benzoxazoles has been researched along with urea in 329 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (0.30) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 84 (25.53) | 29.6817 |
2010's | 207 (62.92) | 24.3611 |
2020's | 37 (11.25) | 2.80 |
Authors | Studies |
---|---|
DeLong, DC; Kisner, K; Paget, CJ; Stone, RL | 1 |
Arch, JR; Chapman, H; Haynes, AC; Jackson, B; Johns, A; Porter, RA; Tadayyon, M | 1 |
Ashmeade, TE; Gartlon, J; Hagan, JJ; Hatcher, JP; Hemmati, P; Hunter, AJ; Johns, A; Jones, DN; Munton, RP; Parker, F; Porter, RA; Routledge, C; Taylor, SG; Upton, N | 1 |
Brough, SJ; Jerman, JC; Jewitt, F; Johns, A; Porter, RA; Sabido-David, C; Smart, D | 1 |
Arch, JR; Blundell, JE; Canto de Souza, AL; Halford, JC; Johns, A; Nunes de Souza, RL; Piper, DC; Porter, RA; Rodgers, RJ; Upton, N | 1 |
Babbs, AJ; Bingham, S; Cutler, L; Davey, PT; Hunter, AJ; Irving, EA; Jeffrey, P; Johns, A; Parsons, AA; Porter, RA; Riba, I; Sammons, MJ; Upton, N; Wyles, M | 1 |
Austin, N; Brough, SJ; Chan, WN; Coldwell, M; Coulton, S; Hadley, MS; Jeffrey, P; Jerman, JC; Jewitt, F; Johns, A; Porter, RA; Smart, D; Widdowson, K | 1 |
Benham, CD; Davies, CH; Evans, ML; Gill, CH; Harries, MH; Soffin, EM | 1 |
Arch, JR; Cawthorne, MA; Chapman, H; Clapham, JC; Haynes, AC; Moore, GB; Tadayyon, M; Taylor, C | 1 |
Arch, JR; Haynes, AC; Smart, D; Williams, G | 1 |
Chiba, T; Nozaki-Taguchi, N; Yamamoto, T | 1 |
Hayashi, H; Kaibara, M; Matsuo, K; Nakane, Y; Taniyama, K; Uezono, Y | 1 |
Duxon, MS; Piper, DC; Smith, MI; Upton, N | 1 |
Buijs, RM; Davies, CH; Lee, K; Nolan, MF; Richardson, PJ; Spanswick, D; van den Top, M | 1 |
Bloom, SR; Coen, CW; Goubillon, ML; Grimshaw, SE; Kalamatianos, T; Kennedy, AR; Murray, JF; Siddiqui, A; Sivanesan, V; Small, CJ; Wilson, CA; Young, H | 1 |
Ehrström, M; Hellström, PM; Kirchgessner, AL; Ma, J; Näslund, E | 1 |
Hirota, K; Kudo, M; Kudo, T; Kushikata, T; Matsuki, A; Smart, D | 1 |
Cheng, JK; Chiou, LC; Chou, RC; Hwang, LL | 1 |
Hirota, K; Jerman, JC; Kudo, M; Kushikata, T; Lambert, DG; Matsuki, A; Smart, D; Yoshida, H | 1 |
Baghdoyan, HA; Bernard, R; Lydic, R | 1 |
Gao, J; Li, Y; Owyang, C; Wu, X; Yan, J | 1 |
Kiwaki, K; Kotz, CM; Lanningham-Foster, L; Levine, JA; Wang, C | 1 |
Brough, SJ; Herdon, HJ; Jerman, JC; Langmead, CJ; Porter, RA; Scott, C | 1 |
Blundell, JE; Halford, JC; Ishii, Y; Johns, A; Porter, R; Rodgers, RJ; Upton, N | 2 |
Brough, SJ; Davies, CH; Gill, CH; Jerman, JC; Soffin, EM | 1 |
Chase, MH; Fung, SJ; Xi, M; Yamuy, J | 1 |
Armstrong, DL; Oomura, Y; Phelix, CF; Wayner, MJ | 1 |
Blundell, JE; Halford, JC; Ishii, Y; Jeffrey, P; Johns, A; Porter, R; Rodgers, RJ; Summerfield, S; Upton, N | 1 |
Gaus, S; Kajiyama, S; Kawamoto, M; Matsunaga, A; Shiraishi, S; Suyama, H; Yuge, O | 1 |
Bray, GA; Ishii, Y; Mendoza, T; Stasi, LP; Upton, N; White, CL; York, DA | 1 |
Kotz, CM; Thorpe, AJ | 1 |
Hirota, K; Kudo, M; Kudo, T; Kushikata, T; Tose, R; Yoshida, H | 1 |
Boutrel, B; de Lecea, L; Kenny, PJ; Koob, GF; Markou, A; Martin-Fardon, R; Specio, SE | 1 |
Hashimoto, S; Khotib, J; Miyatake, M; Nagumo, Y; Nakamachi, T; Narita, M; Sakurai, T; Shioda, S; Suzuki, T; Yanagisawa, M | 1 |
Aimoto, S; Akutsu, H; Ikegami, T; Nagai, K; Nakagawa, A; Nakano, M; Takai, T; Takaya, T | 1 |
Bonci, A; Borgland, SL; Fields, HL; Sarti, F; Taha, SA | 1 |
Dong, HL; Fukuda, S; Higuchi, T; Murata, E; Zhu, Z | 1 |
Chen, F; Cowen, MS; Lawrence, AJ; Oldfield, B; Yang, HJ | 1 |
Azuma, YT; Hata, F; Nakajima, H; Okishio, Y; Satoh, Y; Takeuchi, T | 1 |
Akbari, E; Motamedi, F; Naghdi, N | 2 |
D'Anna, KL; Gammie, SC | 1 |
Hsu, MA; Rasmussen, K; Yang, Y | 1 |
Akerman, S; Goadsby, PJ; Holland, PR | 1 |
Ceregrzyn, M; Kato, I; Korczynski, W; Wolinski, J; Zabielski, R | 1 |
Briski, K; Kale, A; Paranjape, S; Vavaiya, K | 1 |
Branconi, JL; Fenik, VB; Kubin, L; Lu, JW; Mann, GL; Rukhadze, I | 1 |
Akerman, KE; Bengtsson, MW; Flemström, G; Herzig, KH; Mäkelä, K; Sjöblom, M; Uotila, S | 1 |
Libertun, C; Lux-Lantos, V; Silveyra, P | 1 |
Hemrick-Luecke, SK; Hsu, MA; Johnson, BG; Noone, S; Rasmussen, K; Thompson, LK | 1 |
Deng, BS; Fukuda, Y; Kuwaki, T; Nakamura, A; Yanagisawa, M; Zhang, W | 1 |
Fadel, J; Frederick-Duus, D; Guyton, MF | 1 |
Akbari, E; Motamedi, F; Naghdi, N; Noorbakhshnia, M | 1 |
Cools, AR; Ikeda, H; Koshikawa, N; Kotani, A | 1 |
Hirota, K; Kudo, M; Kudo, T; Kushikata, T; Yoshida, H | 1 |
Golden, SA; Nair, SG; Shaham, Y | 1 |
Albericio, F; Armand-Ugón, M; El-Faham, A; Esté, JA | 1 |
Chen, XW; Fan, HX; Gu, JL; Guo, N; Hu, ZA; Huang, W; Lü, J; Ruan, HZ; Xiu, Y; Yan, JA; Yu, ZP; Zhang, CX; Zhou, Z | 1 |
Dileone, RJ; Sarhan, M; Sharf, R | 1 |
Chen, J; Conner, AC; Ramanjaneya, M; Randeva, HS; Stanfield, PR | 1 |
Bartlett, SE; Bonci, A; Borgland, SL; Richards, JK; Simms, JA; Steensland, P; Taha, SA | 1 |
Shono, K; Yamamoto, T | 1 |
Aston-Jones, G; Gompf, HS | 1 |
Bai, YJ; Han, J; Li, YH; Sui, N; Yang, XY; Zheng, XG | 1 |
Gamo, Y; Hanawa, T; Ito, N; Nagai, T; Oikawa, T; Yabe, T; Yamada, H | 1 |
Chen, XW; Ge, L; Huang, W; Song, B; Yan, JA; Yu, ZP | 1 |
Cameron, MD; Hollander, JA; Kamenecka, TM; Kenny, PJ; Lu, Q | 1 |
Bengtsson, MW; Flemström, G; Herzig, KH; Mäkelä, K | 1 |
Baccari, MC; Bani, D; Calamai, F | 1 |
Furukawa, K; Hirota, K; Kudo, M; Kushikata, T; Tose, R; Ueno, S; Yoshida, H | 1 |
Eliassi, A; Naghdi, N; Nazari, M | 1 |
Jochem, J | 1 |
Dias, MB; Li, A; Nattie, EE | 1 |
Douglas, SA; Furukawa, K; Hashiba, E; Hirota, K; Kawaguchi, Y; Kudo, M; Kudo, T; Kushikata, T; Ono, T; Yoshida, H | 1 |
Cannella, N; Ciccocioppo, R; Economidou, D; Heilig, M; Kallupi, M; Massi, M; Stopponi, S | 1 |
Holden, JE; Jeong, Y | 1 |
Brown, JE; Chen, J; Conner, AC; Jöhren, O; Kumar, P; Lehnert, H; Ramanjaneya, M; Randeva, HS; Stanfield, PR | 1 |
Inyushkin, A; Karnas, D; Klisch, C; Meissl, H; Mordel, J; Pévet, P | 1 |
Alcin, E; Ayar, A; Kelestimur, H; Ozcan, M; Sahin, Z; Serhatlioglu, I | 1 |
Boschen, KE; Burk, JA; Fadel, JR | 1 |
Aston-Jones, G; Smith, RJ; Tahsili-Fahadan, P | 1 |
Kirouac, GJ; Li, S; Li, Y; Sui, N | 1 |
Aston-Jones, G; See, RE; Smith, RJ | 1 |
Aston-Jones, G; Moorman, DE | 1 |
Hedou, G; Heidbreder, C; Hutcheson, DM; Quarta, D; Valerio, E | 1 |
Bonci, A; Borgland, SL; Bowers, MS; Chang, SJ; Chen, BT; Chou, J; Floresco, SB; Thompson, JL; Vittoz, N | 1 |
Aston-Jones, G; Chen, J; Gompf, H; Kelz, MB; Sun, Y; Yanagisawa, M | 1 |
Chen, F; Chen, X; Hu, Z; Li, B; Li, Y; Xia, J; Xiong, Y; Yan, J; Ye, J; Zhou, Z | 1 |
Wang, JJ; Yu, L; Zhang, J; Zhang, XY; Zhu, JN | 1 |
Dias, MB; Li, A; Nattie, E | 1 |
Baghdoyan, HA; Lydic, R; Watson, CJ; Watson, SL | 1 |
DiLeone, RJ; Guarnieri, DJ; Sharf, R; Taylor, JR | 1 |
Birnbaum, S; Chuang, JC; Lutter, M; Osborne-Lawrence, S; Perello, M; Rovinsky, SA; Sakata, I; Woloszyn, J; Yanagisawa, M; Zigman, JM | 1 |
Brookshire, BR; España, RA; Jones, SR; Locke, JL; Oleson, EB; Roberts, DC | 1 |
Berrendero, F; de Lecea, L; Maldonado, R; Martín-García, E; Plaza-Zabala, A | 1 |
Benoit, SC; Choi, DL; Davis, JF; Fitzgerald, ME | 1 |
Corrigall, WA; Kotz, CM; LeSage, MG; Perry, JL; Shelley, D | 1 |
Brayton, CE; DiLeone, RJ; Guarnieri, DJ; Sarhan, M; Sharf, R; Taylor, JR | 1 |
Acar, N; Bülbül, M; Gemici, B; Izgüt-Uysal, VN; Ozdem, S; Tan, R; Ustünel, I | 1 |
De Carolis, L; Milella, MS; Nativio, P; Nencini, P; Passarelli, F; Scaccianoce, S; Schepisi, C | 1 |
Dickson, SL; Egecioglu, E; Engel, JA; Jerlhag, E | 1 |
Azizi, H; Mirnajafi-Zadeh, J; Rohampour, K; Semnanian, S | 1 |
Allen, AM; Oldfield, BJ; Verty, AN | 1 |
Babygirija, R; Bülbül, M; Ludwig, K; Takahashi, T | 1 |
Akbari, E; Davoodi, FG; Ghanbarian, E; Motamedi, F; Noorbakhshnia, M | 1 |
Haghparast, A; Hassanpour-Ezatti, M; Safari, MS; Taslimi, Z | 1 |
Chen, X; Kirouac, GJ; Li, S; Li, Y; Qi, K; Sui, N; Wang, H | 1 |
Dezsi, G; Jupp, B; Krstew, E; Lawrence, AJ | 1 |
Pilowsky, PM; Rahman, AA; Shahid, IZ | 1 |
Baghdoyan, HA; Brevig, HN; Lydic, R; Watson, CJ | 1 |
Cunningham, CL; Voorhees, CM | 1 |
Onizuka, S; Shirasaka, T; Tsuneyoshi, I; Yonaha, T | 1 |
Milligan, G; Pediani, JD; Ward, RJ | 1 |
Halbout, B; Heidbreder, C; Hutcheson, DM; Quarta, D; Rigal, A; Valerio, E | 1 |
Cabello, V; Mediavilla, C; Risco, S | 1 |
He, YC; Li, B; Li, HZ; Wang, JJ; Yu, L; Zhang, J; Zhu, JN | 1 |
Cao, J; de Lecea, L; Ikemoto, S | 1 |
Birnbaum, SG; Elmquist, JK; Lutter, M; Marcus, JN; Mochizuki, T; Nestler, EJ; Pettersen, A; Scammell, TE; Scott, MM | 1 |
Kubin, L; Stettner, GM; Volgin, DV | 1 |
Jupp, B; Krivdic, B; Krstew, E; Lawrence, AJ | 1 |
Charnley, JL; Dayas, CV; James, MH; Jones, E; Levi, EM; Smith, DW; Yeoh, JW | 1 |
Gilmour, BP; Perrey, DA; Runyon, SP; Thomas, BF; Zhang, Y | 1 |
DiMicco, JA; Rusyniak, DE; Zaretskaia, MV; Zaretsky, DV | 1 |
Azuma, M; Kang, KS; Kojima, K; Maejima, S; Matsuda, K; Uchiyama, M; Yokobori, E | 1 |
Frohman, MA; Jäntti, MH; Kukkonen, JP; Putula, J; Somerharju, P | 1 |
Gemici, B; İzgüt-Uysal, VN; Tan, R | 1 |
Berrendero, F; Flores, Á; Maldonado, R; Plaza-Zabala, A | 1 |
Chen, Y; Fan, S; Hu, Z; Jia, X; Qi, A; Wang, T; Xia, J; Xiong, J; Yan, J; Yang, N; Ye, J | 1 |
Dossat, AM; Kay, K; Lilly, N; Overton, JM; Parise, EM; Seth, R; Williams, DL | 1 |
Chiou, LC; Fu, SY; Ho, YC; Lee, HJ; Liao, HT; Liao, YY; Mackie, K; Teng, SF; Tung, LW | 1 |
Chaleek, N; Eliassi, A; Haghparast, A; Kermani, M | 1 |
Blasiak, T; Lewandowski, MH; Pekala, D; Raastad, M | 1 |
Cano, G; Madden, CJ; Morrison, SF; Tupone, D | 1 |
Kukkonen, JP; Putula, J | 1 |
Altieri, F; Azzariti, A; Cervoni, L; Crestani, M; Di Giovanni, C; Fracchiolla, G; Gilardi, F; Giudici, M; Guerrini, U; Laghezza, A; Lavecchia, A; Loiodice, F; Mitro, N; Montanari, R; Paradiso, A; Piemontese, L; Pochetti, G; Porcelli, L; Simone, GM; Tortorella, P | 1 |
Fish, EW; Jarrett, TM; Malanga, CJ; McGuigan, MM; Riday, TT; Robinson, JE | 1 |
Cameron, MD; Chan, C; Ghee, SM; Kenny, PJ; Lin, L; See, RE; Zhou, L | 1 |
Aston-Jones, G; Smith, RJ | 1 |
DiMicco, JA; Durant, PJ; Rusyniak, DE; Zaretskaia, MV; Zaretsky, DV | 1 |
Aston-Jones, G; Mahler, SV; Smith, RJ | 1 |
Azizi, H; Fathollahi, Y; Ranjbar-Slamloo, Y; Semnanian, S | 1 |
Fitz, SD; Johnson, PL; Lightman, SL; Lowry, CA; Samuels, BC; Shekhar, A | 1 |
Aston-Jones, GS; Sartor, GC | 1 |
Jäntti, MH; Kukkonen, JP; Turunen, PM | 1 |
Cataldi, NI; Libertun, C; Lux-Lantos, VA | 1 |
Borroni, E; Kilduff, TS; Malherbe, P; Morairty, SR; Moreau, JL; Revel, FG; Valladao, D; Wettstein, JG | 1 |
Martin-Fardon, R; Weiss, F | 2 |
Azhdari-Zarmehri, H; Erami, E; Haghparast, A; Heidari-Oranjaghi, N | 1 |
Aston-Jones, G; Do, PH; See, RE; Smith, RJ; Zhou, L | 1 |
Bhatnagar, S; Heydendael, W; Sengupta, A | 1 |
Dehpour, AR; Esmaeili, B; Ghaffarpour, M; Javadi-Paydar, M; Mirbaha, H; Motiei-Langroudi, R; Tabaeizadeh, M; Tahsili-Fahadan, P | 1 |
Azhdari-Zarmehri, H; Erami, E; Ghasemi-Dashkhasan, E; Haghparast, A; Rahmani, A; Semnanian, S | 1 |
Brieaddy, L; Carroll, FI; Lewin, AH; Mascarella, SW; McElhinny, CJ; Runyon, S | 1 |
Aston-Jones, G; Cason, AM | 3 |
Rodgers, RJ; Snow, NF; Taylor, LJ; Wright, FL | 1 |
Berrendero, F; Flores, Á; Maldonado, R; Martín-García, E; Plaza-Zabala, A; Saravia, R | 1 |
Dai, YW; Huang, SC; Hwang, LL; Lee, YH; Li, TL | 1 |
Chen, F; Chen, H; Hu, B; Hu, ZA; Sui, JF; Wang, YJ; Yan, J; Yang, L; Yang, N; Zhu, ZR | 1 |
Gillman, AG; Kosobud, AE; Leffel, JK; Timberlake, W | 1 |
Liu, XM; Ni, LY; Song, Y; Tang, JY; Zhu, MJ | 1 |
Berrendero, F; Flores, Á; Maldonado, R | 1 |
Kay, K; Lilly, N; Parise, EM; Williams, DL | 1 |
Azhdari-Zarmehri, H; Esmaeili, MH; Haghdoost-Yazdi, H; Sofiabadi, M | 1 |
Billington, CJ; Kotz, CM; Teske, JA | 1 |
de Lecea, L; Farb, CR; Fink, AE; Ledoux, JE; Sears, RM; Wigestrand, MB | 1 |
Amadeo, A; Aracri, P; Banfi, D; Becchetti, A; Pasini, ME | 1 |
Liu, Xm; Ren, Yy; Tang, Jy; Tang, S; Yang, Wx; Zhang, Rx; Zhao, X | 1 |
Cornish, JL; Staples, LG | 1 |
Patrone, A; Perello, M; Reynaldo, M; Valdivia, S | 1 |
Mediavilla, C; Risco, S | 2 |
Fujita, M; Kobashi, M; Matsuo, R; Mitoh, Y; Mizutani, S; Shimatani, Y | 1 |
Cone, JJ; McCutcheon, JE; Roitman, MF | 1 |
Duncan, MJ; Franklin, KM; Legan, SJ; Peng, X; Yun, C | 1 |
Harada, S; Koda, S; Tokuyama, S; Yamazaki, Y | 1 |
Fatahi, Z; Haghparast, A; Sarihi, A; Zarepour, L | 1 |
Chang, X; Guo, L; Ju, SJ; Zhao, Y | 1 |
Adidharma, W; Deats, SP; Lonstein, JS; Yan, L | 1 |
Karasawa, H; Taché, Y; Wang, L; Yakabi, S | 1 |
Berrendero, F; Costa, G; Flores, Á; Maldonado, R; Saravia, R; Valls-Comamala, V | 1 |
Iinuma, N; Konno, N; Matsuda, K; Nakamachi, T; Sakashita, A; Shibata, H; Wada, K | 1 |
Azizi, H; Javan, M; Mirnajafi-Zadeh, J; Mousavi, Y; Semnanian, S | 1 |
Alcaraz-Iborra, M; Carvajal, F; Cubero, I; Lerma-Cabrera, JM; Valor, LM | 1 |
Azizi, H; Ghaemi-Jandabi, M; Semnanian, S | 1 |
Routh, VH; Santiago, AM; Sheng, Z; Thomas, MP | 1 |
Le Foll, C; Levin, BE; Otlivanchik, O | 1 |
Chang, X; Guo, L; Ju, S; Zhao, Y | 1 |
Chen, ZP; Wang, JJ; Yu, L; Zhang, XY; Zhu, JN; Zhuang, QX | 1 |
Fatahi, Z; Haghparast, A; Moradi, M; Rashidy-Pour, A | 1 |
Cornish, JL; Staples, LG; Vanderhaven, MW | 1 |
España, RA; Prince, CD; Rau, AR; Yorgason, JT | 1 |
Kumei, S; Miyagishi, S; Nozu, T; Ohhira, M; Okumura, T; Takakusaki, K | 2 |
Elahdadi Salmani, M; Goudarzi, E; Goudarzi, I; Lashkarbolouki, T | 1 |
Navarro, M; Olney, JJ; Thiele, TE | 2 |
Arezoomandan, R; Fatahi, Z; Haghparast, A; Riahi, E | 1 |
Aston-Jones, G; Bentzley, BS | 1 |
Cui, Y; Guo, SJ; Huang, ZZ; Jiang, JX; Liu, H; Xin, WJ; Zhang, XQ | 1 |
Abbasnejad, M; Amirkhosravi, L; Esmaeili-Mahani, S; Kooshki, R; Rafie, F; Raoof, M; Raoof, R; Sheibani, V | 1 |
Alcaraz-Iborra, M; Carvajal, F; Cubero, I; de la Fuente, L; Lerma-Cabrera, JM; Sanchez-Amate, Mdel C; Valor, LM | 1 |
Chen, QH; He, C; Hu, ZA; Li, C; Xia, JX; Yang, L; Ye, JN; Zhang, J | 1 |
Brown, RM; Jupp, B; Khoo, SY; Kim, AK; Kim, JH; Lawrence, AJ | 1 |
Behrouzvaziri, A; Fu, D; Molkov, YI; Rusyniak, DE; Tan, P; Yoo, Y; Zaretskaia, MV; Zaretsky, DV | 1 |
Chrobok, L; Lewandowski, MH; Palus, K | 1 |
Bernstein, DL; Brodnik, ZD; España, RA; Prince, CD | 1 |
Carfagna, C; Della Ca', N; Fini, F; Gabriele, B; Mancuso, R; Raut, DS | 1 |
Alaii, E; Emam, AH; Komaki, A; Panah, MH; Sarihi, A; Seif, S; Vafaeirad, M | 1 |
Ali Reza, M; Azizi, H; Mirnajafi-Zadeh, J; Mohammad-Pour Kargar, H; Semnanian, S | 1 |
Li, DP; Yuan, F; Zhang, Y; Zhou, JJ | 1 |
Gong, YL; Guo, FF; Peng, XY; Sun, XR; Xu, L | 1 |
Holden, JE; Jeong, Y; Wagner, M; Wardach, J | 1 |
Dunn-Meynell, A; Levin, BE; Otlivanchik, O; Sanders, NM | 1 |
Cole, S; Mayer, HS; Petrovich, GD | 1 |
Joshi, D; Singh, SK | 1 |
Alijanpour, S; Tirgar, F; Zarrindast, MR | 1 |
Aston-Jones, G; Bentzley, BS; Porter-Stransky, KA | 1 |
