beta-carboline-3-carboxylic acid ethyl ester has been researched along with beta-carboline-3-carboxylic acid methyl ester in 28 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 20 (71.43) | 18.7374 |
| 1990's | 6 (21.43) | 18.2507 |
| 2000's | 2 (7.14) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Allen, MS; Cook, JM; Costantino, G; Dorn, LJ; Hagen, TJ; Koehler, KF; LaLoggia, AJ; Martin, MJ; Skolnick, P | 1 |
| Allen, MS; Codding, PW; Hagen, TJ; Koehler, KF; Martin, MJ; Narayanan, K; Schindler, LR; Schultz, C; Tan, YC; Trudell, ML | 1 |
| Chapouthier, G; Dodd, RH; Dorey, G; Poissonnet, G; Potier, MC; Potier, P; Prado de Carvalho, L; Rossier, J; Venault, P | 1 |
| Allen, MS; Codding, PW; Cook, JM; Hagen, TJ; Skolnick, P; Trudell, ML | 1 |
| Eigyo, M; Kawasaki, K; Matsushita, A; Murata, S; Sasatani, T; Shindo, H; Takada, S | 1 |
| Barker, SA; Cain, M; Cook, JM; Crawley, JN; Guzman, F; Paul, SM; Rice, KC; Skolnick, P; Weber, RW | 1 |
| Lippke, KP; Müller, WE; Schunack, WG; Wenning, W | 1 |
| Cain, M; Cook, JM; Guzman, F; Hagen, T; Larscheid, P; Paul, SM; Schweri, M; Skolnick, P | 1 |
| Good, AC; Peterson, SJ; Richards, WG | 1 |
| Platt, DE; Silverman, BD | 1 |
| Karplus, M; So, SS | 1 |
| Ahmad, K; Beg, Y; Cho, SJ; Muddassar, M; Pasha, FA | 1 |
| Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W | 1 |
| Claustre, Y; Dennis, T; Rivy, JP; Scatton, B | 1 |
| Moura, D; Soares-da-Silva, P | 1 |
| Chapouthier, G; de Carvalho, LP; Dodd, RH; Ouannès, C; Potier, P; Rossier, J; Valin, A; Venault, P | 1 |
| Gardner, CR; James, V | 1 |
| Sieghart, W | 1 |
| Cook, JA; Guzman, F; Hagen, TJ; Shannon, HE | 1 |
| Itonaga, M; Kubota, K; Uruno, T | 1 |
| Itonaga, M; Kubota, K | 1 |
| Macdonald, RL; Skerritt, JH | 1 |
| Little, HJ | 1 |
| Bonetti, EP; Haefely, W; Polc, P; Schaffner, R | 1 |
| Paul, SM; Skolnick, P | 1 |
| Barrett, JE; Martin, JV; Mendelson, WB; Paul, SM; Schweri, MM; Skolnick, P | 1 |
| Martin, JV; Mendelson, WB; Paul, SM; Schweri, MM; Skolnick, P; Wagner, RL | 1 |
| Estupinan, LE; France, CP; Gerak, LR | 1 |
1 review(s) available for beta-carboline-3-carboxylic acid ethyl ester and beta-carboline-3-carboxylic acid methyl ester
| Article | Year |
|---|---|
[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid | 1985 |
27 other study(ies) available for beta-carboline-3-carboxylic acid ethyl ester and beta-carboline-3-carboxylic acid methyl ester
| Article | Year |
|---|---|
Predictive binding of beta-carboline inverse agonists and antagonists via the CoMFA/GOLPE approach.
Topics: Animals; Binding, Competitive; Carbolines; Cerebral Cortex; Convulsants; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Mice; Models, Molecular; Models, Statistical; Molecular Conformation; Rats; Receptors, GABA-A; Regression Analysis; Structure-Activity Relationship | 1992 |
Synthetic and computer-assisted analyses of the pharmacophore for the benzodiazepine receptor inverse agonist site.
Topics: Binding Sites; Carbolines; Chemical Phenomena; Chemistry; Computer Simulation; Ligands; Models, Chemical; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 1990 |
Synthesis and benzodiazepine receptor affinities of rigid analogues of 3-carboxy-beta-carbolines: demonstration that the benzodiazepine receptor recognizes preferentially the s-cis conformation of the 3-carboxy group.
Topics: Animals; Carbolines; Chemical Phenomena; Chemistry; In Vitro Techniques; Mice; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 1989 |
Synthesis of novel 3-substituted beta-carbolines as benzodiazepine receptor ligands: probing the benzodiazepine receptor pharmacophore.
Topics: Animals; Carbolines; Chemical Phenomena; Chemistry; Diazepam; Hydrogen Bonding; Indoles; Mice; Pyridines; Receptors, GABA-A; Structure-Activity Relationship | 1988 |
A new thienylpyrazoloquinoline: a potent and orally active inverse agonist to benzodiazepine receptors.
Topics: Administration, Oral; Animals; Anticonvulsants; Indicators and Reagents; Male; Mice; Pentylenetetrazole; Pyrazoles; Quinolines; Receptors, GABA-A; Seizures; Thiophenes | 1987 |
Beta-carbolines: synthesis and neurochemical and pharmacological actions on brain benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Carbolines; Chemical Phenomena; Chemistry; Diazepam; Drug Interactions; Indoles; Male; Mice; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A | 1982 |
beta-Carbolines as benzodiazepine receptor ligands. 1. Synthesis and benzodiazepine receptor interaction of esters of beta-carboline-3-carboxylic acid.
