benzoxazoles has been researched along with l-697661 in 22 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 21 (95.45) | 18.2507 |
2000's | 1 (4.55) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bamberger, DL; Fisher, TE; Goldman, ME; Hoffman, JM; Jones, JH; Rooney, CS; Saari, WS; Smith, AM; Thomas, CM; Wai, JS | 1 |
Condra, JH; Emini, EA; Gotlib, L; Graham, DJ; Lineberger, DW; Long, WJ; Sardana, VV; Schlabach, AJ; Wolfgang, JA | 1 |
Harris, PJ | 1 |
Bender, R; Kirsch, R; Kleim, JP; Meichsner, C; Paessens, A; Riess, G | 1 |
Carroll, SS; Culberson, JC; Kuo, LC; Olsen, DB; Shafer, JA | 1 |
Byrnes, VW; Condra, JH; Emini, EA; Sardana, VV; Schleif, WA | 1 |
Bäckbro, K; Noréen, R; Oberg, B; Unge, T; Vrang, L; Zhang, H | 1 |
Evans, DB; Fan, N; Rank, KB; Sharma, SK; Tarpley, WG; Thomas, RC | 2 |
Byrnes, VW; Emini, EA; Kessler, JA; Lineberger, DW; Massari, F; Staszewski, S; Waterbury, JA | 1 |
Anderson, KW; Bakshi, KK; Durr, S; Göhler, R; Kober, A; Massari, FE; Schneider, CL; Staszewski, S; Taylor, VI; Waterbury, JA | 1 |
Chen, S; Chopra, P; Emini, EA; Hahn, BH; Kappes, JC; McFarland, R; Piatak, M; Saag, MS; Shaw, GM; Yang, LC | 1 |
Goldman, ME; O'Brien, JA; Ostovic, D; Ruffing, TL; Schorn, TW; Siegl, PK; Smith, SJ | 1 |
Chen, IS; Dueweke, TJ; Poppe, SM; Pushkarskaya, T; Stevenson, M; Swaney, SM; Tarpley, WG; Zhao, JQ | 1 |
Byrnes, VW; Douglas, J; Emini, EA; Hildebrand, C; Kappes, JC; Lapidus, WI; Laskin, OL; Saag, MS; Schleif, WA; Whitley, RJ | 1 |
Byrnes, VW; Condra, JH; Long, WJ; Sardana, VV; Schlabach, AJ; Schleif, WA; Schneider, CL; Waterbury, JA; Wolanski, BS; Wolfgang, JA | 1 |
Davey, RT; Dewar, RL; Falloon, J; Haneiwich, SE; Kovacs, JA; Masur, H; Polis, MA; Reed, GF; Vasudevachari, MB; Walker, RE | 1 |
Blaschke, T; Campbell, TB; Collier, A; Kahn, J; Kuritzkes, DR; Messari, F; Phair, J; Pottage, JC; Rosandich, ME; Schooley, RT; Stein, DS | 1 |
Kilby, JM; Saag, MS | 1 |
Baumberger, C; Hirschel, B; Kinloch-de Loës, S; Pechère, M; Perrin, L; Rakik, A; Yerly, S | 1 |
Herold, ML; Lee, LL; Zacchei, AG | 1 |
Dornadula, G; Grobler, JA; Hazuda, DJ; Miller, MD; Rice, MR; Simcoe, AL | 1 |
2 review(s) available for benzoxazoles and l-697661
Article | Year |
---|---|
The genetic and functional basis of HIV-1 resistance to nonnucleoside reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Benzoxazoles; Clinical Trials as Topic; Drug Resistance, Microbial; Genetic Variation; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1994 |
Clinical experience with non-nucleoside reverse transcriptase inhibitors: L-697,661 and nevirapine.
Topics: Benzoxazoles; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1996 |
5 trial(s) available for benzoxazoles and l-697661
Article | Year |
---|---|
Combination therapy with zidovudine prevents selection of human immunodeficiency virus type 1 variants expressing high-level resistance to L-697,661, a nonnucleoside reverse transcriptase inhibitor.