Korim, WS; Llewellyn-Smith, IJ; Verberne, AJ | 1 |
Ebrahimian, F; Haghparast, A; Naghavi, FS; Sadeghzadeh, F; Taslimi, Z; Yazdi, F | 1 |
Abbasnejad, M; Esmaeili-Mahani, S; Kooshki, R; Raoof, M | 2 |
Bícego, KC; Dias, MB; Fonseca, EM; Gargaglioni, LH; Vicente, MC | 1 |
Ayoobi, F; Fatemi, I; Motevalian, M; Roohbakhsh, A; Sanati, MH; Shamsizadeh, A; Taghipour, Z | 1 |
Babapour, V; Ezzatpanah, S; Haghparast, A | 1 |
Azizi, H; Davoudi, M; Mirnajafi-Zadeh, J; Semnanian, S | 1 |
Chang, LY; Chiou, LC; Ho, YC; Hwang, LL; Lee, HJ; Mackie, K; Teng, SF | 1 |
Socała, K; Szuster-Ciesielska, A; Wlaź, P | 1 |
Gong, Y; Guo, F; Hao, H; Luan, X; Sun, X; Xu, L | 1 |
Dong, HL; Liu, Y; Ouyang, PR; Ran, MZ; Tong, L; Yang, C; Zhang, LN; Zhang, ZC | 1 |
Cole, S; Keefer, SE; Petrovich, GD | 1 |
Fatahi, Z; Haghparast, A; Moradi, M; Parsania, S | 1 |
Benedetto, L; Ferreira, A; Rivas, M; Torterolo, P | 1 |
Abdollahi, H; Azizi, H; Ghaemi-Jandabi, M; Semnanian, S | 1 |
Esmaeili, MH; Ezzatpanah, S; Haghparast, A; Reisi, Z | 1 |
Chen, AQ; Chen, H; Chen, L; Chen, WF; Chen, XY; Liu, HX; Liu, HY; Pang, YY; Sheng, Q; Wang, Y; Xue, Y; Yang, YT | 1 |
Hopf, FW; Lei, K; Wegner, SA; Yu, JH | 1 |
Kerr, TM; Martin-Fardon, R; Matzeu, A; Weiss, F | 1 |
Abbasnejad, M; Bahaaddini, M; Esmaeili-Mahani, S; Khatamsaz, S; Raoof, M | 1 |
Herman, MA; Koob, GF; Roberto, M; Schmeichel, BE | 1 |
Kirouac, GJ; Li, S; Wang, H | 1 |
Hayward, LF; Hernandez, ME; Martin, EJ | 1 |
Asadi, S; Fereidoni, M; Kordi Jaz, E; Moghimi, A; Roohbakhsh, A; Shamsizadeh, A | 1 |
Farahmandfar, M; Kadivar, M; Rastipisheh, S | 1 |
Aston-Jones, G; James, MH; Kilroy, EA; Moorman, DE | 1 |
Azizi, H; Hooshmand, B; Javan, M; Semnanian, S | 1 |
Angeli, A; Bartolucci, G; Carta, F; Nocentini, A; Peat, TS; Supuran, CT | 1 |
Kim, MS; Minamino, N; Nakazato, M; Namkoong, C; Sakoda, H; Sasaki, K; Toshinai, K; Ueta, Y; Waise, TMZ | 1 |
Akbari, E; Ardeshiri, MR; Hosseinmardi, N | 3 |
Bowyer, SL; Kassiou, M; O'Brien-Brown, J; Reekie, TA; Werry, EL; Wong, ECN | 1 |
Berrendero, F; Flores, Á; Herry, C; Maldonado, R | 1 |
Doostmohammadi, J; Hooshmandi, M; Hosseinmardi, N; Janahmadi, M; Khakpai, F; Rohampour, K | 1 |
Brailoiu, E; Connelly, KL; Gentile, TA; Muschamp, JW; Simmons, SJ; Watson, MN; Zhang, Y | 1 |
Farahimanesh, S; Haghparast, A; Zarrabian, S | 1 |
Liu, LL; Qiao, SN; Zhang, DQ; Zhong, YM; Zhou, W | 1 |
Alizadeh, AM; Ezzatpanah, S; Haghparast, A; Shafiei, I | 1 |
Chen, AQ; Chen, L; Chu, HY; Liu, C; Liu, YH; Sheng, Q; Wang, Y; Xue, Y | 1 |
Haghparast, A; Karimi-Haghighi, S; Mousavi, Z; Sahafzadeh, M | 1 |
Farahimanesh, S; Haghparast, A; Karimi, S | 1 |
Babapour, V; Haghparast, A; Pourreza, P | 1 |
Kumei, S; Nozu, T; Ohhira, M; Okumura, T; Takakusaki, K | 1 |
Baranowska-Bosiacka, I; Gutowska, I; Kotlińska, J; Listos, J; Listos, P; Talarek, S; Tarnowski, M; Łupina, M | 1 |
Bangasser, DA; Bhatnagar, S; Blume, SR; Luz, S; Nam, H | 1 |
Fujita, T; Kumamoto, E; Wang, C | 1 |
Fazli-Tabaei, S; Haghparast, A; Karimi-Haghighi, S; Rezaee, L | 1 |
Evans, SM; Foltin, RW | 1 |
Abbasnejad, M; Esmaeili-Mahani, S; Raoof, M; Shahsavari, F | 1 |
Azizi, H; Kargar, HM; Mani, AR; Mirnajafi-Zadeh, J; Semnanian, S | 1 |
Aldavert-Vera, L; Álvarez, A; García-Brito, S; Huguet, G; Kádár, E; Segura-Torres, P | 1 |
Edalat, P; Haghparast, A; Kavianpour, M; Zarrabian, S | 1 |
Joshi, D; Sarkar, D; Singh, SK | 1 |
Han, X; Peng, W; Zhou, J | 1 |
Abbasnejad, M; Esmaeili-Mahani, S; Kooshki, R; Mansoori, M; Raoof, M; Soofiabadi, S | 1 |
Hosseini, A; Khazali, H | 1 |
Aston-Jones, G; Bowrey, HE; James, MH; Koll, NE; Stopper, CM; Zimmer, BA | 1 |
Fatahi, Z; Haghparast, A; Hamidi, G; Karimi, S | 1 |
Aston-Jones, G; Bowrey, HE; James, MH; Stopper, CM | 1 |
Guo, F; Han, X; Luan, X; Sun, X; Wang, C; Xu, L | 1 |
Alijanpour, S; Ebrahimi-Ghiri, M; Khakpai, F; Zarrindast, MR | 1 |
Bahramzadeh Zoeram, S; Elahdadi Salmani, M; Goudarzi, I; Lashkarbolouki, T | 1 |
Kaneko, K; Kobayashi, M; Oi, Y; Usui, M | 1 |
Bian, H; Hu, Q; Huang, L; Li, B; Liang, X; Tang, J; Zhang, JH | 1 |
Aston-Jones, G; James, MH; Wiskerke, J | 1 |
Chikahisa, S; Miyatake, Y; Otsuka, A; Sakaue, H; Séi, H; Shiuchi, T | 1 |
Aston-Jones, G; Fragale, JE; James, MH; Pantazis, CB | 1 |
Brojeni, MS; Haghparast, A; Rashvand, M | 1 |
Assar, N; Haghparast, A; Mahmoudi, D; Mousavi, Z; Zarrabian, S | 1 |
Aston-Jones, G; James, MH; Mohammadkhani, A; Pantazis, CB | 1 |
Aston-Jones, G; Bowrey, HE; Fragale, JE; James, MH; Mohammadkhani, A; Pantazis, CB | 1 |
Furukawa, J; Maehara, S; Ota, T | 1 |
Igarashi, S; Ishioh, M; Kumei, S; Nozu, T; Ohhira, M; Okumura, T | 1 |
Haghparast, A; Jamali, S; Motamedi, F; RayatSanati, K; Shirazy, M | 1 |
Cui, C; Jia, M; Li, Y; Ma, H; Miao, D; Wu, L; Yang, M | 1 |
Kim, JS; Martin-Fardon, R | 1 |
Martin-Fardon, R; Matzeu, A | 1 |
Behnaz, M; Haghparast, A; Rahimitabar, N; Rezaee, L; Safari-Sandiani, E | 1 |
Haghparast, A; Matini, T; Rahban, M; Rezaee, L; Tehranchi, A | 1 |
Haghparast, A; Kashfi, K; Manaheji, H; Salehi, S | 1 |
Bayramoğlu, O; Bülbül, M; Sinen, O | 1 |
Abrari, K; Elahdadi Salmani, M; Lashkarbolouki, T; Nasiri, M; Salehabadi, S | 1 |
Matsuura, W; Nakamoto, K; Tokuyama, S | 1 |
Aston-Jones, G; Bentzley, BS; Freeman, LR; James, MH | 1 |
Coiduras, II; Maske, CB; Parise, EM; Williams, DL | 1 |
Joghataei, MT; Komaki, A; Kourosh-Arami, M; Mohsenzadegan, M | 1 |
Haghparast, A; Jamali, S; Karimi-Haghighi, S; Khosrowabadi, E | 1 |
Abbasnejad, M; Esmaeili-Mahani, S; Kooshki, R; Raoof, M; Sheibani, V | 1 |
Gholami, M; Joghataei, MT; Komaki, A; Kourosh-Arami, M; Lavaie, M; Najafi, Z | 1 |
Haghparast, A; Karimi-Haghighi, S; Mahmoudi, M; Maleki-Roveshti, M | 2 |
Aston-Jones, G; Fragale, JE; James, MH | 1 |
Campus, P; Covelo, IR; Flagel, SB; Haight, JL; Johnson, AM; Klumpner, MS; Kuhn, BN; Maria-Rios, CE; Morrow, JD | 1 |
Assar, N; Azizi, P; Haghparast, A; Katebi, SN; Mahmoudi, D; Mousavi, Z | 1 |
Campbell, EJ; Hill, MK; Jin, S; Lawrence, AJ; Maddern, XJ; Pang, TY | 1 |
Akbari, E; Ardeshiri, MR; Khodabande, F | 1 |
Aghajani, N; Azizi, H; Pourhamzeh, M; Semnanian, S | 1 |
Haghparast, A; Hassanlou, AA; Jamali, S; RayatSanati, K | 1 |
Dong, X; Feng, Z; Liu, H; Lu, G; Tang, Y; Wang, J; Xiong, J; Ye, W; Zhong, L | 1 |
Abbasnejad, M; Askari-Zahabi, K; Esmaeili-Mahani, S; Kooshki, R | 1 |
Haghparast, A; Karimi-Haghighi, S; Zargarani, A | 1 |
Haghparast, A; Jamali, S; Zarrabian, S | 1 |
Abbasnejad, M; Esmaeili-Mahani, S; Kooshki, R; Pourrahimi, AM; Raoof, M | 1 |
Askari, K; Ghalebandi, S; Haghparast, A; Mousavi, Z; Zareie, F | 1 |
Durairaja, A; Fendt, M; Steinecke, CS | 1 |
Alibeik, H; Bananej, M; Khakpai, F; Saadati, N; Zarrindast, MR | 1 |
3 review(s) available for benzoxazoles and urea
Article | Year |
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Orexins and the treatment of obesity.
Topics: Animals; Benzoxazoles; Body Weight; Carrier Proteins; Eating; Humans; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Obesity; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2002 |
[Orexin: clinical and therapeutic implications].
Topics: Animals; Arousal; Azepines; Benzoxazoles; Disease Models, Animal; Drug Evaluation, Preclinical; Feeding and Eating Disorders; Feeding Behavior; Humans; Intracellular Signaling Peptides and Proteins; Mice; Mice, Knockout; Mice, Transgenic; Motor Activity; Naphthyridines; Narcolepsy; Neuropeptides; Obesity; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Sleep Disorders, Circadian Rhythm; Sleep Disorders, Intrinsic; Substance-Related Disorders; Triazoles; Urea | 2014 |
Possible Role of CRF-Hcrt Interaction in the Infralimbic Cortex in the Emergence and Maintenance of Compulsive Alcohol-Seeking Behavior.
Topics: Alcoholism; Animals; Benzoxazoles; Compulsive Behavior; Corticotropin-Releasing Hormone; Drug-Seeking Behavior; Humans; Naphthyridines; Orexins; Prefrontal Cortex; Protein Binding; Urea | 2020 |
326 other study(ies) available for benzoxazoles and urea
Article | Year |
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Heterocyclic substituted ureas. II. Immunosuppressive and antiviral activity of benzothiazole- and benzoxazoleureas.
Topics: Animals; Antibody Formation; Antigen-Antibody Reactions; Antiviral Agents; Benzoxazoles; Chemical Phenomena; Chemistry; Coxsackievirus Infections; Erythrocytes; Immunosuppressive Agents; Mice; Sheep; Thiazoles; Urea | 1969 |
A selective orexin-1 receptor antagonist reduces food consumption in male and female rats.
Topics: Animals; Appetite Depressants; Benzoxazoles; Carrier Proteins; Darkness; Eating; Fasting; Female; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Obesity; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2000 |
Effects of centrally administered orexin-B and orexin-A: a role for orexin-1 receptors in orexin-B-induced hyperactivity.
Topics: Animals; Benzoxazoles; Body Temperature; Brain Chemistry; Carrier Proteins; Grooming; Intracellular Signaling Peptides and Proteins; Motor Activity; Naphthyridines; Neuropeptides; Neurosecretory Systems; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reflex, Startle; Urea | 2001 |
SB-334867-A: the first selective orexin-1 receptor antagonist.
Topics: Animals; Benzoxazoles; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Fluorometry; Humans; Naphthyridines; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Transfection; Urea | 2001 |
SB-334867, a selective orexin-1 receptor antagonist, enhances behavioural satiety and blocks the hyperphagic effect of orexin-A in rats.
Topics: Animals; Appetitive Behavior; Benzoxazoles; Body Weight; Carrier Proteins; Eating; Hyperphagia; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Inbred Strains; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Satiety Response; Urea | 2001 |
Orexin-A, an hypothalamic peptide with analgesic properties.
Topics: Abdomen; Analgesics; Anesthesia, Intravenous; Animals; Behavior, Animal; Benzoxazoles; Carrageenan; Carrier Proteins; Female; Ganglia, Spinal; Hyperalgesia; Hypothalamus; Immunohistochemistry; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred ICR; Naloxone; Naphthyridines; Narcotic Antagonists; Neuropeptides; Nociceptors; Orexin Receptors; Orexins; Pain Threshold; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spinal Cord; Urea | 2001 |
1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor.
Topics: Animals; Benzoxazoles; Blood-Brain Barrier; Central Nervous System; CHO Cells; Cricetinae; Humans; Indoles; Infusions, Intravenous; Naphthyridines; Orexin Receptors; Permeability; Quinolines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sensitivity and Specificity; Structure-Activity Relationship; Urea | 2001 |
SB-334867-A antagonises orexin mediated excitation in the locus coeruleus.
Topics: Action Potentials; Animals; Benzoxazoles; Carrier Proteins; Electrophysiology; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Locus Coeruleus; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Receptors, Neuropeptide; Urea | 2002 |
Anorectic, thermogenic and anti-obesity activity of a selective orexin-1 receptor antagonist in ob/ob mice.
Topics: Adipose Tissue, Brown; Animals; Benzoxazoles; Body Composition; Body Weight; Diabetes Mellitus, Type 2; Disease Models, Animal; Eating; Energy Metabolism; Female; Insulin; Mice; Mice, Inbred Strains; Naphthyridines; Obesity; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; RNA, Messenger; Urea | 2002 |
Analgesic effect of intrathecally administered orexin-A in the rat formalin test and in the rat hot plate test.
Topics: Analgesics, Non-Narcotic; Animals; Benzoxazoles; Carrier Proteins; Dose-Response Relationship, Drug; Immunohistochemistry; Injections, Spinal; Intracellular Signaling Peptides and Proteins; Male; Naloxone; Naphthyridines; Neuropeptides; Orexins; Pain Measurement; Rats; Rats, Sprague-Dawley; Urea | 2002 |
Involvement of cholinergic neurons in orexin-induced contraction of guinea pig ileum.
Topics: Acetylcholine; Animals; Atropine; Benzoxazoles; Carrier Proteins; Enteric Nervous System; Female; Ganglionic Blockers; Guinea Pigs; Hexamethonium; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Parasympathetic Nervous System; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Tetrodotoxin; Urea | 2002 |
Evidence implicating a role for orexin-1 receptor modulation of paradoxical sleep in the rat.
Topics: Animals; Benzoxazoles; Carrier Proteins; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep, REM; Urea | 2003 |
Orexins induce increased excitability and synchronisation of rat sympathetic preganglionic neurones.
Topics: Adrenergic Fibers; Animals; Autonomic Fibers, Preganglionic; Benzoxazoles; Carrier Proteins; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; GTP-Binding Proteins; Hypothalamic Area, Lateral; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Male; Membrane Potentials; Microscopy, Confocal; Microscopy, Video; Naphthyridines; Neural Pathways; Neurons; Neuropeptides; Orexins; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Urea | 2003 |
Central orexin A has site-specific effects on luteinizing hormone release in female rats.
Topics: Animals; Benzoxazoles; Carrier Proteins; Cells, Cultured; Estradiol; Female; Gonadotropin-Releasing Hormone; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Luteinizing Hormone; Microinjections; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Ovariectomy; Preoptic Area; Progesterone; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2003 |
Physiological regulation and NO-dependent inhibition of migrating myoelectric complex in the rat small bowel by OXA.
Topics: Animals; Benzoxazoles; Carrier Proteins; Duodenum; Electromyography; Guanethidine; Homeostasis; Immunohistochemistry; Intestine, Small; Intracellular Signaling Peptides and Proteins; Male; Myoelectric Complex, Migrating; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitroarginine; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea; Vagotomy | 2003 |
Effects of central hypocretin-1 administration on hemodynamic responses in young-adult and middle-aged rats.
Topics: Aging; Animals; Benzoxazoles; Blood Gas Analysis; Blood Pressure; Carrier Proteins; Cerebral Cortex; Chromatography, High Pressure Liquid; Disease Models, Animal; Heart Rate; Hemodynamics; Hemoglobins; In Vitro Techniques; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Norepinephrine; Orexins; Potassium Chloride; Rats; Time Factors; Urea | 2003 |
Antiallodynic effects of intrathecal orexins in a rat model of postoperative pain.