Topics: Animals; Carbolines; Cattle; Cerebral Cortex; Indoles; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Biomimetic approach to potential benzodiazepine receptor agonists and antagonists.
Topics: Animals; Benzodiazepines; Cell Membrane; Cerebral Cortex; Diazepam; Indicators and Reagents; Rats; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship | 1984 |
QSAR's from similarity matrices. Technique validation and application in the comparison of different similarity evaluation methods.
Topics: Carbolines; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Imidazoles; Indoles; Molecular Structure; Pyridines; Structure-Activity Relationship | 1993 |
Comparative molecular moment analysis (CoMMA): 3D-QSAR without molecular superposition.
Topics: Adrenal Cortex Hormones; Binding Sites; Mathematics; Models, Molecular; Molecular Conformation; Molecular Structure; Molecular Weight; Predictive Value of Tests; Steroids; Structure-Activity Relationship; Testosterone | 1996 |
Three-dimensional quantitative structure-activity relationships from molecular similarity matrices and genetic neural networks. 2. Applications.
Topics: Cholinesterase Inhibitors; Dopamine beta-Hydroxylase; Drug Design; Enzyme Inhibitors; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Molecular Conformation; Molecular Structure; Neural Networks, Computer; Phosphorylases; Receptors, Aryl Hydrocarbon; Static Electricity; Structure-Activity Relationship | 1997 |
3D and quantum QSAR of non-benzodiazepine compounds.
Topics: Benzodiazepines; Carbolines; Imaging, Three-Dimensional; Imidazoles; Inhibitory Concentration 50; Models, Molecular; Molecular Structure; Pyrimidines; Quantitative Structure-Activity Relationship; Software | 2008 |
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis | 2008 |
Pharmacological studies on stress-induced increase in frontal cortical dopamine metabolism in the rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anti-Anxiety Agents; Carbolines; Dopamine; Electroshock; Fear; Frontal Lobe; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, GABA-A; Stress, Physiological; Swimming; Zolpidem | 1986 |
3-Amino-beta-carboline derivatives and the benzodiazepine receptor. Synthesis of a selective antagonist of the sedative action of diazepam.
Topics: Animals; Carbolines; Convulsants; Diazepam; In Vitro Techniques; Indoles; Male; Mice; Papio; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship | 1985 |
Actions and interactions of benzodiazepine agonists, antagonists and inverse agonists on suprahyoid muscle twitching.
Topics: Amphetamine; Animals; Benzodiazepines; Carbolines; In Vitro Techniques; Male; Muscle Contraction; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Benzodiazepine receptors: multiple receptors or multiple conformations?
Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A | 1985 |
Beta-carbolines as antagonists of the discriminative stimulus effects of diazepam in rats.
Topics: Animals; Carbolines; Diazepam; Discrimination Learning; Harmine; Male; Picrotoxin; Rats; Rats, Inbred F344 | 1988 |
Cholecystokinin antagonism by beta-carboline esters in the central nervous system in mice.
Topics: Animals; Brain; Carbolines; Cholecystokinin; Eating; Male; Mice; Mice, Inbred Strains; Morphine; Nociceptors; Pain; Time Factors | 1988 |
Beta-carbolines selectively antagonize the cholecystokinin action in isolated guinea-pig gallbladder muscle.
Topics: Alkylation; Animals; Carbolines; Cholecystokinin; Dibenzylchlorethamine; Dose-Response Relationship, Drug; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Receptors, Cholecystokinin | 1986 |
Benzodiazepine receptor ligand actions on GABA responses. Beta-carbolines, purines.
Topics: Animals; Carbolines; Cells, Cultured; Diazepam; Drug Interactions; gamma-Aminobutyric Acid; Indoles; Ligands; Mice; Neurons; Purines; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord | 1984 |
The effects of benzodiazepine agonists, inverse agonists and Ro 15-1788 on the responses of the superior cervical ganglion to GABA in vitro.
Topics: Animals; Barbiturates; Benzodiazepinones; Bicuculline; Carbolines; Chlordiazepoxide; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Sympathetic; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
A three-state model of the benzodiazepine receptor explains the interactions between the benzodiazepine antagonist Ro 15-1788, benzodiazepine tranquilizers, beta-carbolines, and phenobarbitone.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Female; Flumazenil; Hippocampus; In Vitro Techniques; Indoles; Male; Mice; Models, Biological; Phenobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord | 1982 |
New concepts in the neurobiology of anxiety.
Topics: Animals; Anxiety; Barbiturates; Behavior; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Central Nervous System; Flumazenil; Humans; Macaca mulatta; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Pharmacokinetic and pharmacodynamic factors contributing to the convulsant action of beta-carboline-3-carboxylic acid esters.
Topics: Animals; Brain; Carbolines; Convulsants; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Indoles; Kinetics; Male; Rats; Rats, Inbred Strains; Saimiri | 1983 |
3-carboethoxy-beta-carboline (beta-CCE) elicits electroencephalographic seizures in rats: reversal by the benzodiazepine antagonist CGS 8216.
Topics: Animals; Benzodiazepines; Brain; Carbolines; Electroencephalography; Indoles; Male; Pyrazoles; Rats; Rats, Inbred Strains; Seizures | 1983 |
Ventilatory effects of negative GABA(A) modulators in rhesus monkeys.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Female; GABA Modulators; Macaca mulatta; Male; Receptors, GABA-A; Respiration, Artificial | 1998 |