Topics: Adult; Antiviral Agents; Base Sequence; Benzoxazoles; CD4 Lymphocyte Count; Double-Blind Method; Drug Resistance, Microbial; Drug Therapy, Combination; Female; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Male; Molecular Sequence Data; Mutation; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sequence Analysis, DNA; Zidovudine | 1995 |
Assessment of antiretroviral therapy by plasma viral load testing: standard and ICD HIV-1 p24 antigen and viral RNA (QC-PCR) assays compared.
Topics: Antiviral Agents; Benzoxazoles; Biomarkers; CD4 Lymphocyte Count; Double-Blind Method; HIV Core Protein p24; HIV Infections; HIV-1; Humans; Immunoassay; Polymerase Chain Reaction; Prospective Studies; Pyridones; Reverse Transcriptase Inhibitors; RNA, Viral; Viremia; Zidovudine | 1995 |
A short-term clinical evaluation of L-697,661, a non-nucleoside inhibitor of HIV-1 reverse transcriptase. L-697,661 Working Group.
Topics: Adult; Antiviral Agents; Base Sequence; Benzoxazoles; CD4-Positive T-Lymphocytes; DNA, Viral; Double-Blind Method; Female; Follow-Up Studies; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Leukocyte Count; Male; Molecular Sequence Data; Pyridones; Reverse Transcriptase Inhibitors; Zidovudine | 1993 |
Plasma viremia as a sensitive indicator of the antiretroviral activity of L-697,661.
Topics: Acquired Immunodeficiency Syndrome; Adult; Antiviral Agents; Benzoxazoles; beta 2-Microglobulin; Biomarkers; CD4 Antigens; Double-Blind Method; Enzyme-Linked Immunosorbent Assay; Female; HIV Core Protein p24; HIV Seropositivity; HIV-1; Humans; Male; Neoplasms; Pyridones; Time Factors; Viremia; Zidovudine | 1993 |
Phase 1 study of combination therapy with L-697,661 and zidovudine. The ACTG 184 Protocol Team.
Topics: Adult; Antipyrine; Antiviral Agents; Base Sequence; Benzoxazoles; Cross-Over Studies; DNA Primers; DNA, Viral; Drug Interactions; Drug Resistance, Microbial; Drug Therapy, Combination; Female; Genes, pol; Genotype; HIV Seropositivity; HIV-1; Humans; Male; Molecular Sequence Data; Pilot Projects; Pyridones; Reverse Transcriptase Inhibitors; Zidovudine | 1996 |
15 other study(ies) available for benzoxazoles and l-697661
Article | Year |
---|---|
Synthesis and evaluation of 2-pyridinone derivatives as HIV-1-specific reverse transcriptase inhibitors. 2. Analogues of 3-aminopyridin-2(1H)-one.
Topics: Aminopyridines; Antiviral Agents; Benzoxazoles; Cells, Cultured; HIV Reverse Transcriptase; HIV-1; Pyridones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 1992 |
Functional analysis of HIV-1 reverse transcriptase amino acids involved in resistance to multiple nonnucleoside inhibitors.
Topics: Amino Acid Sequence; Antiviral Agents; Azepines; Benzodiazepines; Benzoxazoles; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Nevirapine; Pyridines; Pyridones; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship | 1992 |
Possible toxicity associated with L-697,661 administration in a patient with AIDS.
Topics: Acquired Immunodeficiency Syndrome; Antiviral Agents; Benzoxazoles; Humans; Male; Middle Aged; Pyridones; Reverse Transcriptase Inhibitors; Ulcer | 1992 |
Mutational analysis of residue 190 of human immunodeficiency virus type 1 reverse transcriptase.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Delavirdine; DNA Mutational Analysis; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Indoles; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Pyridines; Pyridones; Quinoxalines; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Selection, Genetic; Structure-Activity Relationship | 1994 |
Effect of template secondary structure on the inhibition of HIV-1 reverse transcriptase by a pyridinone non-nucleoside inhibitor.
Topics: Animals; Antiviral Agents; Base Sequence; Benzoxazoles; DNA Primers; Electrophoresis, Polyacrylamide Gel; Globins; HIV Reverse Transcriptase; Molecular Sequence Data; Molecular Structure; Nucleic Acid Conformation; Pyridones; Rabbits; Reverse Transcriptase Inhibitors; RNA, Viral; Templates, Genetic | 1994 |
Enzymatic properties and sensitivity to inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase with Glu-138-->Arg and Tyr-188-->His mutations.