Topics: Animals; Antibodies, Blocking; Benzoxazoles; Carrier Proteins; Exophthalmos; gamma-Aminobutyric Acid; Glycine Agents; Injections, Spinal; Intracellular Signaling Peptides and Proteins; Male; Naloxone; Naphthyridines; Narcotic Antagonists; Neuropeptides; Orexin Receptors; Orexins; Pain Threshold; Pain, Postoperative; Physical Stimulation; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Glycine; Receptors, Neuropeptide; Receptors, Purinergic P2; Strychnine; Suramin; Synaptic Transmission; Urea | 2003 |
Orexinergic neurons and barbiturate anesthesia.
Topics: Animals; Barbiturates; Benzoxazoles; Brain; Carrier Proteins; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Drug Synergism; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Locus Coeruleus; Male; Naphthyridines; Neurons; Neuropeptides; Norepinephrine; Orexin Receptors; Orexins; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, GABA-A; Receptors, Neuropeptide; Urea | 2003 |
Hypocretin-1 causes G protein activation and increases ACh release in rat pons.
Topics: Acetylcholine; Animals; Autoradiography; Benzoxazoles; Carrier Proteins; Dialysis; Dose-Response Relationship, Drug; Drug Interactions; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Pons; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sulfur Isotopes; Time Factors; Urea | 2003 |
Hypothalamus-brain stem circuitry responsible for vagal efferent signaling to the pancreas evoked by hypoglycemia in rat.
Topics: Action Potentials; Animals; Benzoxazoles; Blood Glucose; Brain Stem; Carrier Proteins; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Agonists; Glucose; Hypoglycemia; Hypothalamus; Immunohistochemistry; Insulin; Intracellular Signaling Peptides and Proteins; Kainic Acid; Male; Microinjections; Naphthyridines; Neural Pathways; Neurons, Efferent; Neuropeptide Y; Neuropeptides; Nodose Ganglion; Orexins; Pancreas; Rats; Rats, Sprague-Dawley; Serotonin; Splanchnic Nerves; Urea; Vagus Nerve | 2004 |
Orexin A (hypocretin 1) injected into hypothalamic paraventricular nucleus and spontaneous physical activity in rats.
Topics: Animals; Benzoxazoles; Calorimetry, Indirect; Carbon Dioxide; Carrier Proteins; Dose-Response Relationship, Drug; Feeding Behavior; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Motor Activity; Naphthyridines; Neuropeptides; Orexins; Oxygen Consumption; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Thermogenesis; Urea | 2004 |
Characterisation of the binding of [3H]-SB-674042, a novel nonpeptide antagonist, to the human orexin-1 receptor.
Topics: Animals; Benzoxazoles; CHO Cells; Cricetinae; Humans; Naphthyridines; Orexin Receptors; Protein Binding; Pyrrolidines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Thiazoles; Tritium; Urea | 2004 |
Differential effects of the selective orexin-1 receptor antagonist SB-334867 and lithium chloride on the behavioural satiety sequence in rats.
Topics: Animals; Appetite; Appetite Depressants; Benzoxazoles; Body Weight; Dose-Response Relationship, Drug; Eating; Feeding Behavior; Lithium Chloride; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Inbred Strains; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Satiety Response; Urea | 2004 |
Pharmacological characterisation of the orexin receptor subtype mediating postsynaptic excitation in the rat dorsal raphe nucleus.
Topics: Animals; Benzoxazoles; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Male; Naphthyridines; Orexin Receptors; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2004 |
Hypocretinergic control of spinal cord motoneurons.
Topics: Animals; Benzoxazoles; Carrier Proteins; Cataplexy; Cats; Electric Stimulation; Hypothalamus; Intracellular Signaling Peptides and Proteins; Membrane Potentials; Motor Neurons; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spinal Cord; Sympathomimetics; Urea | 2004 |
Orexin-A (Hypocretin-1) and leptin enhance LTP in the dentate gyrus of rats in vivo.
Topics: Animals; Benzoxazoles; Dentate Gyrus; Dose-Response Relationship, Drug; Intracellular Signaling Peptides and Proteins; Leptin; Long-Term Potentiation; Naphthyridines; Neuropeptides; Orexins; Rats; Rats, Sprague-Dawley; Urea | 2004 |
Anorexia and weight loss in male rats 24 h following single dose treatment with orexin-1 receptor antagonist SB-334867.
Topics: Activity Cycles; Analysis of Variance; Animals; Anorexia; Appetite Depressants; Benzoxazoles; Body Weight; Drug Administration Schedule; Eating; Feeding Behavior; Injections, Intraperitoneal; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Inbred Strains; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Time Factors; Urea; Weight Loss | 2005 |
Satiety enhancement by selective orexin-1 receptor antagonist SB-334867: influence of test context and profile comparison with CCK-8S.
Topics: Analysis of Variance; Animals; Appetite; Behavior, Animal; Benzoxazoles; Body Weight; Drinking; Eating; Food Deprivation; Male; Naphthyridines; Nootropic Agents; Orexin Receptors; Rats; Reaction Time; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Satiety Response; Sincalide; Time Factors; Urea | 2005 |
Spinal orexin-1 receptors mediate anti-hyperalgesic effects of intrathecally-administered orexins in diabetic neuropathic pain model rats.
Topics: Animals; Behavior, Animal; Benzoxazoles; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Dose-Response Relationship, Drug; Drug Interactions; Hyperalgesia; Injections, Spinal; Intracellular Signaling Peptides and Proteins; Male; Naloxone; Naphthyridines; Narcotic Antagonists; Neuropeptides; Orexin Receptors; Orexins; Pain Measurement; Pain Threshold; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spinal Cord; Streptozocin; Time Factors; Urea | 2005 |
Effect of a selective OX1R antagonist on food intake and body weight in two strains of rats that differ in susceptibility to dietary-induced obesity.
Topics: Animals; Benzoxazoles; Body Weight; Diet; Eating; Gene Expression Regulation; Hypothalamus; Male; Naphthyridines; Obesity; Orexin Receptors; Protein Precursors; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; RNA, Messenger; Species Specificity; Urea | 2005 |
Orexin A in the nucleus accumbens stimulates feeding and locomotor activity.
Topics: Animals; Benzoxazoles; Feeding Behavior; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Motor Activity; Naphthyridines; Neuropeptides; Nucleus Accumbens; Orexins; Rats; Rats, Sprague-Dawley; Urea | 2005 |
Lack of interaction between orexinergic and alpha2-adrenergic neuronal systems in rat cerebrocortical slices.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzoxazoles; Cerebral Cortex; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Intracellular Signaling Peptides and Proteins; Locus Coeruleus; Male; Naphthyridines; Neural Pathways; Neurons; Neuropeptides; Norepinephrine; Orexin Receptors; Orexins; Organ Culture Techniques; Potassium; Rats; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep; Urea; Wakefulness; Yohimbine | 2005 |
Role for hypocretin in mediating stress-induced reinstatement of cocaine-seeking behavior.
Topics: Analysis of Variance; Animals; Behavior, Addictive; Benzoxazoles; Brain; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Intracellular Signaling Peptides and Proteins; Male; Models, Statistical; Naphthyridines; Neuropeptides; Orexins; Rats; Rats, Wistar; Reward; Self Administration; Time Factors; Urea | 2005 |
Direct involvement of orexinergic systems in the activation of the mesolimbic dopamine pathway and related behaviors induced by morphine.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Desipramine; Dopamine; Female; Haloperidol; Injections, Intraventricular; Injections, Subcutaneous; Intracellular Signaling Peptides and Proteins; Limbic System; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Knockout; Microdialysis; Microinjections; Morphine; Motor Activity; Naphthyridines; Neuropeptides; Nucleus Accumbens; Orexins; Oxidopamine; Protein Precursors; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Reward; RNA, Messenger; Tyrosine 3-Monooxygenase; Urea; Ventral Tegmental Area | 2006 |
Orexin-A is composed of a highly conserved C-terminal and a specific, hydrophilic N-terminal region, revealing the structural basis of specific recognition by the orexin-1 receptor.
Topics: Amino Acid Sequence; Benzoxazoles; Binding Sites; Conserved Sequence; Humans; Hydrophobic and Hydrophilic Interactions; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Micelles; Models, Molecular; Molecular Sequence Data; Naphthyridines; Neuropeptides; Nuclear Magnetic Resonance, Biomolecular; Orexin Receptors; Orexins; Protein Conformation; Protein Structure, Secondary; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2006 |
Orexin A in the VTA is critical for the induction of synaptic plasticity and behavioral sensitization to cocaine.
Topics: Analysis of Variance; Anesthetics, Local; Animals; Animals, Newborn; Behavior, Animal; Benzoxazoles; Calcium Channel Blockers; Cocaine; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Immunohistochemistry; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Lysine; Male; Motor Activity; N-Methylaspartate; Naphthyridines; Neuronal Plasticity; Neurons; Neuropeptides; Orexins; Patch-Clamp Techniques; Protein Kinase C; Quinoxalines; Rats; Rats, Sprague-Dawley; Synapses; Thionucleotides; Time Factors; Tyrosine 3-Monooxygenase; Urea; Ventral Tegmental Area | 2006 |
Orexins increase cortical acetylcholine release and electroencephalographic activation through orexin-1 receptor in the rat basal forebrain during isoflurane anesthesia.
Topics: Acetylcholine; Anesthetics, Inhalation; Animals; Arousal; Basal Ganglia; Benzoxazoles; Cerebral Cortex; Electric Stimulation; Electroencephalography; Intracellular Signaling Peptides and Proteins; Isoflurane; Male; Microdialysis; Microinjections; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Prosencephalon; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2006 |
The orexin system regulates alcohol-seeking in rats.
Topics: Alcohol Drinking; Animals; Benzoxazoles; Conditioning, Operant; Cues; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexins; Rats; RNA, Messenger; Urea; Ventral Tegmental Area | 2006 |
Orexin A affects ascending contraction depending on downstream cholinergic neurons and descending relaxation through independent pathways in mouse jejunum.
Topics: Acetylcholine; Animals; Arginine; Benzoxazoles; Drug Interactions; Enzyme Inhibitors; Hexamethonium; Immunohistochemistry; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Jejunum; Male; Mice; Mice, Inbred ICR; Models, Biological; Muscle Contraction; Naphthyridines; Neural Pathways; Neurons; Neuropeptides; Nicotinic Antagonists; Nitroarginine; Orexins; Urea | 2006 |
Functional inactivation of orexin 1 receptors in CA1 region impairs acquisition, consolidation and retrieval in Morris water maze task.
Topics: Analysis of Variance; Animals; Benzoxazoles; Discrimination Learning; Dose-Response Relationship, Drug; Escape Reaction; Hippocampus; Intracellular Signaling Peptides and Proteins; Male; Maze Learning; Mental Recall; Microinjections; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Wistar; Reaction Time; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spatial Behavior; Urea | 2006 |
Hypocretin-1 dose-dependently modulates maternal behaviour in mice.
Topics: Aggression; Analysis of Variance; Animals; Behavior, Animal; Benzoxazoles; Dose-Response Relationship, Drug; Female; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Lactation; Maternal Behavior; Mice; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Proto-Oncogene Proteins c-fos; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2006 |
The orexin-1 receptor antagonist SB-334867 blocks the effects of antipsychotics on the activity of A9 and A10 dopamine neurons: implications for antipsychotic therapy.
Topics: Action Potentials; Analysis of Variance; Animals; Antipsychotic Agents; Benzodiazepines; Benzoxazoles; Brain; Dopamine; Drug Interactions; Haloperidol; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Olanzapine; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Time Factors; Urea | 2007 |
Modulation of nociceptive dural input to the trigeminal nucleus caudalis via activation of the orexin 1 receptor in the rat.
Topics: Action Potentials; Afferent Pathways; Animals; Benzoxazoles; Dose-Response Relationship, Drug; Drug Interactions; Facial Nerve; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neural Inhibition; Neurons; Neuropeptides; Nociceptors; Orexin Receptors; Orexins; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Skin; Trigeminal Caudal Nucleus; Trigeminal Nerve; Urea | 2006 |
The selective orexin 1 receptor antagonist SB-334867-A impairs acquisition and consolidation but not retrieval of spatial memory in Morris water maze.
Topics: Animals; Benzoxazoles; Dentate Gyrus; Male; Maze Learning; Memory; Microinjections; Naphthyridines; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spatial Behavior; Swimming; Urea | 2007 |
The effect of orexins on intestinal motility in vitro in fed and fasted rats.
Topics: Animals; Atropine; Benzoxazoles; Drug Interactions; Fasting; Gastrointestinal Motility; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Jejunum; Male; Muscle Contraction; Naphthyridines; Neuropeptides; Orexins; Random Allocation; Rats; Rats, Wistar; Tetrodotoxin; Urea | 2006 |
Role of dorsal vagal motor nucleus orexin-receptor-1 in glycemic responses to acute versus repeated insulin administration.
Topics: Animals; Benzoxazoles; Blood Glucose; Glucagon; Hypoglycemia; Hypoglycemic Agents; Insulin; Intracellular Signaling Peptides and Proteins; Male; Motor Neurons; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Orexin Receptors; Orexins; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Signal Transduction; Urea; Vagus Nerve | 2007 |
Disinhibition of perifornical hypothalamic neurones activates noradrenergic neurones and blocks pontine carbachol-induced REM sleep-like episodes in rats.
Topics: Animals; Benzoxazoles; Bicuculline; Carbachol; Fornix, Brain; GABA Antagonists; Hypothalamus; Injections; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neural Inhibition; Neurons; Neuropeptides; Norepinephrine; Orexin Receptors; Orexins; Pons; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep, REM; Urea | 2007 |
Food-induced expression of orexin receptors in rat duodenal mucosa regulates the bicarbonate secretory response to orexin-A.
Topics: Animals; Atropine; Benzoxazoles; Bethanechol; Bicarbonates; Cerebral Ventricles; Crosses, Genetic; Dose-Response Relationship, Drug; Duodenum; Eating; Food Deprivation; Hydrogen-Ion Concentration; Infusions, Intra-Arterial; Intestinal Mucosa; Intestinal Secretions; Intracellular Signaling Peptides and Proteins; Male; Muscarinic Agonists; Muscarinic Antagonists; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Inbred Lew; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; RNA, Messenger; Time Factors; Up-Regulation; Urea | 2007 |
Both orexin receptors are expressed in rat ovaries and fluctuate with the estrous cycle: effects of orexin receptor antagonists on gonadotropins and ovulation.
Topics: Animals; Benzoxazoles; Dioxanes; Eating; Estrous Cycle; Female; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Gonadotropins; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Ovary; Ovulation; Pentobarbital; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; RNA, Messenger; Urea | 2007 |
The orexin-1 antagonist SB-334867 blocks antipsychotic treatment emergent catalepsy: implications for the treatment of extrapyramidal symptoms.
Topics: Animals; Antipsychotic Agents; Basal Ganglia Diseases; Behavior, Animal; Benzodiazepines; Benzoxazoles; Catalepsy; Haloperidol; Intracellular Signaling Peptides and Proteins; Locomotion; Male; Naphthyridines; Neuropeptides; Olanzapine; Orexins; Prolactin; Rats; Rats, Sprague-Dawley; Risperidone; Urea | 2007 |
Contribution of orexin in hypercapnic chemoreflex: evidence from genetic and pharmacological disruption and supplementation studies in mice.
Topics: Animals; Benzoxazoles; Carbon Dioxide; Chemoreceptor Cells; Disease Models, Animal; Electroencephalography; Electromyography; Hypercapnia; Hypothalamus; Hypoxia; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Pulmonary Ventilation; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reflex; Time Factors; Urea; Wakefulness | 2007 |
Food-elicited increases in cortical acetylcholine release require orexin transmission.
Topics: Acetylcholine; Animals; Benzoxazoles; Cerebral Cortex; Food; Food Deprivation; Hypothalamic Hormones; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Male; Melanins; Microdialysis; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Pituitary Hormones; Prosencephalon; Rats; Rats, Inbred F344; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Synaptic Transmission; Urea | 2007 |
The effect of antagonization of orexin 1 receptors in CA1 and dentate gyrus regions on memory processing in passive avoidance task.
Topics: Animals; Avoidance Learning; Benzoxazoles; Data Interpretation, Statistical; Dentate Gyrus; Dimethyl Sulfoxide; Hippocampus; Male; Memory; Microinjections; Naphthyridines; Orexin Receptors; Psychomotor Performance; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2008 |
Role of orexin receptors in the nucleus accumbens in dopamine-dependent turning behaviour of rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Behavior, Animal; Benzoxazoles; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Functional Laterality; Intracellular Signaling Peptides and Proteins; Male; Motor Activity; Naphthyridines; Neuropeptides; Nucleus Accumbens; Orexin Receptors; Orexins; Quinpirole; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Rotation; Urea | 2008 |
Role of the orexinergic system in acute haemorrhage in the rat.
Topics: Animals; Arterioles; Benzoxazoles; Blood Pressure; Catecholamines; Cerebrovascular Circulation; Heart Rate; Hypotension; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Shock, Hemorrhagic; Sympathetic Nervous System; Up-Regulation; Urea; Vasoconstriction | 2008 |
Differential effects of the hypocretin 1 receptor antagonist SB 334867 on high-fat food self-administration and reinstatement of food seeking in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Benzoxazoles; Caloric Restriction; Conditioning, Operant; Dietary Fats; Dose-Response Relationship, Drug; Eating; Extinction, Psychological; Feeding Behavior; Injections, Intraventricular; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Long-Evans; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Stress, Psychological; Time Factors; Urea; Yohimbine | 2008 |
Use of N-methylpiperazine for the preparation of piperazine-based unsymmetrical bis-ureas as anti-HIV agents.
Topics: Anti-HIV Agents; Benzoxazoles; Carbamates; Cell Line; Cell Survival; HIV Protease; HIV Protease Inhibitors; Humans; Lymphocytes; Methylation; Piperazine; Piperazines; Structure-Activity Relationship; Urea | 2008 |
Reinvestigation of the effect of orexin A on catecholamine release from adrenal chromaffin cells.
Topics: Adrenal Glands; Animals; Benzoxazoles; Catecholamines; Cells, Cultured; Chromaffin Cells; Dose-Response Relationship, Drug; Electrochemistry; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexins; Potassium; Rats; Sympathomimetics; Urea | 2008 |
Orexin mediates the expression of precipitated morphine withdrawal and concurrent activation of the nucleus accumbens shell.
Topics: Analysis of Variance; Animals; Benzoxazoles; Intracellular Signaling Peptides and Proteins; Locus Coeruleus; Male; Mice; Mice, Inbred C57BL; Morphine; Naloxone; Naphthyridines; Narcotic Antagonists; Narcotics; Neuropeptides; Nucleus Accumbens; Orexins; Proto-Oncogene Proteins c-fos; Stilbamidines; Substance Withdrawal Syndrome; Urea; Ventral Tegmental Area | 2008 |
Orexins stimulate steroidogenic acute regulatory protein expression through multiple signaling pathways in human adrenal H295R cells.
Topics: Adrenal Glands; Benzoxazoles; Cell Line; Cell Proliferation; Dose-Response Relationship, Drug; Gene Expression Regulation; Genes, Dominant; GTP-Binding Proteins; Humans; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Peptide Fragments; Phosphoproteins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Signal Transduction; Steroids; Urea | 2008 |
Inhibition of orexin-1/hypocretin-1 receptors inhibits yohimbine-induced reinstatement of ethanol and sucrose seeking in Long-Evans rats.
Topics: Adrenergic alpha-Antagonists; Alcoholism; Animals; Benzoxazoles; Conditioning, Operant; Dose-Response Relationship, Drug; Extinction, Psychological; Male; Motivation; Motor Activity; Naphthyridines; Orexin Receptors; Rats; Rats, Long-Evans; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Sucrose; Taste; Urea; Yohimbine | 2008 |
Orexin-2 receptors inhibit primary afferent fiber-evoked responses of ventral roots in the neonatal rat isolated spinal cord.
Topics: Analysis of Variance; Animals; Animals, Newborn; Benzoxazoles; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Naphthyridines; Nerve Fibers; Neural Inhibition; Neurons, Afferent; Neuropeptides; Orexin Receptors; Orexins; Protein Binding; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Spinal Cord; Spinal Nerve Roots; Urea | 2008 |
Role of orexin input in the diurnal rhythm of locus coeruleus impulse activity.
Topics: Action Potentials; Animals; Axons; Benzoxazoles; Circadian Rhythm; Dorsomedial Hypothalamic Nucleus; Intracellular Signaling Peptides and Proteins; Locus Coeruleus; Male; Microinjections; Naphthyridines; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Synaptic Transmission; Urea; Wakefulness | 2008 |
Orexin A attenuates unconditioned sexual motivation in male rats.
Topics: Animals; Benzoxazoles; Female; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Motivation; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Ovariectomy; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sexual Behavior, Animal; Stereotaxic Techniques; Urea | 2009 |
I.c.v. administration of orexin-A induces an antidepressive-like effect through hippocampal cell proliferation.
