in the mediation of the proconvulsant action of ethyl-beta-carboline-3-carboxylate.
Topics: Animals; Binding Sites; Carbolines; Cerebral Cortex; Drug Synergism; gamma-Aminobutyric Acid; Hippocampus; Indoles; Injections, Intraventricular; Isoniazid; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1984 |
Effects of various 2-amino-6-alkyldithiopurines on brain specific [3H]diazepam binding.
Topics: Animals; Brain; Carbolines; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mercaptopurine; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1984 |
Stress and beta-carbolines decrease the density of low affinity GABA binding sites; an effect reversed by diazepam.
Topics: Animals; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Handling, Psychological; Indoles; Male; Rats; Rats, Inbred Strains; Stress, Physiological | 1984 |
Pharmacokinetic and pharmacodynamic factors contributing to the convulsant action of beta-carboline-3-carboxylic acid esters.
Topics: Animals; Brain; Carbolines; Convulsants; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Indoles; Kinetics; Male; Rats; Rats, Inbred Strains; Saimiri | 1983 |
Ethyl-beta-carboline-3-carboxylate decreases [3H]GABA binding in membrane preparations of rat cerebral cortex.
Topics: Animals; Brain; Carbolines; gamma-Aminobutyric Acid; Indoles; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains | 1983 |
Modulation of GABA binding to rat brain membranes by alkyl beta-carboline-3-carboxylate esters.
Topics: Animals; Brain; Carbolines; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Membranes; Rats | 1982 |
Cardiovascular neurons in cat caudal ventrolateral medulla: location and characterization of GABAergic input.
Topics: Animals; Antibody Specificity; Blood Pressure; Carbolines; Cardiovascular System; Cats; Female; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heart Rate; Ligands; Male; Medulla Oblongata; Microinjections; Muscimol; Neural Pathways; Neurons; Phenylethanolamine N-Methyltransferase; Picrotoxin; Tyrosine 3-Monooxygenase | 1995 |
Enhancement of GABA-activated current by muscarine in rat dorsal root ganglion neurons.
Topics: Acetylcholine; Action Potentials; Animals; Atropine; Bicuculline; Carbachol; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Modulators; Gallamine Triethiodide; gamma-Aminobutyric Acid; Ganglia, Spinal; Ion Channel Gating; Ion Channels; Male; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Nerve Tissue Proteins; Nicotinic Antagonists; Patch-Clamp Techniques; Pentobarbital; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Muscarinic | 1999 |