Topics: Amino Acids; Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Binding, Competitive; Deoxyguanine Nucleotides; Dideoxynucleotides; Foscarnet; HIV Reverse Transcriptase; Humans; Imidazoles; Kinetics; Molecular Sequence Data; Mutation; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sensitivity and Specificity | 1994 |
Mechanism of resistance to U-90152S and sensitization to L-697,661 by a proline to leucine change at residue 236 of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase.
Topics: Amino Acid Sequence; Antiviral Agents; Base Sequence; Benzoxazoles; Delavirdine; DNA Primers; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Indoles; Leucine; Molecular Sequence Data; Piperazines; Point Mutation; Proline; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1995 |
Turnover of circulating virion RNA and of cell-associated viral DNA reflects active viral replication in human immunodeficiency virus type 1-infected individuals.
Topics: Antiviral Agents; Benzoxazoles; Cell Compartmentation; Cell-Free System; DNA, Viral; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; RNA, Viral; Virion; Virus Replication | 1995 |
Simultaneous mutations at Tyr-181 and Tyr-188 in HIV-1 reverse transcriptase prevents inhibition of RNA-dependent DNA polymerase activity by the bisheteroarylpiperazine (BHAP) U-90152s.
Topics: Amino Acid Sequence; Antiviral Agents; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; HIV Reverse Transcriptase; HIV-1; HIV-2; Imidazoles; Indoles; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Point Mutation; Pyridines; Pyridones; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Tyrosine | 1995 |
A rapid bioassay for the determination of non-nucleoside HIV-1 reverse transcriptase inhibitor plasma levels.
Topics: Administration, Oral; Animals; Benzoxazoles; Biological Assay; Chromatography, High Pressure Liquid; HIV Reverse Transcriptase; HIV-1; Macaca mulatta; Pyridones; Reverse Transcriptase Inhibitors | 1993 |
A mutation in reverse transcriptase of bis(heteroaryl)piperazine-resistant human immunodeficiency virus type 1 that confers increased sensitivity to other nonnucleoside inhibitors.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; Drug Resistance; HIV Reverse Transcriptase; Imidazoles; Indoles; Molecular Sequence Data; Mutation; Nevirapine; Oligodeoxyribonucleotides; Piperazines; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1993 |
Comprehensive mutant enzyme and viral variant assessment of human immunodeficiency virus type 1 reverse transcriptase resistance to nonnucleoside inhibitors.
Topics: Acquired Immunodeficiency Syndrome; Antiviral Agents; Benzoxazoles; DNA, Viral; Genetic Variation; HIV Reverse Transcriptase; HIV-1; Humans; Mutation; Nucleosides; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship | 1993 |
Combined therapy with zidovudine and L-697,661 in primary HIV infection.
Topics: Adult; Anti-HIV Agents; Benzoxazoles; CD4 Lymphocyte Count; CD8-Positive T-Lymphocytes; DNA, Viral; Drug Therapy, Combination; HIV Infections; Humans; Pyridones; Reverse Transcriptase Inhibitors; RNA, Viral; Viral Load; Viremia; Zidovudine | 1996 |
High-performance liquid chromatographic method for the determination of an HIV-1 non-nucleoside reverse transcriptase inhibitor (L-696,229) in plasma samples from animals.
Topics: Animals; Antiviral Agents; Benzoxazoles; Chromatography, High Pressure Liquid; Circadian Rhythm; Cohort Studies; Female; HIV-1; Macaca mulatta; Male; Osmolar Concentration; Pyridones; Rats; Reproducibility of Results; Reverse Transcriptase Inhibitors; Spectrophotometry, Ultraviolet; Time Factors | 1996 |
HIV-1 reverse transcriptase plus-strand initiation exhibits preferential sensitivity to non-nucleoside reverse transcriptase inhibitors in vitro.
Topics: Alkynes; Anti-HIV Agents; Benzoxazines; Benzoxazoles; Cyclopropanes; DNA; Dose-Response Relationship, Drug; Drug Resistance, Viral; Enzyme Inhibitors; HIV Reverse Transcriptase; In Vitro Techniques; Inhibitory Concentration 50; Ligands; Models, Genetic; Oxazines; Pyridones; Reverse Transcriptase Inhibitors; Stochastic Processes; Transcription, Genetic; Virus Replication | 2007 |