Topics: Analysis of Variance; Animals; Benzoxazoles; Bromodeoxyuridine; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Doublecortin Protein; Embryo, Mammalian; Exploratory Behavior; Hippocampus; Immobility Response, Tonic; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Mice; Naphthyridines; Nerve Tissue Proteins; Neurogenesis; Neuropeptide Y; Neuropeptides; Neurotransmitter Agents; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Stem Cells; Urea | 2008 |
Orexin affects dorsal root ganglion neurons: a mechanism for regulating the spinal nociceptive processing.
Topics: Action Potentials; Animals; Benzoxazoles; Calcium Signaling; Ganglia, Spinal; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Pain; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Synaptic Transmission; Urea | 2008 |
Insular hypocretin transmission regulates nicotine reward.
Topics: Animals; Benzoxazoles; Cerebral Cortex; Intracellular Signaling Peptides and Proteins; Male; Motivation; Naphthyridines; Neuropeptides; Nicotine; Nicotinic Agonists; Orexin Receptors; Orexins; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Self Administration; Smoking; Synaptic Transmission; Tobacco Use Disorder; Urea | 2008 |
Short food deprivation inhibits orexin receptor 1 expression and orexin-A induced intracellular calcium signaling in acutely isolated duodenal enterocytes.
Topics: Animals; Atropine; Benzoxazoles; Biopsy; Calcium Signaling; Duodenum; Enterocytes; Fluorescent Dyes; Food Deprivation; Fura-2; Humans; In Vitro Techniques; Intestinal Mucosa; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Parasympatholytics; Rats; Rats, Inbred Lew; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reverse Transcriptase Polymerase Chain Reaction; Urea | 2009 |
Evidence for a modulatory role of orexin A on the nitrergic neurotransmission in the mouse gastric fundus.
Topics: Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Electrophysiology; Female; Gastric Fundus; Guanethidine; Guanylate Cyclase; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthyridines; Neuropeptides; NG-Nitroarginine Methyl Ester; Nitric Oxide; Orexins; Oxytocin; Papaverine; Synaptic Transmission; Tetrodotoxin; Urea; Vasoactive Intestinal Peptide | 2009 |
Orexin A decreases ketamine-induced anesthesia time in the rat: the relevance to brain noradrenergic neuronal activity.
Topics: Anesthesia; Anesthetics, Dissociative; Animals; Benzoxazoles; Brain; Cerebral Cortex; In Vitro Techniques; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Ketamine; Male; Microdialysis; Naphthyridines; Neurons; Neuropeptides; Norepinephrine; Orexins; Rats; Receptors, Neuropeptide; Urea | 2009 |
Role of the ventromedial hypothalamic orexin-1 receptors in regulation of gastric Acid secretion in conscious rats.
Topics: Animals; Atropine; Benzoxazoles; Consciousness; Gastric Acid; Gastric Mucosa; Hypothalamus; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Parasympatholytics; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2009 |
Orexin type 1 receptor antagonist SB 334867 inhibits the central histamine-induced resuscitating effect in rats subjected to haemorrhagic shock.
Topics: Animals; Benzoxazoles; Blood Pressure; Heart Rate; Histamine; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Regional Blood Flow; Resuscitation; Shock, Hemorrhagic; Urea | 2009 |
Antagonism of orexin receptor-1 in the retrotrapezoid nucleus inhibits the ventilatory response to hypercapnia predominantly in wakefulness.
Topics: Animals; Benzoxazoles; Hypercapnia; Male; Naphthyridines; Neural Inhibition; Orexin Receptors; Pulmonary Ventilation; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Respiratory Center; Urea; Wakefulness | 2009 |
The effects of benzodiazepines on urotensin II-stimulated norepinephrine release from rat cerebrocortical slices.
Topics: Animals; Benzodiazepines; Benzoxazoles; Calcium Signaling; Cell Line; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Hypnotics and Sedatives; In Vitro Techniques; Male; Midazolam; Naphthyridines; Norepinephrine; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, GABA-A; Receptors, Neuropeptide; Transfection; Urea; Urotensins | 2009 |
Persistent increase of alcohol-seeking evoked by neuropeptide S: an effect mediated by the hypothalamic hypocretin system.
Topics: Alcohol Drinking; Analysis of Variance; Animals; Benzoxazoles; Central Nervous System Depressants; Conditioning, Classical; Cues; Disease Models, Animal; Ethanol; Hypothalamus; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Substance-Related Disorders; Urea | 2009 |
The role of spinal orexin-1 receptors in posterior hypothalamic modulation of neuropathic pain.
Topics: Analgesics; Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Female; Hypothalamus; Naphthyridines; Neurons; Orexin Receptors; Pain; Pain Measurement; Posterior Horn Cells; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sciatic Neuropathy; Spinal Cord; Urea | 2009 |
Orexin-stimulated MAP kinase cascades are activated through multiple G-protein signalling pathways in human H295R adrenocortical cells: diverse roles for orexins A and B.
Topics: Adrenal Cortex; Benzoxazoles; Blotting, Western; Cell Line; Dose-Response Relationship, Drug; Enzyme Activation; GTP-Binding Proteins; Humans; Hydrocortisone; Intracellular Signaling Peptides and Proteins; Mitogen-Activated Protein Kinases; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; p38 Mitogen-Activated Protein Kinases; Protein Isoforms; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Signal Transduction; Urea | 2009 |
Orexin A modulates neuronal activity of the rodent suprachiasmatic nucleus in vitro.
Topics: Animals; Benzoxazoles; Cells, Cultured; Central Nervous System Agents; Circadian Rhythm; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Mice; Mice, Inbred C57BL; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sodium Channel Blockers; Suprachiasmatic Nucleus; Tetrodotoxin; Time Factors; Urea | 2009 |
Orexins activates protein kinase C-mediated Ca(2+) signaling in isolated rat primary sensory neurons.
Topics: Animals; Benzoxazoles; Calcium Signaling; Cells, Cultured; Ganglia, Spinal; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Nociceptors; Orexins; Pain; Protein Kinase C; Rats; Rats, Wistar; Sensory Receptor Cells; Urea | 2010 |
Systemic and intrabasalis administration of the orexin-1 receptor antagonist, SB-334867, disrupts attentional performance in rats.
Topics: Analysis of Variance; Animals; Attention; Behavior, Animal; Benzoxazoles; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Administration Routes; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Long-Evans; Reaction Time; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Time Factors; Urea | 2009 |
Orexin/hypocretin is necessary for context-driven cocaine-seeking.
Topics: Analysis of Variance; Animals; Benzoxazoles; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Disease Models, Animal; Extinction, Psychological; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement, Psychology; Self Administration; Time Factors; Urea | 2010 |
Orexin-A acts on the paraventricular nucleus of the midline thalamus to inhibit locomotor activity in rats.
Topics: Animals; Arousal; Behavior, Animal; Benzoxazoles; Grooming; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Midline Thalamic Nuclei; Morphine; Motor Activity; Naphthyridines; Narcotics; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sympathomimetics; Urea | 2009 |
Orexin/hypocretin signaling at the orexin 1 receptor regulates cue-elicited cocaine-seeking.
Topics: Animals; Behavior, Addictive; Benzoxazoles; Brain; Cocaine; Cocaine-Related Disorders; Cues; Dopamine Uptake Inhibitors; Extinction, Psychological; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement, Psychology; Signal Transduction; Urea | 2009 |
Orexin-1 receptor antagonism decreases ethanol consumption and preference selectively in high-ethanol--preferring Sprague--Dawley rats.
Topics: Alcohol Drinking; Animals; Benzoxazoles; Ethanol; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Urea | 2009 |
The orexin-1 receptor antagonist SB-334867 reduces amphetamine-evoked dopamine outflow in the shell of the nucleus accumbens and decreases the expression of amphetamine sensitization.
Topics: Amphetamine; Amphetamine-Related Disorders; Animals; Benzoxazoles; Dopamine; Dopamine Uptake Inhibitors; Extracellular Fluid; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Microdialysis; Naphthyridines; Neural Pathways; Neuropeptides; Nucleus Accumbens; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Synaptic Transmission; Urea | 2010 |
Orexin A/hypocretin-1 selectively promotes motivation for positive reinforcers.
Topics: Animals; Benzoxazoles; Choice Behavior; Cocaine-Related Disorders; Dietary Fats; Intracellular Signaling Peptides and Proteins; Male; Motivation; Naphthyridines; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement, Psychology; Urea | 2009 |
Halothane-induced hypnosis is not accompanied by inactivation of orexinergic output in rodents.
Topics: Anesthesia, General; Anesthetics, Inhalation; Animals; Benzoxazoles; Circadian Rhythm; Halothane; Hypothalamus; Intracellular Signaling Peptides and Proteins; Isoflurane; Locus Coeruleus; Male; Mice; Mice, Inbred C57BL; Naphthyridines; Neuropeptides; Norepinephrine; Orexins; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Urea | 2009 |
The modulation of orexin A on HCN currents of pyramidal neurons in mouse prelimbic cortex.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Benzoxazoles; Biophysics; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Membrane Potentials; Mice; Mice, Inbred Strains; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Orexin Receptors; Orexins; Patch-Clamp Techniques; Pyramidal Cells; Pyrimidines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sodium Channel Blockers; Tetrodotoxin; Urea | 2010 |
Orexins excite neurons of the rat cerebellar nucleus interpositus via orexin 2 receptors in vitro.
Topics: Action Potentials; Animals; Benzoxazoles; Cerebellar Nuclei; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Organ Culture Techniques; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2010 |
The orexin receptor 1 (OX1R) in the rostral medullary raphe contributes to the hypercapnic chemoreflex in wakefulness, during the active period of the diurnal cycle.
Topics: Analysis of Variance; Animals; Benzoxazoles; Body Temperature; Chemoreceptor Cells; Circadian Rhythm; Electroencephalography; Electromyography; Hypercapnia; Male; Microdialysis; Naphthyridines; Orexin Receptors; Oxygen Consumption; Pulmonary Ventilation; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep Stages; Urea; Wakefulness | 2010 |
Thermal nociception is decreased by hypocretin-1 and an adenosine A1 receptor agonist microinjected into the pontine reticular formation of Sprague Dawley rat.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Aging; Animals; Benzoxazoles; Hot Temperature; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Pain; Pain Measurement; Pons; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reticular Formation; Time Factors; Urea | 2010 |
Orexin mediates morphine place preference, but not morphine-induced hyperactivity or sensitization.
Topics: Animals; Benzoxazoles; Central Nervous System Agents; Cocaine; Conditioning, Classical; Dopamine Uptake Inhibitors; Female; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Motor Activity; Mutation; Naphthyridines; Narcotics; Neuropeptides; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Space Perception; Time Factors; Urea | 2010 |
Ghrelin increases the rewarding value of high-fat diet in an orexin-dependent manner.
Topics: Animals; Benzoxazoles; Brain; Conditioning, Operant; Dietary Fats; Food Preferences; Ghrelin; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naphthyridines; Neuropeptides; Orexins; Proto-Oncogene Proteins c-fos; Receptors, Ghrelin; Reward; Signal Transduction; Urea | 2010 |
The hypocretin-orexin system regulates cocaine self-administration via actions on the mesolimbic dopamine system.
Topics: Animals; Benzoxazoles; Cocaine; Dopamine; Electrochemistry; Intracellular Signaling Peptides and Proteins; Limbic System; Male; Mesencephalon; Mice; Microdialysis; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Signal Transduction; Urea | 2010 |
Hypocretins regulate the anxiogenic-like effects of nicotine and induce reinstatement of nicotine-seeking behavior.
Topics: Animals; Anxiety; Arginine Vasopressin; Behavior, Addictive; Benzoxazoles; Conditioning, Operant; Corticotropin-Releasing Hormone; Extinction, Psychological; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Naphthyridines; Neurons; Neuropeptides; Nicotine; Orexin Receptors; Orexins; Paraventricular Hypothalamic Nucleus; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Tobacco Use Disorder; Urea | 2010 |
The role of orexin-A in food motivation, reward-based feeding behavior and food-induced neuronal activation in rats.
Topics: Animals; Benzoxazoles; Brain; Cacao; Central Nervous System Agents; Cues; Dietary Fats; Eating; Feeding Behavior; Food; Intracellular Signaling Peptides and Proteins; Male; Motivation; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Long-Evans; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Urea | 2010 |
Nicotine self-administration in the rat: effects of hypocretin antagonists and changes in hypocretin mRNA.
Topics: Acetamides; Animals; Arcuate Nucleus of Hypothalamus; Behavior, Animal; Benzoxazoles; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Hypothalamus; Infusions, Intravenous; Intracellular Signaling Peptides and Proteins; Isoquinolines; Male; Naphthyridines; Neuropeptides; Nicotine; Nicotinic Agonists; Orexin Receptors; Orexins; Rats; Rats, Long-Evans; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement, Psychology; RNA, Messenger; Self Administration; Urea | 2010 |
Orexin signaling via the orexin 1 receptor mediates operant responding for food reinforcement.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Data Interpretation, Statistical; Food; Hypothalamic Area, Lateral; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Receptors, Neuropeptide; Reinforcement Schedule; Reinforcement, Psychology; RNA Interference; Urea; Viruses | 2010 |
Endogenous orexin-A modulates gastric motility by peripheral mechanisms in rats.
Topics: Animals; Benzoxazoles; Fasting; Gastric Emptying; Gastrointestinal Motility; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Up-Regulation; Urea; Vagus Nerve | 2010 |
Opposite roles of dopamine and orexin in quinpirole-induced excessive drinking: a rat model of psychotic polydipsia.
Topics: Animals; Benzoxazoles; Cerebral Cortex; Conditioning, Operant; Corticosterone; Disease Models, Animal; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking; Drug Synergism; Haloperidol; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexins; Psychotic Disorders; Quinpirole; Rats; Rats, Sprague-Dawley; Urea | 2010 |
Glutamatergic regulation of ghrelin-induced activation of the mesolimbic dopamine system.
Topics: 2-Amino-5-phosphonovalerate; Alcoholism; Animals; Benzoxazoles; Dopamine; Ghrelin; Limbic System; Male; Mesencephalon; Mice; Mice, Inbred Strains; Motor Activity; Naltrexone; Naphthyridines; Narcotic Antagonists; Nerve Net; Nucleus Accumbens; Orexin Receptors; Peptide Hormones; Receptors, G-Protein-Coupled; Receptors, N-Methyl-D-Aspartate; Receptors, Neuropeptide; Signal Transduction; Urea; Ventral Tegmental Area | 2011 |
Antagonism of orexin type 1 receptors in the locus coeruleus attenuates signs of naloxone-precipitated morphine withdrawal in rats.
Topics: Animals; Benzoxazoles; Injections, Intraventricular; Locus Coeruleus; Male; Morphine; Morphine Dependence; Naloxone; Naphthyridines; Narcotic Antagonists; Narcotics; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Substance Withdrawal Syndrome; Urea | 2010 |
The endogenous actions of hypothalamic peptides on brown adipose tissue thermogenesis in the rat.
Topics: Adipose Tissue, Brown; Animals; Benzoxazoles; Blotting, Western; Body Weight; Eating; Energy Metabolism; Hypothalamic Hormones; Ion Channels; Male; Melanins; Melanocyte-Stimulating Hormones; Mitochondrial Proteins; Naphthyridines; Orexin Receptors; Piperidines; Pituitary Hormones; Pyrimidines; Random Allocation; Rats; Rats, Sprague-Dawley; Receptor, Melanocortin, Type 3; Receptor, Melanocortin, Type 4; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Thermogenesis; Uncoupling Protein 1; Urea | 2010 |
Central orexin-A increases gastric motility in rats.
Topics: Animals; Benzoxazoles; Gastric Emptying; Gastrointestinal Motility; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexins; Postprandial Period; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stress, Physiological; Urea | 2010 |
Orexin-1 receptor mediates long-term potentiation in the dentate gyrus area of freely moving rats.
Topics: Analysis of Variance; Animals; Benzoxazoles; Dentate Gyrus; Electric Stimulation; Electrophysiology; Long-Term Potentiation; Male; Naphthyridines; Neurons; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Synapses; Urea | 2011 |
Chemical stimulation of the lateral hypothalamus induces conditioned place preference in rats: Involvement of OX1 and CB1 receptors in the ventral tegmental area.
Topics: Animals; Benzoxazoles; Carbachol; Choice Behavior; Conditioning, Operant; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Male; Naphthyridines; Neural Pathways; Orexin Receptors; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor Cross-Talk; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Urea; Ventral Tegmental Area | 2011 |
Orexins in the midline thalamus are involved in the expression of conditioned place aversion to morphine withdrawal.
Topics: Animals; Avoidance Learning; Benzoxazoles; Conditioning, Classical; Disease Models, Animal; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Midline Thalamic Nuclei; Morphine; Naloxone; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Substance Withdrawal Syndrome; Urea | 2011 |
Discrete cue-conditioned alcohol-seeking after protracted abstinence: pattern of neural activation and involvement of orexin₁ receptors.
Topics: Alcohol Deterrents; Alcohol Drinking; Alcoholism; Animals; Behavior, Animal; Benzoxazoles; Brain; Conditioning, Operant; Cues; Male; Naphthyridines; Nerve Tissue Proteins; Neurons; Orexin Receptors; Organ Specificity; Proto-Oncogene Proteins c-fos; Rats; Rats, Inbred Strains; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Temperance; Urea | 2011 |
Intrathecal orexin A increases sympathetic outflow and respiratory drive, enhances baroreflex sensitivity and blocks the somato-sympathetic reflex.
Topics: Anesthesia, Spinal; Animals; Baroreflex; Benzoxazoles; Evoked Potentials, Somatosensory; Injections, Spinal; Intracellular Signaling Peptides and Proteins; Kinetics; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Peripheral Nervous System; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Respiration; Splanchnic Nerves; Sympathetic Nervous System; Tachycardia; Urea; Vagotomy | 2011 |
Hypocretin and GABA interact in the pontine reticular formation to increase wakefulness.
Topics: Analysis of Variance; Animals; Behavior, Animal; Benzoxazoles; Bicuculline; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Intracellular Signaling Peptides and Proteins; Isotonic Solutions; Male; Microinjections; Naphthyridines; Neuropeptides; Orexins; Pons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reticular Formation; Ringer's Solution; Sleep Stages; Urea; Wakefulness | 2010 |
Involvement of the orexin/hypocretin system in ethanol conditioned place preference.
Topics: Animals; Behavior, Animal; Benzoxazoles; Conditioning, Classical; Drug-Seeking Behavior; Ethanol; Intracellular Signaling Peptides and Proteins; Male; Mice; Mice, Inbred DBA; Motor Activity; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reward; Self Administration; Urea | 2011 |
Effects of orexin-A on propofol anesthesia in rats.
Topics: Anesthesia, Intravenous; Anesthetics, Intravenous; Animals; Benzoxazoles; Dopamine; Electroencephalography; Infusions, Intravenous; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Microdialysis; Naphthyridines; Neuropeptides; Norepinephrine; Orexin Receptors; Orexins; Postural Balance; Prefrontal Cortex; Propofol; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reflex; Urea | 2011 |
Ligand-induced internalization of the orexin OX(1) and cannabinoid CB(1) receptors assessed via N-terminal SNAP and CLIP-tagging.
Topics: Alkyl and Aryl Transferases; Benzoxazoles; Cell Line; Cell Membrane; Cloning, Molecular; Cyclohexanols; Extracellular Signal-Regulated MAP Kinases; Humans; Intracellular Signaling Peptides and Proteins; Ligands; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Phenylurea Compounds; Phosphorylation; Piperidines; Plasmids; Pyrazoles; Pyrrolidines; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Rimonabant; Thiazoles; Urea | 2011 |
Orexin-1 receptor antagonist SB-334867 reduces the acquisition and expression of cocaine-conditioned reinforcement and the expression of amphetamine-conditioned reward.
Topics: Animals; Behavior, Animal; Benzoxazoles; Cocaine; Conditioning, Operant; Cues; Dextroamphetamine; Discrimination Learning; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement Schedule; Reward; Self Administration; Urea | 2011 |
SB-334867-A, a selective orexin-1 receptor antagonist, enhances taste aversion learning and blocks taste preference learning in rats.
Topics: Animals; Avoidance Learning; Benzoxazoles; Body Weight; Dose-Response Relationship, Drug; Feeding Behavior; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Taste; Urea | 2011 |
A role for orexin in central vestibular motor control.
Topics: Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Benzoxazoles; Drug Interactions; Electric Stimulation; Exploratory Behavior; Hindlimb Suspension; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Membrane Potentials; Microinjections; Motor Activity; Naphthyridines; Neurons; Neuropeptides; Orexins; Patch-Clamp Techniques; Psychomotor Performance; Rats; Receptors, Neuropeptide; Sodium-Calcium Exchanger; Thiourea; Urea; Vestibular Nucleus, Lateral | 2011 |
Intraventricular administration of neuropeptide S has reward-like effects.
Topics: Animals; Behavior, Animal; Benzazepines; Benzoxazoles; Conditioning, Psychological; Dopamine Antagonists; Injections, Intraventricular; Locomotion; Male; Naphthyridines; Neuropeptides; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Neuropeptide; Reward; Self Administration; Urea | 2011 |
Hcrtr1 and 2 signaling differentially regulates depression-like behaviors.
