benzofurans has been researched along with styrylquinoline* in 1 studies
1 other study(ies) available for benzofurans and styrylquinoline
Article | Year |
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Synthesis of styrylbenzofuran derivatives as styrylquinoline analogues for HIV-1 integrase inhibitor.
A series of styrylbenzofuran derivatives (8a-i) as styrylquinoline isosters were efficiently prepared by Wittig reaction and evaluated for inhibitory activity against HIV-1 integrase. In this series, compounds 8g, 8h and 8i containing a free catechol ring showed moderate inhibitory activities (IC50= approximately 40 microM) against HIV-1 integrase, while less than the corresponding styrylquinoline compound (I). Topics: Benzofurans; HIV Integrase; HIV Integrase Inhibitors; Quinolines | 2003 |