Page last updated: 2024-08-21

benzoxazoles and proline

benzoxazoles has been researched along with proline in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's1 (25.00)18.2507
2000's0 (0.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Liberti, JP; Rogers, KS1
Evans, DB; Fan, N; Rank, KB; Sharma, SK; Tarpley, WG; Thomas, RC1
Hamilton, B; Kley, JT; Mack, J; Redemann, N; Scheuerer, S1
Jeon, J; Kim, M; Kim, YH; Lee, KO; Min, KH; Song, J; Suh, KH1

Other Studies

4 other study(ies) available for benzoxazoles and proline

ArticleYear
Inhibition of radiosulfate uptake in rat costal cartilage by lipophilic heterocyclic molecules.
    Biochimica et biophysica acta, 1970, Oct-27, Volume: 222, Issue:1

    Topics: Alcohols; Animals; Benzene Derivatives; Benzoxazoles; Carbon Isotopes; Cartilage; Chemical Phenomena; Chemistry; Chondroitin; In Vitro Techniques; Indoles; Male; Metabolism; Proline; Protein Biosynthesis; Quinolines; Rats; Skatole; Sulfates; Sulfur Isotopes; Sulfuric Acids; Surface Properties; Thiazoles

1970
Mechanism of resistance to U-90152S and sensitization to L-697,661 by a proline to leucine change at residue 236 of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase.
    FEBS letters, 1995, Feb-13, Volume: 359, Issue:2-3

    Topics: Amino Acid Sequence; Antiviral Agents; Base Sequence; Benzoxazoles; Delavirdine; DNA Primers; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Indoles; Leucine; Molecular Sequence Data; Piperazines; Point Mutation; Proline; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase

1995
Discovery of BI 99179, a potent and selective inhibitor of type I fatty acid synthase with central exposure.
    Bioorganic & medicinal chemistry letters, 2011, Oct-01, Volume: 21, Issue:19

    Topics: Administration, Oral; Animals; Benzoxazoles; Caco-2 Cells; Cell Line; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Drug Discovery; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fatty Acid Synthases; High-Throughput Screening Assays; Humans; Hypothalamus; Inhibitory Concentration 50; Injections, Intravenous; Mice; Microsomes, Liver; Molecular Conformation; Molecular Targeted Therapy; Permeability; Proline; Rats; Stereoisomerism; Structure-Activity Relationship; Substrate Specificity

2011
Synthesis of proline analogues as potent and selective cathepsin S inhibitors.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Arthritis; Benzoxazoles; Cathepsin B; Cathepsin K; Cathepsins; Collagen; Disease Models, Animal; Dogs; Enzyme Inhibitors; Half-Life; Humans; Mice; Mice, Inbred ICR; Microsomes; Proline; Protein Binding; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship

2013