Topics: Animals; Anxiety; Benzoxazoles; Choice Behavior; Depression; Disease Models, Animal; Immobility Response, Tonic; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Naphthyridines; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Signal Transduction; Swimming; Urea | 2011 |
Antagonism of orexin 1 receptors eliminates motor hyperactivity and improves homing response acquisition in juvenile rats exposed to alcohol during early postnatal period.
Topics: Animals; Animals, Newborn; Benzoxazoles; Disease Models, Animal; Drug Interactions; Ethanol; Homing Behavior; Hyperkinesis; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2011 |
The orexin₁ receptor antagonist SB-334867 dissociates the motivational properties of alcohol and sucrose in rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Benzoxazoles; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Male; Motivation; Naphthyridines; Orexin Receptors; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Sucrose; Time Factors; Urea | 2011 |
Orexin-1 receptor signalling within the ventral tegmental area, but not the paraventricular thalamus, is critical to regulating cue-induced reinstatement of cocaine-seeking.
Topics: Animals; Benzoxazoles; Cocaine; Cocaine-Related Disorders; Cues; Dopamine Uptake Inhibitors; Extinction, Psychological; Male; Motor Activity; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Thalamus; Urea; Ventral Tegmental Area | 2011 |
Diaryl urea analogues of SB-334867 as orexin-1 receptor antagonists.
Topics: Benzoxazoles; Drug Delivery Systems; Ligands; Molecular Structure; Naphthyridines; Orexin Receptors; Protein Binding; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Structure-Activity Relationship; Urea | 2011 |
The role of orexin-1 receptors in physiologic responses evoked by microinjection of PgE2 or muscimol into the medial preoptic area.
Topics: Animals; Benzoxazoles; Blood Pressure; Body Temperature Regulation; Dinoprostone; Heart Rate; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Muscimol; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2011 |
Stimulatory effect of intracerebroventricular administration of orexin A on food intake in the zebrafish, Danio rerio.
Topics: Animals; Benzoxazoles; Eating; Fasting; Feeding Behavior; Hypothalamus; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Urea; Zebrafish | 2011 |
OX1 orexin/hypocretin receptor activation of phospholipase D.
Topics: Acetophenones; Animals; Benzopyrans; Benzoxazoles; CHO Cells; Cricetinae; Cricetulus; Humans; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Phospholipase D; Protein Kinase C-delta; Protein Kinase Inhibitors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Tetradecanoylphorbol Acetate; Urea | 2012 |
Effect of orexin-A on phagocytic activity of peritoneal macrophage in starved rats.
Topics: Animals; Benzoxazoles; Chondrus; Exudates and Transudates; Fasting; Inflammation; Intracellular Signaling Peptides and Proteins; Macrophages, Peritoneal; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Phagocytosis; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Time Factors; Urea | 2011 |
Hypocretin/orexin signaling in the hypothalamic paraventricular nucleus is essential for the expression of nicotine withdrawal.
Topics: Animals; Antigens, Surface; Benzoxazoles; Intracellular Signaling Peptides and Proteins; Isoquinolines; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Mice, Knockout; Microinjections; Molecular Imaging; Naphthyridines; Neuroanatomical Tract-Tracing Techniques; Neuropeptides; Orexin Receptors; Orexins; Paraventricular Hypothalamic Nucleus; Pyridines; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Substance Withdrawal Syndrome; Tobacco Use Disorder; Urea | 2012 |
Arousal effects of orexin A on acute alcohol intoxication-induced coma in rats.
Topics: Alcoholic Intoxication; Animals; Arousal; Benzoxazoles; Brain; Coma; Consciousness; Electroencephalography; Ethanol; Female; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neurons; Neuropeptides; Orexins; Prazosin; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Neuropeptide; Ritanserin; Urea | 2012 |
Evidence for the role of hindbrain orexin-1 receptors in the control of meal size.
Topics: Animals; Benzoxazoles; Eating; Intracellular Signaling Peptides and Proteins; Islet Amyloid Polypeptide; Male; Motor Activity; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Photoperiod; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Rhombencephalon; Satiation; Urea | 2011 |
Activation of orexin 1 receptors in the periaqueductal gray of male rats leads to antinociception via retrograde endocannabinoid (2-arachidonoylglycerol)-induced disinhibition.
Topics: Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Benzoxazoles; Biphenyl Compounds; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Disease Models, Animal; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Lactones; Male; Morpholines; Naphthalenes; Naphthyridines; Neural Inhibition; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Orlistat; Pain; Pain Measurement; Patch-Clamp Techniques; Periaqueductal Gray; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2011 |
Effects of orexin and glucose microinjected into the hypothalamic paraventricular nucleus on gastric acid secretion in conscious rats.
Topics: Animals; Benzoxazoles; Dose-Response Relationship, Drug; Gastric Acid; Gastric Mucosa; Glucose; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Naphthyridines; Neuropeptides; Orexins; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Urea | 2012 |
The influence of orexins on the firing rate and pattern of rat intergeniculate leaflet neurons--electrophysiological and immunohistological studies.
Topics: Action Potentials; Age Factors; Animals; Benzoxazoles; Enkephalins; Geniculate Bodies; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptide Y; Neuropeptides; Orexins; Rats; Rats, Wistar; Synaptophysin; Urea | 2011 |
An orexinergic projection from perifornical hypothalamus to raphe pallidus increases rat brown adipose tissue thermogenesis.
Topics: Adipose Tissue, Brown; Animals; Benzoxazoles; beta-Galactosidase; Body Temperature; Cholera Toxin; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Gene Transfer Techniques; Globus Pallidus; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Microinjections; N-Methylaspartate; Naphthyridines; Neurons; Neuropeptides; Neurotransmitter Agents; Orexins; Polystyrenes; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Rats, Wistar; Thermogenesis; Urea | 2011 |
Mapping of the binding sites for the OX1 orexin receptor antagonist, SB-334867, using orexin/hypocretin receptor chimaeras.
Topics: Benzoxazoles; Binding Sites; Chimera; HEK293 Cells; Humans; Inositol Phosphates; Models, Molecular; Naphthyridines; Orexin Receptors; Protein Binding; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Transfection; Tritium; Urea | 2012 |
Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity.
Topics: Adipocytes; Animals; Antineoplastic Agents; Benzoxazoles; Body Weight; Calorimetry; Cell Differentiation; Cell Line; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Drug Partial Agonism; Drug Screening Assays, Antitumor; Fibric Acids; Fibroblasts; Gene Expression Profiling; Humans; Insulin Resistance; Intra-Abdominal Fat; Liver; Mice; Mice, Inbred C57BL; Models, Molecular; PPAR alpha; PPAR gamma; Propionates; Stereoisomerism; Structure-Activity Relationship; Urea | 2012 |
Orexin-1 receptor antagonism does not reduce the rewarding potency of cocaine in Swiss-Webster mice.
Topics: Animals; Benzoxazoles; Brain; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Routes; Male; Mice; Motor Activity; Naphthyridines; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement Schedule; Reward; Self Administration; Urea | 2012 |
Orexin-1 receptor mediation of cocaine seeking in male and female rats.
Topics: Animals; Benzoxazoles; Cocaine-Related Disorders; Cues; Extinction, Psychological; Female; Male; Motor Activity; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Sex Characteristics; Urea; Yohimbine | 2012 |
Orexin / hypocretin 1 receptor antagonist reduces heroin self-administration and cue-induced heroin seeking.
Topics: Animals; Behavior, Addictive; Benzoxazoles; Conditioning, Operant; Cues; Heroin; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Urea | 2012 |
The orexin-1 receptor antagonist SB-334867 decreases sympathetic responses to a moderate dose of methamphetamine and stress.
Topics: Animals; Benzoxazoles; Blood Pressure; Body Temperature; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Male; Methamphetamine; Muscimol; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Stress, Psychological; Sympathetic Nervous System; Urea | 2012 |
Interactions between VTA orexin and glutamate in cue-induced reinstatement of cocaine seeking in rats.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzoxazoles; Cocaine; Cues; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Glutamic Acid; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, G-Protein-Coupled; Receptors, N-Methyl-D-Aspartate; Receptors, Neuropeptide; Self Administration; Signal Transduction; Urea; Ventral Tegmental Area | 2013 |
Orexin receptor type-1 antagonist SB-334867 inhibits the development of morphine analgesic tolerance in rats.
Topics: Analgesics, Opioid; Animals; Benzoxazoles; Drug Tolerance; Male; Morphine; Naphthyridines; Nociception; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2012 |
Activation of the orexin 1 receptor is a critical component of CO2-mediated anxiety and hypertension but not bradycardia.
Topics: Animals; Anxiety; Benzoxazoles; Bradycardia; Disease Models, Animal; Hypercapnia; Hypertension; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Respiration; Urea | 2012 |
A septal-hypothalamic pathway drives orexin neurons, which is necessary for conditioned cocaine preference.
Topics: Animals; Baclofen; Benzoxazoles; Cocaine; Conditioning, Psychological; Drug-Seeking Behavior; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Microinjections; Morpholinos; Muscimol; Naphthyridines; Neural Pathways; Neuroanatomical Tract-Tracing Techniques; Neurons; Neuropeptides; Orexins; Rats; Rats, Sprague-Dawley; Septum of Brain; Urea | 2012 |
OX1 orexin/hypocretin receptor signaling through arachidonic acid and endocannabinoid release.
Topics: Animals; Arachidonic Acid; Benzoxazoles; Cannabinoid Receptor Modulators; CHO Cells; Cricetinae; Cricetulus; Endocannabinoids; HEK293 Cells; Humans; Naphthyridines; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Signal Transduction; Urea | 2012 |
Effects of orexins A and B on expression of orexin receptors and progesterone release in luteal and granulosa ovarian cells.
Topics: Animals; Benzoxazoles; Cells, Cultured; Diethylstilbestrol; Dioxanes; Estradiol; Estrogens, Non-Steroidal; Female; Gene Expression; Granulosa Cells; Intracellular Signaling Peptides and Proteins; Luteal Cells; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Ovary; Phenylurea Compounds; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2012 |
Dual hypocretin receptor antagonism is more effective for sleep promotion than antagonism of either receptor alone.
Topics: Aminopyridines; Animals; Benzoxazoles; Dose-Response Relationship, Drug; GABA Agonists; Male; Naphthyridines; Orexin Receptors; Phenylurea Compounds; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep; Sulfonamides; Urea | 2012 |
N-(2-methyl-6-benzoxazolyl)-N'-1,5-naphthyridin-4-yl urea (SB334867), a hypocretin receptor-1 antagonist, preferentially prevents ethanol seeking: comparison with natural reward seeking.
Topics: Analysis of Variance; Animals; Benzoxazoles; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Ethanol; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexins; Rats; Reinforcement, Psychology; Reward; Secondary Prevention; Self Administration; Sweetening Agents; Urea | 2014 |
Antagonism of orexin-1 receptors attenuates swim- and restraint stress-induced antinociceptive behaviors in formalin test.
Topics: Analgesia; Animals; Benzoxazoles; Formaldehyde; Immobilization; Naloxone; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Stress, Physiological; Swimming; Urea | 2012 |
Repeated orexin 1 receptor antagonism effects on cocaine seeking in rats.
Topics: Animals; Benzoxazoles; Cocaine; Drug-Seeking Behavior; Extinction, Psychological; Male; Naphthyridines; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Self Administration; Urea | 2012 |
Putative genes mediating the effects of orexins in the posterior paraventricular thalamus on neuroendocrine and behavioral adaptations to repeated stress.
Topics: Adaptation, Psychological; Animals; bcl-2-Associated X Protein; Benzoxazoles; Intracellular Signaling Peptides and Proteins; Male; Midline Thalamic Nuclei; Naphthyridines; Neuropeptides; Neurosecretory Systems; Orexins; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Recurrence; Stress, Psychological; Urea; Vascular Endothelial Growth Factor A | 2012 |
The differential effects of OX1R and OX2R selective antagonists on morphine conditioned place preference in naïve versus morphine-dependent mice.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Antigens, Surface; Benzoxazoles; Conditioning, Operant; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Isoquinolines; Male; Mice; Morphine; Morphine Dependence; Naphthyridines; Orexin Receptors; Pyridines; Receptors, Cell Surface; Receptors, Neuropeptide; Urea | 2013 |
Blockade of orexin receptor 1 attenuates the development of morphine tolerance and physical dependence in rats.
Topics: Animals; Benzoxazoles; Drug Tolerance; Male; Morphine; Naphthyridines; Opioid-Related Disorders; Orexin Receptors; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2012 |
Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: possible confounding effects on in vivo and in vitro studies.
Topics: Benzoxazoles; Drug Stability; Hydrogen-Ion Concentration; Hydrolysis; Ligands; Molecular Structure; Naphthyridines; Orexin Receptors; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2012 |
Role of orexin/hypocretin in conditioned sucrose-seeking in rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Benzoxazoles; Conditioning, Operant; Drug-Seeking Behavior; Extinction, Psychological; Food Deprivation; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neurons; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Reinforcement Schedule; Reward; Self Administration; Sucrose; Urea | 2013 |
Orexin-1 receptor antagonism fails to reduce anxiety-like behaviour in either plus-maze-naïve or plus-maze-experienced mice.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzoxazoles; Chlordiazepoxide; Intracellular Signaling Peptides and Proteins; Male; Maze Learning; Mice; Naphthyridines; Neuropeptides; Neuropsychological Tests; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2013 |
Attenuation of saccharin-seeking in rats by orexin/hypocretin receptor 1 antagonist.
Topics: Animals; Behavior, Animal; Benzoxazoles; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Extinction, Psychological; Food Deprivation; Male; Naphthyridines; Orexin Receptor Antagonists; Rats; Rats, Sprague-Dawley; Reward; Saccharin; Self Administration; Urea | 2013 |
A role for hypocretin/orexin receptor-1 in cue-induced reinstatement of nicotine-seeking behavior.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Cues; Drug-Seeking Behavior; Extinction, Psychological; Hypothalamus; Isoquinolines; Male; Mice; Microinjections; Naphthyridines; Nerve Tissue Proteins; Neurons; Nicotine; Nicotinic Agonists; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Piperidines; Prefrontal Cortex; Protein Kinase Inhibitors; Pyridines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Self Administration; Signal Transduction; Urea | 2013 |
Blockade of central orexin 2 receptors reduces arterial pressure in spontaneously hypertensive rats.
Topics: Animals; Antibodies, Monoclonal; Arterial Pressure; Benzoxazoles; Cardiovascular System; Heart Rate; Immunoglobulin G; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Paraventricular Hypothalamic Nucleus; Pyridines; Rats; Rats, Inbred SHR; Solitary Nucleus; Urea | 2013 |
Functional inactivation of orexin 1 receptors in the cerebellum disrupts trace eyeblink conditioning and local theta oscillations in guinea pigs.
Topics: Analysis of Variance; Animals; Benzoxazoles; Blinking; Cerebellum; Complement Pathway, Classical; Guinea Pigs; Male; Microinjections; Naphthyridines; Orexin Receptors; Purkinje Cells; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Theta Rhythm; Time Factors; Urea | 2013 |
Behavioral characteristics and pharmacological manipulations of a nicotine-entrainable circadian oscillator.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Behavior, Animal; Benzoxazoles; Circadian Rhythm; Feeding Behavior; Female; Fructose; Light; Motor Activity; Naltrexone; Naphthyridines; Narcotic Antagonists; Nicotine; Nicotinic Agonists; Oscillometry; Rats; Rats, Sprague-Dawley; Time Factors; Topiramate; Urea | 2013 |
Pentylenetetrazol-induced seizures are exacerbated by sleep deprivation through orexin receptor-mediated hippocampal cell proliferation.
Topics: Animals; Benzoxazoles; CA3 Region, Hippocampal; Cell Proliferation; Convulsants; Dentate Gyrus; Hippocampus; Intracellular Signaling Peptides and Proteins; Isoquinolines; Male; Naphthyridines; Neurons; Neuropeptides; Neuroprotective Agents; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pentylenetetrazole; Pyridines; Rats; Rats, Wistar; Seizures; Sleep Deprivation; Time Factors; Urea | 2014 |
The hypocretin/orexin receptor-1 as a novel target to modulate cannabinoid reward.
Topics: Animals; Benzoxazines; Benzoxazoles; Cannabinoid Receptor Agonists; Cannabinoids; Conditioning, Operant; Dopamine; Dronabinol; Hypothalamic Area, Lateral; Male; Marijuana Abuse; Mice; Mice, Knockout; Molecular Targeted Therapy; Morpholines; Naphthalenes; Naphthyridines; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Proto-Oncogene Proteins c-fos; Reinforcement Schedule; Reward; Self Administration; Urea | 2014 |
Hindbrain orexin 1 receptors influence palatable food intake, operant responding for food, and food-conditioned place preference in rats.
Topics: Animals; Benzoxazoles; Choice Behavior; Conditioning, Operant; Eating; Infusions, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; Reinforcement Schedule; Rhombencephalon; Solitary Nucleus; Urea | 2014 |
Orexin receptor type-1 antagonist SB-334867 decreases morphine-induced antinociceptive effect in formalin test.
Topics: Analgesics; Animals; Benzoxazoles; Injections, Intraventricular; Morphine; Naphthyridines; Orexin Receptor Antagonists; Pain Measurement; Rats; Receptors, Neuropeptide; Urea | 2013 |
Mechanisms underlying obesity resistance associated with high spontaneous physical activity.
Topics: Age Factors; Animals; Benzazepines; Benzoxazoles; Body Weight; Dopamine Antagonists; Eating; Electromyography; Eye Movements; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Motor Activity; Naphthyridines; Neuropeptides; Obesity; Orexin Receptor Antagonists; Orexins; Rats; Rats, Sprague-Dawley; Sleep; Substantia Nigra; Urea; Wakefulness | 2014 |
Orexin/hypocretin system modulates amygdala-dependent threat learning through the locus coeruleus.
Topics: Acoustic Stimulation; Amygdala; Animals; Benzoxazoles; Channelrhodopsins; Conditioning, Classical; Fear; Intracellular Signaling Peptides and Proteins; Learning; Locus Coeruleus; Male; Naphthyridines; Neuropeptides; Optogenetics; Orexins; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Urea | 2013 |
Hypocretin (orexin) regulates glutamate input to fast-spiking interneurons in layer V of the Fr2 region of the murine prefrontal cortex.
Topics: Animals; Benzoxazoles; Electrophysiology; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Interneurons; Mice; Mice, Inbred Strains; Naphthyridines; Neural Inhibition; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Patch-Clamp Techniques; Prefrontal Cortex; Pyramidal Cells; Receptors, Ionotropic Glutamate; Synaptic Transmission; Tissue Culture Techniques; Urea; Vesicular Glutamate Transport Protein 1; Vesicular Glutamate Transport Protein 2 | 2015 |
Orexin-A-induced ERK1/2 activation reverses impaired spatial learning and memory in pentylenetetrazol-kindled rats via OX1R-mediated hippocampal neurogenesis.
Topics: Animals; Benzoxazoles; Doublecortin Protein; Enzyme Activation; Hippocampus; Intracellular Signaling Peptides and Proteins; Male; Maze Learning; Memory; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Naphthyridines; Neurogenesis; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pentylenetetrazole; Rats, Wistar; Spatial Learning; Urea | 2014 |
The orexin-1 receptor antagonist SB-334867 attenuates anxiety in rats exposed to cat odor but not the elevated plus maze: an investigation of Trial 1 and Trial 2 effects.
Topics: Animals; Anxiety; Avoidance Learning; Behavior, Animal; Benzoxazoles; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Maze Learning; Naphthyridines; Odorants; Orexin Receptor Antagonists; Rats; Rats, Wistar; Recognition, Psychology; Stress, Psychological; Urea | 2014 |
Blockade of hypocretin receptor-1 preferentially prevents cocaine seeking: comparison with natural reward seeking.
Topics: Analysis of Variance; Anesthetics, Local; Animals; Benzoxazoles; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Disease Models, Animal; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Extinction, Psychological; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Reward; Self Administration; Sweetening Agents; Urea | 2014 |
Acute high fat diet consumption activates the mesolimbic circuit and requires orexin signaling in a mouse model.
Topics: Analysis of Variance; Animals; Benzoxazoles; Diet, High-Fat; Dietary Fats; Immunohistochemistry; Intracellular Signaling Peptides and Proteins; Limbic System; Mice; Naphthyridines; Neural Pathways; Neuroanatomical Tract-Tracing Techniques; Neurons; Neuropeptides; Orexins; Proto-Oncogene Proteins c-fos; Reward; Signal Transduction; Urea; Ventral Tegmental Area | 2014 |
Central orexin inhibits reflex swallowing elicited by the superior laryngeal nerve via caudal brainstem in the rat.
Topics: Animals; Benzoxazoles; Brain Stem; Central Nervous System Agents; Deglutition; Electric Stimulation; Electromyography; Intracellular Signaling Peptides and Proteins; Laryngeal Nerves; Male; Muscle, Skeletal; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats, Sprague-Dawley; Reflex; Solitary Nucleus; Urea | 2014 |
Ghrelin acts as an interface between physiological state and phasic dopamine signaling.
