Page last updated: 2024-08-18

benzotriazole and casein kinase ii

benzotriazole has been researched along with casein kinase ii in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (41.67)29.6817
2010's5 (41.67)24.3611
2020's2 (16.67)2.80

Authors

AuthorsStudies
Bretner, M; Duncan, JS; Graves, LM; Gyenis, L; Haystead, TA; Lenehan, J; Litchfield, DW1
Bretner, M; Kilanowicz, A; Muszyńska, G; Najda-Bernatowicz, A; Sapota, A; Łebska, M1
Bain, J; Cozza, G; Di Maira, G; Elliott, M; Kazimierczuk, Z; Meggio, F; Orzeszko, A; Pagano, MA; Pinna, LA; Ruzzene, M; Sarno, S1
Bretner, M; Kopańska, K; Krzywińska, E; Muszyńska, G; Najda-Bernatowicz, A; Orzeszko, A; Łebska, M1
Kabachinski, G; Klenchin, VA; Loyet, KM; Martin, TF; Nojiri, M1
Poznański, J; Shugar, D; Wąsik, R; Wińska, P1
Kucińska, K; Makowska, M; Poznański, J; Shugar, D; Winiewska, M1
Bugajska, E; Poznański, J; Winiewska, M1
Bretner, M; Chojnacki, K; Skierka, K; Wielechowska, M; Wińska, P1
Bretner, M; Chojnacki, K; Niefind, K; Tölzer, C; Wielechowska, M; Wińska, P; Łukowska-Chojnacka, E1
Marzec, E; Paprocki, D; Poznański, J1
Bretner, M; Kasperowicz, S; Maciejewska, AM; Marzec, E; Mieczkowska, K; Poznański, J; Trzybiński, D; Woźniak, K1

Other Studies

12 other study(ies) available for benzotriazole and casein kinase ii

ArticleYear
An unbiased evaluation of CK2 inhibitors by chemoproteomics: characterization of inhibitor effects on CK2 and identification of novel inhibitor targets.
    Molecular & cellular proteomics : MCP, 2008, Volume: 7, Issue:6

    Topics: Benzimidazoles; Casein Kinase II; Chemistry, Pharmaceutical; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Humans; Inhibitory Concentration 50; Kinetics; Models, Chemical; Mutation; Proteomics; Triazoles; Tumor Suppressor Proteins

2008
New inhibitors of protein kinase CK2, analogues of benzimidazole and benzotriazole.
    Molecular and cellular biochemistry, 2008, Volume: 316, Issue:1-2

    Topics: Benzimidazoles; Casein Kinase II; Humans; Protein Kinase Inhibitors; Triazoles

2008
The selectivity of inhibitors of protein kinase CK2: an update.
    The Biochemical journal, 2008, Nov-01, Volume: 415, Issue:3

    Topics: Animals; Benzimidazoles; Casein Kinase II; Humans; Indazoles; Jurkat Cells; Kinetics; Models, Molecular; Protein Kinase Inhibitors; Rats; Structure-Activity Relationship; Triazoles

2008
Synthesis of new analogs of benzotriazole, benzimidazole and phthalimide--potential inhibitors of human protein kinase CK2.
    Bioorganic & medicinal chemistry, 2009, Feb-15, Volume: 17, Issue:4

    Topics: Benzimidazoles; Casein Kinase II; Humans; Phthalimides; Protein Kinase Inhibitors; Structure-Activity Relationship; Triazoles

2009
CAPS activity in priming vesicle exocytosis requires CK2 phosphorylation.
    The Journal of biological chemistry, 2009, Jul-10, Volume: 284, Issue:28

    Topics: Amino Acid Sequence; Animals; Calcium; Calcium-Binding Proteins; Casein Kinase II; Chlorocebus aethiops; COS Cells; Exocytosis; Humans; Mice; Molecular Sequence Data; PC12 Cells; Phosphorylation; Rats; Sequence Homology, Amino Acid; Serine; Triazoles

2009
Synthesis and physico-chemical properties in aqueous medium of all possible isomeric bromo analogues of benzo-1H-triazole, potential inhibitors of protein kinases.
    The journal of physical chemistry. B, 2012, Jun-21, Volume: 116, Issue:24

    Topics: Bromine; Casein Kinase II; Isomerism; Protein Kinase Inhibitors; Solubility; Thermodynamics; Triazoles; Water

2012
Thermodynamics parameters for binding of halogenated benzotriazole inhibitors of human protein kinase CK2α.
    Biochimica et biophysica acta, 2015, Volume: 1854, Issue:10 Pt B

    Topics: Binding Sites; Calorimetry; Casein Kinase II; Halogenation; Humans; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Protein Kinase Inhibitors; Static Electricity; Thermodynamics; Triazoles

2015
ITC-derived binding affinity may be biased due to titrant (nano)-aggregation. Binding of halogenated benzotriazoles to the catalytic domain of human protein kinase CK2.
    PloS one, 2017, Volume: 12, Issue:3

    Topics: Binding Sites; Calorimetry; Casein Kinase II; Catalytic Domain; Halogenation; Humans; Ligands; Molecular Structure; Protein Binding; Protein Interaction Domains and Motifs; Protein Kinase Inhibitors; Spectrum Analysis; Thermodynamics; Triazoles

2017
Synthesis, in vitro antiproliferative activity and kinase profile of new benzimidazole and benzotriazole derivatives.
    Bioorganic chemistry, 2017, Volume: 72

    Topics: Antineoplastic Agents; Benzimidazoles; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Humans; Molecular Structure; Protein Kinase Inhibitors; Structure-Activity Relationship; Triazoles

2017
Biological properties and structural study of new aminoalkyl derivatives of benzimidazole and benzotriazole, dual inhibitors of CK2 and PIM1 kinases.
    Bioorganic chemistry, 2018, Volume: 80

    Topics: Benzimidazoles; Binding Sites; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Humans; Molecular Dynamics Simulation; Phosphorylation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-pim-1; Recombinant Proteins; Structure-Activity Relationship; Triazoles

2018
Thermodynamic contribution of iodine atom to the binding of heterogeneously polyhalogenated benzotriazoles by the catalytic subunit of human protein kinase CK2.
    IUBMB life, 2020, Volume: 72, Issue:6

    Topics: Casein Kinase II; Catalytic Domain; Humans; Iodine; Magnetic Resonance Spectroscopy; Thermodynamics; Triazoles

2020
A competition between hydrophobic and electrostatic interactions in protein-ligand systems. Binding of heterogeneously halogenated benzotriazoles by the catalytic subunit of human protein kinase CK2.
    IUBMB life, 2020, Volume: 72, Issue:6

    Topics: Casein Kinase II; Catalytic Domain; Crystallography, X-Ray; Humans; Hydrocarbons, Halogenated; Hydrophobic and Hydrophilic Interactions; Ligands; Protein Kinase Inhibitors; Static Electricity; Structure-Activity Relationship; Triazoles

2020