Topics: Action Potentials; Animals; Benzoxazoles; Dopamine; Dose-Response Relationship, Drug; Fasting; Feeding Behavior; Ghrelin; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neural Pathways; Neuropeptides; Nucleus Accumbens; Oligopeptides; Orexins; Rats; Rats, Sprague-Dawley; Signal Transduction; Urea; Ventral Tegmental Area; Wakefulness | 2014 |
Circadian rhythm disruption by a novel running wheel: roles of exercise and arousal in blockade of the luteinizing hormone surge.
Topics: Animals; Arousal; Benzoxazoles; Central Nervous System Agents; Circadian Rhythm; Darkness; Estrus; Female; Gonadotropin-Releasing Hormone; Housing, Animal; Luteinizing Hormone; Mesocricetus; Motor Activity; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Photoperiod; Proestrus; Proto-Oncogene Proteins c-fos; Urea | 2014 |
Hepatic branch vagus nerve plays a critical role in the recovery of post-ischemic glucose intolerance and mediates a neuroprotective effect by hypothalamic orexin-A.
Topics: Animals; Benzoxazoles; Choline O-Acetyltransferase; Glucose Intolerance; Hypothalamus; Infarction, Middle Cerebral Artery; Intracellular Signaling Peptides and Proteins; Liver; Male; Mice; Naphthyridines; Neuropeptides; Neuroprotective Agents; Orexin Receptors; Orexins; Proto-Oncogene Proteins c-fos; Urea; Vagus Nerve | 2014 |
Blockade of orexin-1 receptors in the ventral tegmental area could attenuate the lateral hypothalamic stimulation-induced potentiation of rewarding properties of morphine.
Topics: Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Conditioning, Psychological; Hypothalamic Area, Lateral; Male; Morphine; Motor Activity; Naphthyridines; Narcotics; Orexin Receptor Antagonists; Rats; Rats, Wistar; Reward; Urea; Ventral Tegmental Area | 2014 |
Orexin A protects cells from apoptosis by regulating FoxO1 and mTORC1 through the OX1R/PI3K/AKT signaling pathway in hepatocytes.
Topics: Animals; Apoptosis; Benzoxazoles; Culture Media, Serum-Free; Dose-Response Relationship, Drug; Everolimus; Forkhead Transcription Factors; Gene Expression Regulation; Hepatocytes; Intracellular Signaling Peptides and Proteins; Male; Mechanistic Target of Rapamycin Complex 1; Multiprotein Complexes; Naphthyridines; Nerve Tissue Proteins; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Primary Cell Culture; Proto-Oncogene Proteins c-akt; Pyridones; Pyrimidines; Quinolones; Rats; Rats, Sprague-Dawley; Signal Transduction; Sirolimus; TOR Serine-Threonine Kinases; Urea | 2014 |
Attenuated orexinergic signaling underlies depression-like responses induced by daytime light deficiency.
Topics: Animals; Anxiety; Behavior, Animal; Benzoxazoles; Circadian Rhythm; Depression; Disease Models, Animal; Intracellular Signaling Peptides and Proteins; Light; Male; Motor Activity; Naphthyridines; Neuropeptides; Orexins; Photoperiod; Phototherapy; Rats; Seasonal Affective Disorder; Signal Transduction; Urea | 2014 |
Orexin-1 receptor mediates the increased food and water intake induced by intracerebroventricular injection of the stable somatostatin pan-agonist, ODT8-SST in rats.
Topics: Animals; Benzoxazoles; Drinking; Eating; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Octreotide; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Peptide Fragments; Rats, Sprague-Dawley; Receptors, Somatostatin; Somatostatin; Urea | 2014 |
The hypocretin/orexin system mediates the extinction of fear memories.
Topics: Amygdala; Animals; Benzoxazoles; Extinction, Psychological; Fear; Hippocampus; Intracellular Signaling Peptides and Proteins; Isoquinolines; Male; Memory; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Knockout; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Psychotropic Drugs; Pyridines; Urea | 2014 |
Orexin A enhances locomotor activity and induces anxiogenic-like action in the goldfish, Carassius auratus.
Topics: Animals; Anxiety; Benzoxazoles; Carbolines; Diazepam; Emotions; Goldfish; Hypnotics and Sedatives; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Motor Activity; Naphthyridines; Neuropeptides; Orexins; Urea | 2014 |
Blockade of orexin type-1 receptors in locus coeruleus nucleus attenuates the development of morphine dependency in rats.
Topics: Animals; Benzoxazoles; Locus Coeruleus; Male; Morphine; Morphine Dependence; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Urea | 2014 |
Binge-like consumption of caloric and non-caloric palatable substances in ad libitum-fed C57BL/6J mice: pharmacological and molecular evidence of orexin involvement.
Topics: Animals; Benzoxazoles; Bulimia; Dietary Sucrose; Dose-Response Relationship, Drug; Drinking Behavior; Drinking Water; Energy Intake; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Mice, Inbred C57BL; Mitochondrial Proteins; Motor Activity; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Nuclear Proteins; Orexins; RNA, Messenger; Saccharin; Urea | 2014 |
Blockade of orexin type 1 receptors inhibits the development of morphine tolerance in lateral paragigantocellularis nucleus: an electrophysiological approach.
Topics: Animals; Benzoxazoles; Drug Tolerance; Male; Medulla Oblongata; Morphine; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Urea | 2014 |
Role of orexin/hypocretin in conditioned sucrose-seeking in female rats.
Topics: Animals; Appetitive Behavior; Benzoxazoles; Central Nervous System Agents; Conditioning, Operant; Cues; Dietary Sucrose; Dose-Response Relationship, Drug; Extinction, Psychological; Female; Food Deprivation; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats, Sprague-Dawley; Reward; Self Administration; Sex Characteristics; Spatial Behavior; Urea | 2014 |
Metabolic regulation of lateral hypothalamic glucose-inhibited orexin neurons may influence midbrain reward neurocircuitry.
Topics: Action Potentials; Animals; Benzoxazoles; Glucose; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Mesencephalon; Mice, Inbred C57BL; Naphthyridines; Neurons; Neuropeptides; Orexins; Reward; Synaptic Transmission; Urea; Ventral Tegmental Area | 2014 |
Perifornical hypothalamic orexin and serotonin modulate the counterregulatory response to hypoglycemic and glucoprivic stimuli.
Topics: Animals; Astrocytes; Benzoxazoles; Blood Glucose; Cells, Cultured; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Fornix, Brain; Hypoglycemia; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Midline Thalamic Nuclei; Naphthyridines; Neurons; Neuropeptides; Orexins; Paraventricular Hypothalamic Nucleus; Rats, Sprague-Dawley; Receptors, Neuropeptide; Serotonin; Urea; Ventromedial Hypothalamic Nucleus | 2015 |
Orexin-1 receptor antagonist in central nucleus of the amygdala attenuates the acquisition of flavor-taste preference in rats.
Topics: Animals; Avoidance Learning; Benzoxazoles; Central Amygdaloid Nucleus; Food Preferences; Lithium Chloride; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Saccharin; Taste Perception; Urea | 2014 |
Orexin-A stimulates 3β-hydroxysteroid dehydrogenase expression and cortisol production in H295R human adrenocortical cells through the AKT pathway.
Topics: 3-Hydroxysteroid Dehydrogenases; Adrenocortical Carcinoma; Benzoxazoles; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Gene Expression Regulation, Neoplastic; Humans; Hydrocortisone; Intracellular Signaling Peptides and Proteins; Isoenzymes; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Phosphorylation; Proto-Oncogene Proteins c-akt; Pyridones; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Urea | 2014 |
Orexin excites rat inferior vestibular nuclear neurons via co-activation of OX1 and OX 2 receptors.
Topics: Action Potentials; Animals; Benzoxazoles; Dose-Response Relationship, Drug; Isoquinolines; Naphthyridines; Neurons; Neurotransmitter Agents; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pyridines; Rats, Sprague-Dawley; RNA, Messenger; Sodium Channel Blockers; Tetrodotoxin; Tissue Culture Techniques; Urea; Vestibular Nuclei | 2015 |
Role of intra-hippocampal orexin 1 and orexin 2 receptors in conditioned place preference induced by chemical stimulation of the lateral hypothalamus.
Topics: Animals; Benzoxazoles; CA1 Region, Hippocampal; Carbachol; Cholinergic Agonists; Conditioning, Psychological; Hypothalamic Area, Lateral; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Stimulation, Chemical; Urea | 2015 |
The orexin-1 receptor antagonist SB-334867 decreases anxiety-like behavior and c-Fos expression in the hypothalamus of rats exposed to cat odor.
Topics: Analysis of Variance; Animals; Anxiety; Benzoxazoles; Cats; Disease Models, Animal; Gene Expression Regulation; Hypothalamus; Male; Naphthyridines; Odorants; Proto-Oncogene Proteins c-fos; Random Allocation; Rats; Rats, Wistar; Receptors, Neuropeptide; Urea | 2015 |
Hypocretin/Orexin regulation of dopamine signaling and cocaine self-administration is mediated predominantly by hypocretin receptor 1.
Topics: Analysis of Variance; Animals; Benzoxazoles; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electrochemical Techniques; Intracellular Signaling Peptides and Proteins; Male; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Self Administration; Signal Transduction; Urea | 2015 |
Antinociceptive action against colonic distension by brain orexin in conscious rats.
Topics: Analgesics; Animals; Benzoxazoles; Brain; Colon; Disease Models, Animal; Dose-Response Relationship, Drug; Electrodes, Implanted; Intracellular Signaling Peptides and Proteins; Male; Morphine; Naphthyridines; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pain Threshold; Physical Stimulation; Rats, Sprague-Dawley; Urea; Visceral Pain | 2015 |
Hippocampal orexin receptors inactivation reduces PTZ induced seizures of male rats.
Topics: Animals; Benzoxazoles; Convulsants; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pentylenetetrazole; Pyridines; Rats; Seizures; Urea | 2015 |
Binge-like consumption of ethanol and other salient reinforcers is blocked by orexin-1 receptor inhibition and leads to a reduction of hypothalamic orexin immunoreactivity.
Topics: Animals; Benzoxazoles; Binge Drinking; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Male; Mice; Motor Activity; Naphthyridines; Orexin Receptors; Orexins; Reinforcement, Psychology; Saccharin; Sucrose; Urea | 2015 |
The electrical activity of hippocampal pyramidal neuron is subjected to descending control by the brain orexin/hypocretin system.
Topics: Action Potentials; Animals; Benzoxazoles; Carbachol; Hippocampus; Hypothalamic Area, Lateral; Infusions, Intraventricular; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pyramidal Cells; Rats; Rats, Wistar; Urea | 2015 |
Orexin-1 receptor signaling increases motivation for cocaine-associated cues.
Topics: Animals; Benzoxazoles; Cocaine-Related Disorders; Cues; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Signal Transduction; Urea | 2015 |
Orexin A-mediated AKT signaling in the dentate gyrus contributes to the acquisition, expression and reinstatement of morphine-induced conditioned place preference.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Benzoxazoles; Choice Behavior; Conditioning, Psychological; Dentate Gyrus; Disease Models, Animal; Hypothalamic Area, Lateral; Male; Morphine; Naphthyridines; Opioid-Related Disorders; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Signal Transduction; Urea | 2016 |
Changes in hippocampal orexin 1 receptor expression involved in tooth pain-induced learning and memory impairment in rats.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzoxazoles; Capsaicin; Dental Pulp; Hippocampus; Ibuprofen; Incisor; Learning Disabilities; Male; Maze Learning; Memory Disorders; Naphthyridines; Nerve Tissue Proteins; Nociception; Orexin Receptors; Orexins; Pain Measurement; Random Allocation; Rats; Rats, Wistar; RNA, Messenger; Single-Blind Method; Toothache; Urea | 2015 |
Orexin receptor 1 signaling contributes to ethanol binge-like drinking: Pharmacological and molecular evidence.
Topics: Animals; Benzoxazoles; Binge Drinking; Blood Alcohol Content; Central Nervous System Depressants; Drinking Water; Eating; Ethanol; Hypnotics and Sedatives; Hypothalamic Area, Lateral; Locomotion; Male; Mice, Inbred C57BL; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Reflex; RNA, Messenger; Saccharin; Urea | 2015 |
Functional inactivation of hypocretin 1 receptors in the medial prefrontal cortex affects the pyramidal neuron activity and gamma oscillations: An in vivo multiple-channel single-unit recording study.
Topics: Acetylcholine; Action Potentials; Animals; Benzoxazoles; Chi-Square Distribution; Cholinergic Agonists; Gamma Rhythm; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Urea | 2015 |
Orexin-1 receptor signalling in the prelimbic cortex and ventral tegmental area regulates cue-induced reinstatement of ethanol-seeking in iP rats.
Topics: Animals; Behavior, Animal; Benzoxazoles; Central Nervous System Depressants; Conditioning, Psychological; Cues; Drug-Seeking Behavior; Ethanol; Extinction, Psychological; Limbic Lobe; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Inbred Strains; Signal Transduction; Urea; Ventral Tegmental Area | 2016 |
Orexinergic neurotransmission in temperature responses to methamphetamine and stress: mathematical modeling as a data assimilation approach.
Topics: Animals; Benzoxazoles; Computer Simulation; Dose-Response Relationship, Drug; Hyperthermia, Induced; Male; Methamphetamine; Models, Neurological; Monte Carlo Method; Naphthyridines; Neural Pathways; Orexin Receptors; Rats, Sprague-Dawley; Stress, Physiological; Synaptic Transmission; Temperature; Urea | 2015 |
Orexins/hypocretins modulate the activity of NPY-positive and -negative neurons in the rat intergeniculate leaflet via OX1 and OX2 receptors.
Topics: Animals; Benzoxazoles; Immunohistochemistry; Isoquinolines; Male; Membrane Potentials; Naphthyridines; Neurons; Neuropeptide Y; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Rats, Wistar; Thalamus; Tissue Culture Techniques; Urea | 2015 |
Hypocretin receptor 1 blockade preferentially reduces high effort responding for cocaine without promoting sleep.
Topics: Animals; Appetitive Behavior; Benzoxazoles; Brain; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Hypnotics and Sedatives; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats, Sprague-Dawley; Reinforcement Schedule; Self Administration; Sleep; Urea | 2015 |
Catalytic Oxidative Carbonylation of Amino Moieties to Ureas, Oxamides, 2-Oxazolidinones, and Benzoxazolones.
Topics: Amines; Amino Alcohols; Aminophenols; Benzoxazoles; Catalysis; Imidazoles; Ionic Liquids; Oxamic Acid; Oxazolidinones; Oxidation-Reduction; Palladium; Urea | 2015 |
Effects of activation and blockade of orexin A receptors in the medial preoptic area on food intake in male rats.
Topics: Animals; Benzoxazoles; Eating; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Preoptic Area; Rats, Wistar; Urea | 2015 |
Microinjection of orexin-A into the rat locus coeruleus nucleus induces analgesia via cannabinoid type-1 receptors.
Topics: Analgesics; Analysis of Variance; Animals; Benzoxazoles; Carrier Proteins; Dose-Response Relationship, Drug; Formaldehyde; Locus Coeruleus; Male; Microinjections; Naphthyridines; Orexins; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Wistar; Urea | 2015 |
Upregulation of orexin receptor in paraventricular nucleus promotes sympathetic outflow in obese Zucker rats.
Topics: Action Potentials; Animals; Benzoxazoles; Blood Pressure; Central Nervous System Agents; Disease Models, Animal; Male; Naphthyridines; Neuroanatomical Tract-Tracing Techniques; Neurons; Obesity; Orexin Receptors; Orexins; Paraventricular Hypothalamic Nucleus; Rats, Zucker; Spinal Cord; Sympathetic Nervous System; Tissue Culture Techniques; Up-Regulation; Urea | 2015 |
[Effect of orexin-A and orexin-1 receptor antagonist injected into the fourth ventricle of rats on food-intake and spontaneous physical activity].
Topics: Animals; Benzoxazoles; Diet, High-Fat; Eating; Fourth Ventricle; Motor Activity; Naphthyridines; Obesity; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; Urea | 2015 |
Lateral Hypothalamic Stimulation Reduces Hyperalgesia Through Spinally Descending Orexin-A Neurons in Neuropathic Pain.
Topics: Analgesics, Non-Narcotic; Animals; Benzoxazoles; Carbachol; Female; Hyperalgesia; Hypothalamic Area, Lateral; Naphthyridines; Neuralgia; Orexins; Pain Management; Random Allocation; Rats; Rats, Sprague-Dawley; Spinal Cord Dorsal Horn; Urea | 2016 |
Orexin signaling is necessary for hypoglycemia-induced prevention of conditioned place preference.
Topics: Animals; Arousal; Behavior, Animal; Benzoxazoles; Blood Glucose; Brain; Conditioning, Psychological; Disease Models, Animal; Feeding Behavior; Hypoglycemia; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats, Sprague-Dawley; Reward; Sertraline; Signal Transduction; Time Factors; Urea | 2016 |
Orexin/Hypocretin-1 Receptor Antagonism Selectively Reduces Cue-Induced Feeding in Sated Rats and Recruits Medial Prefrontal Cortex and Thalamus.
Topics: Amygdala; Animals; Benzoxazoles; Cues; Eating; Feeding Behavior; Learning; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Prefrontal Cortex; Rats; Reward; Thalamus; Urea | 2015 |
Localization, expression and role of Orexin A and its receptor in testes of neonatal mice.
Topics: Animals; Animals, Newborn; Anti-Mullerian Hormone; Benzoxazoles; Hypothalamus; Intracellular Signaling Peptides and Proteins; Male; Mice; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Receptors, G-Protein-Coupled; Testis; Tissue Distribution; Urea | 2016 |
Role of dorsal hippocampal orexin-1 receptors in memory restoration induced by morphine sensitization phenomenon.
Topics: Amnesia; Animals; Behavior, Animal; Benzoxazoles; CA1 Region, Hippocampal; Central Nervous System Sensitization; Male; Maze Learning; Morphine; Naphthyridines; Narcotics; Orexin Receptors; Rats; Rats, Wistar; Receptors, Neuropeptide; Spatial Memory; Urea | 2016 |
Individual differences in orexin-I receptor modulation of motivation for the opioid remifentanil.
Topics: Analgesics, Opioid; Animals; Bacterial Outer Membrane Proteins; Behavior, Animal; Benzoxazoles; Conditioning, Operant; Economics, Behavioral; Escherichia coli Proteins; Individuality; Lipoproteins; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Piperidines; Rats; Rats, Sprague-Dawley; Remifentanil; Self Administration; Urea | 2017 |
Activation of Medulla-Projecting Perifornical Neurons Modulates the Adrenal Sympathetic Response to Hypoglycemia: Involvement of Orexin Type 2 (OX2-R) Receptors.
Topics: Adrenal Glands; Animals; Benzoxazoles; Brain; Epinephrine; Fornix, Brain; Hypoglycemia; Hypoglycemic Agents; Hypothalamus; Insulin; Isoquinolines; Medulla Oblongata; Naphthyridines; Neural Pathways; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Urea | 2016 |
Differential roles of orexin receptors within the dentate gyrus in stress- and drug priming-induced reinstatement of conditioned place preference in rats.
Topics: Analgesics, Opioid; Animals; Benzoxazoles; Conditioning, Operant; Conditioning, Psychological; Dentate Gyrus; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Extinction, Psychological; Isoquinolines; Male; Morphine; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Reward; Stress, Psychological; Swimming; Time Factors; Urea | 2016 |
The role of trigeminal nucleus caudalis orexin 1 receptors in orofacial pain transmission and in orofacial pain-induced learning and memory impairment in rats.
Topics: Animals; Benzoxazoles; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Facial Pain; Learning Disabilities; Male; Maze Learning; Memory Disorders; Motor Activity; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Psychomotor Performance; Rats; Rats, Wistar; Reaction Time; Sensory System Agents; Spatial Learning; Trigeminal Nuclei; Urea | 2016 |
Orexinergic system in the locus coeruleus modulates the CO2 ventilatory response.
Topics: Animals; Benzoxazoles; Carbon Dioxide; Hypercapnia; Locus Coeruleus; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pulmonary Ventilation; Rats; Rats, Wistar; Reflex; Sleep; Urea; Wakefulness | 2016 |
Role of orexin-A in experimental autoimmune encephalomyelitis.
Topics: Animals; Attention; Avoidance Learning; Benzoxazoles; Body Weight; Cytokines; Disease Models, Animal; Encephalomyelitis, Autoimmune, Experimental; Exploratory Behavior; Female; Matrix Metalloproteinase 9; Maze Learning; Mice; Mice, Inbred C57BL; Myelin Basic Protein; Myelin-Oligodendrocyte Glycoprotein; Naphthyridines; Nitric Oxide Synthase Type II; Orexin Receptor Antagonists; Orexins; Peptide Fragments; Severity of Illness Index; Spinal Cord; Time Factors; Urea | 2016 |
Differential contribution of orexin receptors within the ventral tegmental area to modulation of persistent inflammatory pain.
Topics: Animals; Benzoxazoles; Carbachol; Hypothalamic Area, Lateral; Isoquinolines; Male; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Pyridines; Rats; Rats, Wistar; Urea; Ventral Tegmental Area | 2016 |
The blockade of GABAA receptors attenuates the inhibitory effect of orexin type 1 receptors antagonist on morphine withdrawal syndrome in rats.
Topics: Animals; Benzoxazoles; Bicuculline; GABA-A Receptor Antagonists; Locus Coeruleus; Male; Microinjections; Morphine; Naloxone; Naphthyridines; Narcotic Antagonists; Orexin Receptor Antagonists; Orexin Receptors; Rats, Wistar; Substance Withdrawal Syndrome; Urea | 2016 |
Levodopa acts centrally to induce an antinociceptive action against colonic distension through activation of D2 dopamine receptors and the orexinergic system in the brain in conscious rats.
Topics: Analgesics; Animals; Benzoxazoles; Brain; Consciousness; Injections, Intraventricular; Injections, Subcutaneous; Levodopa; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pain Threshold; Rats, Sprague-Dawley; Receptors, Dopamine D2; Sulpiride; Urea; Visceral Pain | 2016 |
Stress induces analgesia via orexin 1 receptor-initiated endocannabinoid/CB1 signaling in the mouse periaqueductal gray.
Topics: Analgesics, Opioid; Animals; Benzoxazines; Benzoxazoles; Corticosterone; Hypothalamus; Isoquinolines; Male; Mice, Inbred C57BL; Morpholines; Naloxone; Naphthalenes; Naphthyridines; Neurons; Nociceptive Pain; Orexin Receptors; Pain Perception; Periaqueductal Gray; Proto-Oncogene Proteins c-fos; Pyridines; Receptor, Cannabinoid, CB1; Signal Transduction; Stress, Psychological; Urea | 2016 |
SB 334867, a selective orexin receptor type 1 antagonist, elevates seizure threshold in mice.
Topics: Animals; Anticonvulsants; Benzoxazoles; Brain Chemistry; Convulsants; Electroshock; Male; Mice; Muscle Strength; Myoclonus; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pentylenetetrazole; Psychomotor Performance; Seizures; Urea | 2016 |
Lateral hypothalamic area orexin-A influence the firing activity of gastric distension-sensitive neurons and gastric motility in rats.
Topics: Action Potentials; Animals; Benzoxazoles; Electric Stimulation; Gastrointestinal Motility; Hypothalamic Area, Lateral; Male; Naphthyridines; Neurons; Orexins; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Urea | 2016 |
Orexin-A facilitates emergence of the rat from isoflurane anesthesia via mediation of the basal forebrain.
Topics: Anesthetics, Inhalation; Animals; Basal Forebrain; Benzoxazoles; Isoflurane; Male; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexins; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Urea | 2016 |
Orexin/hypocretin receptor 1 signaling mediates Pavlovian cue-food conditioning and extinction.
Topics: Analysis of Variance; Animals; Association Learning; Benzoxazoles; Conditioning, Classical; Cues; Extinction, Psychological; Food; Locomotion; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; Rats, Long-Evans; Signal Transduction; Urea | 2016 |
Involvement of orexin-1 and orexin-2 receptors within the dentate gyrus of the hippocampus in the acquisition, expression and extinction of lateral hypothalamic-induced conditioned place preference in the rats.
Topics: Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Conditioning, Psychological; Dentate Gyrus; Dose-Response Relationship, Drug; Extinction, Psychological; Hypothalamic Area, Lateral; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Random Allocation; Rats, Wistar; Spatial Behavior; Urea | 2016 |
Hypocretinergic system in the medial preoptic area promotes maternal behavior in lactating rats.
Topics: Animals; Behavior Rating Scale; Benzoxazoles; Female; Hypothalamic Area, Lateral; Hypothalamus, Posterior; Infusions, Intraventricular; Lactation; Maternal Behavior; Microinjections; Naphthyridines; Neurons; Orexin Receptors; Orexins; Preoptic Area; Rats; Rats, Wistar; Statistics, Nonparametric; Urea | 2016 |
The role of orexin type-1 receptors in the development of morphine tolerance in locus coeruleus neurons: An electrophysiological perspective.
Topics: Action Potentials; Animals; Benzoxazoles; Drug Tolerance; Locus Coeruleus; Male; Morphine; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Urea | 2016 |
Functional interaction between orexin-1 and CB1 receptors in the periaqueductal gray matter during antinociception induced by chemical stimulation of the lateral hypothalamus in rats.
Topics: Animals; Benzoxazoles; Carbachol; Disease Models, Animal; Hypothalamic Area, Lateral; Male; Microinjections; Naphthyridines; Orexin Receptors; Orexins; Pain; Pain Measurement; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Stimulation, Chemical; Urea | 2016 |
Orexin-A increases the activity of globus pallidus neurons in both normal and parkinsonian rats.
Topics: Action Potentials; Animals; Benzoxazoles; Globus Pallidus; Haloperidol; Male; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Oxidopamine; Parkinson Disease; Postural Balance; Rats; Rats, Wistar; Urea | 2016 |
Orexin-1 receptor blockade suppresses compulsive-like alcohol drinking in mice.
Topics: Alcohol Deterrents; Alcohol Drinking; Alcohol-Related Disorders; Animals; Benzoxazoles; Choice Behavior; Compulsive Behavior; Dose-Response Relationship, Drug; Isoquinolines; Male; Mice, Inbred C57BL; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Quinine; Urea | 2016 |
Orexin-A/Hypocretin-1 Mediates Cocaine-Seeking Behavior in the Posterior Paraventricular Nucleus of the Thalamus via Orexin/Hypocretin Receptor-2.
Topics: Animals; Benzoxazoles; Cocaine; Drug Interactions; Drug-Seeking Behavior; Extinction, Psychological; Isoquinolines; Male; Naphthyridines; Orexin Receptors; Orexins; Paraventricular Hypothalamic Nucleus; Pyridines; Rats; Rats, Wistar; Urea | 2016 |
The role of trigeminal nucleus caudalis orexin 1 receptor in orofacial pain-induced anxiety in rat.
Topics: Animals; Anxiety; Benzoxazoles; Capsaicin; Disease Models, Animal; Exploratory Behavior; Facial Pain; Formaldehyde; Male; Maze Learning; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pain Measurement; Rats; Rats, Wistar; Time Factors; Trigeminal Nuclei; Urea | 2016 |
Hypocretin Neurotransmission Within the Central Amygdala Mediates Escalated Cocaine Self-administration and Stress-Induced Reinstatement in Rats.
Topics: Animals; Benzoxazoles; Central Amygdaloid Nucleus; Cocaine; Drug-Seeking Behavior; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Reinforcement Schedule; Self Administration; Stress, Psychological; Urea | 2017 |
Role of the orexin (hypocretin) system in contextual fear conditioning in rats.
Topics: Animals; Benzoxazoles; Conditioning, Classical; Electroshock; Fear; Gene Expression Regulation; Hypothalamus; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pyridines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Signal Transduction; Urea | 2017 |
Blockade of orexin receptors attenuates the cardiovascular response to air-jet stress in spontaneously hypertensive rats.
Topics: Acetamides; Air; Animals; Benzoxazoles; Blood Pressure; Brain; Brain-Derived Neurotrophic Factor; Cardiovascular Agents; Dose-Response Relationship, Drug; Heart Rate; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Physical Stimulation; Random Allocation; Rats, Inbred SHR; Rats, Wistar; RNA, Messenger; Species Specificity; Stress, Psychological; Urea | 2016 |
SB-334867, an orexin receptor 1 antagonist, decreased seizure and anxiety in pentylenetetrazol-kindled rats.
Topics: Animals; Anxiety; Benzoxazoles; Dose-Response Relationship, Drug; Kindling, Neurologic; Male; Maze Learning; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pentylenetetrazole; Rats; Rats, Wistar; Seizures; Urea | 2017 |
Blockade of dorsal hippocampal orexin-1 receptors impaired morphine-induced state-dependent learning.
Topics: Animals; Avoidance Learning; Benzoxazoles; Hippocampus; Male; Memory; Mice; Morphine; Motor Activity; Naphthyridines; Narcotics; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Urea | 2016 |
Orexin/hypocretin-1 receptor antagonism reduces ethanol self-administration and reinstatement selectively in highly-motivated rats.
Topics: Alcohol Drinking; Alcohol-Related Disorders; Animals; Animals, Outbred Strains; Benzoxazoles; Central Nervous System Depressants; Conditioning, Operant; Cues; Disease Models, Animal; Drug-Seeking Behavior; Ethanol; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats, Sprague-Dawley; Self Administration; Urea | 2017 |
Intra-LC microinjection of orexin type-1 receptor antagonist SB-334867 attenuates the expression of glutamate-induced opiate withdrawal like signs during the active phase in rats.
Topics: Animals; Benzoxazoles; Disease Models, Animal; Glutamic Acid; Locus Coeruleus; Male; Microinjections; Morphine; Naphthyridines; Orexin Receptor Antagonists; Orexins; Rats, Wistar; Substance Withdrawal Syndrome; Urea | 2017 |
Intramolecular oxidative deselenization of acylselenoureas: a facile synthesis of benzoxazole amides and carbonic anhydrase inhibitors.
Topics: Amides; Benzoxazoles; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Dose-Response Relationship, Drug; Humans; Molecular Structure; Organoselenium Compounds; Oxidation-Reduction; Structure-Activity Relationship; Urea | 2016 |
The Role of Orexin Signaling in the Ventral Tegmental Area and Central Amygdala in Modulating Binge-Like Ethanol Drinking Behavior.
Topics: Animals; Benzoxazoles; Binge Drinking; Central Amygdaloid Nucleus; Ethanol; Injections, Intraventricular; Male; Mice; Mice, Inbred C57BL; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Signal Transduction; Urea; Ventral Tegmental Area | 2017 |
NERP-2 regulates gastric acid secretion and gastric emptying via the orexin pathway.
Topics: Animals; Atropine; Benzoxazoles; Gastric Acid; Gastric Emptying; Injections, Intraventricular; Male; Naphthyridines; Nerve Tissue Proteins; Orexin Receptors; Parasympatholytics; Rats, Sprague-Dawley; Rats, Transgenic; Rats, Wistar; Signal Transduction; Urea; Vagus Nerve | 2017 |
The effect of orexin 1 and orexin 2 receptors antagonisms in the basolateral amygdala on memory processing in a passive avoidance task.
Topics: Animals; Avoidance Learning; Basolateral Nuclear Complex; Benzoxazoles; Dose-Response Relationship, Drug; Isoquinolines; Male; Memory; Mental Recall; Naphthyridines; Orexin Receptor Antagonists; Pyridines; Rats; Rats, Wistar; Reaction Time; Urea | 2017 |
Pharmacological evaluation of a novel series of urea, thiourea and guanidine derivatives as P2X
Topics: Adamantane; Adenosine Triphosphate; Benzoxazoles; Cell Line; Fluorescent Dyes; Guanidines; Humans; Molecular Structure; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Quinolinium Compounds; Thiourea; Urea | 2017 |
Facilitation of Contextual Fear Extinction by Orexin-1 Receptor Antagonism Is Associated with the Activation of Specific Amygdala Cell Subpopulations.
Topics: Animals; Basolateral Nuclear Complex; Benzoxazoles; Calbindins; Extinction, Psychological; Fear; Male; Memory Consolidation; Mice, Inbred C57BL; Naphthyridines; Neural Pathways; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Parvalbumins; Prefrontal Cortex; Psychotropic Drugs; Urea | 2017 |
Antagonism of orexin type-1 receptors (OX1Rs) attenuates naloxone-precipitated morphine withdrawal syndrome in rat dorsal hippocampus.
Topics: Animals; Benzoxazoles; Hippocampus; Male; Microinjections; Morphine; Naloxone; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Urea | 2017 |
Effects of Suvorexant, a Dual Orexin/Hypocretin Receptor Antagonist, on Impulsive Behavior Associated with Cocaine.
Topics: Animals; Azepines; Benzoxazoles; Choice Behavior; Cocaine; Delay Discounting; Impulsive Behavior; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexins; Proto-Oncogene Proteins c-fos; Pyridines; Rats; Triazoles; Urea; Ventral Tegmental Area | 2018 |
Role of orexin receptors in the ventral tegmental area on acquisition and expression of morphine-induced conditioned place preference in the rats.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Isoquinolines; Male; Morphine; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Reward; Urea; Ventral Tegmental Area | 2017 |
Orexin-A Suppresses Signal Transmission to Dopaminergic Amacrine Cells From Outer and Inner Retinal Photoreceptors.
Topics: Amacrine Cells; Animals; Benzoxazoles; Dopamine; Female; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Naphthyridines; Orexin Receptor Antagonists; Orexins; Patch-Clamp Techniques; Photoreceptor Cells, Vertebrate; Pyridines; Retinal Ganglion Cells; Rod Opsins; Signal Transduction; Urea | 2017 |
Blockade of the orexin receptors in the CA1 region of hippocampus decreased the lateral hypothalamic-induced antinociceptive responses in the model of orofacial formalin test in the rats.
Topics: Analgesics; Animals; Benzoxazoles; CA1 Region, Hippocampal; Facial Pain; Formaldehyde; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Urea | 2018 |
The Subthalamic Neurons are Activated by Both Orexin-A and Orexin-B.
Topics: Action Potentials; Animals; Benzoxazoles; Isoquinolines; Male; Motor Activity; Naphthyridines; Neurons; Neurotransmitter Agents; Orexin Receptors; Orexins; Pyridines; Rats, Wistar; Subthalamic Nucleus; Urea | 2018 |
Role of the orexin receptors within the nucleus accumbens in the drug priming-induced reinstatement of morphine seeking in the food deprived rats.
Topics: Animals; Benzoxazoles; Disease Models, Animal; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Food Deprivation; Isoquinolines; Male; Morphine; Morphine Dependence; Naphthyridines; Narcotics; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats, Wistar; Urea | 2018 |
Role of orexin-1 receptors in the dorsal hippocampus (CA1 region) in expression and extinction of the morphine-induced conditioned place preference in the rats.
Topics: Animals; Behavior, Animal; Benzoxazoles; CA1 Region, Hippocampal; Gene Expression Regulation; Male; Morphine; Naphthyridines; Orexin Receptors; Rats; Rats, Wistar; Urea | 2018 |
Role of dorsal hippocampal orexin-1 receptors in modulation of antinociception induced by chemical stimulation of the lateral hypothalamus.
Topics: Analgesics; Animals; Benzoxazoles; CA1 Region, Hippocampal; Carbachol; Catheters, Indwelling; Cholinergic Agonists; Dose-Response Relationship, Drug; Formaldehyde; Hypothalamic Area, Lateral; Inflammation; Male; Naphthyridines; Nociceptive Pain; Orexin Receptor Antagonists; Orexin Receptors; Pain Perception; Rats, Wistar; Stimulation, Chemical; Urea | 2018 |
Orexin 1 and orexin 2 receptor antagonism in the basolateral amygdala modulate long-term potentiation of the population spike in the perforant path-dentate gyrus-evoked field potential in rats.
Topics: Action Potentials; Animals; Basolateral Nuclear Complex; Benzoxazoles; Dentate Gyrus; Electric Stimulation; Isoquinolines; Long-Term Potentiation; Naphthyridines; Neural Pathways; Neurons; Orexin Receptor Antagonists; Perforant Pathway; Pyridines; Rats; Urea | 2018 |
Ghrelin acts centrally to induce an antinociceptive action during colonic distension through the orexinergic, dopaminergic and opioid systems in conscious rats.
Topics: Analgesics; Analgesics, Opioid; Animals; Benzoxazoles; Brain; Consciousness; Dopamine; Ghrelin; Male; Naphthyridines; Orexins; Rats, Sprague-Dawley; Receptors, Dopamine D1; Urea; Visceral Pain | 2018 |
SB-334867 (an Orexin-1 Receptor Antagonist) Effects on Morphine-Induced Sensitization in Mice-a View on Receptor Mechanisms.
Topics: Animals; Astrocytes; Benzoxazoles; Brain; Male; Mice; Microglia; Morphine; Motor Activity; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Receptor, Adenosine A1; Receptor, Adenosine A2A; RNA, Messenger; Urea | 2018 |
Sex- and Age-dependent Effects of Orexin 1 Receptor Blockade on Open-Field Behavior and Neuronal Activity.
Topics: Age Factors; Animals; Benzoxazoles; Brain; Exploratory Behavior; Female; Male; Naphthyridines; Neurons; Orexin Receptors; Rats; Rats, Sprague-Dawley; Sex Characteristics; Urea | 2018 |
Modulation by orexin A of spontaneous excitatory and inhibitory transmission in adult rat spinal substantia gelatinosa neurons.
Topics: Animals; Benzoxazoles; Dioxanes; Excitatory Postsynaptic Potentials; GABAergic Neurons; Glycine; Inhibitory Postsynaptic Potentials; Male; Naphthyridines; Neurons; Orexin Receptors; Orexins; Patch-Clamp Techniques; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Substantia Gelatinosa; Synaptic Transmission; Urea | 2018 |
Effects of intrathecal administration of orexin-1 receptor antagonist on antinociceptive responses induced by chemical stimulation of lateral hypothalamus in an animal model of tonic nociception.
Topics: Analgesics; Animals; Benzoxazoles; Hypothalamic Area, Lateral; Injections, Spinal; Male; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Rats, Wistar; Spinal Cord; Urea | 2018 |
Hypocretin/orexin antagonists decrease cocaine self-administration by female rhesus monkeys.
Topics: Animals; Behavior, Addictive; Benzoxazoles; Central Nervous System Stimulants; Cocaine; Dose-Response Relationship, Drug; Female; Macaca mulatta; Naphthyridines; Orexins; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Urea | 2018 |
Orexin-1 receptors in the rostral ventromedial medulla are involved in the modulation of capsaicin evoked pulpal nociception and impairment of learning and memory.
Topics: Animal Experimentation; Animals; Benzoxazoles; Capsaicin; Dental Pulp; Dose-Response Relationship, Drug; Male; Medulla Oblongata; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; Rats, Wistar; Sensory System Agents; Spatial Learning; Spatial Memory; Urea | 2018 |
Orexin A presynaptically decreases inhibitory synaptic transmission in rat locus coeruleus neurons.
Topics: Animals; Benzoxazoles; Dose-Response Relationship, Drug; Inhibitory Postsynaptic Potentials; Locus Coeruleus; Male; Naphthyridines; Neural Inhibition; Neurons; Orexins; Presynaptic Terminals; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Synaptic Transmission; Urea | 2018 |
Increased training compensates for OX1R blockage-impairment of spatial memory and c-Fos expression in different cortical and subcortical areas.
Topics: Animals; Benzoxazoles; Brain; Male; Maze Learning; Memory Consolidation; Memory Disorders; Naphthyridines; Orexin Receptors; Practice, Psychological; Proto-Oncogene Proteins c-fos; Psychotropic Drugs; Rats, Wistar; Reversal Learning; Spatial Memory; Urea | 2018 |
Role of orexin-1 and orexin-2 receptors in the CA1 region of hippocampus in the forced swim stress- and food deprivation-induced reinstatement of morphine seeking behaviors in rats.
Topics: Animals; Benzoxazoles; CA1 Region, Hippocampal; Drug-Seeking Behavior; Extinction, Psychological; Food Deprivation; Isoquinolines; Male; Morphine Dependence; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats, Wistar; Stress, Psychological; Swimming; Urea | 2018 |
The hypothalamic neuropeptide orexin A- a possible regulator in glucose homeostasis and germ cell kinetics in adult mice testes.
Topics: Animals; Benzoxazoles; Blotting, Western; Cell Cycle; Cell Proliferation; Cell Survival; Flow Cytometry; Glucose; Glucose Transport Proteins, Facilitative; Glucose Transporter Type 3; Homeostasis; Hypothalamus; In Situ Nick-End Labeling; L-Lactate Dehydrogenase; Male; Mice; Naphthyridines; Orexin Receptors; Orexins; Spermatozoa; Urea | 2018 |
Orexins Facilitates Osteogenic Differentiation of MC3T3-E1 Cells.
Topics: Alkaline Phosphatase; Animals; Benzoxazoles; Calcification, Physiologic; Carbazoles; Cell Differentiation; Cell Line; Core Binding Factor Alpha 2 Subunit; Culture Media; Dose-Response Relationship, Drug; Mice; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Osteoblasts; Osteogenesis; p38 Mitogen-Activated Protein Kinases; Urea | 2018 |
Activation of orexin-1 receptors in the ventrolateral periaqueductal grey matter (vlPAG) modulates pulpal nociception and the induction of substance P in vlPAG and trigeminal nucleus caudalis.
Topics: Animals; Benzoxazoles; Bicuculline; Capsaicin; Dental Pulp; Fluorescent Antibody Technique; Male; Naphthyridines; Nociception; Orexins; Periaqueductal Gray; Rats; Rats, Wistar; Substance P; Trigeminal Nuclei; Urea | 2019 |
Central Orexin A Affects Reproductive Axis by Modulation of Hypothalamic Kisspeptin/Neurokinin B/Dynorphin Secreting Neurons in the Male Wistar Rats.
Topics: Animals; Benzoxazoles; Dioxanes; Dynorphins; Gene Expression Regulation; Gonadotropin-Releasing Hormone; Hypothalamus; Injections, Intraventricular; Kisspeptins; Luteinizing Hormone; Male; Naphthyridines; Neurokinin B; Neurons; Orexins; Phenylurea Compounds; Random Allocation; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; Reproduction; Sexual Behavior, Animal; Testosterone; Urea | 2018 |
Increased Number and Activity of a Lateral Subpopulation of Hypothalamic Orexin/Hypocretin Neurons Underlies the Expression of an Addicted State in Rats.
Topics: Animals; Benzoxazoles; Cell Count; Cocaine; Drug-Seeking Behavior; Extinction, Psychological; Gene Knockdown Techniques; Hypothalamic Area, Lateral; Hypothalamic Hormones; Male; Melanins; Microinjections; Morpholinos; Motivation; Naphthyridines; Neurons; Orexins; Pituitary Hormones; Rats; Self Administration; Urea | 2019 |
Orexin 1 receptors in the anterior cingulate and orbitofrontal cortex regulate cost and benefit decision-making.
Topics: Animals; Benzoxazoles; Cost-Benefit Analysis; Decision Making; Gyrus Cinguli; Male; Motor Activity; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Prefrontal Cortex; Psychotropic Drugs; Rats, Wistar; Reward; Urea | 2019 |
Demand elasticity predicts addiction endophenotypes and the therapeutic efficacy of an orexin/hypocretin-1 receptor antagonist in rats.
Topics: Animals; Behavior, Addictive; Benzoxazoles; Cocaine; Dose-Response Relationship, Drug; Endophenotypes; Forecasting; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Sprague-Dawley; Self Administration; Treatment Outcome; Urea | 2019 |
Orexin-A signaling in the paraventricular nucleus modulates spontaneous firing of glucose-sensitive neurons and promotes food intake via the NPY pathway in rats.
Topics: Animals; Benzoxazoles; Dihydropyridines; Eating; Glucose; Male; Naphthyridines; Neurons; Neuropeptide Y; Orexin Receptors; Orexins; Paraventricular Hypothalamic Nucleus; Phenylurea Compounds; Proto-Oncogene Proteins c-fos; Rats, Sprague-Dawley; Receptors, Neuropeptide Y; Signal Transduction; Urea | 2018 |
The basolateral amygdala orexin 1 and 2 receptors' involvement in modulating spatial reference memory.
Topics: Animals; Basolateral Nuclear Complex; Benzoxazoles; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Spatial Memory; Urea | 2019 |
The effect of CA1 administration of orexin-A on hippocampal expression of COX-2 and BDNF in a rat model of orofacial pain.
Topics: Animals; Benzoxazoles; Brain-Derived Neurotrophic Factor; Capsaicin; Cyclooxygenase 2; Disease Models, Animal; Facial Pain; Hippocampus; Male; Naphthyridines; Neurons; Orexin Receptors; Orexins; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Urea | 2018 |
Co-administration of the low dose of orexin and nitrergic antagonists induces an antidepressant-like effect in mice.
Topics: Animals; Antidepressive Agents; Benzoxazoles; Depression; Dose-Response Relationship, Drug; Drug Therapy, Combination; Hindlimb Suspension; Locomotion; Male; Mice; Naphthyridines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Orexins; Swimming; Treatment Outcome; Urea | 2019 |
Hippocampal orexin receptor blocking prevented the stress induced social learning and memory deficits.
Topics: Animals; Anxiety; Benzoxazoles; Hippocampus; Isoquinolines; Male; Maze Learning; Memory; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats, Wistar; Social Behavior; Stress, Psychological; Urea | 2019 |
Orexin facilitates GABAergic IPSCs via postsynaptic OX
Topics: Animals; Animals, Genetically Modified; Benzoxazoles; Cerebral Cortex; GABAergic Neurons; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Isoquinolines; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Patch-Clamp Techniques; Protein Kinase C; Pyramidal Cells; Pyridines; Rats; Urea | 2019 |
The arousal effect of hyperbaric oxygen through orexin/hypocretin an upregulation on ketamine/ethanol-induced unconsciousness in male rats.
Topics: Animals; Arousal; Benzoxazoles; Dioxanes; Ethanol; Hyperbaric Oxygenation; Ketamine; Male; Naphthyridines; Orexin Receptor Antagonists; Orexins; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Reflex, Righting; Unconsciousness; Up-Regulation; Urea | 2020 |
The orexin-1 receptor antagonist SB-334867 reduces motivation, but not inhibitory control, in a rat stop signal task.
Topics: Animals; Benzoxazoles; Drug-Seeking Behavior; Executive Function; Inhibition, Psychological; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats, Sprague-Dawley; Reward; Urea | 2020 |
Role of orexin in exercise-induced leptin sensitivity in the mediobasal hypothalamus of mice.
Topics: Animals; Benzoxazoles; Exercise Test; Hypothalamus; Leptin; Male; Mice, Inbred C57BL; Naphthyridines; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Phosphorylation; Physical Conditioning, Animal; Receptors, Leptin; STAT3 Transcription Factor; Urea | 2019 |
The role of orexin-1 receptor signaling in demand for the opioid fentanyl.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Benzoxazoles; Conditioning, Operant; Cues; Drug-Seeking Behavior; Economics, Behavioral; Extinction, Psychological; Fentanyl; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Sprague-Dawley; Self Administration; Urea | 2019 |
Role of orexin receptors within the dentate gyrus of the hippocampus in antinociception induced by chemical stimulation of the lateral hypothalamus in the tail-flick test as a model of acute pain in rats.
Topics: Acute Pain; Analgesics; Animals; Benzoxazoles; Carbachol; Dentate Gyrus; Dose-Response Relationship, Drug; Isoquinolines; Male; Motor Activity; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pain Measurement; Pyridines; Rats; Rats, Wistar; Stimulation, Chemical; Urea | 2019 |
Role of orexin-1 and -2 receptors within the nucleus accumbens in the acquisition of sensitization to morphine in rats.
Topics: Animals; Benzoxazoles; Conditioning, Classical; Conditioning, Operant; Conditioning, Psychological; Drug Interactions; Drug Tolerance; Isoquinolines; Male; Morphine; Morphine Dependence; Naphthyridines; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pyridines; Rats; Rats, Wistar; Reward; Urea | 2019 |
Persistent effects of the orexin-1 receptor antagonist SB-334867 on motivation for the fast acting opioid remifentanil.
Topics: Analgesics, Opioid; Animals; Basal Forebrain; Benzoxazoles; Conditioning, Operant; Drug-Seeking Behavior; Male; Motivation; Naphthyridines; Rats, Sprague-Dawley; Remifentanil; Reward; Urea | 2020 |
Orexin-1 Receptor Signaling in Ventral Pallidum Regulates Motivation for the Opioid Remifentanil.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Benzoxazoles; Cues; Drug-Seeking Behavior; Economics, Behavioral; Globus Pallidus; Male; Motivation; Motor Activity; Naphthyridines; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Recurrence; Remifentanil; Reward; Urea | 2019 |
Orexin 2 receptor is involved in orexin A-induced hyperlocomotion in rats.
Topics: Aminopyridines; Animals; Benzoxazoles; Locomotion; Male; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Sulfonamides; Urea | 2019 |
Brain orexin improves intestinal barrier function via the vagal cholinergic pathway.
Topics: Animals; Antimetabolites; Atropine; Benzoxazoles; Colon; Deoxyglucose; Efferent Pathways; Intestinal Mucosa; Lipopolysaccharides; Muscarinic Antagonists; Naphthyridines; Orexin Receptor Antagonists; Orexins; Permeability; Rats; Subarachnoid Space; Urea; Vagotomy; Vagus Nerve | 2020 |
Role of orexinergic receptors in the dentate gyrus of the hippocampus in the acquisition and expression of morphine-induced conditioned place preference in rats.
Topics: Animals; Behavior, Animal; Benzoxazoles; Conditioning, Classical; Dentate Gyrus; Isoquinolines; Male; Morphine; Naphthyridines; Narcotics; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Reward; Urea | 2020 |
The role of the nucleus accumbens OXR1 in cocaine-induced locomotor sensitization.
Topics: Animals; Behavior, Animal; Benzoxazoles; Central Nervous System Sensitization; Cocaine; Dopamine Uptake Inhibitors; Locomotion; Male; Mitochondrial Proteins; Naphthyridines; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Urea | 2020 |
Targeting the orexin system for prescription opioid use disorder: Orexin-1 receptor blockade prevents oxycodone taking and seeking in rats.
Topics: Analgesics, Opioid; Animals; Benzoxazoles; Drug-Seeking Behavior; Isoquinolines; Male; Naphthyridines; Opioid-Related Disorders; Orexin Receptors; Orexins; Oxycodone; Prescription Drug Misuse; Pyridines; Rats; Rats, Wistar; Self Administration; Urea | 2020 |
The contribution of orexin receptors within the ventral tegmental area to modulation of antinociception induced by chemical stimulation of the lateral hypothalamus in the animal model of orofacial pain in the rats.
Topics: Animals; Benzoxazoles; Carbachol; Dose-Response Relationship, Drug; Facial Pain; Hypothalamic Area, Lateral; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pain Measurement; Pyridines; Rats; Urea; Ventral Tegmental Area | 2020 |
Involvement of Orexinergic System Within the Nucleus Accumbens in Pain Modulatory Role of the Lateral Hypothalamus in Orofacial Pain Model.
Topics: Analgesics, Non-Narcotic; Animals; Benzoxazoles; Carbachol; Facial Pain; Formaldehyde; Hypothalamic Area, Lateral; Isoquinolines; Male; Naphthyridines; Nociception; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats, Wistar; Urea | 2020 |
Chemical stimulation of the lateral hypothalamus induces antiallodynic and anti-thermal hyperalgesic effects in animal model of neuropathic pain: Involvement of orexin receptors in the spinal cord.
Topics: Animals; Benzoxazoles; Carbachol; Disease Models, Animal; Dose-Response Relationship, Drug; Hot Temperature; Hyperalgesia; Hypothalamic Area, Lateral; Isoquinolines; Naphthyridines; Neuralgia; Orexin Receptor Antagonists; Orexin Receptors; Pain Management; Pain Threshold; Pyridines; Rats; Rats, Wistar; Spinal Cord; Urea | 2020 |
Central neuropeptide-S administration alleviates stress-induced impairment of gastric motor functions through orexin-A.
Topics: Animals; Benzoxazoles; Gastric Emptying; Hypothalamus; Naphthyridines; Neuropeptides; Orexins; Postprandial Period; Pyloric Antrum; Rats; Restraint, Physical; Stress, Physiological; Urea; Vagus Nerve | 2020 |
Investigating the role of the amygdala orexin receptor 1 in memory acquisition and extinction in a rat model of PTSD.
Topics: Amygdala; Animals; Anxiety; Behavior, Animal; Benzoxazoles; Disease Models, Animal; Elevated Plus Maze Test; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Hypothalamus; Memory; Naphthyridines; Open Field Test; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats; RNA, Messenger; Stress Disorders, Post-Traumatic; Urea | 2020 |
Involvement of descending pain control system regulated by orexin receptor signaling in the induction of central post-stroke pain in mice.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Benzoxazoles; Brain; Brain Ischemia; Hyperalgesia; Isoquinolines; Male; Mice; Mitochondrial Proteins; Naphthyridines; Neuralgia; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Piperazines; Pyridines; Serotonin Antagonists; Signal Transduction; Urea; Yohimbine | 2020 |
Sex Differences in Demand for Highly Palatable Foods: Role of the Orexin System.
Topics: Animals; Behavior, Animal; Benzoxazoles; Eating; Economics, Behavioral; Feeding Behavior; Female; Male; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexins; Rats; Rats, Sprague-Dawley; Sex Characteristics; Urea | 2021 |
Hindbrain orexin 1 receptors blunt intake suppression by gastrointestinal nutrients and cholecystokinin in male rats.
Topics: Animals; Benzoxazoles; Chocolate; Cholecystokinin; Eating; Feeding Behavior; Male; Naphthyridines; Neurons; Nutrients; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Rats, Wistar; Rhombencephalon; Urea | 2020 |
Phospholipase Cβ3 in the hippocampus may mediate impairment of memory by long-term blockade of orexin 1 receptors assessed by the Morris water maze.
Topics: Animals; Benzoxazoles; Hippocampus; Male; Maze Learning; Memory; Naphthyridines; Orexin Receptors; Orexins; Phospholipase C beta; Rats; Rats, Wistar; Urea | 2020 |
Differential Roles of Intra-accumbal Orexin Receptors in Acquisition and Expression of Methamphetamine-Induced Conditioned Place Preference in the Rats.
Topics: Animals; Benzoxazoles; Central Nervous System Stimulants; Conditioning, Classical; Drug-Seeking Behavior; Isoquinolines; Male; Methamphetamine; Naphthyridines; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats, Wistar; Urea | 2020 |
Activation orexin 1 receptors in the ventrolateral periaqueductal gray matter attenuate nitroglycerin-induced migraine attacks and calcitonin gene related peptide up-regulation in trigeminal nucleus caudalis of rats.
Topics: Animals; Benzoxazoles; Calcitonin Gene-Related Peptide; Male; Microinjections; Migraine Disorders; Naphthyridines; Nitroglycerin; Orexin Receptor Antagonists; Orexin Receptors; Periaqueductal Gray; Rats; Rats, Wistar; Trigeminal Nuclei; Up-Regulation; Urea | 2020 |
Persistent effects of the orexin-1 receptor antagonist SB-334867 on naloxone precipitated morphine withdrawal symptoms and nociceptive behaviors in morphine dependent rats.
Topics: Animals; Behavior, Animal; Benzoxazoles; Disease Models, Animal; Morphine; Morphine Dependence; Naloxone; Naphthyridines; Narcotic Antagonists; Narcotics; Nociceptive Pain; Orexin Receptor Antagonists; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Urea | 2022 |
Chemical stimulation of the lateral hypothalamus induced seeking behaviors in rats: Involvement of orexin receptors in the ventral tegmental area.
Topics: Animals; Behavior, Animal; Benzoxazoles; Carbachol; Conditioning, Operant; Dose-Response Relationship, Drug; Exploratory Behavior; Extinction, Psychological; Hypothalamic Area, Lateral; Isoquinolines; Male; Microinjections; Muscarinic Agonists; Naphthyridines; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Reward; Stimulation, Chemical; Urea; Ventral Tegmental Area | 2020 |
Intermittent self-administration of fentanyl induces a multifaceted addiction state associated with persistent changes in the orexin system.
Topics: Animals; Benzoxazoles; Drug-Seeking Behavior; Economics, Behavioral; Fentanyl; Male; Motivation; Naphthyridines; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Self Administration; Urea | 2021 |
The lateral hypothalamus and orexinergic transmission in the paraventricular thalamus promote the attribution of incentive salience to reward-associated cues.
Topics: Animals; Benzoxazoles; Choice Behavior; Conditioning, Classical; Cues; Hypothalamic Area, Lateral; Isoquinolines; Male; Midline Thalamic Nuclei; Motivation; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Sprague-Dawley; Reward; Urea | 2020 |
The orexin receptors in the ventral tegmental area are involved in the development of sensitization to expression of morphine-induced preference in rats.
Topics: Animals; Benzoxazoles; Brain; Carbachol; Conditioning, Classical; Conditioning, Operant; Conditioning, Psychological; Drug-Seeking Behavior; Hypothalamic Area, Lateral; Isoquinolines; Male; Morphine; Naphthyridines; Nucleus Accumbens; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Pyridines; Rats; Rats, Wistar; Reward; Urea; Ventral Tegmental Area | 2020 |
Orexin-1 receptor signaling within the lateral hypothalamus, but not bed nucleus of the stria terminalis, mediates context-induced relapse to alcohol seeking.
Topics: Alcohol Drinking; Alcoholism; Animals; Behavior, Addictive; Behavior, Animal; Benzoxazoles; Conditioning, Operant; Disease Models, Animal; Lateral Thalamic Nuclei; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Punishment; Rats; Septal Nuclei; Signal Transduction; Urea | 2020 |
The modulation of the spatial reference memory by the orexinergic system of the dorsal raphe nucleus.
Topics: Animals; Benzoxazoles; Dorsal Raphe Nucleus; Male; Morris Water Maze Test; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Spatial Memory; Urea | 2021 |
Blockade of orexin receptors in the ventral tegmental area reduced the extinction period of the lateral hypothalamic-induced conditioned place preference in rats.
Topics: Animals; Benzoxazoles; Carbachol; Cholinergic Agonists; Conditioning, Classical; Dose-Response Relationship, Drug; Hypothalamic Area, Lateral; Isoquinolines; Male; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Reward; Urea; Ventral Tegmental Area | 2021 |
Central blockade of orexin type 1 receptors reduces naloxone induced activation of locus coeruleus neurons in morphine dependent rats.
Topics: Action Potentials; Analgesics, Opioid; Animals; Benzoxazoles; Injections, Intraperitoneal; Injections, Intraventricular; Locus Coeruleus; Male; Morphine; Morphine Dependence; Naloxone; Naphthyridines; Narcotic Antagonists; Neurons; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Urea | 2021 |
Blockade of orexin receptors in the hippocampal dentate gyrus reduced the extinction latency of morphine-induced place preference in male rats.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Dentate Gyrus; Drug-Seeking Behavior; Extinction, Psychological; Isoquinolines; Male; Morphine; Naphthyridines; Narcotics; Orexin Receptor Antagonists; Pyridines; Rats; Rats, Wistar; Urea | 2021 |
Wakefulness-Promoting Effects of Lateral Hypothalamic Area-Deep Brain Stimulation in Traumatic Brain Injury-Induced Comatose Rats: Upregulation of α1-Adrenoceptor Subtypes and Downregulation of Gamma-Aminobutyric Acid β Receptor Expression Via the Orexins
Topics: Anesthesia; Animals; Benzoxazoles; Brain Injuries, Traumatic; Coma; Consciousness; Deep Brain Stimulation; Delta Rhythm; Electroencephalography; Female; Functional Laterality; Hypothalamic Area, Lateral; Injections, Intraventricular; Male; Naphthyridines; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, GABA; Signal Transduction; Urea; Wakefulness | 2021 |
Orexin one receptors within the basolateral amygdala are involved in the modulation of cognitive deficits associated with a migraine-like state in rats.
Topics: Animals; Basolateral Nuclear Complex; Benzoxazoles; Cognitive Dysfunction; Male; Migraine Disorders; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Rats; Rats, Wistar; Urea | 2021 |
Role of hippocampal orexin receptors in antinociception elicited by chemical stimulation of the lateral hypothalamus in the tail-flick test.
Topics: Animals; Behavior, Animal; Benzoxazoles; CA1 Region, Hippocampal; Carbachol; Dimethyl Sulfoxide; Hypothalamic Area, Lateral; Isoquinolines; Male; Muscarinic Agonists; Naphthyridines; Nociception; Orexin Receptor Antagonists; Orexin Receptors; Pyridines; Rats; Rats, Wistar; Stimulation, Chemical; Urea | 2021 |
Similar role of mPFC orexin-1 receptors in the acquisition and expression of morphine- and food-induced conditioned place preference in male rats.
Topics: Animals; Benzoxazoles; Conditioning, Operant; Drug-Seeking Behavior; Food; Male; Morphine; Morphine Dependence; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Prefrontal Cortex; Rats; Rats, Wistar; Reward; Urea | 2021 |
The involvement of orexin 1 and cannabinoid 1 receptors within the ventrolateral periaqueductal gray matter in the modulation of migraine-induced anxiety and social behavior deficits of rats.
Topics: Animals; Anxiety; Behavior, Animal; Benzoxazoles; Male; Migraine Disorders; Naphthyridines; Orexin Receptors; Periaqueductal Gray; Piperidines; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Neuropeptide; Social Behavior; Urea | 2021 |
Orexin receptors in the CA1 region of hippocampus modulate the stress-induced antinociceptive responses in an animal model of persistent inflammatory pain.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Benzoxazoles; CA1 Region, Hippocampal; Cyclophosphamide; Disease Models, Animal; Doxorubicin; Etoposide; Inflammation; Isoquinolines; Male; Microinjections; Naphthyridines; Orexin Receptor Antagonists; Orexin Receptors; Pain; Pain Measurement; Prednisone; Pyridines; Rats, Wistar; Stress, Psychological; Urea; Vincristine | 2022 |
Intracerebroventricular infusion of the selective orexin 1 receptor antagonist SB-334867 impairs cognitive flexibility in a sex-dependent manner.
Topics: Animals; Benzoxazoles; Cognition; Female; Infusions, Intraventricular; Male; Mice; Mice, Inbred C57BL; Naphthyridines; Orexin Receptors; Orexins; Urea | 2022 |
Synergistic antidepressant effects of citalopram and SB-334867 in the REM sleep-deprived mice: Possible role of BDNF.
Topics: Animals; Antidepressive Agents; Benzoxazoles; Brain-Derived Neurotrophic Factor; Citalopram; Depression; Male; Mice; Naphthyridines; Orexins; Sleep Deprivation; Sleep, REM; Urea | 2022 |